Patents in Class 544/52

Matches 1 - 50 out of 165

1 2 3 4 >

Match	Document	Document Title
1	8178671	Methods of treating or preventing autoimmune diseases with 2, 4-pyrimidinediamine compounds The present invention provides methods of treating or preventing autoimmune diseases with 2,4-pyrimidinediamine compounds, as well as methods of treating, preventing or ameliorating symptoms...
2	8129369	Antifungal compounds containing benzothiazinone, benzoxazinone or benzoxazolinone and process thereof The present invention discloses novel compounds of the Formula (1), comprising benzothiazinone, benzoxazinone or benzoxazolinone moieties having antifungal activity, method for preparing these...
3	8071600	Derivatives of 4-piperazin-1-yl-4-benzo[B]thiophene suitable for the treatment of CNS disorders A heterocyclic compound or a salt thereof represented by the formula (1): where R2 represents a hydrogen atom or a lower alkyl group; A represents a lower alkylene group or lower alkenylene group;...
4	7981886	Antibiotics derivatives The invention relates to antibiotic derivatives of formula I wherein: A represents —O—, S, —C(═O)—, —C(═NOR6)—;Z—B represents NCH2CH2, NCOCH2, NCH2CO, NCH2CH(OH), CHN(R8)CH2 or CHN(R8)CO;D repre...
5	7960376	Benzo-fused heterocycles The present invention provides benzo-fused heterocyclic compounds having the structure of formula I, as well as prodrugs, stereoisomers, racemates, salts, hydrates, solvates, acid salt hydrates and...
6	7879845	Bicyclic sulfonamide derivatives which are L-CPT1 inhibitors The invention is concerned with novel heterobicyclic derivatives of formula (I) wherein R1, R2, R3, R4, R5, R6, V, W, X and Y are as defined in the description and in the claims, as well as...
7	7863268	Benzothiazinone derivatives and their use as antibacterial agents Disclosed are benzothiazin derivatives of formula (I), preparation methods therefore, and treatment methods employing such compounds as antibacterial agents in treating infectious diseases of...
8	7842686	CGRP receptor antagonists The present invention relates to CGRP receptor antagonists, pharmaceutical compositions thereof, and methods therewith for treating CGRP receptor-mediated diseases and conditions.
9	7790726	Monocyclic and bicyclic compounds and methods of use Compounds are provided that act as potent antagonists of the CCR1 receptor, and have in vivo anti-inflammatory activity. The compounds are generally monocyclic and bicyclic compounds and are useful...
10	7786105	Pyrimidine compounds and use thereof The invention relates to pyrimidine compounds of general formula (I), and to the use of these compounds of general formula (I) and of the physiologically compatible acid addition salts of compounds...
11	7576078	Tetrahydroquinoline analogues as muscarinic agonists The present invention relates to tetrahydroquinoline compounds as muscarinic receptor agonists; compositions comprising the same; methods of inhibiting an activity of a muscarinic receptor with...
12	7531534	Heterocyclic antiviral compounds Compounds having the formula Ia or Ib wherein R1, R2, R3 and R4 are as defined herein are Hepatitis C virus NS5b polymerase inhibitors. Also disclosed are compositions and methods for treating an...
13	7491714	Quinolines and nitrogenated derivatives thereof and their use as antibacterial agents Quinoline and naphthridine derivatives useful in the treatment of bacterial infections in mammals, particularly humans.
14	7479489	Heterocyclic antiviral compounds Compounds having the formula I wherein A, m and R1 are herein defined are Hepatitis C virus polymerase inhibitors. Also disclosed are compositions and methods for treating diseases mediated by HCV...
15	7348426	Substituted bicyclic heterocycles, process for their preparation and their use as antiobesity and hypocholesterolemic agents The present invention relates to novel antiobesity and hypocholesterolemic compounds, their derivatives, their analogs, their tautomeric forms, their stereoisomers, their polymorphs, their...
16	7205408	Quinolines and nitrogenated derivative thereof substituted in 4-position by a piperidine-containing moiety and their use as antibacterial agents Piperidine derivatives and pharmaceutically acceptable derivatives thereof useful in methods of treatment of bacterial infections in mammals, particularly in man.
