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7317124 Ortho-substituted pentafluorosulfanylbenzenes, process for their preparation and their use as valuable synthetic intermediates  
Pentafluorosulfanyl-benzenes according to Formula (I): a process for their preparation and their use as valuable synthetic intermediates for preparing, for example, medicaments, diagnostic...
7238830 N-alkylaspartyl dipeptide ester compounds  
The present invention provides N-alkylaspartyl dipeptideester compounds and salts thereof, such as N-[N-[3-(3-hydroxy-4-methoxyphenyl)-3-methylbutyl]-L-α-aspa rtyl]-L-phenylalanine 1-methyl ester,...
7217832 5-amidino-2-hydroxybenzenesulfonamide derivatives, pharmaceutical compositions containing the same and intermediates for their preparation  
The present invention relates to a 5-amidino-2-hydroxybenzenesulfonamide derivative represented by the general formula: wherein R 1 is a hydrogen atom or an optionally substituted lower alkyl...
7196229 Benzoylcyclohexenone derivatives  
The invention relates to benzoylcyclohexenone derivatives of general formula (I) wherein the variables R 1 to R 10 and n have the designation cited in claim 1 . The invention also relates to the...
7041844 Irreversible non-steroidal antagonist compound and its use in the treatment of prostate cancer  
The present invention relates to an antiandrogen compound and a method of treating prostate cancer in a patient utilizing the compound. The present invention also relates to a pharmaceutical...
6541670 Aminobenzophenones as inhibitors of IL 1β and TNF-α  
A compound of the general formula I wherein R 1 represents a substituent selected from the group consisting of halogen, hydroxy, mercapto, trifluoromethyl, amino, (C 1 -C 3 )alkyl, (C 2 -C 3...
6541422 Method for improving the selectivity of 1,3-cyclohexanedione herbicide  
A method of selectively controlling undesirable vegetation in crops by using a postemergent application of an herbicidally effective amount of a metal chelate of a 2-(substituted...
6344505 Mono- and bis-benzotriazolyldihydroxybiaryl UV absorbers  
Provided is a composition which contains a mono- or bis-benzotriazole compound, an N-oxide thereof, or a mixture of at least two of the preceding compounds. Representative bis-benzotriazole...
6218431 Substituted biphenyls  
Substituted biphenyls having glucagon receptor antagonistic activity. Claimed compounds have the formula ##STR1## wherein R 1a and R 1b independently represent (C 1 -C 6 ) alkyl; R 2 ...
RE37087 Insecticidal triffluormethyl alkane derivatives  
There are provided new alkane and alkoxyalkane derivatives of the general formula I ##STR1## in which R 1 , R 2 , R 3 , R 4 and A have the meanings given in the description, processes for their...
6150412 Catechol derivatives  
The invention relates to compounds of formula (I) ##STR1## wherein R 1 is an electronegative substituent, preferably nitro, cyano, formyl or carboxy, R 2 is --A--R 4 , wherein A is a branched or...
6057358 Amine derivatives, processes for producing them and a use of them as antiarrhythmic drugs  
Novel amine derivatives of the following general formula (I): ##STR1## (wherein) A may denote --(CH 2 )--O--, --(CH 2 ) 2 --O--, or --(CH 2 ) 2 --NH--; B may denote --(CH 2 ) 2 --; R 1 ...
6040339 Urea derivatives having ACAT inhibitory activity, their preparation and their therapeutic and prophylactic use  
Compounds of formula (I): ##STR1## wherein: R 1 is alkyl; R 2a , R 2b , R 2c and R 2d are the same or different and each is hydrogen, optionally substituted alkyl or various other organic...
5880147 Amide derivatives having ACAT inhibitory activity, their preparation and their therapeutic and prohylactic use  
Compounds of formula (I): ##STR1## wherein: R 1 is alkyl; R 2a , R 2b , R 2c and R 2d are the same or different and each is hydrogen, optionally substituted alkyl, --(CO)--B 1 (wherein B 1 ...
5849796 Ortho-substituted benzoil acid derivatives  
Ortho-substituted benzoic acid derivatives of the formula I ##STR1## in which R 1 , R 2 and R 3 have the given meanings, and Q is guanidyl, and also their physiologically harmless salts, exhibit...
5739374 Processes of preparing diphenylheteroalkyl derivatives  
Diphenylheteroalkyl derivatives of the formula I ##STR1## where A and R 1 -R 6 have the meanings specified in the description, and the preparation thereof are described. The substances are...
