Patents in Class 546/100

Matches 1 - 50 out of 90

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Match	Document	Document Title
1	RE39265	Heteroarylpiperidines, and their use as antipsychotics and analgetics Heteroarylpiperidines, pyrrolidines, and piperazines are useful as antipsychotic and analgesic agents. The compounds are especially useful for treating psychoses by administering to a mammal a...
2	6890377	Thermochromic rylene dyes Rylene dyes of the general formula I where R is hydrogen; unsubstituted or substituted C 1 -C 30 -alkyl, aryl or hetaryl; R′ is unsubstituted or substituted C 2 -C 30 -alkyl or C 5 -C 8...
3	6768010	Organophotoreceptor with an epoxy-modified charge transport compound having an azine group Organophotoreceptors comprise an electrically conductive substrate and a photoconductive element on the electrically conductive substrate, the photoconductive element comprising: a) a charge...
4	6559306	Dye compounds This invention relates to new fluorescent or non-fluorescent dye compounds having a terminal hydroxy, carboxylic acid/ester or amino group and a process for their preparation. The new fluorescent...
5	6486319	Thermochromic rylene dyes The invention relates to rylene dyes of the general formula (I), wherein the variables have the following meanings: R represents hydrogen; optionally substituted C 1 -C 30 alkyl-C 5 -C 8...
6	6410505	Dimeric non-azo naphthalimides and uses for the same A class of predominantly hydrophilic 1,8-naphthalimide dyes. The dye contains at least two 1,8-naphthalimide ring systems, joined by a spacer moiety. Each of the 1,8-naphthalimide ring system has a...
7	RE37729	4-Heteroaryl-1-piperidinealkylamines and derivatives thereof and their therapeutic utility Heteroarylpiperidines, pyrrolidines, and piperazines are useful as antipsychotic and analgesic agents. The compounds are especially useful for treating psychoses by administering to a mammal a...
8	6358746	Fluorescent compounds for use in industrial water systems Fluorescent compounds of the formula: wherein R 1 and R 2 are either both SO 3 M, or one of R 1 and R 2 is SO 3 M and the other is COOM, where M is selected from the group consisting of H,...
9	6248890	Naphthalimide diester fluorescent tracers having improved solubility and fluorescence A fluorescent naphthalimide diester dye that is miscible or soluble in a variety of organic compounds such as, for example, mineral oil, polyalkylene glycols, polyolesters, motor oil, gear oil,...
10	6177570	Method for producing aromatic bisimides
11	6150306	Fluorescent tracer dyes A dye composition has the formula: ##STR1## where R 1 and R 2 are the same or different and are selected from (A) C 2 -C 12 alkyloxyalkyl, and (B) C 9 -12 alkyl, (A) comprising from about 30 to...
12	5998621	Aryloxy-poly(oxyalkylene) naphthalimide derivative colorants This invention relates to colorants comprising naphthalimide base groups with specific water-solubilizing pendant moieties attached. These pendant moieties are based upon aryloxypolyoxyalkylene...
13	5981753	Bis-naphthalimides for the treatment of cancer Disclosed herein are compounds pharmaceutical compositions containing same of the formula 1. A compound of the Formula ##STR1## wherein X, X', X" and X'", A, B, D, R, and R' are as identified in...
14	5918269	Naphthalimide colorants with improved compatibility in refrigeration and air conditioning lubricants Novel naphthalimide-derivative colorants are provided which are present in a neat liquid state at ambient temperature and pressure. Such colorants are produced through the reaction between 4-chloro...
15	5858930	Liquid Benz-iso-Quinoline derivatives 1,8-Naphthalimide derivatives of Formula (I) are useful as fluorescent dyes: ##STR1## wherein R 1 and R 2 are each independently selected from the group consisting of branched alkyl groups...
16	5840903	4-aminomethyl-1-azaadamantane derived benzamides This invention relates to compounds of the formula: ##STR1## or a pharmaceutically acceptable salt thereof wherein Z is selected from the group consisting of ##STR2## R 1 is alkoxy of one to six...
17	5817820	Quinolone derivatives and processes for the preparation thereof The present invention relates to optical isomers of quinoline compounds of Formula (IA) or Formula (IA'), their pharmaceutically acceptable salts and their intermediates: ##STR1## In the above...
18	5776963	3-(heteroaryl)-1- (2,3-dihydro-1h-isoindol-2-yl)alkyl!pyrrolidines and 3-(heteroaryl)-1- (2,3-dihydro-1h-indol-1-yl)alkyl!pyrrolidines and related compounds and their therapeutic untility Heteroarylpiperidines, pyrrolidines, and piperazines are useful as antipsychotic and analgesic agents. The compounds are especially useful for treating psychoses by administering to a mammal a...