17	7141564	Nitrogen-containing bicyclic heterocycles for use as antibacterials Cyclohexane and cyclohexene derivatives and pharmaceutically acceptable derivatives thereof useful in methods of treatment of bacterial infections in mammals, particularly man.
18	7141566	Benzoxazine and benzothiazine derivatives and the use thereof in medicaments The invention relates to compounds of formula (I), the tautomeric and isomeric forms and salts thereof, in addition to a method for production and use thereof in medicaments.
19	7049312	Benzothiazinone and benzoxazinone compounds Q is —N=or CR2 X is S, O or NOR3 Y is —O—, —S—, —SO— or —SO2—R and R1 are each, independently, H, a substituted or unsubstituted aliphatic, aromatic, heteroaromatic or aralkyl groupR2 is H or a...
20	6900204	Antimicrobial agents and uses thereof The invention features compounds that act as antimicrobial agents and/or antimicrobial enhancer agents, compositions that include the antimicrobial enhancer agents of the invention, and methods for...
21	6740649	Cyclic hydroxamic acids as inhibitors of matrix metalloproteinases and/or TNF- α converting enzyme (TACE) The present application describes novel cyclic hydroxamic acids of formula I: or pharmaceutically acceptable salt forms thereof, wherein ring B is a 5-7 membered cyclic system containing from 0-2...
22	6683101	Bicyclic cyclohexylamines and their use as NMDA receptor antagonists Described are heterocycle-substituted cyclohexylamines of formula (I), and their pharmaceutically acceptable salts thereof. The compounds of the formula (I) are antagonists of NMDA receptor channel...
23	6573218	Fused-benzene derivatives useful as herbicides A compound of the formula (Ia): or its salts, in which the variables are as described in the disclosure; herbicidal compositions of said compounds, herbicidal processes using said compounds,...
24	6448246	Substituted 4H-1,4-benzothiazine-2-carboxamide: GABA brain receptor ligands Disclosed are 4H-1,4-Benzothiazine-2-carboxamides. These compounds are highly selective agonists, antagonists or inverse agonists for GABAa brain receptors or prodrugs of agonists, antagonists or...
25	6410484	6-Hydroxy-5,6-dihydrouracil compound and herbicidal composition containing thereof A 5,6-dihydrouracil compound given by the formula [I]: wherein, R1 represents C1-C2 haloalkyl group and Q represents Q1 of the formula below, etc.: wherein, R3 is hydrogen atom or halogen atom, R15...
26	RE37556	Superoxide radical inhibitor A superoxide radical inhibitor containing, as an effective ingredient, an azole derivative represented by the general formula (1), [wherein R1 represents a phenyl group which may have 1-3 lower...
27	RE37555	Process and composition for multicomponent one hundred percent solid fabric softeners The invention relates to a method of producing a mixture of a quaternary ammonium compound, fatty acid, fatty acid ester and tertiary amine salt in situ which is a highly functional mixture that is...
28	6339155	Process for producing 3-phenyluracil compounds The uracil compounds represented by the formula [V]: wherein R1 represents C1-C5 perfluoroalkyl group and Q represents an aromatic group,can be produced by making the amide compounds represented by...
29	6339084	Process for the production of thiazine-indigo pigments A process of forming the cis- or the trans-isomers of thiazine-indigo compounds comprising the step of reacting o-aminomercapto-carbocyclic or -heterocyclic compounds with a maleic acid or fumaric...
30	6333413	Production of pyridazine herbicides Carboxylic acids of formula (1):##STR1## wherein R2 and R3 are independently hydrogen or C1 -C3 alkyl, and Q is optionally substituted phenyl, can be easily converted by ring closing into...
31	6303542	Herbicidal 3-substituted-phenyl-1,2,3-benzotriazin-4-ones This invention relates to 3-substituted-phenyl-1,2,3-benzotriazin-4-ones which have activity as herbicides, to compositions which contain these compounds and to methods of use of these compounds.
32	6300342	Antithrombotic phenylalkyl derivatives Antithrombotic phenylalkyl derivatives of the formula ##STR1##Exemplary compounds are: (a) 1-[3-(4-amidino-phenyl)propionyl]-6-(4-fluoro-phenylsulphona mido)-1,2,3,4- tetrahydro-quinoline, (b)...
33	6232310	Fused 1,4-thiazine-2-carbonitrile derivatives, their preparation and use The present invention relates to fused 1,4-thiazine-2-carbonitrile derivatives, compositions thereof and methods for preparing the compounds.The compounds are useful in the treatment of diseases of...
