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8138216 |
Cannabinoid receptor antagonists/inverse agonists useful for treating metabolic disorders, including obesity and diabetes
The present invention provides novel pyrazoles that are useful as cannabinoid receptor antagonists and pharmaceutical compositions thereof and methods of using the same for treating obesity,...
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8101749 |
Process for the preparation of onium salts with a tetrafluoroborate anion having a reduced halide content
The invention relates to a method for producing onium salts with tetrafluoroborate anion by reacting an onium halide with an oxonium tetrafluoroborate, sulfonium tetrafluoroborate, or...
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8003626 |
Pyrazole-4-carboxamide derivatives as microbiocides
Compounds of the formula I in which the substituents are as defined in claim 1 are suitable for use as microbiocides.
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7998996 |
Substituted pyrazoline compounds for reducing triglycerides in blood
The present invention relates to substituted pyrazoline compounds, methods for their preparation, medicaments comprising these compounds as well as their use for the preparation of a medicament for...
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7968582 |
5(S)-substituted pyrazoline compounds, their preparation and use as medicaments
The present invention relates to substituted pyrazoline compounds, methods for their preparation, medicaments comprising these compounds as well as their use for the preparation of a medicament for...
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7718687 |
Prodrugs of mitotic kinesin inhibitors
The present invention relates to prodrugs of dihydropyrazole compounds that are useful for treating cellular proliferative diseases, for treating disorders associated with KSP kinesin activity, and...
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7705160 |
Method for preparing 3-halo-4,5-dihydro-1H-pyrazoles
This invention relates to a method for preparing a 3-halo-4,5-dihydro-1H-pyrazole compound of Formula I comprising contacting with HX1 a different 4,5-dihydro-1H-pyrazole compound of Formula II...
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7504519 |
Derivatives of pyrazoline, procedure for obtaining them and use thereof as therapeutic agents
The invention relates to derivatives of general formula (I), and to their pharmaceutically acceptable salts, their stereoisomeric forms, preferably their pure enantiomeric or diastereomeric forms...
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7335780 |
Method for preparing 3-halo-4,5-dihydro-1H-pyrazoles
This invention relates to a method for preparing 3-halo-4,5-dihydro-1H-pyrazole compound of Formula (I), comprising contacting with HX1 a different 4,5-dihydro-1H-pyrazole compound of Formula (II),...
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RE39681 |
1-(4-sulfamyaryl)-3-substituted-5-aryl-2-pyrazolines and inhibitors of cyclooxygenase-2
Compounds of the formula wherein: X is selected from the group consisting of trihalomethyl, C1-C6 alkyl, and a group of formula II: wherein: R3 and R4 are independently selected from the group...
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6852750 |
Benzenedicarboxylic acid derivatives
New benzenedicarboxylic acid derivative compounds; pharmaceutical compositions, diagnostic methods, and diagnostic kits that include those compounds; and methods of using those compounds for...
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6831075 |
Heterocyclic substituted pyrazolones
The present invention is directed to novel heterocyclic substituted pyrazolones, including pharmaceutical compositions, diagnostic kits, assay standards or reagents containing the same, and methods...
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6774229 |
Coupling condensation synthesis of heterocycles
The invention relates to a process for the preparation of heterocycles, characterised in that the following components: i) a propargyl derivative of the general structural formula I a wherein Het...
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6689770 |
Aryl sulfonyls as factor Xa inhibitors
The present application describes aryl sulfonyls of formula I: or pharmaceutically acceptable salt or prodrug forms thereof, wherein D, E, and M are defined below, are effective factor Xa inhibitors.
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6617342 |
Hypoglycemic sulfonyl pyrazolones and pyrazolines
This invention provides compounds and their pharmaceutically acceptable salts, pharmaceutical formulation of said compounds and methods for treating hyperglycemia associated with non-insulin...
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6376519 |
1-(4-sulfamylaryl)-3-substituted-5-aryl-2-pyrazolines and inhibitors of cyclooxygenase-2
Compounds of the formula wherein:X is selected from the group consisting of trihalomethyl, C1-C6 alkyl, and a group of formula II: wherein:R3 and R4 are independently selected from the group...
