Patents in Class 544/52

Matches 1 - 50 out of 157

1 2 3 4 >

Match	Document	Document Title
1	7576078	Tetrahydroquinoline analogues as muscarinic agonists The present invention relates to tetrahydroquinoline compounds as muscarinic receptor agonists; compositions comprising the same; methods of inhibiting an activity of a muscarinic receptor with...
2	7531534	Heterocyclic antiviral compounds Compounds having the formula Ia or Ib wherein R 1 , R 2 , R 3 and R 4 are as defined herein are Hepatitis C virus NS5b polymerase inhibitors. Also disclosed are compositions and methods for...
3	7491714	Quinolines and nitrogenated derivatives thereof and their use as antibacterial agents Quinoline and naphthridine derivatives useful in the treatment of bacterial infections in mammals, particularly humans.
4	7479489	Heterocyclic antiviral compounds Compounds having the formula I wherein A, m and R 1 are herein defined are Hepatitis C virus polymerase inhibitors. Also disclosed are compositions and methods for treating diseases mediated by...
5	7348426	Substituted bicyclic heterocycles, process for their preparation and their use as antiobesity and hypocholesterolemic agents The present invention relates to novel antiobesity and hypocholesterolemic compounds, their derivatives, their analogs, their tautomeric forms, their stereoisomers, their polymorphs, their...
6	7253164	Bicyclic compounds and compositions as PDF inhibitors This invention is directed to novel bicyclic compounds, to the uses of these compounds in various medicinal applications, including treating disorders amenable to treatment by peptidyl deformylase...
7	7205408	Quinolines and nitrogenated derivative thereof substituted in 4-position by a piperidine-containing moiety and their use as antibacterial agents Piperidine derivatives and pharmaceutically acceptable derivatives thereof useful in methods of treatment of bacterial infections in mammals, particularly in man.
8	7141566	Benzoxazine and benzothiazine derivatives and the use thereof in medicaments The invention relates to compounds of formula (I), the tautomeric and isomeric forms and salts thereof, in addition to a method for production and use thereof in medicaments.
9	7141564	Nitrogen-containing bicyclic heterocycles for use as antibacterials Cyclohexane and cyclohexene derivatives and pharmaceutically acceptable derivatives thereof useful in methods of treatment of bacterial infections in mammals, particularly man.
10	7067513	Phenylpiperazines The invention relates to a novel group of phenylpiperazines having interesting pharmacological properties such as a high affinity for the dopamine D 2 receptor and/or the serotonin reuptake site,...
11	7049312	Benzothiazinone and benzoxazinone compounds Q is —N=or CR 2 X is S, O or NOR 3 Y is —O—, —S—, —SO— or —SO 2 — R and R 1 are each, independently, H, a substituted or unsubstituted aliphatic, aromatic, heteroaromatic or...
12	6900204	Antimicrobial agents and uses thereof The invention features compounds that act as antimicrobial agents and/or antimicrobial enhancer agents, compositions that include the antimicrobial enhancer agents of the invention, and methods for...
13	6740649	Cyclic hydroxamic acids as inhibitors of matrix metalloproteinases and/or TNF- α converting enzyme (TACE) The present application describes novel cyclic hydroxamic acids of formula I: or pharmaceutically acceptable salt forms thereof, wherein ring B is a 5-7 membered cyclic system containing from...
14	6683101	Bicyclic cyclohexylamines and their use as NMDA receptor antagonists Described are heterocycle-substituted cyclohexylamines of formula (I), and their pharmaceutically acceptable salts thereof. The compounds of the formula (I) are antagonists of NMDA receptor channel...
15	6573218	Fused-benzene derivatives useful as herbicides A compound of the formula (Ia): or its salts, in which the variables are as described in the disclosure; herbicidal compositions of said compounds, herbicidal processes using said compounds,...
16	6448246	Substituted 4H-1,4-benzothiazine-2-carboxamide: GABA brain receptor ligands Disclosed are 4H-1,4-Benzothiazine-2-carboxamides. These compounds are highly selective agonists, antagonists or inverse agonists for GABAa brain receptors or prodrugs of agonists, antagonists or...
