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7465721 |
2-hydroxytetrahydrofuran derivatives and use thereof as medicaments
A hydroxytetrahydrofuran of formula
wherein A is
with the substituents as defined in the specification, having a calpain inhibiting activity and/or an activity which traps the reactive...
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7384933 |
Derivatives of 2-hydroxytetrahydrofuran and their use as medicaments
A hydroxytetrahydrofuran of formula
wherein A is
with the substituents as defined in the specification, having a calpain inhibiting activity and/or an activity which traps the reactive...
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7358358 |
Electrochromic compound
A compound for use in electrochromic devices.
The compound includes (1) β-(10-phenothiazyl)propoxy phosphonic acid; (2) β-(10-phenothiazyl)propyl-phosphonic acid; and (3)...
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7160874 |
Phenylalanine derivatives
Specified phenylalanine derivatives and analogues thereof have an antagonistic activity to α4 integrin. They are used as therapeutic agents for various diseases concerning α4 integrin.
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7083884 |
Organophotoreceptor with charge transport material having a hydrazone group linked to an epoxy group and a heterocyclic ring
Improved organophotoreceptor comprises an electrically conductive substrate and a photoconductive element on the electrically conductive substrate, the photoconductive element comprising:
...
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6992082 |
Phenothiazine kinesin inhibitors
Phenothiazine derivatives of formula (I) are disclosed. The compounds are inhibitors of the mitotic kinesin KSP and are useful in the treatment of cellular proliferative diseases, such as cancer,...
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6800618 |
Chemosensitizing agents against chloroquine resistant plasmodium falciparum and methods of making and using thereof
A compound having the structural formula or a pharmaceutically acceptable salt or prodrug thereof, wherein X is a substituted or unsubstituted alkyl or a heteroatom; n is 4, 5 or 6; Y is a...
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6583138 |
Heterocyclic-ring condensed benzothiazine compound
The invention provides a novel heterocyclic ring condensed benzothiazine compound which is effective for prevention or remedy of disease, in which histamine, leukotriene and the like participate....
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6083651 |
Phenothiazine or phenoxazine derivative, charge-transporting material comprising the same, and electrophotographic photoreceptor
A phenothiazine or phenoxazine derivative represented by the following general formula (1), a charge-transporting material comprising the derivative, and an electrophotographic photoreceptor...
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5861394 |
Use of N-substituted phenothiazines
The invention relates to the use of N-substituted phenothiazines for the production of medicaments for the treatment of cerebral disorders. The invention likewise relates to novel active compounds...
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5597819 |
Phenothiazine cytokine inhibitors
New benzothiazine derivatives corresponding to the general formula I: ##STR1## in which: X represents halogen, n represents 0, 1, or 2, B represents the following formula: ##STR2## in which:...
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5321026 |
Phenothiazine derivatives, their preparation and pharmaceutical compositions containing them
New phenothiazine derivatives of general formula (I) in which R represents 4- to 6-membered cycloalkyl, or represents --CH 2 R" in which R" is hydrogen, alkyl containing 1 to 5 carbon atoms,...
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5308840 |
Substituted or unsubstituted benzhydryl heteroalkyl-substituted aminophenol compounds and pharmaceutical compositions thereof
Aminophenol derivatives of the following formula (I) ##STR1## wherein X is hydrogen atom, lower alkyl or a protecting group for phenolic hydroxy, Y is hydrogen atom or lower alkyl, Z is hydrogen...
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5269954 |
Nitrogenous additives with an antioxidant action and lubricating compositions containing the said additives
The present invention relates to the preparation of antioxidant additives to lubricants and to their use in lubricating compositions. The additives according to the invention have the formula: ...
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5049669 |
Analgesic phenothiazine derivatives
Phenothiazine derivatives of general formula (I), in which R is a linear or branched (1 to 6 C) alkyl radical and R 1 and R 2 , which may be identical or different, are linear or branched (1 to 4...
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5024774 |
Nitrogen containing anti-oxidant compositions
This invention describes compositions containing nitrogen, sulfur and optionally oxygen which are useful as antioxidants for lubricants.
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4912105 |
Derivatives of phenothiazine and the compositions which contain them
Phenothiazine derivatives of formula ##STR1## in which R represents --NR 1 R 2 in which R 1 and R 2 , which may be identical or different, are alkyl, hydroxyalkyl or acetyloxyalkyl radicals, or...
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4798895 |
Process for preparing levomepromazine hydrogen maleate
Levomepromazine hydrogen maleate is prepared by resolving (±)-10-(3-dimethylamino-2-methylpropyl)-2-methoxyphenothiaz
ine with (-)-di(p-toluoyl)-L-tartaric acid to produce the neutral salt of the...
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4705854 |
Phenothiazine compounds
The present invention relates to compounds of the formula (I): ##STR1## or a salt, ester or amide thereof; wherein R 1 is a C 1 -7 bivalent aliphatic hydrocarbon group or a single bond; R 2 ...
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4681878 |
Fluoropheno-thiazine and pharmaceutical use
The compound 2-[10-(2-Dimethylaminopropyl)-7-fluoro-2-phenothiazinyl]-2-m
ethylpropionic acid or a pharmaceutically acceptable salt thereof. The compound or salt are useful as antihistamines.