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6242609 |
Method for manufacturing a color coupler used in a silver halide photographic light-sensitive material
A method for manufacturing a color coupler used in a silver halide photographic light-sensitive material using an ammonium trihalide.Said method for manufacturing the color coupler comprising the...
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6004903 |
2-Anylocyclohexanediones having improved herbicidal properties
Benzoyl derivatives of the formula I ##STR1## where Z is a 5-membered or 6-membered heterocyclic, saturated or unsaturated radical containing one to three hetero atoms selected from the group...
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5789597 |
Process for the preparation of compounds having ACE inhibitory action and intermediates in said process
There is disclosed a process for the preparation of compounds having ACE inhibitory action of the formula ##STR1## wherein R has the meanings as in claim 1, wherein the stereospecific amino acid N-...
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5783576 |
Benzoyl guanidine derivatives, the preparation thereof and their use in pharmaceutical compositions
New compounds of general formula (I) are provided: ##STR1## which are explained in the specification can be prepared by a variety of methods. The compounds may be used in pharmaceutical compositions.
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5728839 |
Metal complexes with heterocycles carbenes
A complex of the formula La Mb Xc !n (A)n Ias described in the application useful as homogenous catalysts.
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5510361 |
Di-tert-butylphenol compounds with heterocyclic moiety, useful as anti-inflammatory agents
The subject invention relates to compounds having the structure: ##STR1## wherein a) each R is independently alkyl having from 1 to about 7 carbon atoms; b) Z is O or N--X; c) X is selected from...
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5366991 |
Pyrazolecarboxamides exhibiting insecticide and acaricide activity
5-pyrazolecarboxylic acid amide-based insecticide and acaricide compounds of general formula (I): ##STR1## in which: R1 represents a hydrogen atom, a linear or branched C1 -C4 alkyl group or a...
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5208251 |
Styryl pyrazoles, isoxazoles and analogs thereof having activity as 5-lipoxygenase inhibitors, pharmaceutical compositions and methods of use therefor
The present invention is 3,5-substituted, isoxazoles, pyrazoles, isothiazoles, and analogs thereof having 5-lipoxygenase or cyclooxygenase inhibiting activity or as a sunscreen.
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5152824 |
Sulfamidosulfonamide derivatives and herbicides
A sulfamidosulfonamide derivative of the formula (1) and an agriculturally suitable salt thereof: ##STR1## wherein Q is ##STR2## X is an oxygen atom or a sulfur atom; and G is ##STR3## which are...
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4992203 |
Non-linear optics
Optical elements having non-linear optical properties comprising a compound of the formula: ##STR1## wherein D is an electron donor A is an electron acceptor;and W, X, Y and Z are each...
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4897223 |
Tri-phenyl methyl color-forming agents
Color-forming agents of the general formula ##STR1## wherein X denotes hydroxyl, alkoxy, alkenyloxy, aralkoxy, cycloalkoxy, aryloxy, acyloxy, alkoxycarbonyloxy, alkylamino, dialkylamino, acylamino,...
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4788293 |
Preparation of 1-pyrazolines
1-Pyrazolines are prepared by oxidation of a 1,3-diamine with sodium hypochlorite and a peroxide in aqueous solution.
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4749701 |
Aminostyryl compound, leukotriene antagonistic composition containing the same as effective ingredients and method of antagonizing SRS by employing the same
Disclosed are an aminostyryl compound represented by Formula I: ##STR1## wherein A represents a linking group having 3 to 4 chain members; B represents an unsubstituted or substituted 5 to...
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4654431 |
Photopolymerizable thioacrylate monomers
A novel photocurable monomer having the formula: ##STR1## wherein: Ar is arylene; R1 is H, alkyl, alkoxy, amino, halogen, sulfide, sulfoxide, sulfonate, aryl or heterocyclic; R2 is H, alkyl, aryl...
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4551528 |
Carrying out organic condensation reactions at elevated temperatures by feeding the starting materials into the bottom of a reactor charged with mineral oil followed by product distillation
Organic condensation reactions are carried out at elevated temperatures by a method in which the starting material or materials are fed in, in gaseous form, at the bottom of a reactor charged with...
