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7598416 |
4-((phenoxyalkyl)thio)-phenoxyacetic acids and analogs
The invention features 4-((phenoxyalkyl)thio)-phenoxyacetic acids and analogs, compositions containing them, and methods of using them as PPAR modulators to treat or inhibit the progression of, for...
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7598292 |
4-((phenoxyalkyl)thio)-phenoxyacetic acids and analogs
The invention features 4-((phenoxyalkyl)thio)-phenoxyacetic acids and analogs, compositions containing them, and methods of using them as PPAR delta modulators to treat or inhibit the progression...
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7597825 |
Method of quenching electronic excitation of chromophore-containing organic molecules in photoactive compositions
The photostabilizing electronic excited state energy—particularly singlet state energy from a UV-absorbing molecule has been found to be readily transferred to (accepted by)...
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7588702 |
Method of quenching electronic excitation of chromophore-containing organic molecules in photoactive compositions
The photostabilizing electronic excited state energy—particularly singlet state energy from a UV-absorbing molecule has been found to be readily transferred to (accepted by)...
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7560585 |
Process for preparing (S)- alpha-cyano-3-phenoxybenzyl-(S)-2-(4-chlorophenyl)-isovalerate
The present invention relates to an environmentally benign process for the preparation of (S)-α-cyano-3-phenoxybenzyl-(S)-2-(4-chlorophenyl)isovalera
te from its diastereomeric mixture...
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7517896 |
Aminodicarboxylic acid derivatives having pharmaceutical properties
The invention relates to compounds of formulae (II), (IV), and (VI) as shown below,
wherein the several variable groups are as defined in the specification and claims. Processes for making...
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7507852 |
Process for preparing gamma-cyhalothrin
A process for the preparation of gamma-cyhalothrin comprising steps of a) chlorinating 1R cis-Z 3-(2-chloro-3,3,3-trifluoro-1-propenyl)-2,2-dimethyl cyclopropanecarboxylic acid to give 1R cis-Z...
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7476759 |
Matrix metalloproteinase inhibitors
Compounds of Formula (I):
wherein: R 1 is optionally substituted —C 4-12 alkyl, —C 2-10 alkylcycloalkyl, —C 2-6 alkylheterocycloalkyl, —C 2-6 alkylaryl, optionally substituted 5-...
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7470723 |
Diphenylethylene compounds and uses thereof
The present invention relates to Diphenylethylene Compounds and compositions comprising a Diphenylethylene Compound. The present invention also relates to methods for preventing or treating various...
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7425649 |
4-((phenoxyalkyl)thio)-phenoxyacetic acids and analogs
The invention features 4-((phenoxyalkyl)thio)-phenoxyacetic acids and analogs, compositions containing them, and methods of using them as PPAR modulators to treat or inhibit the progression of, for...
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7368479 |
Alpha-sulfonylamino-acetonitriles
The invention relates to α-sulfonylamino-acetonitrile derivatives of the general formula (I) including the optical isomers thereof and mixtures of such isomers, wherein Ar 1 , and Ar 2 ...
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7297816 |
Sulfonamide compounds
Certain sulfonamide compounds are dual CCK1/CCK2 inhibitors useful in the treatment of CCK1/CCK2 mediated diseases.
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7279478 |
Cathepsin cysteine protease inhibitors
This invention relates to class of compounds which are cysteine protease inhibitors, including but not limited to, inhibitors of cathepsins K, L, S and B. These compounds are useful for treating...
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7232923 |
Method of hydroaminating N-alkenoylcarbamates with primary aromatic amines
The invention provides methods for hydroaminating N-alkenoyl carbamates with aromatic amines.
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7223988 |
Color tunable photoluminescent blends
Embodiments of the present invention are directed toward a photoluminescent article comprising at least one host material and at least one color tunable photoluminescent dye. In certain...
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7166746 |
N-bisaryl- and n-aryl-cycloakylidenyl-αhydroxy-and α-alkoxy acid amides
The invention relates to N-bisaryl- and N-aryl-cycloalkylidenyl-a-hydroxy- and a-alkoxy acetic acid amides of the general formula (I) including the optical isomers thereof and mixtures of such...
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7153813 |
Substituted aryl ketones
The invention relates to novel substituted aryl ketones of the formula (I)
in which Z, X, R and n are as defined in the disclosure, to processes for their preparation and to their use as...