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4634699 |
Branched chain phenothiazine
The compound 2-[10-(2-Dimethylaminopropyl)-2-phenothiazinyl]-2-methylprop
ionic acid or a pharmaceutically acceptable salt thereof. The compound and salt are useful as antihistamines.
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4628087 |
Process for the preparation of pharmacologically active compounds containing a sulfoxide group
Process for the preparation of pharmacologically active compounds containing a sulfoxide group by oxidation of a thioether with hypochlorite in an alkaline medium at a pH higher than 10 and at a...
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4366314 |
Dimethine dyestuffs, their preparation and their use for dyeing synthetic and natural materials
Styryl dyestuffs of the general formula ##STR1## wherein Het represents a pyridinium radical having the structure ##STR2## R and R 1 independently of one another designate lower alkyl or alkenyl...
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4349679 |
Pyrrolidino and piperidino benz ring substituted phthalides
Phthalide compounds of the formula ##STR1## wherein A and B, independently of the other, represent a monovalent radical of the formula ##STR2## wherein X 1 represents an amino group of the formula...
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4258182 |
Quaternized amino-substituted styryl dyestuffs
Styryl dyestuffs of the formula ##STR1## wherein Q♁ represents a grouping containing a quaternary nitrogen atom and A represents a bridge member, at least one of the radicals R and R 1 ...
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4160099 |
Labile, non-heterocyclic quaternary ammonium salt/esters as transient derivatives
Labile quaternary ammonium salts of the following formula (I) and (II) are provided: ##STR1## wherein ##STR2## represents a tertiary aliphatic amine; wherein ##STR3## represents an unsaturated...
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4155874 |
Phenothiazinyl sulfides
A new group of compounds, generically classed as phenothiazinyl sulfides, are described having the formula: ##STR1## wherein n is 1 or 2, x and/or y and/or z represent 0, 1 or 2; R 1 may be H,...
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4065471 |
N-(4-Amino-2-butynyl)imides
N-(4-Amino-2-butynyl)imides are prepared from N-propargylimides, paraformaldehyde and the appropriate secondary amine. The compounds are useful as stimulants or depressants of the central nervous...
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4029783 |
N-substituted 1-amino-3-phenoxy-propan-2-ol compounds and therapeutic compositions containing them
New N-substituted 1-amino-3-phenoxy-propan-2-ol compounds of the formula: ##STR1## wherein R 1 and R 2 are, individually, hydrogen or, taken together, represent a sulfur linkage, an ethylene...
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3966930 |
Phenothiazine derivatives, compositions thereof and methods of preparation thereof
Fluoro-substituted phenothiazine derivatives as well as their non-toxic pharmaceutically acceptable acid addition salts having pronounced neuroleptic properties and a relatively low degree of...
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3905981 |
N-dealkylation of tertiary amines
A method for the N-dealkylation of tertiary amines which involves replacing an N-alkyl group of the tertiary amine with a vinyloxycarbonyl group by reaction with, for example, vinyl chloroformate...
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3882044 |
Antioxidant composition of a rearrangement product of a tetra-aryl hydrazine and sulfur or a sulfurizing agent
Antioxidant compositions are prepared by thermally rearranging tetra-aryl hydrazines and then heating the rearrangement product with sulphur or sulphurising agents.
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3719671 |
10-IMIDOYLPHENOTHIAZINES
Novel 10-imidoylphenothiazines are prepared by reacting a phenothiazine which may have hydrogen, trifluoromethyl, methylthio, alkyl, alkoxy or halogen substituents in the 2 or 4 position with a...
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3625963 |
PROCESS FOR THE PREPARATION OF 3-METHANESULPHONYL-PHENTHIAZINES
3-Methanesulphonyl-phenthiazines (Beilstein nomenclature) unsubstituted or substituted on the nitrogen atom of the phenthiazine nucleus are prepared by oxidizing the methylthio group of a...
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3535316 |
PHENOTHIAZINES AND PROCESS FOR THEIR PRODUCTION
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3534030 |
PHENOTHIAZINE DERIVATIVES
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3525736 |
SUBSTITUTED DIAZIRIDINES AND DIAZIRINES
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3501497 |
(1-INDOLINYL)-LOWER ALKYLAMIDOXIMES AND -AMIDINE
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3484444 |
INTERNAL SALT OF SCOPOLAMINE
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3472872 |
INDOLYL-LOWER-ALKYL-AMIDOXIMES
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3454598 |
NOVEL PROCESS FOR PREPARING DIHYDROBENZOXAZEPINES
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3453269 |
NOVEL CHLORPROMAZINE SALTS
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3431270 |
CERTAIN AMINOXYETHYL DERIVATIVES OF 2(1H)-PYRIDONES
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3419553 |
Fluorinated phenothiazine compounds
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3409713 |
Phenothiazinyl aminocyclopropanes
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3354174 |
1-and 2-benzimidazolyl-lower-alkylamidoximes, amidines-, and guanidines
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3347857 |
Organic compounds
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3346573 |
Process for aminoalkylation of phenothiazine and derivatives thereof
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3345361 |
Certain n, n'-substituted diaminoethane compounds
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3320249 |
Adamantyl derivatives of phenothiazines
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