Patents in Class 564/381

Matches 1 - 50 out of 145

1 2 3 >

Match	Document	Document Title
1	7589127	Aminoalkylphenols, methods of using and making the same The present invention relates to Mannich base antimalarial aminoalkylphenol compounds and their use against protozoa of the genus Plasmodium , particularly emerging strains of drug-resistant...
2	6861561	Substituted aromatic policyclic tertiary-heteroalkylamines useful for inhibiting cholesteryl ester transfer protein activity The invention relates to substituted aromatic polycyclic tertiary-heteroalkylamine compounds useful as inhibitors of cholesteryl ester transfer protein (CETP; plasma lipid transfer protein-I) and...
3	6852891	Method of inhibiting methaphetamine synthesis A method of inhibiting or preventing the use of anhydrous ammonia as a solvent in a dissolving metal reduction process comprises adding to anhydrous ammonia a chemical reagent which is capable of...
4	6803466	HIV/FIV protease inhibitors having a small P3 residue With the help of X-ray structural analyses of drug-resistant HIV proteases and molecular modeling, a new type of inhibitor with a small P3 residue has been developed. These inhibitors are effective...
5	6765023	Use of substituted N, N-disubstituted reverse aminoalcohol compounds useful for inhibiting cholesteryl ester transfer protein activity The invention relates to substituted polycyclic aryl and heteroaryl tertiary-heteroalkylamine compounds useful as inhibitors of cholesteryl ester transfer protein (CETP; plasma lipid transfer...
6	6723753	Substituted n-benzyl-n-phenyl aminoalcohol compounds useful for inhibiting cholesteryl ester transfer protein activity The invention relates to substituted polycyclic aryl and heteroaryl tertiary-heteroalkylamine compounds useful as inhibitors of cholesteryl ester transfer protein (CETP; plasma lipid transfer...
7	6723752	(R)-chiral halogenated substituted n-benzyl-n-phenyl aminoalcohol compounds useful for inhibiting cholesteryl ester transfer protein activity The invention relates to substituted aryl and heteroaryl (R)-Chiral Halogenated 1-Substitutedamino-(n+1 )-Alkanol compounds useful as inhibitors of cholesteryl ester transfer protein (CETP; plasma...
8	6683113	(R)-chiral halogenated substituted N,N-Bis-benzyl aminioalcohol compounds useful for inhibiting cholesteryl ester transfer protein activity The invention relates to substituted aryl and heteroaryl (R)-Chiral Halogenated 1-Substitutedamino-(n+1)-Alkanol compounds useful as inhibitors of cholesteryl ester transfer protein (CETP; plasma...
9	6683099	Substituted N,N-disubstituted cycloalkyl aminoalcohol compounds useful for inhibiting cholesteryl ester transfer protein activity The invention relates to substituted polycyclic aryl and heteroaryl tertiary-heteroalkylamine compounds useful as inhibitors of cholesteryl ester transfer protein (CETP; plasma lipid transfer...
10	6677380	Substituted N, N-disubstituted mercapto amino compounds useful for inhibiting cholesteryl ester transfer protein activity The invention relates to substituted polycyclic aryl and heteroaryl tertiary-heteroalkylamine compounds useful as inhibitors of cholesteryl ester transfer protein (CETP; plasma lipid transfer...
11	6482859	Microbicidal N-sulfonylglycin alkynyloxyphenethyl amide derivatives The invention relates to novel pesticidally active compounds of the general formula I as well as possible isomers and mixtures of isomers thereof, wherein n is a number zero or one; and R 1 is...
12	6469005	Propargylether derivatives Propargylether derivatives of formula I including the optical isomers thereof and mixtures of such isomers, wherein R 1 is hydrogen, alkyl, cycloalkyl or optionally substituted aryl, R 2 and R...
13	6399828	Preparation of amphetamines from phenylpropanolamines A process for making compound of formula I from a phenylpropanolamine salt of formula II wherein: R 1 is hydrogen or a lower alkyl group; each R 2 is independently a hydrogen, halogen, lower...
14	6277849	N-sulphonyl and N-sulphinyl amino acid amides as microbiocides The invention relates to novel pesticidally active compounds of the general formula I ##STR1## as well as possible isomers and isomeric mixtures thereof, wherein n is a number zero or one; and ...
