Patents in Class 546/26

Matches 1 - 50 out of 84

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Match	Document	Document Title
1	8163749	Six-membered heterocycles useful as serine protease inhibitors The present invention provides compounds of Formula (I): or a stereoisomer, tautomer, pharmaceutically acceptable salt or solvate form thereof, wherein the variables A, B, R3 and R11 are as defined...
2	8158376	Bisubstrate fluorescent probe binding to protein kinases This invention relates to fluorescent probes for identification of compounds binding to protein kinases, for measurement of the affinity of inhibitors of protein kinases, and determination of the...
3	8115001	Zeolite ITQ-30 The invention relates to a laminar microporous crystalline zeolite material known as ITQ-30 which, as when synthesized, has a chemical composition in the anhydrous state with the following molar...
4	8088922	Dibenzorylenetetracarboximides as infrared absorbers Dibenzorylenetetracarboximides of the general formula I in which the variables are each defined as follows: R′ are identical or different radicals: hydrogen; optionally substituted aryloxy, a...
5	8084610	Compositions and methods for detecting and treating tumors containing acidic areas Improved compositions have been developed which are selectively sequestered in acidic areas of tumors. When the compositions contain a radioisotope effective to report the presence of the...
6	8083971	Use of rylene derivatives as active components in solar cells and photodetectors The invention relates to compounds of general formula (I) and to the use thereof as active materials in solar cells and photodetectors. The variables in formula (I) are defined in the...
7	8071775	Substituted rylene derivatives Rylene derivatives of the general formula I in which the variables are each defined as follows: Rylene is a polycyclic conjugated ring system which comprises at least one perylene unit may comprise...
8	8072137	Fused heterocyclic compound and organic light emitting device To provide a material for an organic light emitting device showing a light emission hue with an extremely good purity and outputting light having high luminance and a long lifetime with high...
9	8058457	Star-shaped oligothiophene-arylene derivatives and organic thin film transistors using the same A star-shaped oligothiophene-arylene derivative in which an oligothiophene having p-type semiconductor characteristics is bonded to an arylene having n-type semiconductor characteristics positioned...
10	8052899	Heptarylene-and octarylenetetracarboximides and preparation thereof The present invention relates to heptarylene- and octarylenetetracarboximides of the general formula (I) to precursors thereof or mixtures thereof, and to processes for their preparation and to...
11	8030346	Heterocyclic quinolone derivatives that inhibit prolyl hydroxylase activity Compounds of Formula I are useful inhibitors of HIF prolyl hydroxylases. Compounds of Formula I have the following structure: where the definitions of the variables are provided herein.
12	7989583	Process to obtain dimers, trimers and up to polymers from pyridinmethanol derivatives compounds The dimerization or polymerization reaction of pyridinic alcohols is carried out in order to produce novel products. The process is carried out in the absence or presence of some solvent, during...
13	7972789	Dye compounds The present disclosure provides compounds that may be used as chromogens, fluorochromes, or as both. Said compounds may further be used as substrate for at least one enzyme, wherein said enzyme is...
14	7932463	Quinacridine derivatives and organic electronic devices using the same The present invention relates to a novel quinacridine derivative and an organic electronic device using the same.
15	7888863	Organic electroluminescent compounds and organic electroluminescent device using the same The present invention relates to novel organic electroluminescent compounds, and organic electroluminescent devices employing the same as electroluminescent material. Specifically, the organic...
16	7858636	Hexarylene and pentarylene tetracarboxylic acid diimides Rylenetetracarboximides of the general formula I in which the variables are defined as follows: R are identical or different radicals: hydrogen; alkyl, cycloalkyl, aryl or hetaryl, each substituted...
17	7799778	5-substituted 2-aminopyridine analogs for treating allergic and inflammatory diseases Methods for treating an allergic or inflammatory disease or other Syk-mediated disease or Syk-mediated condition characterized by administering a composition which contains a therapeutically...
18	7795468	Functionalized higher diamondoids This invention is directed to functionalized higher diamondoids having at least one functional group. Preferably these derivatives have the following Formula I: wherein D is a higher diamondoid...