5736579 Substituted spiro compounds for the treatment of inflammation  
A class of substituted spiro compounds is described for use in treating inflammation and inflammation-related disorders. Compounds of particular interest are defined by Formula III: ##STR1##...
5731351 Alkenyl-benzoylguanidine derivatives  
Alkyl-benzoylguanidines of the formula I ##STR1## wherein R 1 , R 2 and R 3 have the meanings given, and physiologically acceptable salts thereof show antiarrhythmic properties and act as...
5688945 Compounds  
The present invention relates to novel derivatives of 3-hydroxyanthranilic acid, 3-HANA, of the general formula I ##STR1## wherein R 1 and R 2 are the same or different and selected from H and...
5665777 Biphenyl hydroxamate inhibitors of matrix metalloproteinases  
Compounds of formula ##STR1## or a pharmaceutically acceptable salt thereof inhibit matrix metalloproteinases and TNFα secretion and are useful in the treatment of inflammatory disease states....
5661183 3-hydroxy anthanilic acid derivatives  
The present invention relates to novel derivatives of 3-hydroxyanthranilic acid, 3-HANA of general formula (I), wherein R 1 and R 2 are the same or different and selected from H and alkyl; X is...
5571842 Perfluoroalkyl-substituted, benzoylguanidines, a process for their preparation, their use as a medicament or diagnostic agent, and a medicament containing them  
Perfluoroalkyl-substituted benzoylguanidines, a process for their preparation, their use as a medicament or diagnostic agent, and a medicament containing them A description is given of...
5514642 Cyclohexenone oxime ethers, their preparation and their use  
Cyclohexenone oxime ethers of the formula I ##STR1##
5493053 Method for preparing desferrioxamine B and homologs thereof  
A new and versatile route to N'-[5-[[4-[[5-(acetylhydroxyamino)pentyl]amino]-1,4-dioxobut yl]hydroxyamin o]pentyl]-N-(5-aminopentyl)-N-hydroxybutanediamide, desferrioxamine B (DFO) is described....
5482942 (3,4-dioxocyclobuten-1-yl)chromene, indene, and dihydronaphthalenone derivatives as smooth muscle relaxants  
This invention relates to novel 4-(3,4-dioxocyclobuten-1-yl)chromenes and dihydronaphthalenones and 3-(3,4-dioxocyclobuten-1-yl)indenes and salts thereof having smooth muscle relaxing activity, to...
5480668 N-substituted derivatives of aspartame useful as sweetening agents  
Lower alkyl esters of compounds of the formula ##STR1## wherein Z is hydrogen or hydroxyl and R is a hydrocarbyl group optionally substituted by hydroxy and/or alkoxy group, are useful as...
5338886 Process for preparation of aromatic thiols  
Disclosed is a process for preparation of an aromatic thiol corresponding to the structure A-(SH)n wherein A is a substituted or unsubstituted aromatic radical and n is 1, 2, 3, 4, 5 or 6...
5321169 Cyclohexane derivatives  
A novel tetracyclic cyclohexylcyclohexene derivatives represented by formula: ##STR1## wherein ##STR2## n, X and Y are as defined in the specifications, are disclosed. The compounds are useful as...
5238818 Oxidizable color producing reagent  
This amount of an oxidative substance or a peroxidase-like substance can be determined by using a combined color former comprising 4-aminoantipyrine or a derivative thereof, etc., as a main color...
5185375 Thioformamide derivatives  
Therapeutically useful thioformamide derivatives of the formula: ##STR1## wherein R represents alkyl, Ar represents optionally substituted phenyl group, Y represents ethylene, methylene or a...
5180744 Aralkyl-N-terminal amino hydroxy  
Non-peptidyl compounds characterized generally as aralkyl-N-terminal amino hydroxy β-amino acid derivatives are useful as renin inhibitors for treatment of hypertension. Compounds of particular...
5136081 Process for the preparation of cyclopentene, cyclopentane and cyclohexane derivatives  
The invention provides a process for the preparation of fungicidally active cyclopentene derivatives of the general formula ##STR1## cyclopentane derivatives of the general formula ##STR2## and...
5131945 Certain glyoxyl-cyclohexendiones as herbicides  
Compounds of formula I ##STR1## are useful as herbicides, effective against dicotyledonous weeds.
5132326 Cyclopropanethiocarboxamides  
Cyclopropanethiocarboxamides I ##STR1## (R 1 , R 2 =H, CN, NO 2 , halogen, C 1 -C 4 -alkyl, C 1 -C 4 -alkoxy, C 1 -C 4 -haloalkyl, C 1 -C 4 -haloalkoxy; R 3 , R 4 =H, C 1 -C 4 -alkyl;...
