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3980655 Basically substituted 1,4-dihydro-2H-isoquinoline derivatives and process for preparing them  
1,4-Dihydro-2H-isoquinoline derivatives of the general formula I ##SPC1## in which R 1 represents hydrogen or straight chain or branched alkyl of 1 to 6 carbon atoms, R 2 represents low...
3957791 Hydroxyalkyl-piperazino-quinoline nitrates  
Disclosed are compounds of the class of quinolines substituted at the 2-, 3- or 4- position by an amino function bearing a hydroxyalkyl nitrate moiety, e.g. 4-(2-hydroxyethylpiperazino)-quinoline...
3948898 1,3-Dioxo-2-aminoalkyl-4,4-dimethyl-isoquinolines and salts thereof  
Compounds of the formula ##SPC1## Wherein R 1 is hydrogen, halogen, methoxy or methylthio R 2 is hydrogen or methoxy, n is 2 or 3, and A is ##SPC2## Or ##SPC3## Where R 3 is...
3948917 1,4-Dithiino(2,3-c)pyrrole derivatives  
New compounds of the formula: ##SPC1## Wherein A is a phenyl, pyridyl, pyridazinyl, 2-, 3- or 4-quinolyl or naphthyridinyl radical, or a said radical substituted by one or two atoms or radicals...
3944551 N-Coumaranyl and chromanyl -methyl-or sulfur analogs thereof-N'- thiazolyl piperazines  
Disubstituted piperazines of the formula: ##SPC1## Wherein: n is 1 or 2; X is oxygen or sulfur; R is hydrogen or lower alkyl; Het is pyridyl, pyrimidinyl, pyridazinyl, pyrazinyl,...
3932412 1-(4-Hydroxyalkylpiperazino)-isoquinoline nitrates  
Disclosed are compounds of the class of isoquinolines substituted at the 1-position by an amino function bearing a hydroxy-alkyl nitrate moiety, e.g.,...
3932416 N-tetrazolyl quinaldamides  
Compounds of the general formula (I): ##SPC1## in which R 1 , R 2 and R 3 may be the same or different and each represents a hdyrogen atom, an alkyl group, a nitro group, a halogen atom or a...
3929791 2 Substituted-10[4-(2-oxazolidi none-lower alkyl)]-piperazine-dibenzo[b,f]t  
Dibenzothiepin derivatives of the general formula ##SPC1## Wherein m, n, R 1 , R 2 , R 3 and X are as hereinafter set forth, And salts thereof as well as processes for their manufacture are...
3917593 N-alkenyl and N-alkynyl (2-quinolyl)thio-acetamides  
The compounds are N-alkenyl and N-alkynyl thioamides, for example N-allyl and N-propargyl 2-(2-pyridyl)thioacetamide, which are inhibitors of gastric acid secretion.
3915965 2-Alkoxy(and 2-amino)-3-amino-2-heterocyclic-thiopropanamides  
The compounds are 2-alkoxy(and 2-amino)-3-amino-2-heterocyclic-thiopropanamides, for example 2-methoxy-N-methyl-3-morpholino-2-(2-pyridyl)thiopropanamide , which are inhibitors of gastric acid...
3914231 (-)(Cis-1,2-epoxypropyl)-phosphonic acid and salts thereof  
(-) (Cis-1,2-epoxypropyl)-phosphonic acid, a water soluble acidic substance, and its salts are active against both gram-positive and gram-negative bacteria. The antibiotic is produced by growing...
3910915 1-Aryl-2-[(substituted amino)alkanoyl]-1,2,3,4-tetrahydroisoquinolines  
1-Aryl-2-[(substituted amino)alkanoyl]-1,2,3,4-tetrahydroisoquinolines having anti-arrhythmic, anti-bacterial, anti-fungal, anti-algal, anti-protozoal and anthelmintic activity are described...
3905982 1-Aryl-n-dialkylaminoalkyl-3,4-dihydro-2(1H)-isoquinolinecarboxamides and related compounds  
1-Aryl-N-dialkylaminoalkyl-3,4-dihydro-2(1H)-isoquinolinecar boxamides and related N-substituted amides having anti-arrhythmic, anti-bacterial, anti-fungal, anti-algal and anthelmintic activity are...
3886163 1,3(2H,4H)-dioxoisoquinoline-4-carboxamides  
1,3(2H,4H)-Dioxoisoquinoline-4-carboxamides, nuclear unsubstituted and substituted, are prepared by reacting the appropriate homophthalimide with potassium cyanate. Secondary carboxamides are...
3884921 Isoindoline derivatives  
Isoindolin-1-one derivatives substituted in the 2-position by an unsubstituted or substituted quinolyl radical, substituted in the 3-position by a 4-methylpiperazin-1-ylcarbonyloxy or...
3876645 Pyridine thioacetamide derivatives  
Compounds of the formula ##SPC1## Wherein R 1 is hydrogen, lower alkyl, lower alkoxy or halogen and n is an integer of 1 to 4, or wherein (R 1 ) n is a divalent straight chain hydrocarbon radical...
3860592 2-ALKOXY-3-AMINO-2-HETEROCYCLIC-THIOPROPANAMIDES  
The compounds are 2-alkoxy(and 2-amino)-3-amino-2-heterocyclic-thiopropanamides, for example 2-methoxy-N-methyl-3-morpholino-2-(2-pyridyl)thiopropanamide , which are inhibitors of gastric acid...
