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7202367 Process for arylating or vinylating or alkynating a nucleophilic compound  
The present invention concerns a process for arylating or vinylating or alkynating a nucleophilic compound. More particularly, the invention concerns arylating nitrogen-containing organic...
7084178 Antiamyloid phenylsulfonamides: N-cycloalkylcarboxamides derivatives  
A series of N-cycloalkylcarboxamide derivatives of N-benzyl benzenesulfonamides of Formula I are described. The compounds inhibit β-amyloid peptide (β-AP) production and are useful in the...
6864373 Stable amorphous celecoxib composite and process therefor  
A process is provided for preparing a celecoxib-crystallization inhibitor composite wherein at least a detectable amount of celecoxib is in amorphous form. Also provided are compositions prepared...
6838458 5-(alkylidene-cycloalkyl)-and 5-(alkylidene-heterocyclyl)-pyrazoles  
The present invention relates to 5-(alkylidene-cycloalkyl)-pyrazoles and 5-(alkylidene-heterocyclyl)-pyrazoles of the formula I: wherein the ring of the formula (R 5 )-A-(SO m R 4 ), m, B,...
6689805 Pyrazole-3-one derivative, method for preparing the same, and pharmaceutical composition containing the same  
A pyrazole-3-one derivative of formula 1 or a non-toxic salt thereof, a preparation method thereof, and a pharmaceutical composition containing the derivative or the salt as an active ingredient...
6562856 Pyrazolyl benzyl ether deriviatives having a fluoromethoxy group and the use thereof as pesticides  
The invention relates to novel pyrazolyl benzyl ethers, to a process for their preparation and to their use for controlling harmful organisms.
6518266 1- Aryl-3-thioalkyl pyrazoles, the synthesis thereof and the use thereof as insecticides  
The present invention is directed to novel pyrazole derivatives and their use as pesticidal agents. The pyrazole derivatives have Formula I: or a salt thereof, where R 1 represents R 5 O, R 5...
6322775 Cosmetic compositions containing pyrazolin-4,5-diones, novel pyrazolin-4,5-diones, preparation methods therefor and uses thereof  
The present invention relates to novel cosmetic compositions, in particular for coloring the skin and/or the hair, comprising, in a cosmetically acceptable support, at least one...
6242612 Process for making substituted pyrazoles  
This invention relates to a novel process of preparing selected 5-substituted pyrazoles useful as p38 kinase and COX-2 inhibitors.
H001942 Herbicidal 3-(pyrazolylphenyl)propanoic acids and derivatives  
Novel herbicidal compounds, compositions containing them, and methods for their preparation and use in controlling weeds are disclosed. The novel herbicidal compounds are...
6133451 Method for producing 2-(3-pyrazolyl-oxymethylene) nitrobenzenes  
2-(3-Pyrazolyloxymethylene)nitrobenzene [sic] derivatives of the formula I ##STR1## where the substituents and indices have the meanings given in the description, are prepared by bromination of an...
6107487 Methine and azamethine dyes based on 5-membered heterocycles with a trifluoromethyl group  
Dyes of the formula Q-X=Het where X is nitrogen or CH, Q is a 5- or 6-membered carbocyclic or heterocyclic radical and Het is a radical of the formula ##STR1## where Y is oxygen, sulfur,...
6054592 2-((Dihydro) pyrazol-3'-yloxymethylenes  
2-[(Dihydro)pyrazol-3'-yloxymethylene]anilides of the formula I ##STR1## processes and intermediates for their preparation and their use as pesticides and fungicides.
6040458 Method for producing N-substituted 3-hydroxypyrazoles  
6028093 Fungicide compositions  
5958838 Arylheterocycles with herbicidal activity  
Arylheterocycles having the general formula (I): ##STR1## and process for preparing them. The arylheterocycles having the general formula (I) display high herbicidal activity.
5935986 Azolyl oxybenzyl alkoxyacrylic acid esters, process for producing them and their use  
There are described compounds of the general formula I ##STR1## in which the index and the substituents have the following meanings: n is 0, 1, 2, 3 or 4; R is nitro, cyano, halogen, ...
5886175 7-(substituted)-8-(substituted)-9-(substitued amino)-6-demethyl-6-deoxytetracyclines  
The invention provides compounds of the formulas ##STR1## which are useful as intermediates for the preparation of 6-demethyl-6-deotetracycline antibiotic agents.
