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7595337 |
Mitotic kinesin inhibitors
The present invention relates to tricyclic pyrazoles that are useful for treating cellular proliferative diseases, for treating disorders associated with KSP kinesin activity, and for inhibiting...
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7595320 |
Hydrazinocarbonyl-thieno[2,3-C]pyrazoles, process for preparing them, compositions containing them and use thereof
The present invention concerns hydrazinocarbonyl-thieno[2,3- c ]pyrazoles of formula (I):
wherein R1, R3, R4, are R5 are as defined in the disclosure; their preparation method, compositions...
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7576087 |
Heterocyclyl-3-sulfonylazaindole or -azaindazole derivatives as 5-hydroxytryptamine-6 ligands
The present invention provides a compound of formula I and the use thereof for the treatment of a central nervous system disorder related to or affected by the 5-HT6 receptor.
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7501449 |
2H -or 3H-benzo[e]indazol-1-yl carbamate derivatives, the preparation and therapeutic use thereof
Compounds corresponding to the formula (I)
as defined in the disclosure as well as methods for making such compounds, intermediates employed in such methods, pharmaceutical compositions...
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7485660 |
Non-steroidal ligands for the glucocorticoid receptor, compositions and uses thereof
The invention provides non-steroidal ligands for the glucocorticoid receptor, methods for making non-steroidal ligands of the glucocorticoid receptor, compositions of non-steroidal ligands of the...
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7470717 |
Indazole derivatives
The present invention provides a compound represented by Formula (I):
[wherein R 1 represents CONR 1a R 1b (wherein R 1a and R 1b may be the same or different and each represents a hydrogen...
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7468371 |
Tricyclic pyrazole kinase inhibitors
Compounds of the present invention are useful for inhibiting protein tyrosine kinases. Also disclosed are methods of making the compounds, compositions containing the compounds, and methods of...
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7449586 |
Processes for the preparation of CGRP-receptor antagonists and intermediates thereof
The invention relates to novel processes for the preparation of small molecule antagonists of calcitonin gene-related peptide receptors (“CGRP-receptor”) and intermediates thereof.
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7449488 |
Pyrazolopyrimidines as protein kinase inhibitors
In its many embodiments, the present invention provides a novel class of pyrazolo[1,5-a]pyrimidine compounds as inhibitors of protein and/or checkpoint kinases, methods of preparing such compounds,...
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7446210 |
Factor Xa compounds
The present invention is directed to novel compounds of Formula I:
and forms and pharmaceutical compositions thereof, and the use thereof as inhibitors of Factor Xa.
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7425572 |
Use of dioxindoindazoles and dioxoloindazoles for treating glaucoma
Novel dioxinoindazole compounds and dioxoloindazole compounds are disclosed. Also disclosed are methods for the lowering and controlling of normal or elevated intraocular pressure as well as a...
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