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7468382 Pyridine derivatives useful as inhibitors of PKC-theta  
Disclosed are novel compounds of formula (I): wherein R 1 , R 2 and R 3 are as defined herein, which are useful as inhibitors of PKC-theta and are thus useful for treating a variety of...
7304161 Diaclhydrazine ligands for modulating the expression of exogenous genes in mammalian systems via an ecdysone receptor complex  
The present invention relates to non-steroidal ligands for use in nuclear receptor-based inducible gene expression system, and a method to modulate exogenous gene expression in which an ecdysone...
7300991 Cationic conductor, its intermediate, and lithium secondary battery using the conductor  
The disclosure discloses a polymer represented by the general formula, wherein R p is a residue of a polymer of a compound having a polymerizable unsaturated bond, Q is an organic residue of...
7279470 Compounds and uses thereof for decreasing activity of hormone-sensitive lipase  
Use of compounds to inhibit hormone-sensitive lipase, pharmaceutical compositions comprising the compounds, methods of treatment employing these compounds and compositions, and novel compounds. The...
7273867 Phenyl derivatives  
Novel compounds of the formula I in which W, X, Y, T, R 1 and R 2 are as defined in Patent claim 1 , are inhibitors of coagulation factor Xa and can be employed for the prophylaxis and/or...
6992192 Carboline derivatives as PDE5 inhibitors  
Compounds of the general structural formula (I), and use of the compounds and salts and solvates thereof, as therapeutic agents.
6949539 Admantane derivatives  
The invention provides compounds of general formula (I) in which m, A, R 1 and Ar have the meanings defined in the specification; a process for their preparation; pharmaceutical compositions...
6815556 Compounds having fungicidal activity and processes to make and use same  
A compound according to formula one that is useful as a fungicide is provided. Additionally, processes to make and use same are provided.
6727265 Phenoxyethyl-thiourea-pyridine compounds and their use for treatment of HIV-infections  
The invention provides compounds which inhibit reverse transcriptase (RT) and which inhibit replication of a retrovirus, such as human immunodeficiency virus-1 (HIV-1). The compound of the...
6713492 N-acyloxylated cycloalkyl compounds, composition containing the same and methods of use therefor  
Drugs or reagents containing as the active ingredient N-acyloxylated cycloalkyl compounds represented by general formula (I): wherein A is optionally substituted C 4 or C 5 cycloalkyl which...
6667327 Pyridine amido derivatives  
Disclosed are pyridine amido derivatives of the formula wherein X, Y, and R 1 to R 6 are as defined herein. These compounds are selective MAO-B inhibitors and are useful in treating diseases...
6608204 Aromatic heterocyclic derivatives as enzyme inhibitors  
The present invention discloses peptide aldehydes which are potent and specific inhibitors of thrombin, their pharmaceutically acceptable salts, pharmaceutically acceptable compositions thereof,...
6603044 Phthalamide derivatives, or salt thereof agrohorticultural insecticide, and method for using the same  
The present invention provides a phthalamide derivative of the formula (I): wherein A 1 is (substituted) C 1 -C 8 alkylene, (substituted) C 3 -C 8 alkenylene, (substituted) C 3 -C 8 ...
6452008 Pyridone derivatives and process for preparing the same  
A process for preparing a pyridone derivative ( 4 ), which comprises reacting the compound ( 1 ) with a hypochlorite or a hypobromite or with lead tetraacetate to give the compound ( 2 ), and...
6342504 Aromatic heterocyclic derivatives as enzyme inhibitors  
The present invention discloses peptide aldehydes which are potent and specific inhibitors of thrombin, their pharmaceutically acceptable salts, pharmaceutically acceptable compositions thereof,...
6339045 N-(unsubstituted or substituted)-4-substituted-6-(unsubstituted or substituted)phenoxy-2-pyridinecarboxamides or thiocarboxamides, processes for producing the same, and herbicides  
N-(substituted or unsubstituted)-4-substituted-6-(substituted or unsubstituted) phenoxy-2-pyridine carboxamide or thiocarboxamide represented by the general formula (I) and a process for producing...
6329360 Hetero-linked phenylglycinolamides  
The hetero-linked phenylglycinolamides are prepared by reaction of the corresponding hetero-linked phenylacetic acids with appropriate phenylglycinols. The hetero-linked phenylglycinolamides are...