17	6410484	6-Hydroxy-5,6-dihydrouracil compound and herbicidal composition containing thereof A 5,6-dihydrouracil compound given by the formula [I]: wherein, R 1 represents C1-C2 haloalkyl group and Q represents Q1 of the formula below, etc.: wherein, R 3 is hydrogen atom or halogen...
18	RE37555	Process and composition for multicomponent one hundred percent solid fabric softeners The invention relates to a method of producing a mixture of a quaternary ammonium compound, fatty acid, fatty acid ester and tertiary amine salt in situ which is a highly functional mixture that is...
19	RE37556	Superoxide radical inhibitor A superoxide radical inhibitor containing, as an effective ingredient, an azole derivative represented by the general formula (1), [wherein R 1 represents a phenyl group which may have 1-3...
20	6339084	Process for the production of thiazine-indigo pigments A process of forming the cis- or the trans-isomers of thiazine-indigo compounds comprising the step of reacting o-aminomercapto-carbocyclic or -heterocyclic compounds with a maleic acid or fumaric...
21	6339155	Process for producing 3-phenyluracil compounds The uracil compounds represented by the formula [V]: wherein R 1 represents C1-C5 perfluoroalkyl group and Q represents an aromatic group, can be produced by making the amide compounds...
22	6333413	Production of pyridazine herbicides Carboxylic acids of formula (1): ##STR1## wherein R 2 and R 3 are independently hydrogen or C 1 -C 3 alkyl, and Q is optionally substituted phenyl, can be easily converted by ring closing...
23	6303542	Herbicidal 3-substituted-phenyl-1,2,3-benzotriazin-4-ones This invention relates to 3-substituted-phenyl-1,2,3-benzotriazin-4-ones which have activity as herbicides, to compositions which contain these compounds and to methods of use of these compounds.
24	6300342	Antithrombotic phenylalkyl derivatives Antithrombotic phenylalkyl derivatives of the formula ##STR1## Exemplary compounds are: (a) 1-[3-(4-amidino-phenyl)propionyl]-6-(4-fluoro-phenylsulphona mido)-1,2,3,4- tetrahydro-quinoline, ...
25	6232310	Fused 1,4-thiazine-2-carbonitrile derivatives, their preparation and use The present invention relates to fused 1,4-thiazine-2-carbonitrile derivatives, compositions thereof and methods for preparing the compounds. The compounds are useful in the treatment of diseases...
26	6200971	Bicyclic heterocyclic compounds The bicyclic heterocyclic compounds are prepared by reaction of correspondingly substituted carboxylic acids with amines, in particular with phenylglycinolamine. The bicyclic heterocyclic compounds...
27	6191127	Substituted heterocycles and their use in medicaments
28	6127357	N-((phenyl, benzodioxinyl or N-heteroarylpiperazinyl)alkyl)-N-(N-heteroaryl)substituted carboxamides Piperazine derivatives of formula I ##STR1## and their pharmaceutically acceptable acid addition salts are 5-HT 1A binding agents, particularly 5-HT 1A antagonists and may be used, for example,...
29	6071860	2,4-Diamino-1, 3,5-triazines, their preparation, and their use as herbicides and plant growth regulators Compounds of the formula (I) and salts thereof ##STR1## where R 1 to R 5 , A, Z, X, X', n and m are as defined in claim 1 are suitable as herbicides and plant growth regulators. They can be...
30	6069114	2-amino-4-bicycloamino-1,3,5-Triazines, their preparation, and their use as herbicide and plant growth regulators Compounds of the formula (I) and their salts ##STR1## in which R 1 to R 6 , Y 1 , to Y 2 , Y 3 , m and n are as defined in claim 1 are suitable as herbicides and plant growth regulators. They can...
31	6015774	Pyrazin-2-one derivatives, their use, and intermediates for their production Novel pyrazin-2-one derivatives of formula [1] are provided, ##STR1## which are useful as active ingredients of herbicides, wherein R 1 is hydrogen or alkyl; R 2 is haloalkyl; R 3 is optionally...
32	6011033	Phenylene derivatives This invention relates to a phenylene derivative represented by the following formula (1) or a salt thereof and also to a medicine containing it as an effective ingredient. ##STR1## wherein R 1 ...
33	6008218	N-phenyl carbamate compounds, process for producing the same, and agricultural or horticultural bactericides This invention relates to An N-phenyl carbamate compound which is represented by the following formula (1): wherein R 1 represents a hydrogen atom, an alkoxyalkyl group having 2 to 5 carbon atoms,...