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6949669 |
Organic compounds
Compounds of general formula (I) wherein the substituents are as defined in claim 1 are suitable for use as herbicides
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6768019 |
3,4-dihydro-1H-naphthalene derivatives as a highly selective cyclooxygenase-2 inhibitor
The present invention relates to a novel 3,4-dihydro-1H-naphthalene derivative having a structure of formula 1 or formula 2, its pharmaceutically acceptable salts and their geometric isomers as a...
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6686493 |
3,4-dihydro-1H-naphthalene derivatives as a highly selective cyclooxygenase-2 inhibitor
The present invention relates to a novel 3,4-dihydro-1H-naphthalene derivative having a structure of formula 1 or formula 2, its pharmaceutically acceptable salts and their geometric isomers as a...
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6667412 |
Nitrile compound
The present invention provides a novel nitrile compound useful as an intermediate for the production of, for example, N,N-substituted cyclic amine derivatives or phenylacetonitrile derivatives that...
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6444838 |
Process for the preparation of 1,4-diaryl-2-fluoro-4-cyano-2-butenes and intermediates useful therefor
The present invention provides a process for the preparation of pesticidal 1,4-diaryl-2-fluoro-4-cyano-2 -butene compounds having the structural formula I and intermediates useful therefor.
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6399776 |
Processes and intermediates in the synthesis of 5-(3-exo-bicyclo&lsqb 2.2.1&rsqb hept-2-yloxy-4-methoxyphenyl)-3,4,5,6-tetrahydropyrimidine-2(1H)-one
This invention relates to novel processes for preparing the pharmaceutically active compound 5-(3-[(2S)-exo-bicyclo[2.2.1]hept-2-yloxy]-4-methoxyphenyl)-
3,4,5,6-tetrahydropyrimidin-2(1H)-one and...
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6242634 |
Pyrimidin-4-one derivatives, their use, intermediates for their production, and processes for producing these intermediates
Novel pyrimidin-4-one derivatives of formula [1] are provided, which are useful as active ingredients of herbicides, wherein R 1 is hydrogen or alkyl; R 2 is alkyl optionally substituted with...
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6225491 |
Method for preparing certain acetonitriles
The invention relates to a process for making certain acetonitriles.
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6207837 |
Process for producing dibenzo[b,f]thiepine derivatives
Efficient synthesis of diaryl sulfide derivatives useful as intermediates for pharmaceutical compounds. Provision of a convenient process for producing large quantities of dibenzo[b,f]thiepine...
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6197993 |
Naphthyloxyacetic acid derivatives and a pharmaceutical composition comprising them as an active ingredient
The naphthyloxyacetic acid derivatives of the formula (I) ##STR1## wherein A is H, -(alkylene)COOR 1 , -(alkylene)CONR 2 R 3 , -(alkylene)OH, -(alkylene)tetrazole, -(alkylene)CN; E is single bond...
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RE37087 |
Insecticidal triffluormethyl alkane derivatives
There are provided new alkane and alkoxyalkane derivatives of the general formula I ##STR1## in which R 1 , R 2 , R 3 , R 4 and A have the meanings given in the description, processes for their...
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5968908 |
Restricted 9-cis retinoids
The invention is novel analogs of 9-cis-retinoic acid which are useful for the treatment and prevention of coronary artery disease and to protect against premature atherosclerosis by increasing HDL...
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5846999 |
Substituted N-arylmethylamino derivatives of cyclobutene-3,4-diones
The compounds of the formula: ##STR1## wherein R 1 is straight chain alkyl, branched chain alkyl, cycloalkyl, hydroxyalkyl, fluoroalkyl or polyfluoroalkyl; R 2 and R 3 are, independently,...
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5760275 |
Cyanoacetals by hydroformlation of unsaturated nitriles in the presence of orthoesters
Disclosed is an improved process for producing cyanoaldehydes and acetals wherein an α, β-unsaturated nitrile is reacted with carbon monoxide and hydrogen in the presence of a Group 8 metal...
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5633405 |
Asymmetric synthesis of (-)-6-chloro-4-cyclopropyl-ethynyl-4-trifluoromethyl-1,4-dihydro-2H-3,1- benzoxanzin-2-one
An improved synthesis of a highly potent HIV reverse transcription inhibitor is disclosed, involving an acetylide and a trifluoromethyl ketone which produces a chiral product in the presence of a...
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5627284 |
Process for producing (E)-alkoxyimino or hydroxyiminoacetamide compounds and intermediates therefor
The present invention relates to a process for producing (E)-alkoxyiminoacetamide compounds useful as agricultural fungicides and a process for producing (E)-hydroxyiminoacetamide compounds useful...
