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7951602 |
Mass defect labeling and methods of use thereof
Mass defect labeled peptides and methods of identifying peptides are provided. In particular, embodiments of the present disclosure include mass defect labels for polypeptides that include at least...
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7709548 |
Method for manufacturing monosulfonium salt, cationic polymerization initiator, curable composition, and cured product
A monosulfonium salt in which very little unreacted raw material remains, which has a purity of at least 96%, and which has one sulfonio group in its molecule is manufactured without a refining...
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7659317 |
Methods to prepare carbon-isotope labeled organohalides with high specific radioactivity from carbon-isotope monoxide
Methods and reagents for labeling synthesis of organohalides by transition metal mediated carbonylation reactions using carbon-isotope labeled carbon monoxide are provided. The resultant...
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7339081 |
Route to prepare 4-bromo-1-oxypentafluorosulfanylbenzene
A process for preparing bromo-1-oxypentafluorosulfanylbenzene is provided, the process including the step of brominating pentafluorosulfanyloxybenzene with a bromination agent to provide the...
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7323602 |
Preparation process of some halogeno-substituted monosulfides and their hydroxy-monosulfide or isothiouronium bromide equivalents as intermediates
A process for preparing an intermediate compound of formula (II) where n is an integer of from 3 to 14; R1 is haloC1-10alkyl, C1-10alkyl, C2-10alkenyl, C2-10cycloalkyl, carboxyC1-10alkyl,...
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7087789 |
Methods for nucleophilic fluoromethylation
A novel, convenient and efficient method for trifluoromethylation of substrate compounds is disclosed. Particularly, alkoxide and hydroxide induced nucleophilic trifluoromethylation of carbonyl...
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7087764 |
Process for producing arylsulfenyl halide
A process for producing a compound of the formula (II): wherein Hal1 represents halogen and R1 and R2 each independently represents halogen, alkyl, alkoxy, nitro or cyano, which comprises allowing...
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6770776 |
Synthesis of fluorocarbon compounds
Fluorocarbon compounds are synthesized by reacting a substrate hydrocarbyl compound containing at least one sp3-hybridized halophoric carbon atom bearing at least two halogen atom substituents, at...
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6596905 |
Method for preparing aromatic diphenyl thioethers
The invention concerns a method for preparing aromatic diphenyl thioethers. More particularly the invention concerns the preparation of 4-chloro-4′-thiomethyldiphenylether. The inventive method f...
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6518460 |
Processes for preparing 3-arylsulfur hydroxamic acids
This invention provides processes for the preparation of a compound of Formula I: Y—C(═O)—C(R1)(R2)—CH2—S(O)nR3 wherein:Y is hydroxy or XONX, where each X is independently hydrogen, lower alkyl or ...
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6506286 |
Reactant, compound and process for the perfluoroalkylation of a nucleophile, and the derivatives obtained
A reagent comprising a compound of formula (I): Rf—M(X)(Z)n—Y—R, wherein R is a hydrocarbon radical advantageously having at most 10 carbon atoms and being selected from alkyls and aryls; Rf is a ...
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6379590 |
Method for making unsymmetrically substituted fluorenyl compounds for nonlinear optical applications
A new method for producing unsymmetrically substituted fluorenyl compounds, one step of which is the preparation of 2,7-disubstituted fluoren-9-one derivatives via the nucleophilic substitution of...
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6369275 |
Process for making diaryl pyridines useful as cox-2 inhibitors
The invention encompasses a process for making compounds of Formula I useful in the treatment of cyclooxygenase-2 mediated diseases.
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6326519 |
Diallylic sulfides and processes for preparing the same
Diallylic sulfides represented by Formula I ##STR1##wherein: R1 and R2 are independently chosen from the group consisting of --CHO, --CH2 Cl, --CH2 Br, --CH2 I, --CH2 OH, CH2 OSO2 CF3, --CH2 OSO2...
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6326337 |
Perfluoropolyalkylether lubricant formulation with improved stability
An oxidation-corrosion additive for enhancing the stability of PFPAEs which has the formula: ##STR1##wherein Q is --Rf or --S--Rf, Rf is a perfluoroalkyl or perfluoroalkylether group having 1 to 30...
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6225505 |
Trifluoro methylthiomethyl benzene derivatives and process for production same
The present invention lies in a process for producing a trifluoromethylthiomethylbenzene derivative represented by the following general formula (2): ##STR1##(wherein R is a hydrogen atom, a...
