Patents in Class 548/261

Matches 1 - 50 out of 264

1 2 3 4 5 6 >

Match	Document	Document Title
1	8133515	Alkynes and methods of reacting alkynes with 1,3-dipole-functional compounds 1,3-Dipole-functional compounds (e.g., azide functional compounds) can be reacted with certain alkynes in a cyclization reaction to form heterocyclic compounds. Useful alkynes (e.g., strained,...
2	8088801	Aryloazol-2-yl cyanoethylamino compounds, method of making and method of using thereof The present invention relates to novel aryloazol-2-yl-cyanoethylamino derivatives of formula (I): wherein R3, R4, R5, R6, R7, P, Q, V, W, X, Y, Z and a are as defined in the description,...
3	8043607	UV-absorbers for ophthalmic lens materials Dihydroxybenzotriazole UV absorbing compounds that are particularly useful in ophthalmic devices are disclosed.
4	8008290	Compounds A first aspect of the invention relates to a compound of formula (I), or a pharmaceutically acceptable salt, hydrate, complex or pro-drug thereof, wherein:R3 is selected from cyclopentyl and...
5	7968578	Indole amide derivatives as EP4 receptor antagonists The invention is directed to indole amide derivatives as EP4 receptor antagonists useful for the treatment of EP4 mediated diseases or conditions, such as acute and chronic pain, osteoarthritis,...
6	7964621	Thioamide compounds, method of making and method of using thereof The present invention relates to novel thioamide derivatives of formula (I) and formula (Ia): wherein, R3, R4, R5, R6, R7, P, Q, T, V, W, X, Y, Z, a, m and n are as defined in the description,...
7	7923568	Estrogen receptor modulators The present invention relates to compounds and derivatives thereof, their synthesis, and their use as estrogen receptor modulators. The compounds of the instant invention are ligands for estrogen...
8	7897625	Carbamoylbenzotriazole derivatives as inhibitors of lipases and phospholipases The invention relates to carbamoylbenzotriazole derivatives of general formula (I), which are defined as cited in the description, to their pharmaceutically applicable salts and to their use as...
9	7851491	Modified bio-related substance, process for producing the same, and intermediate A modified bio-related substance, wherein at least one poly(alkylene glycol)oxy group represented by the following formula (1) is combined in a molecule: wherein R is a hydrocarbon group having 1...
10	7795315	N-(2-amino-phenyl)-amide derivatives The present invention provides novel compounds of the general formula (I) and pharmaceutically acceptable salts thereof, processes for the manufacture of these novel compounds and medicaments...
11	7763184	Light stabilizing liquid matter containing 2- (2-hydroxy-3-α-cumyl-5-tert-octylphenyl) -2h-benzotriazole A light stabilizing liquid matter, that can be added to a composition to be stabilized and that has a storage stability high enough for storage before being added to the composition, includes a...
12	7514457	Substituted aryloxymethyl bicyclicmethyl acetamide compounds Compounds of the general formula (I): pharmaceutical compositions comprising a compound of general formula (I); and methods of treating disease conditions caused by overactivation of the VR1...
13	7511042	Triazole compounds Disclosed are compounds of formula (I) Where Ar1, X, R3, R4, R5 and R6 are defined herein. The compounds of the invention inhibit production of cytokines and are thus useful for treating cytokine...
14	7402606	Derivatives of 1-(oxoaminoacetyl) pentylcarbamate as cathepsin K inhibitors for the treatment of bone loss Heterocycle substituted ketoamide derivatives of Formula (I), wherein the substitutes A, D, A and R are defined as in claim in, which are useful as cathepsin K inhibitors are described herein. The...
15	7388006	Non-steroidal progesting The present invention relates to non-steroidal progestins of the general formula (I) wherein R1 and R2 are independently of each other —H or —F,R3 is —CH3 or —CF3, andAr is or a pharmac...
16	7361767	N-sulfonyldicarboximide containing tethering compounds Compounds having two reactive functional groups are described that can be used as a tethering compound to immobilize an amine-containing material to a substrate. The first reactive functional group...
17	7157586	Bloom-resistant benzotriazole UV absorbers and compositions stabilized therewith Benzotriazole UV absorbers substituted with a ultra long ester or amide moiety wherein the ester or amide group is a hydrocarbyl group of 25 to 100 carbon atoms or is a group of alkyl of 25 to 100...