34	5981436	Substituted diazacyclohexanedi (thi) ones The invention relates to new substituted diazacyclohexanedi(thi)ones of the general formula (I) ##STR1## in which Q 1 , Q 2 , R 1 , R 2 , R 3 , R 4 , R 5 , R 6 and R 7 have the meanings given in...
35	5919784	Heterocyclic aminomethyl compounds A compound of general formula (I): ##STR1## where A, X, R 1 , Y, n and Ar are defined in the description. Medicinal products containing the same are useful as D 4 receptor Ligands.
36	5883049	Hydantoin derivatives and herbicides containing said derivatives as active ingredient This invention provides with novel hydantoin derivatives, processes for preparing them, and herbicides containing said derivatives as active ingredient. The hydantoin derivative of this invention...
37	5830890	Fungicidal acrylate derivatives Compounds, useful as plant fungicides, having the formula (I): ##STR1## or a stereoisomer thereof, wherein A is CH or N, B is OCH 3 or NHCH 3 , X is CH 2 , CH 2 O, O or S, Y is R 1 --CC--R 2 ...
38	5739130	Heterotricyclic derivatives, process for their preparation and pharmaceutical compositions containing them Heterotricyclic derivatives of the formula: ##STR1## wherein R 1 is hydrogen, lower alkyl, lower alkoxy, lower alkylthio, halogen, nitro, amino or protected amino, R 2 is hydroxy, protected...
39	5726307	Benzo-fused lactams promote release of growth hormone There are disclosed certain novel compounds identified as benzo-fused lactams which promote the release of growth hormone in humans and animals. This property can be utilized to promote the growth...
40	5719141	2,9-diamino- and 2-amino-8-carbamoyl-4-hydroxy-alkanoic acid amide derivatives Compounds of the formula I ##STR1## in which R 1 is arylamino, N-aryl-N-(lower alkoxy-lower alkyl)-amino, N-aryl-N-aryl-lower alkyl-amino or heterocyclyl bonded via a ring carbon atom, X is a...
41	5712225	Oxa-and thia(di)azabicyclic compounds The present invention relates to oxa(di)azabicyclic and thia(di)azabicyclic compounds, a method for their preparation and their use as herbicides.
42	5661107	Heterocyclic compounds and their use as herbicides Compounds of the formula ##STR1## wherein m represents 1 or 2, X represents O, S, CH 2 or substituted CH 2 , R 1 -R 4 represent hydrogen or substituted or unsubstituted hydrocarbon groups, and Q...
43	5599815	Antipsychotic benzoisothiazolyl piperazine derivatives Compounds represented by the formula (I) and pharmacologically acceptable salts thereof: ##STR1## These compounds have little extrapyramidal effect and thus are effective as an anti-psychotic agent...
44	5597819	Phenothiazine cytokine inhibitors New benzothiazine derivatives corresponding to the general formula I: ##STR1## in which: X represents halogen, n represents 0, 1, or 2, B represents the following formula: ##STR2## in which:...
45	5547952	3-oxo-1,4-benzothiazine derivatives This invention relates to the compounds of the formula [I] which are useful for the treatment of cataracts, and the synthetic intermediates of the formula [II], ##STR1## wherein R 1 is hydroxy...
46	5530126	Process for the preparation of substituted 6-(pyrazol-3yl)-1,4-benzoxazin-3-ones The disclosure herein relates to a process for the preparation of compounds according to Formula N ##STR1## which comprises using a compound of Formula M ##STR2## as starting material for...
47	5521145	Iminothiazoline derivatives and herbicides containing them as active ingredients There is disclosed an iminothiazoline derivative of the general formula: ##STR1## wherein R 1 is (halo)alkyl, (halo)alkenyl, (halo)alkynyl or the like; R 2 is (halo)alkyl, optionally substituted...
48	5496815	Thiazine (or oxazine) derivatives and preparation thereof Thiazine derivatives of the formula [I]: ##STR1## wherein R 1 , R 2 , R 4 and R 5 are each hydrogen atom; R 3 is hydrogen atom or a halogen atom; X is sulfur atom; R 6 is naphthyl, a...
49	5440035	Heterocyclic amide derivatives The invention concerns novel, pharmaceutically useful, amide derivatives of certain benzoheterocyclylalkanoic acids (and related tetrazoles and acylsulphonamides) of the formula I and salts...
50	5416084	Benzo-fused thiomorpholinyl-terminated alkylamino ethynyl alanine amino diol compounds for treatment of hypertension Compounds characterized generally as benzo-fused thiomorpholinyl-terminated alkylamino ethynyl alanine amino diol derivatives are useful as renin inhibitors for the treatment of hypertension....

Matches 1 - 50 out of 157

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