Patents in Class 560/168

Matches 1 - 50 out of 162

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Match	Document	Document Title
1	7527733	Chelating agents for heavy metal removal The present invention provides for Troika acids attached to a macroporous resin and Methods of preparing the same, including direct attachment of a Troika acid, and attachment of a Troika acid...
2	7449446	Combination product comprising melagatran and dexamethasone There is provided a combination product comprising; (A) melagatran or a pharmaceutically acceptable derivative thereof; and (B) dexamethasone or a pharmaceutically acceptable derivative there of,...
3	7354905	Prodrugs of thrombin inhibitors There is provided compounds of formula I, R 1 O(O)C—CH 2 —(R)Cgl-Aze-Pab-R 2 I
4	7223745	Proteasome inhibitors and methods of using the same The present invention provides boronic acid compounds, boronic esters, and compositions thereof that can modulate apoptosis such as by inhibition of proteasome activity. The compounds and...
5	7135587	Urea and urethane derivatives as integrin inhibitors Novel urea and urethane derivatives of general formula (I) in which R1, R2, R3, R5, R5′, X, Y, B, m, n and o are as defined in Patent Claim 1 , and physiologically acceptable salts or solvates...
6	7015348	Method for producing an optically active β-amino acid To provide a producing method of an optically active β-amino acid useful as intermediate for the production of medicines, agricultural chemicals and physiologically active substances, by means of...
7	6962905	Pharmaceutical formulation comprising a low molecular weight thrombin inhibitor and its prodrug A kit of parts containing (a) a pharmaceutical formulation including a low molecular weight thrombin inhibitor, or a pharmaceutically acceptable derivative thereof, in admixture with a...
8	6919449	Process for the preparation of cephalosporin intermediate and its use for the manufacture of cephalosporin compounds The present invention relates to a method for the preparation of cephalosporin antibiotic of the formula (II), which comprises hydrolyzing and halogenating the ester of formula (III) by...
9	6888022	Methods and compounds for inhibiting β-amyloid peptide release and/or its synthesis Disclosed are compounds which inhibit β-amyloid peptide release and/or its synthesis, and, accordingly, have utility in treating Alzheimer's disease. Also disclosed pharmaceutical compositions...
10	6784311	Method of producing 3-aminoalkanoic acid esters Process for the preparation of 3-aminoalkanoic acid esters of the general formula: in which R is C 1-6 -alkyl and R 1 is hydrogen, C 1-6 -alkyl or phenyl, or their salts, by catalytic...
11	6660246	Ligands and metal complexes thereof Novel compounds of the formula and novel complexes of these compounds with metals are useful in diagnostic and therapeutic methods.
12	6608196	Process for solid supported synthesis of pyruvate-derived compounds Provided are processes for synthesizing structurally diverse pyruvate-derived compounds using a parallel approach on a solid phase support. Examples of such a solid phase support include resins...
13	6605688	Low Viscosity imine reactive diluents and coating compositions made therefrom This invention concerns low viscosity aldimine and ketimine reactive diluents having multi-imine functionality, which are useful in automotive refinish coating compositions, including a process for...
14	6465686	Halogenated 2-amino-5,6 heptenoic acid derivatives useful as nitric oxide synthase inhibitors The present invention discloses halogenated 2-amino-5,6 heptenoic acid derivatives useful as nitric oxide synthase inhibitors.
15	6420592	Amino acid-derived phosponamidic anhydrides and methods of preparing the same Phosphonamide compounds and methods of forming those compounds are provided. The inventive methods comprise forming a template opened-ring phosphonamide compound and optionally subjecting the...
16	6365673	Low viscosity imine reactive diluents and coating compositions made therefrom This invention concerns low viscosity aldimine and ketimine reactive diluents having multi-imine functionality, which are useful in automotive refinish coating compositions, including a process for...
17	6348617	Method for purifying pyruvic acid compounds The present invention is directed to a method for purifying pyruvic acid compounds, which method comprises reacting a pyruvic acid compound of general formula (I): wherein R 1 is an optionally...
