Patents in Class 564/440

Matches 1 - 50 out of 333

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Match	Document	Document Title
1	7449594	Process for preparing 4-pentafluorosulfanylbenzoylguanidines A process for preparing 4-pentafluorosulfanylbenzoylguanidines of formula I wherein R1 to R4 have the meanings indicated in the specification. The compounds of formula I are NEH1 inhibitors and...
2	7446226	Capsaicin derivates and the production and use thereof The invention relates to new compounds, namely capsaicin derivates, a new method for their production, and their use as micro-organism-repellent agents in paints and coatings, in particular for...
3	7365231	Compound with antitumor activity and preparation method therefor The present invention provides the diaminophenyladamantane derivatives with antitumor activities and the preparation method therefore. The method includes a step of reacting an aromatic diol with...
4	7351389	Aminocarboxylate ligands having substituted aromatic amide moieties Novel metal-chelate complexes comprising aminocarboxylate ligands including substituted aromatic amide moieties, such as those having the formula wherein R 13 , A 1 , R 1 and R 2 are as...
5	7347879	Sulfur-containing secondary para-phenylenediamines dye compositions comprising such para-phenylenediamines, processes, and uses thereof The present disclosure relates to a novel family of sulfur-containing secondary para-phenylenediamines, to processes for preparing them, to compositions for dyeing keratin fibers, for example...
6	7338958	Sulfoximine-substituted pyrimidines as CDK-and/or VEGF inhibitors, their production and use as pharmaceutical agents This invention relates to pyrimidine derivatives of general formula I in which Q, R 1 , R 2 , R 3 , R 4 , R 5 , X, and m have the meanings that are contained in the description, as inhibitors...
7	7297820	Stilbene derivatives and their use for binding and imaging amyloid plaques This invention relates to a method of imaging amyloid deposits and to labeled compounds, and methods of making labeled compounds useful in imaging amyloid deposits. This invention also relates to...
8	7196229	Benzoylcyclohexenone derivatives The invention relates to benzoylcyclohexenone derivatives of general formula (I) wherein the variables R 1 to R 10 and n have the designation cited in claim 1 . The invention also relates to the...
9	7015176	Process for the synthesis of aryl sulfurpentafluorides A process is described for the synthesis of an aryl sulfur pentafluoride compound. In one embodiment of the present invention, there is provided a process for preparing an aryl sulfurpentafluoride...
10	6989036	Reactive dyes and use thereof for dyeing substrates containing nucleophilic groups The present invention relates to novel reactive dyes of the formula (I) where R 1 to R 4 are independently hydrogen, C 1 –C 8 -alkyl, C 2 –C 8 -alkyl, wherein nonadjacent CH 2 groups may...
11	6806388	Polyfluorinated aromatic or heterocyclic derivatives with sulphurpentalfluoride group(s) The invention provides polyfluorinated aromatic or heterocyclic compounds comprising at least three ring substituents, at least one of which comprises a sulfurpentafluoride group and at least one...
12	6780891	Tramadol analogs and uses thereof Compounds of formula I are effective in treating disorders modulated by opiate receptor activity and/or monoamine activity. In formula I, R 1 is selected from alkyl, aryl, alkylaryl,...
13	6747149	Glucamine salts for treating hepatitis virus infections N-Substituted glucamine compounds of formula I are effective in treatment of hepatitis infections, including hepatitis B and hepatitis C. In treating hepatitis infections the compounds of formular...
14	6677380	Substituted N, N-disubstituted mercapto amino compounds useful for inhibiting cholesteryl ester transfer protein activity The invention relates to substituted polycyclic aryl and heteroaryl tertiary-heteroalkylamine compounds useful as inhibitors of cholesteryl ester transfer protein (CETP; plasma lipid transfer...
15	6489511	Azomethine compound manufacture Disclosed is a process for forming an azomethine compound, comprising: (a) reacting a compound “A” having an active methylene group or methine group with an arylprimaryamine compound “B”;...
16	6486351	Method for condensation of aromatic derivative(s) and a sulphinic derivative The invention concerns a method for the condensation of aromatic derivative(s) or a sulphinic derivative by a perhalogenated, advantageously perfluorinated, carbon atom. Said method is...
17	6476248	Hydroxythiol grignard reaction synthesis A method for the preparation of hydroxythiol compounds by reacting a hydroxyl-protected halide compound having the structure: X—R—OPg with magnesium in a Grignard-suitable solvent to form a...
