Patents in Class 560/119

Matches 1 - 50 out of 273

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Match	Document	Document Title
1	8076502	2-amino-bicyclo(3.1.0) hexane-2,6-dicarboxylic ester derivative A drug effective for the treatment and prevention of psychiatric disorders such as schizophrenia, anxiety and related ailments thereof, depression, bipolar disorder and epilepsy. The drug...
2	8043789	Photosensitive compound and photoresist composition including the same A photosensitive compound whose size is smaller than conventional polymer for photoresist, and which has well-defined (uniform) structure, and a photoresist composition including the same are...
3	7960579	2-amino-bicyclo [3.1.0] hexane-2,6-dicarboxylic ester derivative A drug effective for the treatment and prevention of psychiatric disorders such as schizophrenia, anxiety and related ailments thereof, depression, bipolar disorder and epilepsy. The drug...
4	7816476	Polymerizable cyclopropyl acrylates Cyclopropyl acrylate of general formula (1), constitutional and stereoisomers thereof and their mixtures in which A is selected from:
5	7786314	Processes for preparing bicyclo [3.1.0] hexane derivatives, and intermediates thereto Processes for the preparation of certain [3.1.0]hexane derivatives which are useful as mGluR agonists, and intermediates prepared during such processes.
6	7659358	Binders containing ortho ester groups A process for preparing polymers containing polyortho ester groups and optionally NCO groups by reacting A) and B) where A) is a polyortho ester containing at least one isocyanate-reactive group...
7	7655695	Illudin analogs useful as anticancer agents Acylfulvene analogs, which inhibit tumor growth, especially solid tumor growth, and which have an adequate therapeutic index to be effective for in vivo treatment are provided herein. The compounds...
8	7534475	Liquid crystal compound comprising two condensed and substituted rings A new liquid crystal compound comprises two condensed and substituted rings. The ring preferably is a five-membered heterocyclic ring. The heterocyclic ring is preferably condensed with benzene...
9	7501222	Photoresist monomer polymer thereof and photoresist composition including the same A polymer including a monomer represented by the following Formula and a photoresist composition including the same are disclosed. The polymer and photoresist composition can improve the resolution...
10	7425644	Method of purifying pravastatin The present invention provides pure pravastatin compositions and pure compactin compositions, and methods for the preparation thereof.
11	7157594	6-Fluorobicyclo[3.1.0]hexane derivatives An antidepressant comprising, as an active ingredient, a compound having an antagonistic effect on group II metabotropic glutamate receptors, as well as a...
12	7078558	Crystals of the sodium salt of pravastatin Lovastatin, pravastatin, simvastatin, mevastatin, atorvastatin, fluvastatin and cervastatin and derivatives and analogs thereof are known as HMG-CoA reductase inhibitors and are used as...
13	7071359	Neuropathy improvers containing nitrogenous compounds as the active ingredient A compound represented by the Formula below, and an agent for the remedy of neural damage having the said compound as the active ingredient. [Here, G represents G1 shown below R4 represents,...
14	7018818	Intermediates in the preparation of therapeutic fused bicyclic amino acids The invention presents compounds of formula (I), where R represents H or a suitable carboxylic acid protecting group, which are intermediates in the preparation of therapeutic fused bicyclic amino...
15	6965026	Nanoscale faceted polyhedra The subject invention pertains to nanoscale polyhedron-shaped molecules having molecular building blocks connected at their vertices. The subject invention also concerns methods of producing...
16	6936731	Pravastatin sodium substantially free of pravastatin lactone and epi-pravastatin, and compositions containing same The present invention provides pravastatin sodium substantially free of pravastatin lactone and epiprava, the C-6 epimer of pravastatin. The present invention further provides a novel process for...
17	6875867	Process for preparing chiral diol sulfones and dihydroxy acid HMG CoA reductase inhibitors A process is provided for preparing chiral diol sulfones of the structure where R3 is preferably where R4a is preferably aryl such as phenyl, and R1a is preferably alkyl such as t-butyl, which are...