RE37087 Insecticidal triffluormethyl alkane derivatives  
There are provided new alkane and alkoxyalkane derivatives of the general formula I ##STR1## in which R 1 , R 2 , R 3 , R 4 and A have the meanings given in the description, processes for their...
6133442 Aryl- and hetaryl-sulfonamide derivatives, their preparation and their use as endothelin antagonists  
Compounds of formula I ##STR1## wherein R 1 signifies phenyl, substituted phenyl or heterocyclyl; R 2 signifies phenyl or substituted phenyl; R 3 signifies hydrogen, lower-alkyl, cyano,...
6017937 Pyridine derivative, anti-ulcer drug, and antibacterial drug  
A pyridine derivative or a salt thereof expressed by the following formula 1: ##STR1## wherein W represents a group expressed by the following formula 2 or formula 3; ##STR2## wherein R 1 ...
6015905 Process for the preparation of 2-(6-substituted pyrid-2-yloxymethyl) phenylacetate  
5972975 Substituted 2-aminopyridines as inhibitors of nitric oxide synthase  
Substituted 2-aminopyridine compounds of Formula (I) and pharmaceutically acceptable salts which have been found useful in the treatment of nitric oxide synthase mediated diseases and disorders....
5959116 Pyridine-2, 3-dicarboximides their preparation and their use for controlling undesired plant growth  
A pyridine-2,3-dicarboxylic acid diester of the formula Va ##STR1## where the radicals R 2 and R 4 have the meanings set out in the specification and where R 8 is a C 1 -C 4 -alkyl, C 3 -C 5 ...
5883282 3-(3-aryloxyphenyl)-1-(substituted methyl-s-triazine-2,4,6-oxo or thiotrione herbicidal agents  
There is provided a 3-(3-aryloxyphenyl)-1-(substituted methyl)-s-triazine-2,4,6-oxo or thiotrione compound having the structural formula I ##STR1## Further provided are a composition and a method...
5877297 Boronic compound complexing reagents and highly stable complexes  
Boron compound completing reagents, intermediate reagents of those reagents and methods of synthesizing these reagents. These reagents, including those shown as General Formula CII may be used,...
5872224 Boronic compound complexing reagents and highly stable complexes  
Boron compound complexing reagents, boron compound complexes, and methods of synthesizing these reagents and complexes are disclosed. These reagents and complexes include those shown in General...
5869623 Boronic compound complexing reagents and complexes  
Boron compound complexing reagents, intermediate reagents of those reagents, and methods of synthesizing these reagents are disclosed. These reagents, including those shown as General Formula II...
5859210 Boronic compound complexing reagents and complexes  
Boron compound complexing reagents, boron compound complexes, and methods of synthesizing these reagents and complexes are disclosed. These reagents and complexes include those shown in General...
5849361 Methine dyes based on formylaminopyridones  
Methine dyes of the formula ##STR1## where K is a carbocyclic or heterocyclic radical, X is nitrogen or a radical of the formula C--Q 1 , and Q 1 , Q 2 and Q 3 are hydrogen, substituted or...
5811370 Azamethine dyes  
Azamethine dyes of the formula ##STR1## where W is oxygen, sulfur or a radical of the formula --NH--CO--, --NH--COO-- oder --NH--SO 2 --, Z 1 is C 1 -C 4 -alkyl with or without substitution,...
5792779 Pyridinone thrombin inhibitors  
Compounds of the invention are useful in inhibiting thrombin and associated thrombotic occlusions and have the following structure: ##STR1## for example: ##STR2##
5773623 Methine dyes containing a 5- or 6- membered carbocyclic or heterocyclic radical  
Methine dyes of the formula ##STR1## where K is a 5- or 6-membered carbocyclic or heterocyclic radical, X is nitrogen or a radical of formula C--Q 1 , and Q 1 , Q 2 and Q 3 are each...
5760063 Arylhydrazone derivatives useful as antibacterial agents  
The subject invention, provides arylhydrazone compounds having the Formula 1: ##STR1## wherein A and B are independently aryl or heteroaryl and A and B independently are substituted with at least...
5756524 Anilide derivatives as fungicides  
A compound of formula I ##STR1## X is O or S; A is 6-alkoxy-3-pyridyl optionally substituted by halogen; Y is hydrogen or alkyl; R 3 is alkyl or a metal salt complex thereof. This invention...