18	6433021	Indane compounds and their pharmaceutical use Indane compounds of general formulae (1) to (4) and their pharmaceutical use, particularly to achieve mast cell stabilising activity and/or anti-inflammatory activity are described. In these...
19	6372945	Process for the synthesis of vinyl sulfoxides The present invention is directed to a new process for the synthesis of vinyl sulfoxides, in particular diarylvinyl sulfoxides
20	6344558	1-phenyl-3-dimethylaminopropane compounds with a pharmacological effect 1-phenyl-3-dimethylaminopropane compounds corresponding to the formula I a method of preparing them, and the use of these substances as analgesic active ingredients in pharmaceutical compositions.
21	6320079	Process for the preparation of S(ω-aminoalkylamino) alkyl aryl sulfide dihydrochlorides A process for preparing S-(ω-aminoalkylamino) alkyl aryl sulfide dihydrochlorides includes the steps of (a) reacting aryl mercaptan and (ω-aminoalkylamino) alkylbromide dihydrobromide to cause...
22	6313348	Crosslinking aromatic diamines for polyimide optical alignment layers The invention provides novel crosslinking aromatic diamines useful in preparing polyamic acids and polyimides for optical alignment layers. The novel compositions comprise crosslinking diamines...
23	6306179	Method for the synthesis of 2-hydroxyalkyl-para-phenylenediamines, new 2-hydroxyalkyl-para-phenylenediamines, their use for oxidation dyeing, dyeing compositions and methods of dyeing The present invention relates to a new method for the synthesis of 2-hydroxyalkyl-para-phenylenediamines which are substituted or unsubstituted at the 5-position of the benzene ring, new...
24	6291702	Azulenyl nitrone spin trapping agents, methods of making and using same The present invention relates to chromotropic nitrone spin trapping agents, methods of making these agents, compositions comprising same, and methods of their use. In particular, azulenyl nitrones...
25	6262277	Intermediates and processes for the preparation of benzothiepines having activity as inhibitors of ileal bile acid transport and taurocholate uptake Provided are novel benzothiepines, derivatives, and analogs thereof; pharmaceutical compositions containing them; and methods of using these compounds and compositions in medicine, particularly in...
26	6175042	Process for preparing perfluoroalkyl aryl sulfides and novel perfluoroalkyl aryl sulfides This invention relates to a process for preparing perfluoroalkyl aryl sulfides by reaction of disulfides with alkali metal salts of aliphatic perfluorocarboxylic acids in the presence of a...
27	6169206	4-(n,n-dialkylamino)aniline compound, photographic processing composition containing the same and color image-forming method 4-(N,N-Dialkylamino)aniline compounds of the following general formula (I): ##STR1## wherein R 1 represents an alkyl group, an aryl group or a heterocyclic group, R 2 to R 5 each represent a...
28	5973178	Dye intermediates A compound of the formula: ##STR1## wherein: A is hydrogen, a substituted or unsubstituted C 1 to C 4 alkyl, a substituted or unsubstituted C 1 to C 4 alkoxy or a substituted or unsubstituted...
29	5959152	Substituted benzenedithiol metal complex A novel substituted benzenedithiol metal complex represented by the general formula (1) is provided. The substituted benzenedithiol metal complex is useful as a singlet oxygen quencher and as an...
30	5874618	2-nitro-para-phenylenediamines substituted by sulphur in the 5-position, the process for their preparation, dyeing compositions in which they are present and their use in the dyeing of keratin fibers Novel nitrobenzene compounds of the nitroparaphenylene-diamine type substituted by sulphur in the 5-position are disclosed. These compounds are intended especially for the dyeing of keratin fibers...
31	5872300	Process for the preparation of 2-amino-6-chlorophenyl-alkylsulfanes, and 2-amino-6-chlorophenyl-isopropylsulfane 2-Amino-6-chlorophenyl-alkylsulfanes are prepared in a particularly advantageous manner by hydrogenating 2-chloro-6-nitrophenyl-alkylsulfanes catalytically in the presence of a solvent without the...
32	5869506	Fluoropropene compound, an insecticide containing the same and an intermediate for production thereof The present invention provides a fluoropropene compound represented by Formula I: ##STR1## wherein R 1 represents a C 1 -C 10 alkyl group or other groups, Z represents an oxygen atom or other...
33	5854409	Pro-thiol aryl azide labelling of nucleic acids Reagents and methods for multi-step labeling of nucleic acids allow the addition of relatively insoluble or unstable labels to nucleic acid in the final step. Nucleic acids can be stored as a...