15	RE37087	Insecticidal triffluormethyl alkane derivatives There are provided new alkane and alkoxyalkane derivatives of the general formula I ##STR1## in which R 1 , R 2 , R 3 , R 4 and A have the meanings given in the description, processes for their...
16	6127550	Stereospecific preparation of chiral 1-aryl-and 1-heteroaryl-2-substituted ethyl-2-amines This invention is directed to methods for stereospecifically preparing [(1-optionally substituted aryl)- or (1-optionally substituted heteroaryl)]-2-substituted ethyl-2-amines, having chirality at...
17	6087346	Sigma receptor ligands and the use thereof
18	6046351	Process for preparing racemic phenethylamines
19	5976812	Activated amphetamines The invention concerns activated amphetamine derivatives, a process for their production as well as their use for producing immunogens or detection conjugates carrying amphetamine groups. A further...
20	5969186	Process for racemizing of optically active amines The present invention provides a process for effectively racemizing an amine compound in which an asymmetric carbon is located at the β-position of the amino group or more distant therefrom, which...
21	5847216	Preparation of selegiline A process for preparing selegiline hydrochloride by reaction of R-(-)-N,α-dimethylphenylethylamine with 3-bromo-1-propyne is described, which consists in reacting the substances in a molar ratio...
22	5808156	Process for the production of the isomers (R) and (S)-α-methyl-3(trifluoromethyl)benzeneethanamine Process for the production of the isomers (R) and (S)-α-methyl-3-(trifluoromethyl)benzeneethanamine, the second being useful as intermediate in the synthesis of the anorexic drug dexfenfluramine...
23	5527830	Drugs for the treatment of cardiac arrest and other shock states The invention relates to new drugs for augmenting perfusion pressure administered during cardiopulmonary resuscitation and other shock states. The compounds include phenylethanolamines and...
24	5470997	Amphetamine derivatives and protein and polypeptide amphetamine derivative conjugates and labels The present invention is directed to novel amphetamine derivatives which are synthesized for the covalent attachment to antigens (proteins or polypeptides) for the preparation of antibodies or...
25	5449828	Process for the preparation of propargyl ammonium-chloride The present invention relates to a process for the preparation of L-isomer of propargyl-ammonium-chloride derivatives of the formula (I) ##STR1## by decomposing D-tartarte of L-isomer of the amine...
26	5442120	Production of dobutamine compounds The invention relates to a process for the production of an acid addition salt of a dobutamine compound of the general formula ##STR1## wherein R is a hydrogen atom or a methyl group, and n is 1 or...
27	5292956	Hydroxyphenyl-substituted amine antioxidants Tertiary amines corresponding to the formula Z 2 Z'N in which Z is a 3,5-dihydrocarbyl-4-hydroxyphenalkyl group having the structure: ##STR1## wherein R is hydrogen or an alkyl group of 1-3...
28	5274002	Trisubstituted phenyl analogs having activity for congestive heart failure Novel trisubstituted phenyl analogs are now found to have activity as for the treatment of congestive heart failure.
29	5220068	Psychostimulant agent The present invention relates to a pharmaceutical composition comprising as active ingredient a compound of the Formula I ##STR1## wherein R 1 stands for straight or branched chain alkyl...
30	5198587	Phenethylamine derivatives Phenethylamine derivatives shown by the general formula ##STR1## wherein Ro represents a lower alkyl group; R 1 represents a lower alkyl group or a lower alkoxy group; R 2 represents hydrogen...
31	5106713	Photoconductive imaging members with unsymmetrical squaraine compositions The cyclized squaraines essentially as represented by the formula ##STR1## wherein R 1 and R 2 are independently selected from alkyl and hydrogen; R 3 and R 4 are independently selected from...
32	5087753	Process for recovering α-aminoalcohols Process for recovering α-aminoalcohols by extraction from aqueous solutions, in which process an aromatic aldehyde is added at elevated pH to an aqueous solution of an aminoalcohol in an at least...
33	5047433	N-alkyl derivatives of 2-amino-6,7-dimethoxy tetraline and pharmaceutical compositions having antihypertensive activity containing same N-alkyl derivatives of 2-amino-6,7-dimethoxy tetraline having general formula (I) ##STR1## wherein R is selected from hydrogen, ethyl, n-propyl and methyl cyclopropyl; R 1 is selected from...