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RE37087 |
Insecticidal triffluormethyl alkane derivatives
There are provided new alkane and alkoxyalkane derivatives of the general formula I ##STR1##in which R1, R2, R3, R4 and A have the meanings given in the description, processes for their preparation...
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6175042 |
Process for preparing perfluoroalkyl aryl sulfides and novel perfluoroalkyl aryl sulfides
This invention relates to a process for preparing perfluoroalkyl aryl sulfides by reaction of disulfides with alkali metal salts of aliphatic perfluorocarboxylic acids in the presence of a...
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6140515 |
Process of making 3-aryloxy, 4-aryl furan-2-ones useful as inhibitors of COX-2
Described is a process of preparing 3-aryl, 4-aryloxy furan-5-ones which are useful as inhibitors of cyclooxygenase-2 (COX-2). Such compounds are useful as anti-inflammatory agents. The process is...
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6121496 |
Aromatic thioether acylation method
The present invention relates to a process for the acylation of an aromatic thioether. In its preferred variant, the invention resides in a process for the condensation of acetic anhydride or...
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6080790 |
Tri-substituted phenyl derivatives and processes for their preparations
Compounds of formula (1) ##STR1## are described wherein Y represents a halogen atom or a group --OR1, where R1 is an optionally substituted alkyl group; R2 represents an optionally substituted...
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5998667 |
Substituted biphenyl oxazolines
The invention relates to new substituted biphenyloxazolines of the formula (I) ##STR1## in which R1 represents C1 -C6 -halogenoalkylthio and R2 represents hydrogen, or R1 and R2 together with the...
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5962483 |
Trisubstituted phenyl derivatives and processes for their preparation
Compounds of general formula (1) ##STR1## are described wherein Y is a halogen atom or a group --OR1, where R1 is an optionally substituted alkyl group; X is --O--, --S-- or --N(R7)--, where R7 is...
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5942648 |
Naphthalene derivatives
Naphthalene derivatives of the fomula I ##STR1## in which: R1 is an alkyl or alkenyl radical which is unsubstituted, monosubstituted by CH or CF3 or monosubstituted by halogen and has 1 to 15...
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5907063 |
Aromatic bromination process
Activated aromatic compounds are more economically ring brominated by reacting the compounds with a sulfoxide/HBr brominating agent while removing water from the reaction mixture. The water removal...
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5874656 |
Process for preparing o-alkylfluorobenzenes
o-Alkylfluorobenzenes are advantageously prepared by heating the corresponding chloroformates to from 70° to 200° C. in the liquid phase in the presence of hydrogen fluoride and in the presence o...
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5861540 |
Substituted 1,1,1-triaryl-2,2,2-trifuoroethanes and processes for their synthesis
Synthetic procedures to tetraalkyls, tetraacids and dianhydrides substituted 1,1,1-triaryl-2,2,2-trifluoroethanes which comprises: (1) 1,1-bis(dialkylaryl)-1-aryl-2,2,2 -trifluoroethane, (2)...
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5808164 |
Process for producing aromatic sulfides
A process which can be used to produce an aromatic sulfide compound having the formula of (R4-n)(Xn)(W)Ar--S--R' is provided. The process comprises contacting, in the presence of a surfactant, a...
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5798396 |
Sulfonium salt-containing compounds and initiators of polymerization
The present invention is directed to sulfonium salt-containing compounds represented by a following general formula; ##STR1## wherein R1 is alkyl containing from 1 to 18 carbon atoms, hydroxy,...
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5760269 |
4,4,4-Trichlorobutyl methanesulfonate
The invention provides the novel compound 4,4,4-trichlorobutyl methanesufonate, useful as an intermediate in the production of certain agricultural pesticides, and a process for its manufacture.
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5756849 |
Process for grafting a substituted difluoromethyl group onto a compound containing an electrophilic functional group
The invention relates to a process and a nucleophilic reagent which is useful for grafting a substituted difluoromethyl group onto a compound containing at least one electrophilic function,...
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5731477 |
Method for synthesis of aryl difluoromethyl ethers
This invention relates to a method for preparing difluoromethyl ethers, thiols and amines without using chlorofluorocarbon gases. The intermediates prepared by this method can be used to make...
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5639887 |
MDR reversal agents
Compounds of the general formula: ##STR1## wherein R1, R2, R3, R4 and R5 are herein described, A is a straight or branched (C2 -C12)alkyl or a phenyl moiety and B is a moiety of the formula:...
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5557008 |
Process for the introduction of fluoro substituents
A one pot process for the perfluoroalkylation and/or perfluoroacyloxylation of organic substrates is provided. The process comprises contacting a substrate with a perfluoroalkanoic anhydride in the...