19	7795433	Methods for preparing perylene/perinone pigments A method for preparing a perylene pigment or perinone pigment involves a condensation reaction between perylene tetracarboxylic acid or naphthalene tetracarboxylic acid, or anhydrides or imides...
20	7741487	Method for producing quaterrylene-3,4:13, 14-tetracarboxy diimides by direct synthesis A process for preparing quaterrylene-3,4:13,14-tetracarboximides of the general formula I in which R, R′ are each independently hydrogen or optionally substituted C1-C30-alkyl, C5-C8-cycloalkyl o...
21	7692029	Star-shaped oligothiophene-arylene derivatives and organic thin film transistors using the same A star-shaped oligothiophene-arylene derivative in which an oligothiophene having p-type semiconductor characteristics is bonded to an arylene having n-type semiconductor characteristics positioned...
22	7678807	Isoquinoline and benzo[H] isoquinoline derivatives, preparation and therapeutic use thereof as antagonists of the histamine H3 receptor The invention concerns a compound of formula (I): Wherein A, l, m, n, R1 and R2 are as defined herein. The compounds of this invention are useful as medicaments, particularly, in the treatment of...
23	7674797	2-phenoxy- and 2-phenylsulfonamide derivatives with CCR3 antagonistic activity for the treatment of asthma and other inflammatory or immunological disorders The present invention relates to a benzenesulfonamide derivative of formula (I), which is useful as an active ingredient of pharmaceutical preparations. The benzenesulfonamide derivatives of the...
24	7671198	Process for preparing intermediates to 5-HT4 receptor agonist compounds The invention provides 8-azabicyclo[3.2.1 ]octyl intermediates useful for the preparation of 5-HT4 receptor agonist compounds. The invention also provides processes for the preparation of such...
25	7659281	HMG-CoA reductase inhibitors Compounds are provided of the following structure are HMG CoA reductase inhibitors and thus are active in inhibiting cholesterol biosynthesis, modulating blood serum lipids, for example, lowering...
26	7619086	HIV integrase inhibitors Compounds of Formula I are inhibitors of HIV integrase and inhibitors of HIV replication: wherein Z, R1, R2, R3, R4, R5, R6, R7, R8 and R9 are defined herein. The compounds are useful in the...
27	7553959	Fluorescent dye composition and target labeled therewith This invention provides for labeling reagents, labeled targets and processes for preparing labeling reagents. The labeling reagents can take the form of cyanine dyes, xanthene dyes, porphyrin dyes,...
28	7521556	1,6,9,14-tetrasubstituted terrylene tetracarboxylic acid diimides 1,6,9,14-Tetrasubstituted terrylenetetracarboxylic diimides are particularly useful for absorbing and emitting in the long-wavelength red and near infrared region of the electromagnetic spectrum.
29	7495111	Compounds useful as serotonin inhibitors and 5-HT1A agonists and antagonists 3-Amino chroman and 2-amino tetralin derivatives and compositions containing such compounds are disclosed. Such compounds are useful for modulating activity of a 5-HT1A receptor (agonizing or...
30	7449488	Pyrazolopyrimidines as protein kinase inhibitors In its many embodiments, the present invention provides a novel class of pyrazolo[1,5-a]pyrimidine compounds as inhibitors of protein and/or checkpoint kinases, methods of preparing such compounds,...
31	7427693	Polar liquid crystal Compounds that are useful in compositions for flat panel displays, for example, are provided. The compounds provided are polar, and are useful in low threshold voltage mixtures. The compounds...
32	7408061	Rylene dyes Rylene dyes of the general formula I where the variables are defined as follows: R is hydrogen; optionally substituted C1-C30-alkyl, C5-C8-cycloalkyl, aryl or hetaryl;R′ is bromine; cyano; —...
33	7358362	Method for the production of terylene-3,4:11,12-tetracarboxydiimides by direct synthesis A process for preparing terylene-3,4:11,12-tetracarboximides I where the variables are each defined as follows: R, R′ are each independently hydrogen; if desired substituted alkyl or c...
34	7273938	Preparation of novel substituted haloarene compounds This invention relates to a new process for the preparation of novel substituted haloarene compounds of the formula I or IV: respectively, wherein R1, R2, R3, R4, R5, X, and Y are as defined...