18	7084280	Benzotriazol-1-yl-aminoacetonitrile compounds and their use in the control of parasite disease The invention relates to benzotriazol-1-yl-aminoacetonitrile compounds and optionally the enantiomers thereof. The active ingredients have advantageous pesticidal properties. They are especially...
19	7019003	Peptide deformylase inhibitors Novel PDF inhibitors and novel methods for their use are provided.
20	6949556	Acylated 1,2,3,4-tetrahydronaphthyl amines and their use as pharmaceutical agents The present invention relates to compounds of general formula (I), wherein R1-R4 have the meanings given in the specification, A is CH2, CHOH or CH—(C1-C3-alkyl), B and C are independently CH2 or C...
21	6930136	Adhesion promoters containing benzotriazoles Benzotriazole adducts contain a benzotriazole segment and a segment with a curable and polymerizable functionality, or an adhesion promoting functionality, particularly suitable for use on metal...
22	6869913	Pyridazin-3-one derivatives, their use and intermediates for their production Novel pyridazin-3-one derivatives of formula [1] are provided, which are useful as active ingredients of herbicides, wherein R1 is haloalkyl; R2 and R3 are hydrogen, alkyl, haloalkyl, or...
23	6800676	Benzotriazoles containing phenyl groups substituted by heteroatoms and compositions stabilized therewith 2H-Benzotriazole UV absorbers substituted at the 3-position and/or the 5-position of the phenyl ring by a phenyl moiety which is substituted by a heteroatom are particularly photostable in...
24	6790955	Processes for the preparation of aminophenylsulfonyl-ureas and intermediate products for the processes The invention relates to the preparation of compounds (I) in which A═H or acyl and R1, R2, R3, R, n, X, Y and Z are as defined in claim 1 by halogenation and rearrangement of compounds (II) (...
25	6664395	Benzotriazoles anti-inflammatory compounds The present invention relates to novel benzotriazoles of the formula I wherein Het is an optionally substituted 5-membered heterocycle containing one to two heteroatoms selected from nitrogen,...
26	6653484	Polyoxyalkylene substituted and bridged benzotriazole derivatives Triazine, benzotriazole and benzophenone derivatives which are substituted or bridged with polyoxyalkylene groups, according to claim 1, and their use as UV absorbers, especially in photographic...
27	6562972	Method for preparing heterocyclic-carboxylic acids The present invention relates to a method for preparing quinoxaline-5- and 6-carboxylic acids. The method comprises contacting an aqueous alkaline suspension of a 5- or 6-halomethyl quinoxaline...
28	6559308	Method for preparing heterocyclic-carboxylic acids The present invention relates to a method for preparing quinoxaline-5- and 6-carboxylic acids. The method comprises contacting an aqueous suspension of a 5- or 6-hydroxymethyl quinoxaline with...
29	6548525	Nitrogen containing heteroaromatics with ortho-substituted P1's as factor Xa inhibitors The present application describes nitrogen containing heteroaromatics with ortho-substituted P1's and derivatives thereof of formula I: or pharmaceutically acceptable salt or prodrug forms thereof,...
30	6548678	Method for producing 5-phenoxycarbonylbenzotriazole Disclosed is a method for producing 5-phenoxycarbonylbenzotriazole (I): by reacting 1H-benzotriazole-5-carboxylic acid (II): with diphenyl carbonate (III):
31	6541423	4-(3′,4′-heterocyclyl benzoyl) pyrazoles as herbicidal agents The invention relates to pyrazolyl derivatives of benzo-condensated, unsaturated 5-membered nitrogen heterocycles of the general formula (I), wherein X represents N or a group C—R3; Y is O, S, S...
32	6515124	Dehydroamino acids Aromatic dehydroamino acids are disclosed that are active as LFA-1 arnagonists This activity enables these compounds to prevent inflammation which is a consequence of T cell activation and...
33	6498004	Silver halide light sensitive emulsion layer having enhanced photographic sensitivity This invention provides a photographic element comprising at least one silver halide emulsion layer in which the silver halide is sensitized with a compound of the formula (a): Δ−(t)m−XY′ (a)XY′...
34	6489383	2H-benzotriazole UV absorbers substituted with 1,1-diphenylalkyl groups and compositions stabilized therewith 2H-Benzotriazole UV absorbers substituted at the 3-position or at the 5-position of the phenyl ring by a 1,1-diphenylalkyl moiety, particularly a 1,1-diphenylethyl group, are particularly...