18	6770676	Dicarboxylic acid derivatives The present invention relates to 2-amino-6-fluorobicyclo[3.1.0]hexane-2,6-dicarboxylic acid derivatives represented by the formula: the pharmaceutically acceptable salts thereof, or the hydrates...
19	6756507	Process for the preparation of sodium salts of statins A process for the preparation of sodium salts of statins, namely Compactin, Lovastatin and Pravastatin.
20	6746728	Compound having tetrahydronaphthalene skeleton and liquid crystal composition containing same A tetrahydronaphthalene derivative represented by the general formula (I) and a liquid crystal composition containing the same. A compound represented by the general formula (I) shows superior...
21	6740775	Crystalline sodium salt of pravastatin A crystalline form of the sodium salt of pravastatin, which is known by the chemical name 1-naphthaleneheptanoic acid, 1,2,6,7,8,8a-hexahydro-β, δ,6-trihydroxy-2-methyl-8-(2-methyl-1-oxobutoxy)-, m...
22	6689590	Process for recovering statin compounds from a fermentation broth A composition comprising pravastatin sodium substantially free of pravastatin lactone is described.
23	6541515	HIV integrase inhibitors Compounds useful in the inhibition of HIV integrase, the prevention or treatment of infection by HIV and the treatment of AIDS, either as compounds, pharmaceutically acceptable salts,...
24	6506929	Process to manufacture simvastatin and intermediates A process is disclosed for the preparation of simvastatin which enables highly regio selective C-methylation of the 2′-position group of lovastatin without requiring protection/deprotection of 1...
25	6392086	Intermediates and process for producing fluorine-containing amino acid compound by using the same The present inventions relate to a (1S,5R,6S)- or (1SR, 5RS, 6SR)-3-fluoro-2-oxobicyclo[3.1.0]hex-3-ene-6-carboxylic acid derivative represented by Formula (1): [in the formula, R represents OR1 or...
26	6376700	Alicyclic compound An alicyclic compound of the formula (1) is disclosed: wherein R1 and R2 each independently is a hydroxyl group, a C1-8 hydroxyalkyl group, or a C3-8 hydroxycycloalkyl group; R3, R4 and R5 each...
27	6369194	Vicinyl tricarbonyl compounds and combinatorial libraries containing same The invention relates to compounds of formula where R is a structural diversity element selected from the group consisting of alkyl, cycloalkyl, aryl, heteroaryl, peptidyl, heteroatom-substituted...
28	6365382	Biotechnological process for preparing hydroxylated ML-236B derivatives, known as M-4 and M-4′, and analogues thereof The very effective conversion of ML-236B substances and derivatives thereof into 6′-hydroxylated products with the microorganisms of species Amycolatopsis orientalis, or with an extract or a h...
29	6326369	Bicyclic quinone compounds, their production and use A compound of the formula: ##STR1##wherein R1 and R2 each represents a lower alkyl, or R1 and R2 may be bonded together to form a ring; X represents a spacer of which the number of atoms...
30	6316498	Fluorine-containing amino acid derivatives Fluorine-containing amino acid derivatives represented general formula (I), pharmaceutically acceptable salts thereof or hydrates of the same, wherein X1 represents hydrogen or fluorine; and R1 and...
31	6306629	Microorganism streptomyces exfoliatus yj-118 and a method for producing pravastatin sodium by using the strain The present invention is related to a new microorganism Streptomyces exfoliatus YJ-118 and a method for producing pravastatin sodium by using this microorganism which shows a strong tolerance to...
32	6217793	Acetylene compound, liquid crystal composition and liquid crystal element Provided are novel acetylene compounds which are useful as a component for a liquid crystal composition used for a liquid crystal element, a liquid crystal composition containing said compounds and...
33	6177586	Vitamin D3 derivative and production process thereof The starting materials for a production process of a vitamin D3 derivative are disclosed, e.g., a cyclopentene derivative represented by the formula (1-2): ##STR1##wherein R11 is a hydrogen atom,...
34	6160009	Excitatory amino acid receptor modulators Compounds of the formula ##STR1## in which R1 and R2 are as defined in the specification, and non-toxic metabolically labile ester and amides thereof are useful as modulators of metabotropic...