18	6130246	Pesticides The compounds of formula I ##STR1## wherein: a) X is O, and Y is OC 1 -C 4 alkyl; or b) X is O or S, and Y is NHCH 3 have fungicidal properties and can be used in plant protection for...
19	6090974	Alkyl 3-oxoalkanoate and process for the preparation thereof This invention includes an alkyl 3-oxoalkanoate, and processes for its preparation and use for the synthesis of fatty hydroxylated amino acids, fatty amino alcohols and ceramides.
20	6034137	Cationic lipids for gene therapy This invention provides novel cationic lipids, particularly guanidino lipids, and methods for their preparation. Also provided are polyanionic-lipid complexes comprising the lipids of the...
21	5977025	1,3-oxazin-4-one derivative, herbicide containing same, and intermediate for preparing same This invention provides 1,3-oxazin-4-one derivatives represented by following general formula (I): ##STR1## in which R 1 represents a phenyl group which may be substituted; R 2 represents a...
22	5948931	Preparation and use of α-(hydroxyimino) phosphonoacetic acids α-(hydroxyimino)phosphonoacetic acids (also referred to as "α,α-disubstituted trifunctional oximes" and "Troika Acids") and their derivatives, and methods to prepare them are disclosed. Also...
23	5945408	Hydroxyanidino derivatives useful as nitric oxide synthase inhibitors The current invention discloses hydroxyamidino derivatives useful as nitric oxide synthase inhibitors.
24	5939392	Method of thrombin inhibition The invention relates to new competitive tripeptide inhibitors of trypsin-like serine proteases, their synthesis, pharmaceutical compositions containing the compounds as active ingredients, and the...
25	5935988	Tolerability of pharmaceutically active β-amino acids The present invention relates to mixtures of α-amino acids and/or derivatives thereof and cyclopentane-β-amino acids and/or derivatives thereof, dipeptides of the abovementioned α-amino acids...
26	5863931	Amidino derivatives and their use as nitric oxide synthase inhibitors Amidino derivatives of formula (I) and salts, and pharmaceutically acceptable esters and amides thereof, in which: R 1 is a C 1 -6 straight or branched chain alkyl group, a C 2 -6 alkenyl group, a...
27	5861533	Process for nitrosation of C-H-acidic compounds A process for nitrosating C-H-acidic compounds. The process substantially avoids producing polluted wastewater.
28	5847195	Process for the production of compounds containing aspartate and aldimine groups The present invention relates to a process for preparing compounds containing aspartate and aldimine groups corresponding to the formula ##STR1## by a) reacting 50 to 95 mole % of the primary amino...
29	5710324	Inhibitors of nitric oxide biosynthesis The present invention is directed to a new class of compound which are useful as inhibitors of the biosynthesis of nitric oxide.
30	5707967	Pain relief compositions Disclosed are compositions containing either aspartame or monosodium glutanate combined with an amino acid.
31	5696283	Preparation of methyl isoproylideneaminooxyacetoxyacetate Process for preparing methyl isopropylideneaminooxyacetoxyacetate I ##STR1## by reacting in an integrated process, a) acetone with hydroxylammonium sulfate and sodium hydroxide solution to give...
32	5616764	Functionalization of polymers via enamine of acetoacetate The present invention relates to the preparation of polymers bearing reactive functional groups. More particularly, this invention relates to the preparation of polymers containing functional...
33	5399590	Quaternary ammonium salts and pharmaceutical compositions containing them The invention relates to the field of organic chemistry and more particularly to that of therapeutic chemistry. More particularly it relates to new quaternary ammonium salts of general formula (I):...
34	5359128	Malic acid derivatives and compositions for the treatment of psoriasis The invention comprises compositions and methods for the treatment of psoriasis. The compositions comprise compounds of the formula: ##STR1##
35	5312962	Process for the production of compounds containing aldimine or ketimine groups and the compounds obtained by this process The invention relates to a process for the production of organic compounds containing aldimine or ketimine groups by the reaction of compounds containing β-ketoester groups with bis-aldimines or...
