Patents in Class 544/298

Matches 51 - 100 out of 627

Match	Document	Document Title
51	6794336	Herbicidal substituted pyridines, their preparation, and their use as herbicides and plant growth regulators The present invention relates to a compound of the formula (I) or salt thereof in which R 1 is identical or different at each occurrence and is H, halogen, CN, nitro, SF 5 , (C 1 -C 8 )alkyl,...
52	6787561	Benzimidazole compounds A benzimidazole compound or a salt thereof which has an inhibitory action of forming of macrophages and is useful as an active ingredient of an orally available medicament for preventive and/or...
53	6746731	Ferroelectric active matrix displays with wide operating temperature range The active-matrix display contains a chiral smectic liquid-crystal mixture comprising at least one compound of the formula (I) R 1 —(A 1 —M 1 ) a —(A 2 —M 2 ) b —A 3 —X—B 1 —(B 2 )...
54	6727254	Heteroaryl tropane derivatives as superior ligands for nociceptin receptor ORL-1 Novel compounds of the formula wherein R is optionally substituted heteroaryl or R 1 is H or C 1 -C 6 alkyl; and R 2 and R 3 are —CH 3 , —OCH 3 or halo; or a pharmaceutically...
55	6723753	Substituted n-benzyl-n-phenyl aminoalcohol compounds useful for inhibiting cholesteryl ester transfer protein activity The invention relates to substituted polycyclic aryl and heteroaryl tertiary-heteroalkylamine compounds useful as inhibitors of cholesteryl ester transfer protein (CETP; plasma lipid transfer...
56	6720322	Butyne diol derivatives The present invention relates to novel butyne diol derivatives of the general formula I and their use as active ingredients in the preparation of pharmaceutical compositions. The invention also...
57	6720327	Lactone integrin antagonists The present invention relates to a class of compounds represented by the Formula I. or a pharmaceutically acceptable salt thereof, pharmaceutical compositions comprising compounds of the Formula...
58	6706745	Biphenylamidine derivatives The present invention relates to a biphenylamidine derivative of the general formula (1): or a pharmaceutically acceptable salt thereof, which is a novel compound functioning as a clinically...
59	6686367	Polyhydroxylated monocyclic N-heterocyclic derivatives as anti-coagulants This invention is directed to poly-hydroxylated monocyclic N-heterocyclic derivatives selected from the following formulae: wherein Z 1 , Z 2 , R 1 , R 2 , R 3 , R 4 , R 5 , R 6 , and R 7 are...
60	6686364	Benzamidine derivatives and their use as anti-coagulants This invention is directed to benzamidine derivatives which are useful as anti-coagulants. This invention is also directed to pharmaceutical compositions containing the compounds of the invention,...
61	6685995	Ester compounds, liquid crystal compositions and liquid crystal display devices Liquid crystalline compounds suitable for driving at a low voltage and at a wide temperature range, and suitable for high speed response, liquid crystal compositions comprising the compound, and...
62	6677339	Phenylalanine derivatives Phenylalanine derivatives of formula (1) are described: in which: Ar 1 is an aromatic or heteroaromatic group; L 1 is a linker atom or group; R is a carboxylic acid or a derivative thereof; Ar...
63	6670367	Azinyloxy, and phenoxy-diaryl-carboxylic acid derivatives, their preparation and use as mixed ETA/ETB endothelin receptor antagonists The invention relates to carboxylic acid derivatives of the formula I where the radicals have the meanings stated in the description, and to their use as drugs.
64	6667326	Pesticidal aminoheterocyclamide compounds The invention relates to compounds of the general formula wherein R 1 , R 2 , R 3 , R 4 , R 5 , X 1 , X 2 , X 3 , m and n have the significances given in claim 1 , and optionally the...
65	6653258	Hetero-aryl compounds having herbicidal, fungicidal and insecticidal activity Fungicidal compounds of the formula (I): and stereoisomers thereof, wherein R 1 is optionally substituted aryl or optionally substituted heteroaryl; Y is oxygen, sulphur or NR 4 ; R 2 , R 3 ...
66	6642230	Imidazopyrimidines and imidazopyridines for the treatment of neurological disorders Corticotropin releasing factor (CRF) antagonists of formula (I): and their use in treating psychiatric disorders and neurological diseases, anxiety-related disorders, post-traumatic stress...
67	6616990	Chiral 1, 3-dioxane compounds The present invention relates to chiral 1,3-dioxane compounds and diastereomers thereof of the general formula I where R 1 , R 2 and R 3 are as defined in the description, and the use of these...