19	5663449	Intermediate compounds in the synthesis of heteroarylpiperidines, pyrrolidines and piperazines Heteroarylpiperidines, pyrrolidines, and piperazines are useful as antipsychotic and analgesic agents. the compounds are especially useful for treating psychoses by administering to a mammal a...
20	5654319	N-[(4-heteroaryl-1-piperidinyl)alkyl]-2,3-naphthalimides and related compounds and their therapeutic utility Heteroarylpiperidines, pyrrolidines, and piperazines are useful as antipsychotic and analgesic agents. the compounds are especially useful for treating psychoses by administering to a mammal a...
21	5641782	3-aromatic and 3-heteroaromatic substituted bisnaphthalimides This invention relates to 3-Pyrimidinyl Bisnaphthalimides as Anticancer Agents and pharmaceutically acceptable salts thereof, of the formula: ##STR1## and processes for the preparation of such...
22	5639764	2-[(4-heteroaryl)-1-piperidinyl)alkyl]-1,3-indandiones and related compound and their therapeutic utility Heteroarylpiperidines, pyrrolidines, and piperazines are useful as antipsychotic and analgesic agents, the compounds are especially useful for treating psychoses by administering to a mammal a...
23	5637710	Intermediate compounds in the synthesis of heteroarylpiperidines and piperazines Heteroarylpiperidines, pyrrolidines, and piperazines are useful as antipsychotic and analgesic agents. the compounds are especially useful for treating psychoses by administering to a mammal a...
24	5633265	*WITHDRAWN PATENT AS PER THE LATEST USPTO WITHDRAWN LIST* Heteroarylpiperidines, pyrrolidines and piperazines and their use as antipsychotics and analgetics Heteroarylpiperidines, pyrrolidines, and piperazines are useful as antipsychotic and analgesic agents. The compounds are especially useful for treating psychoses by administering to a mammal a...
25	5614543	1-(aryloxyalkyl)-3- (heteroaryl) pyrrolidines and related compounds useful as antipsychotics and analgesics Heteroarylpiperidines, pyrrolidines, and piperazines are useful as antipsychotic and analgesic agents. The compounds are especially useful for treating psychoses by administering to a mammal a...
26	5612342	*WITHDRAWN PATENT AS PER THE LATEST USPTO WITHDRAWN LIST* [(4-heteroaryl-1-piperindyl)alkoxy]-3,4-dihydro-1(2H)-naphthalenones and related compounds and their therapeutic utility Heteroarylpiperidines, pyrrolidines, and piperazines are useful as antipsychotic and analgesic agents. The compounds are especially useful for treating psychoses by administering to a mammal a...
27	5612343	N-[(4-heteroaryl-1-piperazinyl)alkyl]-2,3-naphthalimides and related compounds and their therapeutic utility Heteroarylpiperidines, pyrrolidines, and piperazines are useful as antipsychotic and analgesic agents. the compounds are especially useful for treating psychoses by administering to a mammal a...
28	5597842	3-heteroaryl-1-pyrrolidinealkanols and derivatives thereof and their therapeutic utility Heteroarylpiperidines, pyrrolidines, and piperazines are useful as antipsychotic and analgesic agents. the compounds are especially useful for treating psychoses by administering to a mammal a...
29	5585497	Substituted 1-naphthyl-3-pyrazolecarboxamides which are active on neurotensin The invention relates to substituted 1-naphyl-3-pyrazolecarboxamides of formula I: ##STR1## These compounds are useful for the treatment of neuropsychiatric disorders, especially those associated...
30	5578624	Heteroarylpyrrolidines and their use as antipsychotics and analgesics Heteroarylpiperidines, pyrrolidines, and piperazines are useful as antipsychotic and analgesic agents. The compounds are especially useful for treating psychoses by administering to a mammal a...
31	5552544	5-nitrobenzo[de]isoquinoline-1,3-diones their preparation and their use An antitumor 5-nitrobenzo[de]isoquinoline-1,3-dione of the formula I ##STR1## where n is 1 or 2, R 1 and R 2 are identical or different and are each hydrogen, C 1 -C 6 -alkyl, C 1 -C 6 ...
32	5488110	Highly water soluble bis-naphthalimides useful as anticancer agents This invention relates to bis-naphthalimides, including 2,2'-[1,2-ethanediylbis(methylimino-2,1-ethanediyl)]-bis[5-n itro-1H-benz[d e]isoquinoline-1,3(2H)-dione],...
33	5420136	Eradication of pathogenic biological contaminants using non-azo naphthalimide dyes A class of predominantly hydrophobic non-azo N-substituted 1,8-naphthalimide compounds, each bearing, at its 3-position, a nucleofuge and, at its 4-position, a heteroatomic electron-releasing...