35	6143783	Excitatory amino acid receptor modulators The present invention relates to compounds of the formula ##STR1## in which R1 is defined in the specification, and non-toxic metabolically labile esters and amides thereof are useful as modulators...
36	6118019	3-alkoxypropionic ester derivative A 3-alkoxypropionic ester derivative, an olefin polymerization solid catalyst component using the same, an olefin polymerization catalyst using the same, and a process for the preparation of a...
37	RE36520	HMG-CoA reductase inhibitors Novel 3-hydroxy-3-methylglutaryl-coenzyme A (HMG-CoA) reductase inhibitors are useful as antihypercholesterolemic agents and are represented by the following general structural formula (II): ##STR1##
38	5925782	Synthetic excitatory amino acids The present invention provides novel compounds that affect certain excitatory amino acid receptors, and are useful in the treatment of neurological disorders and psychiatric disorders.
39	5916920	3-substituted Bicyclo 3.1.0!hexane-6-carboxylic acids Compounds of the formula ##STR1## in which X represents a bond, S, O or NRa ; and R is as defined in the specification are useful as modulators of metabotropic glutamate receptor function.
40	5834404	Substituted bicycloheptanedione derivative and herbicide The present invention is directed to substituted bicycloheptanedion e derivatives represented by a general formula I!; ##STR1## wherein R represents C1 -C4 alkyl, R1 represents hydrogen, C1 -C10...
41	5827855	Hexahydronaphthalene ester derivatives their preparation and their therapeutic uses Compounds of formula (I): ##STR1## wherein R1 represents a group of formula (II) or (III): ##STR2## R2 is alkyl, alkenyl or alkynyl; R3 and R4 are each hydrogen, alkyl, alkenyl or alkynyl; R5 is...
42	5741925	Transvinylation of naphthenic acids Vinyl naphthenate monomer mixtures are prepared by transvinylation of naphthenic acid in the presence of a catalyst of a palladium carboxylate complexed with one or more aryl N-containing ligands...
43	5700833	Isocarbacyclin derivatives The present invention provides novel isocarbacyclin derivatives useful for search and study of prostacyclin receptor and as a therapeutic drug for central nervous system diseases, which derivatives...
44	5532408	α-chain-modified isocarbacyclins and process for the production thereof Provided are α-chain-modified isocarbacyclins of which the α-chain is modified with a phenylene group, a cycloalkylene group or a thiophendiyl group, and these α-chain-modified isocarbacyclins sh...
45	5489613	Carbacyclin derivatives, process for their preparation and compositions containing them Compounds of formula (I): ##STR1## have valuable platelet-aggregation inhibitory activities and may be used for the prophylaxis and treatment of such diseases as thrombosis.
46	5468905	Bicyclo[4,1,0]heptane-2,4-dion derivatives, its synthetic intermediates and process for the manufacture thereof Compounds represented by general formulas (I) and (II), useful as the intermediates for agricultural chemicals, particularly herbicidal compounds, wherein R1 and R2 represent each hydrogen, alkyl...
47	5449684	Cytotoxic compounds Compounds isolated from a marine sponge, and derivatives thereof, have the formulae: ##STR1## in which R1 is H or lower alkyl; R2 is OH or CH3 ; R3 is OH or CH3, and R4 H or MPTA. The compounds...
48	5405870	Carbacyclin compounds; pharmaceutical compositions and method of use Compounds of formula (Ic): ##STR1## having valuable platelet-aggregation inhibitory activities useful for the prophylaxis and treatment of such diseases as thrombosis and pharmaceutical...
49	5386039	Process for the preparation of a bicyclic decalin ketone Perhydro-5,5-8a-trimethyl-2-naphthalenone is prepared by acid cyclization of carboxylic esters of formula ##STR1## having a double bond in one of the positions indicated by the dotted lines and...
50	5374654	9-substituted carbacyclin derivatives, processes for their preparation, and their use as medicinal agents The invention relates to carbacyclin derivatives of Formula I ##STR1## wherein the various substituents are defined herein, including, inter alia, if R2 is a hydrogen atom, their salts with...

Matches 1 - 50 out of 273

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