35	6469004	Benzoheterocycles and their uses as MEK inhibitors The invention provides compounds having formula (I), wherein W is OH, or derivatives of the carboxylic acid, and Q is a heterocyclo-condensed ortho-phenylene residue. These compounds are useful as...
36	6451887	Benzotriazoles containing α-cumyl groups substituted by heteroatoms and compositions stabilized therewith 2H-Benzotriazole UV absorbers substituted at the 3-position and/or the 5-position of the phenyl ring by α-cumyl moiety which is substituted by a heteroatom are particularly photostable in ...
37	6452018	2-(2′-hydroxyphenyl) benzotriazoles containing a 2,4-imidazolidinedione group and process for their preparation 2-(2′-hydroxyphenyl)benzotriazoles having general formula (I). The above 2-(2′-hydroyzphenyl)benzotriazoles having general formula (I) are useful as heat, oxygen and light stabilizers for org...
38	6407254	2-(2′-hydroxyphenyl)benzotriazoles used as U.V. stabilizers 2-(2′-hydroxyphenyl)benzotriazoles having general formula (I). The above 2-(2′-hydroxyphenyl)benzotriazoles are useful as light stabilizers for organic polymers.
39	6392056	2H-benzotriazole UV absorders substituted with 1,1-diphenylalkyl groups and compositions stabilized therewith 2H-Benzotriazole UV absorbers substituted at the 3-position or at the 5-position of the phenyl ring by a 1,1-diphenylalkyl moiety, particularly a 1,1-diphenylethyl group, are particularly...
40	6387992	Substituted 5-heteroaryl-2-(2-hydroxyphenyl)-2h-benzotriazole UV absorbers, a process for preparation thereof and compositions stabilized therewith Compounds of formula I or II where R is a heteroaryl moiety, such as 3-pyridyl, or T is a heteroaryl moiety, such as thien-2,5-diyl, and E1 and E2 are independently hydrogen, alkyl, aralkyl and the...
41	6376065	Fluorochemical benzotriazoles The invention provides compounds having the formula: wherein Rf is CnF2n+1—(CH2)m—, wherein n is 1 to 22 and m is 0, or an integer from 1 to 3; X is —CO2—, —SO3—, —CONH—, —O—, —S— a covalent bond...
42	6337402	Asymmetrical bisbenzotriazoles substituted by a perfluoroalkyl moiety and compositions stabilized therewith Asymmetrical bisbenzotriazoles of the formula I where G2′ is perfluoroalkyl of 1 to 12 carbon atoms, preferably CF3, and where G2 does not contain said group are red-shifted and due to the a...
43	6268505	2-(2'Hydroxyphenyl) benzotriazoles and process for their preparation 2-(2'-hydroxyphenyl)benzotriazoles having general formula (I): ##STR1##The above 2-(2'-hydroxyphenyl)benzotriazoles can be used as light stabilizers for organic polymers.
44	6261676	Amide functional ultraviolet light absorbers for fluoropolymers An ultraviolet light absorbing material that resists blooming and migration is made up of a fluoropolymer and an amide functional ultraviolet light absorbing compound, wherein the polymer and the...
45	6248899	Transesterification catalysts fixed to solid support materials A description is given of a process for the transesterification of carboxylic esters, characterized in that the catalyst used is a tin(IV) compound comprising a radical of the formula ##STR1##bound...
46	6239151	Compounds as inhibitor of tumor necrosis factor alpha release The invention provides hydrazine derivatives of the formula ##STR1##wherein R1 is lower alkyl, lower alkenyl, lower cycloalkyl, lower cycloalkyl-lower alkyl, aryl or aryl-lower alkyl; R2 is an acyl...
47	6229011	N-aroylphenylalanine derivative VCAM-1 inhibitors Compounds of the formula: ##STR1##are disclosed which have activity as inhibitors of binding between VCAM-1 and cells expressing VLA-4. Such compounds are useful for treating diseases whose...
48	6201134	Diaminorhodamine derivatives
49	6197795	Preparation and use of ortho-sulfonamido heteroaryl hydroxamic acids as matrix metalloproteinase and tace inhibitors The present invention relates to the discovery of novel, low molecular weight, non-peptide inhibitors of matrix metalloproteinases (e.g. gelatinases, stromelysins and collagenases) and TNF-α ...
50	6190777	Ultraviolet absorbing material and ultraviolet absorbing plate An ultraviolet absorbing material prepared by reacting (a) an aminosilane compound of general formula (1) or a derivative thereof wherein R1 is C1 -C10 alkylene or --(CH2)m --NH-- (wherein m is an...

Matches 1 - 50 out of 264

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