68	6610695	Aryloxy substituted pyrimidine imidazole compounds Novel 2,4,5-triaryl substituted imidazole compounds and compositions for use in therapy of CSBP/RK/p38 mediated diseases.
69	6610678	CRF antagonistic quino-and quinazolines This invention concerns compounds of formula including the stereoisomers and the pharmaceutically acceptable acid addition salt forms thereof, wherein R 1 is C 1-6 alkyl, NR 6 R 7 , OR 6 or SR...
70	6605611	Base analogues Nucleoside analogues or base analogues having structure (I), where X=O or NH or S, Y=N or CHR 6 or CR 6 , W=N or NR 6 or CHR 6 or CR 6 or S, n=1 or 2; each R 6 is independently H or O or alkyl...
71	6600044	Process for recovery of the desired cis-1,3-oxathiolane nucleosides from their undesired trans-isomers A process for the preparation of 1,3-oxathiolane nucleoside analogues in predominantly the cis-form, from mixture of cis-/trans-1,3-oxathiolane nucleosides or their protected derivatives thereof,...
72	6596727	Substituted pyrimidines, processes for their preparation, and their use as pesticides and fungicides Substituted 4-amino- and 4-alkoxy-cycloalkylpyrimidines, processes for their preparation, and their use as pesticides and fungicides The invention relates to compounds of the formula in which R 1...
73	6586441	Adenosine receptor ligands and their use in the treatment of disease The invention relates to cyclic heteroaromatic compounds, containing at least one nitrogen atom, and to their use in the manufacture of medicaments for the treatment of diseases, related to...
74	6576303	Liquid crystal compounds exhibiting negative anisotropy of permittivity Novel liquid crystal compound having a negative and absolutely large value of dielectric anisotropy, being excellent in compatibility with other liquid crystalline compounds at a low temperature...
75	6552030	Polyhydroxylated monocyclic N-heterocyclic derivatives as anti-coagulants This invention is directed to poly-hydroxylated monocyclic N-heterocyclic derivatives selected from the following formulae: wherein Z 1 , Z 2 , R 1 , R 2 , R 3 , R 4 , R 5 , R 6 , and R 7 are...
76	6548504	Compounds The present invention therefore provides, in a first aspect, a compound of formula (I) or a salt thereof: in which the group D is selected from a group of formula (A), (B) or (C) below: in...
77	6545154	Method for the production of N-(5-amino-2-cyano-4-fluoro-phenyl)-sulphonamides and new intermediate products The invention relates to a process for preparing N-(5-amino-2-cyano-4-fluoro-phenyl)-sulphonamides in which, in a first step, 2-amino-4,5-difluoro-benzonitrile is reacted with sulphonyl halides in...
78	6528455	Phenoxy-and thiophenoxy acrylic acid compounds as herbicides Phenoxy- and thiophenoxyacrylic acid compounds of the formula I in which Het, R 1 , R 2 , R 3 , V, W and Z are as defined in claim 1 and processes for their preparation, intermediates for...
79	6492366	Cyano-indole serotonin-reuptake inhibitor compound A compound selected from those of formula (I): wherein: R 1 and R 2 each independently represent hydrogen or, alkyl, T 1 and T 2 each independently represent alkylene, G represents a...
80	6482829	Substituted heterocyclic siprodecane compound active as an antagonist of neurokinin 1 receptor The invention relates to compounds of the formula as described herein and pharmaceutically acceptable acid addition salts thereof. The described compounds have a good affinity to the NK1 receptor.
81	6469167	Process for the preparation of thiazolidine-2,4-dione derivatives An improved process for the preparation of 5-[4-[[3-Methyl-4-oxo-3,4-dihydroquinazolin-2-yl]methoxy]ben zyl]thiazolidine-2,4-dione of formula (1) which comprises: reducing the compound of formula...
82	6458433	Difluorophenyl derivatives, liquid-crystal compounds, and liquid-crystal composition Disclosed are liquid crystalline compounds which (i) are characterized in that the compounds have a wide temperature range in which the compounds exhibit a liquid crystal phase, are low in...
83	6448242	Cyclic amide compounds The invention relates to compounds represented by the following general formula (1): wherein A is an aromatic compound which may be substituted, or the like, B is a nitrogen atom or CH, X is a...
84	6444278	2,6-di-tert-butylphenols The present invention relates to 2,6-di-tert-butylphenols of the formula I in which R, A 1 A 2 , Z 1 , Z 2 m and n are as defined herein, and their use as stabilizers or antioxidants.
85	6444679	4-phenyl-4-heteroarylpiperidine derivatives The present invention relates to compounds of the formula I, wherein Z 1 , X, Y, ( ) n , R 1 , R 2 and R 3 are defined as in the specification, pharmaceutical compositions containing such...