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5534634 |
Process for preparing trifluoroethyl sulfur compounds from thiolates and 1-chloro-2,2,2-trifluoroethane
Process for preparing trifluoroethyl sulfur compounds from thiolates and 1-chloro-2,2,2-trifluoroethane. The invention relates to the preparation of trifluoroethyl sulfur compounds of the formula...
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5534557 |
Onium salt, photopolymerization initiator, energy ray-curing composition containing the initiator, and cured product
The composition of the present invention is excellent in compatibility, transparency and curability and give a cured coat of excellent gloss and of less smell, and cured products of excellent...
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5498730 |
Fluorinated alkyl compound derivatives and process for preparing same
The present invention provides fluorinated alkyl compound derivatives represented by formula of: ##STR1## wherein: R is C2-4 lower alkyl, cyclohexyl or thiophene; phenyl substituted with hydrogen,...
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5492917 |
Endothelin antagonists incorporating a cyclobutane
Novel compounds of the general structural formula I: ##STR1## have endothelin antagonist activity and are therefore useful in treating cardiovascular disorders, such as hypertension, pulmonary...
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5478959 |
Method for preparing 1,2-dithiins and precursors of 1,2-dithiins
A method for preparing 1,4-(Z,Z)-disubstituted-1,4-disulfurated-1,3-butadienes is disclosed. The butadienes can be further elaborated to provide 3,6-unsymmetrically-substituted-1,2-dithiins. Also...
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5463088 |
Process for preparing perfluoroalkoxy (alkylthio) benzenes
A process for preparing perfluoroalkoxy(alkylthio)benzenes from perfluorochloroalkoxy(alkylthio)-benzenes by reaction with hydrogen fluoride in the gas phase and in the presence of a catalyst.
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5463138 |
Process for preparing difluoromethoxyarenes and difluoromethylthioarenes
Difluoromethoxyarenes and difluoromethylthioarenes of the general formula (I), Ar--Q--CHF2 (I)in which Ar represents optionally substituted aryl, and Q represents oxygen or sulphur,(which can be...
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5449801 |
Reactive distillation process for free radical halogenation
A process for the selective high yield halogenation R--CH3 wherein R is ##STR1## Si(Cl)m (CH3)n, wherein m is 1 to 3, n is 1 to 3 and m+n is 3; phenyl; or phenyl substituted with Cl, Br, F, OR1,...
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5446186 |
Structure and synthesis of nitrophenyl-EGTA, a caged calcium, intermediates thereof and a method of producing a high photochemical yield of liberated calcium
The synthesis and compound of a new caged calcium which is an ortho-nitrophenyl derivative of EGTA and various intermediates. It is synthesized in ten steps and 24% overall yield. The...
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5393776 |
Tocotrienol analogs in the treatment of hypercholesterolemia and hyperlipidemia
This invention relates to structurally novel acyclic tocotrienol analogs, which are useful for cholesterol/lipid lowering in cases of hypercholesterolemia and hyperlipidemia, and for...
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5382686 |
Process for preparing nitrodiphenyl (thio) ethers
Nitrodiphenyl(thio) ethers in which the nitro group is in the ortho- or para-position with respect to the ether oxygen or ether sulphur can be prepared from halonitrobenzones in which the nitro...
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5380923 |
Polymeric sulfonium salts and method of preparation thereof
Polymeric triarylsulfonium salts are provided having a repeating structural unit with the formula: ##STR1## where R represents a substituted or unsubstituted aryl group, X- represents a...
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5321046 |
Hypocholesterolemic unsymmetrical dithiol ketals
Disclosed herein are novel unsymmetrical dithiol ketals which are useful in the treatment or prevention of hypercholesterolemia, hyperlipoproteinemia, and atherosclerosis.
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5302757 |
Ultraviolet light sensitive onium salts
A composition of matter including an onium salt and a method of forming images. The onium salt has a chromophore which absorbs ultraviolet radiation, an S, Se, As, N or P atom which is free of...
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RE34423 |
Substituted benzenes useful as intermediates
A process for producing a 4-benzoyl-5-hydroxylpyrazole of the formula III: ##STR1## which comprises reacting carbon monoxide and a 5-hydroxypyrazole of the formula II: ##STR2## with a substituted...
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5231221 |
Process for the preparation of acylals
Compounds of the formula ##STR1## can advantageously be prepared by reacting compounds the formula II ##STR2## in which the substituents R1 -R4 have the meanings given, with the anhydride of the...
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