RE33989 Oxime ethers and fungicides containing these compounds  
Oxime ethers of the formula ##STR1## where R 1 and R 2 are hydrogen or alkyl, X(m=1 to 5) is halogen, cyano, trifluoromethyl, nitro, allyl, alkoxy, unsubstituted or substituted phenyl,...
5089046 Aryl and heteroaryl diones  
Cyclic 1-one-2-ene-3-ol compounds substituted in 2-position by an aroyl or heteroaroyl group bearing a hydrocarbylsulfonyloxy or hydrocarbylsulfonylamino substituent exhibiting herbicidal activity.
5072034 Preparation of 4-alkoxy-2-hydroxybenzophenone-5-sulfonic acids  
4-alkoxy-2-hydroxybenzophenone-5-sulfonic acids of the general formula I ##STR1## where R 1 is C 1 -C 20 -alkyl which is unsubstituted or substituted by halogen, cyanao, hydroxyl, C 1 -C 20 ...
5055223 Aryl-sulfur pentafluorides  
Aryl-sulfur pentafluorides of the formula I ##STR1## wherein R, A, Z, n, m and X° have the meaning indicated in claim 1 are suitable for use as components of liquid-crystal phases for field-effect...
5047426 Fungicidal compositions  
The invention provides fungicidal compositions which comprise a carrier and, as active ingredient, a compound of the general formula ##STR1##
5047425 Amine derivatives having cardiovascular activity  
Compounds of the formula ##STR1## wherein Ar, R, R 1 , R 2 , R 3 , R 4 , X and n have the meanings mentioned in the description, processes and intermediates for their preparation, pharmaceutical...
5021414 Phenol derivatives  
A phenol derivative of the formula NU--A--X--R 1 wherein NU is a defined bis-phenolic nucleus including a hydroxyphenyl-hydroxynaphthyl; hydroxyphenyl-hydroxyindanyl,...
5006158 Certain 2-(2-substituted benzoyl)-1,3-cyclohexanediones  
Compounds of the formula ##STR1## wherein R 1 is hydrogen or C 1 -C 4 alkyl; R 2 is hydrogen, C 1 -C 4 alkyl or ##STR2## wherein R a is C 1 -C 4 alkyl; R 1 and R 2 together are alkylene...
5003101 Acrylates and fungicides containing them  
and fungicides containing these compounds.
5001152 Use of catechol-O-methyl transferase (COMT) inhibitors and their physiologically acceptable salts for ulcer treatment  
The invention is concerned with the new use of known catechol derivatives of the formula ##STR1## wherein R 1 and R 2 are each hydrogen, alkyl having 1 to 4 carbon atoms or alkanoyl having 2 to 5...
4983628 Leukotriene antagonists  
Compounds having the formula: ##STR1## are antagonists of leukotrienes of C 4 , D 4 and E 4 , the slow reaction substance of anaphylaxis. These compounds are useful as anti-asthmatic,...
4954160 Oximino ether compounds  
The invention provides compounds of the general formula ##STR1## wherein R represents a hydrogen atom, or an optionally substituted alkyl or acyl group, or an alkenyl or alkynyl group or an...
4939170 Substituted aminophenyl carbamates  
Fungicidal substituted aminophenyl carbamates of the formula ##STR1## in which X represents --CO--NR 8 R 9 ; --CO--OR 9 ; --CO--SR 9 ; --CO R 10 ; --SO 2 R 9 or hydrogen, in which R 8 ...
4935517 Sweetening agents derived from N-hydrocarbon-substituted L-aspartic and L-glutamic acids  
Sweetening agents of the general formula: ##STR1## wherein R is a saturated or unsaturated, acyclic, cyclic or mixed hydrocarbon group having 5 to 13 carbon atoms, wherein R' is, in a preferred...
4933367 Carboxylic acid derivatives, processes for the preparation thereof, the use thereof, and pharmaceutical compositions which contain these compounds  
This invention relates to carboxylic acid derivatives and their use thereof. The compounds are useful in treatment of various diseases such as diabetes, prediabetic conditions, adipositas ailments...
4921632 Liquid crystal compounds and compositions  
Liquid Crystal compounds represented by the following formula are disclosed. ##STR1## wherein R and R' are independently selected from alkyl groups containing 1.about.20 carbon atoms; X is --O--,...
Matches 1 - 50 out of 138 1 2 3 >