34	5008292	Pesticidal method The invention relates to N-[2-(4-fluorophenyl)-1-methyl]-ethyl-N-methyl-N-propynyl amine of the Formula I ##STR1## and isomers and salts thereof. The compound of the Formula I is useful as an...
35	4996316	Process for the preparation of tertiary N, N-dimethylamines A process for the preparation of tertiary N,N-dimethylamines by the reaction of primary amines, formaldehyde, and hydrogen under pressure and at elevated temperature in the presence of a...
36	4967003	Propylamines, and their use as fungicides N-Arylpropyl-substituted secondary amines of the formula ##STR1## where R 1 and R 2 are each hydrogen, alkyl, cycloalkyl, haloalkyl, alkoxy, chlorine, bromine or fluorine, m is 0, 1 or 2, R 3 ...
37	4960797	N-2[(4-fluoro-phenyl)-1-methyl]-2-ethyl-N-methyl-N-propynyl amine and the method of use thereof The invention relates to the new N-[2-/4-fluorophenyl/-1-methyl]-ethyl-N-methyl-N-propynyl amine of the Formula I ##STR1## and isomers and salts thereof. The compound of the formula I is useful as...
38	4959488	Polyfunctional hexasubstituted benzene derivatives Polyfunctional hexasubstituted benzene derivatives wherein at least three of the substituents are saturated carbon chains having from 1 to 21 carbon atoms and functional groups containing hetero...
39	4913891	Positron emitter labeled enzyme inhibitors This invention involves a new strategy for imaging and mapping enzyme activity in the living human and animal body using positron emitter-labeled suicide enzyme inactivators or inhibitors which...
40	4880841	Process of producing phenethylamine derivatives Phenethylamine derivatives shown by the general formula ##STR1## wherein Ro represents a lower alkyl group; R 1 represents a lower alkyl group or a lower alkoxy group; R 2 represents hydrogen...
41	4725602	Acetylene amines and their use as vasodilators and antihypertensives Acetylenes of the following formula (I): ##STR1## wherein Y, m, R 1 , R 2 , R 3 , n and R 4 are defined herein and R 5 is hydrogen, alkyl, cycloalkyl or substituted alkyl are useful vasodilators...
42	4704407	Soluble dobutamine salts Hydroxyalkanoic or alkandioic acid salts of dobutamine having desirable water solubility, useful in preparing intravenous solution for treatment of cardiogenic shock.
43	4695589	Alpha-(aminoalkyl-4-hydroxy-3-(alkylthio)benzenemethanols Alpha-(aminoalkyl)-4-hydroxy-3-(alkylthio)benzenemethanols useful as intermediates and as antihypertensive agents are prepared by reduction of the corresponding aminoalkyl...
44	4647699	New diamines and a process for their production New aminoalkyl anilines having the formula: ##STR1## wherein k is 0 or 1; QNH 2 is a residue of formula ##STR2## which is situated in one of the positions of the benzene ring ortho or para to the...
45	4622218	Testicular-specific drug delivery Testicularly acting drug species are site-specifically/sustainedly delivered to the testes by administering to a male in need of such treatment a pharmacologically effective amount of the target...
46	4564706	Process for the preparation of propargyl amines The invention relates to a new process for the preparation of propargyl ammonium chlorides of the Formula I ##STR1## by alkaline decomposition of the d-tartarate of the 1-isomer of an amine of the...
47	4490392	Benzylalcohol derivative and process for preparing A benzylalcohol derivative of the formula: ##STR1## wherein R is hydroxy, benzyloxy, halogen or alkoxy having one to four carbon atoms, and Ring A is monomethoxyphenyl, dimethoxyphenyl,...
48	4486602	Valienamine derivatives, their production and use A compound of the formula: ##STR1## wherein A is a chain hydrocarbon group having 1 to 10 carbon atoms optionally substituted by hydroxyl, phenoxy, thienyl, furyl, pyridyl, cyclohexyl or an...
49	4473586	Aminoalkyl dihydronaphthalenes Disclosed herein are 1-aminoalkyl-3,4-dihydronaphthalenes represented by the formula ##STR1## wherein n is 1 or 2; R, R 1 , and R 2 are independently selected from hydrogen, hydroxy, loweralkoxy...
50	4376125	Aminobenzlpropranolol and pharmaceutical preparation thereof 1-(p-Amino-α,α-dimethylphenethylamino)-3-(1-naphthoxy)-2-p ropan ol, 1-(p-hydroxy-α,α-dimethylphenethylamino)-3-(1-naphthoxy)-2 -pro panol,...

Matches 1 - 50 out of 145

1 2 3 >