34	5420137	Amonafide salts The monohydrochloride and the monomethanesulfonate of amonafide are described. The salts have good pharmaceutical properties besides their antitumor action.
35	5308773	Non-azo 1,8-naphthalimide dyes for the detection and quantitation of a paramagnetic metal cation in a non-aqueous medium The use of a class of non-azo 1,8-naphthalimide dyes for the detection and quantitation of a paramagnetic metal cation in a non-aqueous medium and some of the dyes that will complex with a...
36	5283355	Benzoquinone compounds Compounds of the Formula (5) and processes for their preparation and use, particularly in the manufacture of unsymmetrical triphenodioxazine dyes: ##STR1## wherein: Y is H, alkyl, substituted...
37	5266569	Azatricyclo carboxylic acids useful as anti-bacterial agents Quinolone carboxylic acids 7-substituted by azabicyclo groups have antibacterial activity.
38	5202318	Tricyclic compounds acting at serotonin receptor subtypes Compounds of Formula I: ##STR1## in which Z is CH 2 or CO; X and Y are independently selected from hydrogen, halogen, hydroxy, lower alkoxy, lower alkyl, nitro, amino, aminocarbonyl, (lower...
39	5202333	Tricyclic 5-HT.sub.3 receptor antagonists The present invention is directed to 5-HT 3 receptor antagonist compounds of formula I: ##STR1## in which the dashed line denotes an optional double bond; n is 1, 2 or 3; p is 0, 1, 2 or 3; ...
40	5183821	Method for treating leukemias using N-(2-dimethylaminoethyl)-3-amino-1,8-naphthalimide for treating leukemias and solid tumors N-(2-dimethylaminoethyl)-3-amino-1,8-naphthalimide (amonafide) is an effective agent for the treatment of leukemias and solid tumors.
41	5162335	Di- and tetrahydroisoquinoline derivatives The invention relates to new di- and tetrahydroisoquinoline derivatives having interesting cytostatic properties, to the preparation of the said new compounds, and to compositions comprising such a...
42	5082938	Organic materials containing poly(oxyalkylene) moieties having enhanced functionality and their preparation Enhanced branched chain hydroxyl compounds are provided of formula Y--(Z) 1 -6 wherein Y is the residue of a nucleophile devoid of conjugated divalent linking moieties, and each Z is a...
43	5066800	Qunoline intermediates useful therein for synthesizing antibacterial compounds A novel process and intermediates used therein for linking a cephalosporin compound to a quinolone are disclosed. According to the disclosed process, the 2-carboxylic acid moiety of the...
44	4990517	7-(1-pyrrolidinyl)-3-quinolone- and -naphthyridonecarboxylic acid derivatives as antibacterial agents and feed additives 7-(1-Pyrrolidinyl)-3-quinolone- and -naphthyridonecarboxylic acid derivatives as antibacterial agents and feed additives, of the formula ##STR1## in which X 1 is halogen, X 2 is hydrogen,...
45	4892950	Process for the preparation of naphthalene-1,8-dicarboximides Process for the preparation of naphthalene-1,8-dicarboximide which is optionally substituted in the naphthalene ring, characterized in that naphthalene-1,8-dicarboxylic anhydride which is...
46	4874863	Bisnaphthalimides Bisnaphthalimides of the formula I ##STR1## where X 1 to X 4 and R have the meanings stated in the description, and their preparation are described. The compounds are cytotoxic towards human...
47	4816453	N-heterocyclic derivatives of benzamides and their use in treating gastric and intestinal disorders Compounds of formula (i) and pharmaceutically acceptable salts thereof: ##STR1## wherein: m and n are independently 1 or 2 and p is 0, 1 or 2 such that m+n+p≥3; R 1 and R 2 are independently...
48	4782064	2-heteroaryl-alkyl-1H-benz[de]-isoquinoline-1,3(2H)-diones This invention concerns novel 2-heteroarylalkyl-1H-benz[de]isoquinoline-1,3(2H)-diones which are useful as inhibitors of thromboxane synthetase and/or as hypotensive agents in the treatment of...
49	4659834	Process for the preparation of fluoromethyl-quinoline derivatives A process is disclosed for preparing a compound of the Formula (I) ##STR1## wherein R 2 is trifluoromethyl or chloro; R 3 is hydrogen or chloro; and X is halogen; wherein a compound of the...
50	4473693	Aminonaphthalimide dyes for intracellular labelling Fluorescent yellow dyes of the aminonaphthalimide type which have the following structures: ##STR1## In the formula above alk (alkali metal) may be substituted for Li + and thus alk may be Li + ,...

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