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4273937 |
Organic amine compositions
Organic amine compositions which are substantially free of nitrosamine contaminants are provided which comprise an organic amine and an inhibiting amount of an inhibitor additive selected from the...
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4239901 |
Pyrazol-1-ylphenylacetic acids
Pyrazol-1-ylphenylacetic acids of the formula ##STR1## wherein R1, R2 and R3 are the same or different and denote a hydrogen atom or a halogen atom, R4 denotes a hydrogen atom or an alkyl group, A...
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4152517 |
Synthesis of 6-(2-hydroxyphenyl)-3(2H)-pyridazinones from trihalocarbinols
A new synthesis for the preparation of 6-(2-hydroxyphenyl)-3-pyridazinones whose key reaction is cyclizing a 1,1,1-trihalo-2-hydroxy-4-(2-hydroxyphenyl)-1-butanone with hydrazine....
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4115413 |
Triaryl-methane dyestuffs
Triaryl-methane dyestuffs which are free from sulfonic acid and carboxylic acid groups and are selected from the group consisting of dyestuffs having one of the following four formulae: ##STR1##...
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4112231 |
Process for the condensation of epoxides with organic compounds having an active hydrogen
A process is provided for the condensation of epoxides with organic compounds having an active hydrogen atom, such as alcohols, polyols, and amines, in the presence of a neutral inorganic salt...
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3931406 |
Pyrazolidine fungicides
There is provided a method for protecting plants from attack by fungi by applying to said plants a fungicidally effective amount of a pyrazolidine and acid salt derivatives thereof.
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3925408 |
Pyrazolinium compounds as herbicides
This invention provides for 1,2-dialkyl-3,5-disubstituted and -3,4,5-trisubstituted pyrazolinium salts, a method for the preparation of the said compounds, and a method for controlling undesirable...
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3896143 |
Substituted pyrazolyl phenylacetic acid derivatives
Substituted pyrazolyl phenylacetic acid derivatives, e.g. 2-pyrazolin-3-yl and pyrazol-3-yl-phenyl acetic acids and phenyl acetamides are prepared by reacting a crotonoyl or cinnamoyl phenylacetic...
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3871898 |
PROCESS FOR THE OPTICAL BRIGHTENING OF ORGANIC FIBRE MATERIAL
A process for the non-aqueous optical brightening of organic fibre material, especially fibre material made from cellulose, natural or synthetic polyamide, by the exhaustion method, is disclosed,...
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3697501 |
BASIC INDAZOLE AZO DYE SUBSTITUTED BY A SULFONAMIDE GROUP
A basic azo dye of the formula ##SPC1## Wherein: R1 is methyl or ethyl, R2 is amino or a substituted amino radical, X is an anion, Y is the radical of the formula ##SPC2## R3 being cyclohexyl,...
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3666772 |
PREPARATION OF PYRAZOLINES BY CYCLIZATION OF AN AZINE
Alkyl substituted pyrroles and pyrazolines are prepared by treating a ketazine or aldazine with a metal halide of the formula MX2 where M is cobalt or nickel and X is a halogen at a temperature of...
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3530183 |
DIBENZOCYCLOHEPTENES
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3772328 |
PREPARATION OF PYRROLES BY CYCLIZATION OF AZINES
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3833655 |
AMINO-DIBENZO(A,D)CYCLOHEPTA(1,4)DIEN-5-ONE COMPOUNDS
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3657231 |
OLIGOMERIC OPTICAL BRIGHTENING COMPOUNDS
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3826800 |
BASIC INDAZOLE AZO COMPOUNDS
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3560216 |
LIGHT SENSITIVE FREE RADICAL IMAGING MATERIAL CONTAINING PYRAZOLINE SENSITIZERS
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3686162 |
MONOAZO DYESTUFFS CONTAINING A BENZTHIAZOLYL RADICAL
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3478048 |
2,3;3A,12B - TETRAHYDRO - 8H - DIBENZO (3,4;6,7)CYCLOHEPT(1,2-D)OXAZOLES AND DERIVATIVES
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