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5563161 |
Alcohols and ethers with aromatic substituents as tachykinin-antagonists
Compounds of formula (I), and salt and prodrugs thereof, wherein Q is optionally substituted phenyl or benzhydryl; R 1 is H; optionally substituted C 1 -6 alkyl; optionally substituted phenyl(C 1...
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5536865 |
Process for the preparation of 5,6-dihydroxyindole and intermediate compounds
Process for the preparation of 5,6-dihydroxyindole, wherein the compound of formula: ##STR1## in which R' denotes a hydrogen atom or an optionally substituted benzyl radical, is subjected either to...
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RE35230 |
Enantiomeric enrichment of cyanohydrins
A method of enantiomerically enriching chiral cyanohydrins is disclosed that involves selective cleavage of the unwanted enantiomer into its cleavage products HCN and the corresponding aldehyde or...
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5446067 |
Oxime ethers and fungicides containing them
Oxime ethers of the formula ##STR1## wherein m, G, R, R 1 , X, Y, and Z are as defined herein and fungicides containing these compounds.
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5442063 |
Process for producing (E)-alkoxyimino or hydroxyimino-acetamide compounds and intermediates therefor
The present invention relates to a process for producing (E)-alkoxyiminoacetamide compounds useful as agricultural fungicides and a process for producing (E)-hydroxyiminoacetamide compounds useful...
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5380755 |
Alkyl and alkylbenzyl ethers of substituted hydroquinones
The present invention provides alkyl and alkylbenzyl ethers of substituted hydroquinones and pharmaceutical compositions containing them. The present invention further provides methods of using...
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5329023 |
Method of preparing optically active alcohols which consist substantially or entirely of one enantiomer
The invention relates to a method of preparing optically active alcohols which consist substantially (at least 75% e.e.) or entirely of one enantiomer of formula 4 ##STR1## wherein R and A are as...
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5312957 |
Enantioselective hydrocyanation of aromatic vinyl compounds
The invention provides a process for enantioselective hydrocyanation of aromatic vinyl compounds which produces nonracemic mixtures of chiral, arylpropionitriles; novel carbohydrate phosphorus and...
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5248834 |
Pesticides
Pesticidal compounds of formula I I: R A CR 3 CR 4 CHDR B in which formula: R A represents a group ArCR 1 R 2 - in which Ar represents a phenyl or naphthyl group optionally...
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5234894 |
Carbonyl acetonitrile derivative and herbicide containing it as an active component
A cyanoketone derivative of the following formula (1) ##STR1## wherein A 1 is a substituted or unsubstituted phenyl or naphthyl group or a substituted or unsubstituted heterocyclic group; each...
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5223536 |
1,4-diaryl-1-cyclopropyl-4-substituted butanes as insecticides and acaricides
The 1,4-diaryl-1-cyclopropyl-4-substituted butane pesticides of the following formula are effective as insecticides and acaricides: ##STR1## in which X and Y are independently hydrogen, halogen,...
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5220048 |
Substituted benzocyclobutenes, a process for their preparation and their use
Benzocyclobutene-1,2-dichlorides, -bromides and -iodides which are substituted in the benzene ring are accessible in good yields and short reaction times by reacting substituted 1,2-(dichloromethyl...
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5204468 |
Substituted 4,5,6,7-tetrahydrothiens[2,3-C]pyridine compounds
This invention provides the single species (-)-(S)-4-(3,4-dihydroxyphenyl)-7, 8-dihydroxy-1,2,3,4-tetrahydroisoquinoline hydrochloride hydrate, which is useful as a nephrovascular dilator.
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5196562 |
Substituted 1,3,5-triazinetriones, for use against parasitic protozoa
Protecting against parasitic protozoa with substituted 1,3,5-triazinetriones of the formula ##STR1## in which R 1 represents aromatic or heteroaromatic radicals, each of which is optionally...
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5187296 |
Cyanohydrination process
A process for the assymetric cyanohydrination of m- phenoxybenzaldehyde with HCN, using a catalytically effective amount of enantiomeric cyclo(phenylalanylhistidine) absorbed on a solid support...
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5169991 |
Compound
A compound is a condensate of 1,2,3-trihydroxybenzene with an aldehyde. The condensate is a macrocyclic compound such as a cyclic tetramer. The aldehyde is preferably a long-chain aldehyde such as...
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5147892 |
Benzyl ketones and fungicides containing them
Benzyl ketones of the formula ##STR1## where X is CH or N, Y is O or NR 4 , R 1 , R 2 are H or alkyl, R 3 is halogen, cyano, nitro, alkyl, cycloalkyl, alkoxy, haloalkyl, arylalkyl,...
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