34	5840984	Stabilization of (hydrocarbylthio) aromatic amines against odor formation Odor formation during storage of (hydrocarbylthio)aromatic amines due to formation and release of odoriferous sulfur-containing species such as dihydrocarbyldisulfides, is suppressed. To accomplish...
35	5801201	1-phenyl-2-dimenthylaminomethyl-cyclohexan-1-ol compounds as pharmaceutical active ingredients 1-phenyl-2-dimethylaminomethyl-cyclohexan-1-ol compounds, methods of preparing them and the use of these compounds in drugs are described.
36	5696167	4-mercaptobenzoylguanidine derivatives 4-Mercaptobenzoylguanidines of the formula I ##STR1## in which A, R 1 , R 2 and R 3 have the meanings given, and the physiologically unobjectionable salts thereof exhibit antiarrhythmic...
37	5686642	Compounds useful for the preparation of bi-and polyfunctional reactive dyestuffs Reactive dyestuffs which, in the form of the free acid, correspond to the following formula ##STR1## wherein D is the radical of an organic dyestuff of the mono-azo, polyazo or metal complex azo...
38	5672759	Dye composition for keratinic fibres containing sulfured metaphenylenediamines, dyeing process and new sulfured metaphenylenediamines and preparation method thereof The invention relates to a dye composition for keratinic fibers comprising an oxidation colorant precursor of the type ortho and/or para and a sulfured metaphenylenediamine having formula (I)...
39	5652271	Therapeutic agents Compounds of formula I ##STR1## and pharmaceutically acceptable salts thereof in which m is 0, 1 or 2; n is 2, 3, 4 or 5; X is carbonyl or a group of formula II ##STR2## in which R 5 is H or...
40	5616809	Sulfated metaaminophenol compounds Sulfated metaaminophenols are disclosed and have the formula ##STR1## where: Z is alkyl, aralkyl, monohydroxyalkyl, polyhydroxyalkyl, aryl, aminoalkyl; R 1 is hydrogen, alkyl, monohydroxyalkyl,...
41	5599813	Thiazolopyrimidine derivatives Thiazolopyrimidine derivatives represented by the formula ##STR1## and salts thereof are provided, which are characterized by a carboxamide residue substituted with R 4 and R 5 . The derivatives...
42	5585522	Amino substituted bishalomethyl benzene compounds Novel amino substituted bishalomethyl benzene compounds, which are precurs to phenylene polymers are disclosed having non-linear optical properties, and which can be converted to electrically...
43	5510532	Stable conducting polymer and processes for the preparation thereof Conductive polymers having repeating units of formula (II) ##STR1## formed by chemical or electrochemical oxidation of aniline derivatives of formula (I) ##STR2## wherein R 1 denotes --(CH 2 ) n ...
44	5484953	O-phenylenediamines containing fluoroalkyl(ene) groups Novel o-phenylenediamines of the formula containing fluoroalkyl(ene) groups ##STR1## in which the symbols used have the meaning given in the description, processes for their preparation and their...
45	5466871	Process for preparing nitroaniline derivatives A process for preparing a nitroaniline derivative comprising a step of reacting an aromatic nitro compound with an O-alkylhydroxylamine or a salt thereof in the presence of a base and optionally a...
46	5446134	Bis(perfluorosulfonyl)methane salts, and a process for preparing same Bis(perfluorosulphonyl)methanes, process for preparing same and uses thereof. The compounds of the invention are based on the formula (1/nM)+[(R F SO 2 ) 2 CY] - in which Y denotes an...
47	5414131	Process for preparing [5-amino-2-(2-hydroxyethylamino)-phenyl](2-hydroxyethyl)sulphone A process for preparing the sulphone of the formula ##STR1## consists in reductive cleavage of disazo/disazoxy dyestuffs of the formula ##STR2## in which B is a direct bond or a bridging member and...
48	5410081	Process for the preparation of amino-substituted thioethers Compounds of the formula (I) ##STR1## are prepared by reacting 2-mercaptoethanol with compounds of the general formula (II) ##STR2## the substituents having the definition given in the description.
49	5405947	Triazine ring-containing reactive dyestuffs, their preparation and use Reactive dyestuffs which, in the form of the free acid, have the following formula ##STR1## in which X denotes fluorine, chlorine or bromine and SO 2 -Z denotes a specific reactive radical, the...
50	5393776	Tocotrienol analogs in the treatment of hypercholesterolemia and hyperlipidemia This invention relates to structurally novel acyclic tocotrienol analogs, which are useful for cholesterol/lipid lowering in cases of hypercholesterolemia and hyperlipidemia, and for...

Matches 1 - 50 out of 333

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