5883112 Synergistic compositions comprising pesticidal 5-amino-4-ethylsulfinyl-1-arylpyrazoles and piperonyl butoxide  
The invention relates to a synergistic pesticidal composition comprising: (a) a pesticidally effective amount of a compound having the formula: ##STR1## wherein X is chlorine or bromine, Y is...
5869517 2- (dihydro)pyrazol-3'-yloxymethylene!anilides, their preparation and their use  
The invention concerns 2- (dihydro)pyrazolyl-3'-oxymethylene!-anilides of formula (I) in which -- is a single or double bond and the subscripts and substituents are as follows: n 0, 1, 2, 3 or 4; m...
5859259 Activated esters of 1-phenylpyrazolin-5-one for labeling amine-functionalized molecules  
The disclosed invention is drawn to pyrazolinone derivatives, and methods of use thereof, for non-radioactive labeling of amine-functionalized molecules, especially biomolecules such as DNA, RNA,...
5795907 Gastin and CCK receptor ligands  
Compounds of formula (Ia), (Ib), or (Ic), wherein A represents a group having two fused rings, or a group of formula (Id), R 1 (m) represents up to 6 substituents, K represents --O--, --S--, --CH 2...
5789618 Synthetic method for a halogen-containing condensation product  
A method for synthesizing a halogen-containing condensation product, the method comprising the step of: reacting a compound represented by Formula (I) with a compound represented by Formula (II)...
5739083 Pyrazole derivatives and insecticidal compositions containing the derivative as active component  
A pyrazole derivative represented by the formula (1) is low in toxicity and persistence and yet has an extremely high insecticidal efficacy ##STR1## wherein A is CH, N or C-halogen atom, R 1 is...
5707936 Methyl α-phenylbutenoates  
Methyl α-phenylbutenoates of the formula I ##STR1## where -- is a single or double bond and the index and the substituents have the following meanings: n is 0, 1, 2, 3 or 4; R 1 is nitro,...
5663365 Process for the preparation of pyrazolones  
A process for the preparation of pyrazolone derivatives represented by the general formula ##STR1## wherein R is a hydrogen atom, an alkyl group, an allyl group, an aryl group or an aralkyl group,...
5591833 Colorants and intermediates therefor having branched poly(oxyalkylene)moieties, and their manufacture  
Colorants and compositions useful as a fugitive or permanent colorant for a variety of substrates, or as intermediates for their manufacture, and having one or more improved properties of enhanced...
5559244 Preparation of 1-(het) aryl-3-hydroxypyrazoles  
A process for preparing 1-(het)aryl-3-hydroxypyrazoles of the formula I ##STR1## where R is an unsubst. or subst. aromatic or heteroaromatic radical, n is 0, 1 or 2 and R' is a group which is...
5495032 Process for producing 7-(substituted)-8-(substituted-9-[(substituted glycyl)amido]-6-demethyl-6-deoxytetracyclines  
The invention provides a process for the production of compounds of the formula: ##STR1## wherein, R, R 3 , R 4 , X and W are defined in the specification in which a compound of the following...
5430158 Pyrazole derivatives  
An anilin derivative which corresponds to the following formula: ##STR1## wherein, R 2 is hydrogen, lower alkoxy group, a nitro group, or one or more halogen atoms selected from fluorine, chlorine...
5306562 Xanthenylamide handle for use in peptide synthesis  
The preparation and properties of xanthenylamide handles for use in peptide synthesis is disclosed. The compounds, omega-(9-(9-fluorenylmethyloxycarbonyl)aminoxanthan-2-oxy)al kanoic acid...
5250700 Phenyl pyrazolidinones as bronchodilators and anti-inflammatory agents  
There are disclosed compounds of the formula ##STR1## wherein R 1 is hydrogen or lower alkyl; R 2 is C 3 -7 alkyl or C 3 -7 cycloalkyl; R 3 is hydrogen, lower alkyl, carboxyloweralkyl,...
5233044 Active esters for solid phase peptide synthesis  
Derivatives of 1-phenyl pyrazolin-5-one have many applications for biomolecule synthesis. Enol esters of protected amino acids made by the present process provide efficient coupling in solid-phase...
5206242 Diaryl-substituted pyrazole compounds and drugs and cosmetics obtained therefrom  
Compounds of formula I ##STR1## where R 1 and R 2 are each hydrogen or methyl, A is en ethylene or methylene radical which is unsubstituted or substituted by methyl, hydroxyl or oxo, L is a...