35	7223864	2-hydroxyethidium, methods of preparation and uses thereof The inventors have purified the fluorescent product in the hydroethidine-based supeorxide detection assays and further identified the product as 2-hydroxyethidium. Methods for synthesizing...
36	7220856	Substituted quinoline CCR5 receptor antagonists The present invention relates to CCR5 receptor antagonists of formulae (1a) or (1b): enantiomers, diastereomers, salts and solvates thereof wherein R1, R2, R3, R4, R5, and R7 are as defined herein....
37	7196111	Pyrazolo[1,5a]pyrimidine compounds as antiviral agents The invention relates to the inhibition of hepatitis C virus (HCV) replication. In particular, embodiments of the invention provide compounds and methods for inhibiting HCV RNA-dependent RNA...
38	7166726	Aryl substituted 3,4-dihydroanthracene derivatives having retinoid antagonist or retinoid inverse agonist type biological activity Disclosed herein are compounds of the formula wherein R1 is independently H or alkyl of 1 to 6 carbons; R2 is optional and is defined as lower alkyl of 1 to 6 carbons, F, Cl, Br, I, CF3, fluoro...
39	7145010	Tert-alkylphenoxy-substituted polycyclic compounds Tert-alkylphenoxy-substituted polycyclic compounds of the general formula I where P is a conjugated polycyclic radical which is stable to bases and nucleophiles, optionally bears aryl substituents...
40	7138522	Rylene derivatives and their use as dyes Rylene derivatives of the general formula I where the variables have the following meanings: R is hydrogen or substituted or unsubstituted C1–C30-alkyl, aryl or hetaryl;R1 is hydrogen or b...
41	7033541	Bicarbonate receptor compounds The present invention relates to compounds and more particularly to compounds which are useful for the determination of bicarbonate and the delivery of bicarbonate to a non-aqueous solution. The...
42	7018840	Fluorescent metal sensors, and methods of making and using the same The present invention is directed, in part, to fluorescent metal sensors for detecting metal ions, and methods of making and using the same.
43	6890377	Thermochromic rylene dyes Rylene dyes of the general formula I where R is hydrogen; unsubstituted or substituted C1-C30-alkyl, aryl or hetaryl;R′ is unsubstituted or substituted C2-C30-alkyl or C5-C8-cycloalkyl, or s...
44	6881867	Method for hydroformylation, xanthene-bridged ligands and catalyst comprising a complex of said ligands In a process for the hydroformylation of ethylenically unsaturated compounds, at least one complex of a metal of transition group VIII. with at least one phosphorus-, arsenic- or...
45	6818149	Ligand and complex for catalytically bleaching a substrate The present invention provides a bleaching composition comprising a [3.3.1] bicyclo compound carrying at least one tertiary amine group the bleaching composition substantially devoid of a peroxygen...
46	6803129	Organic light emitting diode and organic luminescent materials thereof The present invention relates to an organic light emitting diode (OLED) device, comprising an anode disposed on a substrate, an organic EL layer disposed on the anode and a cathode disposed on the...
47	6756497	Benzoic acid derivatives and processes for the preparation thereof Benzoic acid derivatives useful as intermediates for the preparation of drugs and agricultural chemicals, particularly compounds having herbicidal activity; and easy and economical processes for...
48	6706698	α-Substituted β-aminoethyl phosphonate derivatives The present invention relates to novel α-substituted-β-aminoethylphosphonate and α-substituted-β-aminovinylphosphonate derivatives and their uses for lowering plasma levels of apo (a), Lp(a), apo...
49	6703504	Conformationally constrained compounds as dendrimer cores There are provided novel chemical compounds and their uses in the preparation of polymers and oligomers, and the preparation of such compounds. In certain embodiments there are provided dendritic...
50	6689770	Aryl sulfonyls as factor Xa inhibitors The present application describes aryl sulfonyls of formula I: or pharmaceutically acceptable salt or prodrug forms thereof, wherein D, E, and M are defined below, are effective factor Xa inhibitors.

Matches 1 - 50 out of 84

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