34	6200971	Bicyclic heterocyclic compounds The bicyclic heterocyclic compounds are prepared by reaction of correspondingly substituted carboxylic acids with amines, in particular with phenylglycinolamine. The bicyclic heterocyclic compounds...
35	6191127	Substituted heterocycles and their use in medicaments
36	6127357	N-((phenyl, benzodioxinyl or N-heteroarylpiperazinyl)alkyl)-N-(N-heteroaryl)substituted carboxamides Piperazine derivatives of formula I ##STR1## and their pharmaceutically acceptable acid addition salts are 5-HT1A binding agents, particularly 5-HT1A antagonists and may be used, for example, as...
37	6071860	2,4-Diamino-1, 3,5-triazines, their preparation, and their use as herbicides and plant growth regulators Compounds of the formula (I) and salts thereof ##STR1## where R1 to R5, A, Z, X, X', n and m are as defined in claim 1 are suitable as herbicides and plant growth regulators. They can be prepared...
38	6069114	2-amino-4-bicycloamino-1,3,5-Triazines, their preparation, and their use as herbicide and plant growth regulators Compounds of the formula (I) and their salts ##STR1## in which R1 to R6, Y1, to Y2, Y3, m and n are as defined in claim 1 are suitable as herbicides and plant growth regulators. They can be...
39	6015774	Pyrazin-2-one derivatives, their use, and intermediates for their production Novel pyrazin-2-one derivatives of formula [1] are provided, ##STR1## which are useful as active ingredients of herbicides, wherein R1 is hydrogen or alkyl; R2 is haloalkyl; R3 is optionally...
40	6011033	Phenylene derivatives This invention relates to a phenylene derivative represented by the following formula (1) or a salt thereof and also to a medicine containing it as an effective ingredient. ##STR1## wherein R1...
41	6008218	N-phenyl carbamate compounds, process for producing the same, and agricultural or horticultural bactericides This invention relates to An N-phenyl carbamate compound which is represented by the following formula (1): wherein R1 represents a hydrogen atom, an alkoxyalkyl group having 2 to 5 carbon atoms,...
42	5981436	Substituted diazacyclohexanedi (thi) ones The invention relates to new substituted diazacyclohexanedi(thi)ones of the general formula (I) ##STR1## in which Q1, Q2, R1, R2, R3, R4, R5, R6 and R7 have the meanings given in the description, a...
43	5919784	Heterocyclic aminomethyl compounds A compound of general formula (I): ##STR1## where A, X, R1, Y, n and Ar are defined in the description. Medicinal products containing the same are useful as D4 receptor Ligands.
44	5883049	Hydantoin derivatives and herbicides containing said derivatives as active ingredient This invention provides with novel hydantoin derivatives, processes for preparing them, and herbicides containing said derivatives as active ingredient.The hydantoin derivative of this invention...
45	5830890	Fungicidal acrylate derivatives Compounds, useful as plant fungicides, having the formula (I): ##STR1## or a stereoisomer thereof, wherein A is CH or N, B is OCH3 or NHCH3, X is CH2, CH2 O, O or S, Y is R1 --CC--R2 or R1 -...
46	5739130	Heterotricyclic derivatives, process for their preparation and pharmaceutical compositions containing them Heterotricyclic derivatives of the formula: ##STR1## wherein R1 is hydrogen, lower alkyl, lower alkoxy, lower alkylthio, halogen, nitro, amino or protected amino, R2 is hydroxy, protected hydroxy,...
47	5726307	Benzo-fused lactams promote release of growth hormone There are disclosed certain novel compounds identified as benzo-fused lactams which promote the release of growth hormone in humans and animals. This property can be utilized to promote the growth...
48	5719141	2,9-diamino- and 2-amino-8-carbamoyl-4-hydroxy-alkanoic acid amide derivatives Compounds of the formula I ##STR1## in which R1 is arylamino, N-aryl-N-(lower alkoxy-lower alkyl)-amino, N-aryl-N-aryl-lower alkyl-amino or heterocyclyl bonded via a ring carbon atom, X is a...
49	5712225	Oxa-and thia(di)azabicyclic compounds The present invention relates to oxa(di)azabicyclic and thia(di)azabicyclic compounds, a method for their preparation and their use as herbicides.
50	5661107	Heterocyclic compounds and their use as herbicides Compounds of the formula ##STR1## wherein m represents 1 or 2, X represents O, S, CH2 or substituted CH2, R1 -R4 represent hydrogen or substituted or unsubstituted hydrocarbon groups, and Q...

Matches 1 - 50 out of 165

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