86	6441175	1-(N'-arylalkylaminoalkyl)aminoisoquinolines: a new class of dopamine receptor subtype Disclosed are compounds of the formula or the pharmaceutically acceptable salts thereof wherein the variables R 5 , R 11 , R 12 , R 13 , R 1 , R 11 , Ar, n, m and L are defined herein. These...
87	6440965	Substituted pyrimidine derivatives, their preparation and their use in the treatment of neurodegenerative or neurological disorders of the central nervous system The present invention relates to novel derivatives of a series of substituted pyrimidines, to pharmaceutical compositions which contain them, to methods for their preparation and to their use in...
88	6441169	Pyrimidin-2-oxy-4-one and pyrimidin-2-oxy-4-thione derivatives Novel pyrimidin-4-one and pyrimidin-4-thione derivatives of formula (I) wherein A is phenyl, thienyl (including all 3 isomers), thiazolyl or pyridyl; X is oxygen or sulfur; R 1 is hydrogen,...
89	6417359	Pharmaceutical compositions and methods for use A compound having the formula: wherein X′ is nitrogen or carbon bonded to a substituent species characterized as having a sigma m value greater than 0, less than 0 or 0; X is nitrogen or...
90	6403794	Substituted 2-amino-4-alkylamino-1,3,5-triazines as herbicides The invention relates to novel substituted 2-amino-4-alkylamino-1,3,5-triazines of the formula (I) in which R 1 represents in each case optionally substituted alkyl having 2 to 6 carbon atoms...
91	6376428	Dihalopropene compounds, insecticidal/acaricidal agents containing same, and intermediates for their production The dihalopropene compounds of the general formula [I] have excellent insecticidal/acaricidal activity, so that they are satisfactorily effective for the control of noxious insects, mites and ticks.
92	6362180	Imidazopyridines for the treatment of neurological disorders Corticotropin releasing factor (CRF) antagonists of formula (I): and their use in treating psychiatric disorders and neurological diseases, anxiety-related disorders, post-traumatic stress...
93	6362192	2-(Pyrazolyloxy) -pyridin-3-ylacetic acid derivatives, agents containing the same and use thereof against noxious fungi and animal parasites Compounds of the formula I and salts thereof, in which the substituents and the index n have the following meanings: Q is —C(═CHCH 3 )—COOCH 3 , —C(═CHOCH 3 )—COOCH 3 , —C(═NOCH...
94	6333082	Liquid crystalline (E,E)-butadiene compounds and mixtures and devices containing such compounds Liquid crystalline compounds useful in super twisted nematic liquid crystal displays are described and have the formula: ##STR1## wherein n is 1-5; m is 0-5; p is 0, 1 or 2; q is 0, 1...
95	6333080	Liquid-crystal alkenyltolan derivative, liquid-crystal composition, and liquid-crystal display element A liquid crystalline alkenyltolan derivative expressed by the general formula C t H 2t -1 --G--(CH 2 ) m --A 1 --B 1 --(A 2 --B 2 ) n --(A 3 --B 3 ) p --A 4 --X wherein A 1 , A 2 , A 3 ,...
96	6326065	Pyrimidine derivative, liquid crystal composition comprising the derivative, and liquid crystal display device fabricated by using the composition Liquid crystalline compounds having a comparatively high voltage holding ratio, high Δn and high Δε, and excellent miscibility with known liquid crystalline compounds at low temperatures. The...
97	6312538	Chemical compound suitable for use as an explosive, intermediate and method for preparing the compound A new compound, 1,1-diamino-2,2-dinitroethylene suitable for use as an explosive, as well as an intermediate for preparing the compound consisting of a heterocyclic 5- or 6-ring of the general...
98	6310071	2-(0-(Pyrimidin-4-yl)methyleneoxy)phenylacetic acid derivatives and their use for controlling harmful fungi and animal pests 2-(O-[pyrimidin-4-yl]methylenoxy)phenylacetic acid derivatives of the general formula I ##STR1## and the salts and N-oxides thereof where the radicals R 1 to R 4 and Q have the following...
99	6303569	Trialkyl-lock-facilitated polymeric prodrugs of amino-containing bioactive agents The present invention is directed to double prodrugs containing polymeric-based transport forms. These polymeric compounds comprise the formula: ##STR1## wherein: B is H, OH, OSiR 13 , a...
100	6291467	Heteroaromatic derivatives An aromaheterocyclic derivative represented by the formula: ##STR1## wherein Z is a group represented by the following formula: ##STR2## wherein Ar 1 is a phenyl group or a phenyl group...

Matches 51 - 100 out of 627

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