5202442 Process for preparing pyrazolecarboxylic acid compounds  
A process for preparing a pyrazolecarboxylic acid compound of the formula (II): ##STR1## wherein Y and Z each represent a hydrogen, a halogen, a nitro, a cyano, COOR 1 , NR 1 R 2 , CONR 1 R 2 ,...
5136045 Pyrazole containing methine compounds  
A methine compound represented by the following formula and an agent containing the same for coloring resins such as polystyrene, ABS. ##STR1## wherein R 1 is a hydrogen atom, a lower alkyl group,...
5134142 Pyrazole derivatives, and pharmaceutical composition comprising the same  
The present invention concerns pyrazole derivatives of formula: ##STR1## used for the treatment of inflammation, pain, thrombosis and rheumatism.
5122611 Method of producing azomethine or indoaniline series dyes  
A method for producing an azomethine or indoaniline series dye, which comprises oxidatively condensing an active methylene- or methine-containing compound, except those containing a sulfonic or...
4950678 Substituted N-(heterocyclic-substituted phenyl)-N'-benzylureas  
Novel substituted N-(heterocyclic-substituted phenyl)-N'-benzoyl-ureas, processed for producing these compounds, intermediates therefor, compositions thereof and the use of the compounds for the...
4909827 Herbicidal compositions based on substituted pyrazolin-5-one derivatives and use thereof  
The invention relates to the use of partly known substituted pyrazolin-5-one derivatives of the formula (I) ##STR1## as herbicides and fungicides, new substituted pyrazolin-5-one derivatives and...
4826867 Substituted 1-aryl-3-tert.-butyl-pyrazoles  
Insecticidally and acaricidally active novel 1-aryl-3-tert.-butyl-pyrazoles of the formula ##STR1## in which R 1 represents nitro or halogen, R 2 represents halogen or the --NR 3 R 4 group,...
4808210 Herbicidal method of using 5-pyrazolones  
A 5-pyrazolone of the formula ##STR1## wherein R is selected from the group consisting of mono- and polycyclic aromatic of 6 to 14 carbon atoms, heterocyclic optionally substituted with phenyl,...
4643757 Herbicidal 4-benzoyl-1-methyl-5-hydroxypyrazoles  
Pyrazole derivatives, selective herbicidal compositions containing said derivatives and the use of said derivatives are provided. The pyrazole derivatives having selective herbicidal activity are...
4567139 Chromogen for measuring the formation of hydrogen peroxide based on 1-substituted-aminoantipyrin compounds  
Compounds of the general formula ##STR1## wherein R represents an alkyl group of 1 to 3 carbon atoms or the group N(R 2 ) 2 , in which R 2 represents a hydrogen atom, an alkyl group of 1 to 3...
4545806 5-(Oxo or thio heterocycle) cyclohexane-1,3-dione derivatives and their use for controlling undesirable plant growth  
Cyclohexane-1,3-dione derivatives of the formula ##STR1## where A is an unsubstituted or substituted, saturated or unsaturated 4-membered to 7-membered heterocyclic structure which contains from 1...
4522917 Photographic silver halide light-sensitive material  
A photographic silver halide light-sensitive material is disclosed. The material is comprised of a support and a photographic layer or layers on the support. The photographic layer contains at...
4515801 Fungicidally active pyrano-pyrazole derivatives  
Pyrano-pyrazole derivative of the formula ##STR1## in which R 1 represents hydrogen, alkyl, alkanoyl, alkoxycarbonyl, optionally substituted phenyl or optionally substituted phenylalkyl, R 2 ...
4489002 Azo compound and an azomethine compound and having a tertiary N-dative bond  
Compounds of the general formula I ##STR1## where E is --CH or --N, K is the radical of an amine or of a coupling component of the benzene, naphthalene, pyrazole, pyridine, pyrimidine,...
4451398 Dyes containing imidazolymethylene groups  
Dyes of the formula ##STR1## where R 1 is hydrogen, C 1 -C 6 -alkyl or C 2 -C 6 -alkenyl, R 2 and R 3 independently of one another are hydrogen, C 1 -C 5 -alkyl or C 2 -C 5 -alkenyl, R 4...
4450114 Process for production of sulfuric acid semiesters  
A compound having at least one --SO 2 CH 2 CH 2 OSO 3 M group in the molecule, wherein M is hydrogen or an alkali metal, which is useful as a reactive dye for dying cellulose fiber materials or...
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