5750547 Certain carbanate anti-cancer agents  
The present invention is concerned with novel anticancer agents having potent antineoplastic activity without systemic toxicity and mutagenicity. The novel anticancer agents of the present...
5726314 Pyridinium compounds  
Novel quaternary pyridinium compounds useful in inhibiting acetylcholinesterase in mammals of the general structure: ##STR1## or pharmaceutically acceptable salts thereof, where R 5 is...
5721366 Platelet aggregation inhibitors  
This invention relates to compounds having the following formula ##STR1## or a pharmaceutically acceptable salt thereof which are useful in the inhibition of platelet aggregation, to pharmaceutical...
5721222 Heterocyclic ketones  
The present invention relates to certain novel heterocyclic ketones which are 1-pyridylacetamide ketones of formula I, set out herein, which are inhibitors of human leukocyte elastase (HLE), also...
5721259 Method of using 2-formylpyridine thiosemicarbazone compounds  
A method of treatment of tumors is provided based upon a compound of the formula ##STR1## wherein one of R 1 is NHR 4 or NR 4 R 5 or R 3 is NHR 4 , NR 4 R 5 or OH, and the other is hydrogen;...
5688817 Di(aromatic) compounds and their use in human and veterinary medicine and in cosmetics  
Di(aromatic) compounds corresponding to the following formula: ##STR1## in which: Ar represents either ##STR2## n=1 or 2 or: ##STR3## X represents a divalent radical, Z represents O, S or a...
5684198 Method of preparing therapeutic amides  
Amides having formula I: ##STR1## wherein E, X, R 2 and R 3 have the meanings given in the specification, and pharmaceutically acceptable salts and pharmaceutically acceptable in vivo...
5654301 Amino acid derivative anticonvulsant  
The present invention relates to compounds of the formula ##STR1##
5620996 Sulfonamidocarbonyl pyridine-2-carboxesteramides and their pyridine-N-oxide compounds and their use as pharmaceuticals  
The invention relates to sulfonamidocarbonylpyridine-2-carboxesteramides and their pyridine-N-oxides according to the formula I ##STR1## Said compounds are used as pharmaceuticals against fibrotic...
5563159 Dithiocarbonimide derivatives useful as acaricidal, fungicidal, and insecticidal agents  
There is disclosed a dithiocarbonimide derivative of the formula: ##STR1## wherein B is a C 1 -C 6 alkyl group; X is an NH group or an oxygen atom and Y is a nitrogen atom or a CH group, A is a...
5547951 Pyrido[2,3-b][1,4]benzoxazepin (and thiazepin)-6(5H)-ones and -thiones and their use in the prevention or treatment of HIV-1 infection  
Compounds of the class of pyrido[2,3-b][1,4]benzoxazepin (and thiazepin)-6(5H)-ones and -thiones, having the following general structural formula ##STR1## wherein either X or Z is sulfur and the...
5530014 Cyclohexadiene derivatives  
The cyclohexadiene derivatives are prepared by reaction of cyclohexanones with amines and subsequent dehydration. The compounds are suitable as active compounds in medicaments on account of their...
5486529 Certain pyridyl ketones for treating diseases involving leukocyte elastase  
The present invention relates to certain novel heterocyclic ketones which are 1-pyridylacetamide ketones of formula I, set out herein, which are inhibitors of human leukocyte elastase (HLE), also...
5476924 Protecting group for acetals and methods of using the same in the activation of saccharides  
The present invention relates to a method of protecting the hemiacetal or acetal group at the anomeric carbon of a saccharide molecule comprising forming a 4-alkenyl glycoside or 4-alkenoyl...
5464622 Antimicrobial compositions comprising iodopropargyl butylcarbamate and 2-mercaptopyridine n-oxide and method of controlling microbes  
A synergistic antimicrobial composition comprising 2-mercaptopyridine N-oxide, and salts thereof, and iodopropargyl butylcarbamate in a ratio to each other which exhibits synergism is disclosed.
5389652 3-cycloalkyl-prop-2-enamides  
A compound selected from the group consisting of a compound of the formula ##STR1## wherein R 1 is hydrogen or alkyl of 1 to 3 carbon atoms, W is selected from the group consisting of --O--,...
Matches 1 - 50 out of 196 1 2 3 4 >