3856796 HYDROXYALKYL-SUBSTITUTED-AMINO-QUINOLINES AND NITRATES THEREOF  
Disclosed are compounds of the class of quinolines substituted at the 2-, 3- or 4- position by an amino function bearing a hydroxyalkyl nitrate moiety, e.g. 4-(2-hydroxyethylpiperazino)-quinoline...
3759924 1-AMINO-3(OR4)-PHENYL-3,4-DEHYDROISOQUINOLINES  
3,4-Dihydroisoquinoline derivatives of the formula:- ##SPC1## Wherein the symbols R represent hydrogen, halogen or methoxy, or together form the methylenedioxy radical, the symbols R 1 and R 2 ...
3723434 PIPERAZINO ISOQUINOLINE BRONCHODILATORS  
A series of novel 4-piperazino-6,7-dialkoxyquinazolines and 1-piperazino-6,7-dialkoxyisoquinolines have been prepared, including their acid addition salts. These compounds are useful in therapy as...
3692790 5-(AMINOALKYLAMINO)-6(OR)-HALO-8-QUINOLINEMETHANOLS, THEIR ALKYL ETHERS AND ALKANOYL ESTERS  
5-(Aminoalkylamino)-6(or 7)-halo-8-quinolinemethanols, their lower-alkyl ethers and lower-alkanoyl esters, having schistosomacidal activity, are prepared by reducing the corresponding lower-alkyl...
3682920 (PHENYL PIPERAZYL ALKYL) 3,4-DIHYDROCARBOSTYRIL  
1-Substituted derivatives of 3,4-dihydrocarbostyril that are useful as analgesic agents. These compounds are prepared by reacting a 3,4-dihydrocarbostyril or substituted 3,4-dihydrocarbostyril with...
3682927 5,7-BICHLORO-8-HYDROXY-2-ACETYLAMINO QUINOLINE  
An extensive series of quinoline derivatives is disclosed, more particularly several 5,7-bichloro-8-hydroxy-quinolines carrying various substituents in the 2-position. The most interesting...
3671518 BENZODIAZEPIN-2-ONES AND PROCESSES FOR THEIR PREPARATION  
3-substituted benzodiazepin-2-ones, derivatives thereof and processes for their preparation are described. These compounds are useful as anti-convulsants, muscle relaxants and sedatives.
3668207 2-AMINO-4-ARYL-QUINOLINES  
2-Amino-4-aryl-quinolines, e.g. those of the formula ##SPC1## Acyl derivatives, quaternaries and salts thereof, exhibit antiinflammatory effects.
3625969 6-SULFAMYL-4-HYDROXY-3-CARBOXY-QUINOLINES  
Compounds of the formula ##SPC1## In which R = disubstituted amino group R 3 = lower aliphatic hydrocarbon radical, lower alkoxy group, lower alkenyloxy group, hydroxy group, halogen,...
3622457 PROCESS FOR PREPARING 5-(AMINOALKYLAMINO)-6 (OR 7)-HALO-8-QUINOLINE METHANOLS  
5-(aminoalkylamino)-6(or 7)-halo-8-quinolinemethanols, having schistosomacidal activity, are prepared by subjecting the correspoonding 6(or 7)-halo-5-(aminoalkylamino)-8-methylquinoline to the...
3551413 BENZO-LACTAMS  
3542785 2-HYDROXY-4-ARYL-QUINOLINES  
3538101 4 PHENOL DIHYDROQUINOLINES  
3517005 CERTAIN 2- AND 4-SUBSTITUTED QUINAZOLINES  
3493570 QUINOLINE DERIVATIVES  
3488728 N-(NITRO-FURFURYLIDENE-METHYL-HETEROCYCLYL)-AMIDINES  
3472857 N-(3-PYRAZOLYL-PROPYL)-N'-PHENYL PIPERAZINES  
3444173 SUBSTITUTED 8-HYDROXY-QUINOLINE DERIVATIVES  
3399199 Nitroalkyl-piperazines  
3393195 1, 2, 3, 6, 7, 11b-hexahydro-4h-pyrazino-2, 1-a-isoquinolines  
3387001 Novel aminoacyl esters of desacetyl vincaleukoblastine  
3374231 Hydrazones of 1-amino-4-(xanthenyl and thioxanthenyl)piperazines  
3367936 4-(PIPERAZINOALKYL)-PYRAZOLES  
3362956 1-[(heterocyclyl)-lower-alkyl]-4-substituted-piperazines  
3351525 Coccidiostatic compositions and methods of using same  
3341519 Novel benzoxazines, benzothiazines, benzoxazepins and benzothiazepins  
3331843 1-substituted-4-substituted aminoalkylene piperazines  
3330823 N-amino-loweralkylene-benzo-lactams  
3324129 Quinoline derivatives  
3311632 3-acetyl-cinchoninic acid compounds  
3275628 4-substituted-aliphatic-2, 2-dialiphatic-1, 2-dihydroquinolines  
3272807 Unsymmetrical disubstituted aminoalkyl hydrazines  
3272824 4-amino-6, 7-di(lower) alkoxyquinolines