36	5268501	Process for preparing haloketo acid derivatives Process for preparing haloketo acid derivatives [I]: ##STR1## wherein R is H or C 1 -6 alkyl, and X is chlorine or bromine, which comprises reacting β-oxo-acid ester [II]: ##STR2## wherein R 1 is...
37	5245060	Terpene derivatives and process for preparing the same A terpene derivative represented by the general formula (I): ##STR1## wherein R 1 represents a lower alkyl group; R 2 represents an alkyl group, a cycloalkyl group, a cycloalkylalkyl group, an...
38	5241101	Pesticidal substituted oxime ethers Pesticidal substituted oxime ethers of the formula ##STR1## in which R represents in each case unsubstituted or substituted alkyl, cycloalkyl, aryl or heterocyclyl and X represents nitrogen or a...
39	5196450	Method of inhibiting protozoal growth This invention relates to the use of α- halomethyl, α-acetylenic or α-allenic derivatives of arginine and agmatine, or their dehydro analogs, in the treatment of Chagas disease and Coccidiosis.
40	5100655	Arginine derivatives and cosmetic compositions containing the same Emulsifier compositions capable of forming an emulsion which is stable over a wide range of temperatures and contains at least one of a N α -long-chain acyl arginine higher alkyl ester of the...
41	5055588	Process for preparing N-substituted amino acid esters A process for preparing N-substituted amino acid esters having the formula (I): ##STR1## wherein R 1 and R 4 , the same or different, are an alkyl, aralkyl, cycloalkyl or aryl group; and R 2 and...
42	5030732	Aminoethylphosphinic acid derivatives Disclosed are some new aminoethylphosphinic acid derivatives useful as antibacterial agents.
43	5011854	Hydroxamic acid derivatives and use thereof in combatting lipoxygenase-mediated diseases A hydroxamic acid compound represented by the general formula (I) or a salt thereof; ##STR1## wherein R 1 represents a hydrogen atom, or a substituted or unsubstituted alkanoyl group, R 2 ...
44	5010189	Processes for the preparation of 5-amino-4-hydroxy-valeric acid derivatives The invention relates to novel processes and intermediates for the preparation of 5-amino-4-hydroxyvaleric acid derivatives of the formula ##STR1## in which R 1 represents hydrogen, optionally...
45	4990649	Azulenesquaric acid dyes that contain urethane groups Azulenesquaric acid dyes of the formula ##STR1## where L is substituted or unsubstituted C 1 -C 12 -alkylene, R 1 is C 1 -C 20 -alkyl, C 5 -C 7 -cycloalkyl or substituted or unsubstituted...
46	4959495	Process for the preparation of intermediates used to produce aminothiazoloximino cephalosporins A process is disclosed for the preparation of intermediates useful in the synthesis of aminothiazoloximino cephalosporins.
47	4933486	Process for the preparation of 4-halo-3-oxo-2-alkoxyaminobutyric esters A process for the preparation of 4-halo-3-oxo-2-alkoxyiminobutyric esters. A process for the preparation of 4-halo-3-oxo-2-alkoxyiminobutyric esters by solvent-free halogenation of the liquid...
48	4927965	N-(N-succinyl-L-leucyl)agmatine, related compounds and use in pharmacology Compounds having the formula: ##STR1## wherein R 1 is --NH(CO)OR 5 , --NH(CNH)NH 2 or --NH(CN--NO 2 )HN 2 ; R 2 is hydrogen, C 1 -8 alkyl or C 6 -8 aryl; n is 2 to 6; and R 5 is...
49	4927964	Method for production of 2-oxyimino-3-oxobutyric acids An advantageous method of producing in large amounts on a commercial scale 2-substituted oxyimino-3-oxobutyric acids, which are useful as intermediates in the synthesis of e.g. aminothiazole...
50	4898977	Processes for the preparation of 5-amino-4-hydroxyvaleric acid derivatives The invention relates to novel processes and intermediates for the preparation of 5-amino-4-hydroxyvaleric acid derivatives of the formula ##STR1## in which R 1 represents hydrogen, optionally...

Matches 1 - 50 out of 162

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