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4292312 Method for preparing alloxan stable aqueous solutions and solutions resulting therefrom  
Stable aqueous injectable solutions comprising alloxan stabilized with a reducing sugar selected from the group consisting of levulose, glucose and lactose are disclosed.
4288147 Electro-optical composition of the guest-host type  
The electro-optical composition comprises a host liquid crystal and guest dichroic dye which is characterized generally as a linear, noncondensed aromatic compound including one or more quinonoid...
4288442 Inhibiting adrenergic β-receptors with piperidinopropyl derivatives  
A piperidinopropyl derivative of the formula ##STR1## in which R 1 and R 2 each independently is hydrogen or a lower alkyl radical, or together are an alkylene radical, R 3 is hydrogen,...
4287342 2,4,6-Trihalo-5-alkyl-and 5-alkenylsulphonylpyrimidines  
There are described compounds of the formulae I and II ##STR1## and also salts of compounds of the formula I, wherein X represents optionally substituted alkyl or alkenyl, and the Y's represent...
4269873 2-, 5-, and 6-Substituted-1-carbadethiapen-2-em-3-carboxylic acids  
Disclosed are 2-, 5- and 6-substituted-1-carbadethiapen-2-em-3-carboxylic acids having the structure: ##STR1## wherein R 6 , R 7 , R 8 and R 9 are, inter alia, independently selected from the...
4213899 Reactive dyestuffs containing chlorine or fluorine substituents and one or more pyridine radicals linked to the dyestuff at the 2-, 4- or 6-position  
A dyestuff of the formula ##STR1## where D is a chromophoric residue n is 1 or 2 Z is ##STR2## where R is H, C 1 -4 alkyl, C 1 -4 alkyl substituted by OH, OSO 3 H, CN or SO 3 H or is phenyl...
4210583 Azo dyes of the 2,6-di(substituted) amino pyridine series  
An azo dye of the general formula ##STR1## where A is cyano or carbamoyl, R is hydrogen, alkyl or phenyl, R 1 is hydrogen, bromine, chlorine or nitro, R 2 is hydrogen, chlorine, bromine,...
4196288 Ergoline derivatives and a process for their preparation  
New ergoline derivatives are disclosed which are compounds of formula (I) having the structure: ##STR1## wherein R 1 is hydrogen or methoxy; R 2 is hydrogen or methyl; and X is hydroxy, R 3 COO,...
4188483 5-Alkylsulphonyl- and 5-alkenylsulphonylbarbituric acids and derivatives thereof  
There are described compounds of the formulae I and II ##STR1## and also salts of compounds of the formula I, wherein X represents optionally substituted alkyl or alkenyl, and the Y's represent...
4179562 2,4-Diamino-5-alkyloxy-pyrimidines  
Compounds of the formula ##STR1## and pharmaceutically acceptable salts thereof and antimalarial and antibacterial compositions containing an effective amount of active agent and a pharmaceutically...
4166852 Piperazino-pyrimidines and their use as spasmolytic agents  
The compounds of the formula: ##STR1## in which R represents a methyl or methylthio group, X represents a halogen atom or an alkoxy group containing 1 to 5 carbon atoms, Y represents an acylamino...
4152426 Pesticidally active O-alkyl-O-[1,6-Dihydro-1-substituted-6-oxo-pyrimid in-4-yl]-(thiono) (thiol) phosphoric (phosphonic) acid esters and ester-amides  
O-alkyl-O-[1,6-dihydro-1-substituted-6-oxo-pyrimidin-4-yl]-( thiono) (thiol) phosphoric (phosphonic) acid esters and ester-amides of the formula ##STR1## in which R represents alkyl, R 1 ...
4147789 6-Methyl-8-thiomethyl-ergolene derivatives  
This invention provides new compounds of formula I, ##STR1## wherein X Y IS THE GROUP ##STR2## and R is hydrogen, cyano, a 5- or 6-membered unsaturated heterocyclic radical attached through a ring...
4061643 Certain 16-aryloxy-11,12-seco-prostaglandins  
This invention relates to aryloxy-, alkoxy-, arylthio-, and alkylthio-11,12-seco-prostaglandins and to processes for their manufacture. These compounds have prostaglandin-like activity and are...
4059548 Hexahydropyrimidine-1,3-diacetonitriles and processes for preparing the same  
N,N'-Dicarboxymethyl-1,3-propanediamine (designated PDDA) is prepared by reacting 1,3-propanediamine with formaldehyde and HCN to form hexahydropyrimidine-1,3-diacetonitrile, which is hydrolyzed...
4058528 5-Hydroxyhexahydropyrimidine  
N,N'-Dicarboxymethyl-1,3-propanediamine (designated PDDA) is prepared by reacting 1,3-propanediamine with formaldehyde and HCN to form hexahydropyrimidine-1,3-diacetonitrile, which is hydrolyzed...
4052386 Reactive phthalocyanine dyestuffs containing a fluoropyrimidinyl group  
Reactive dyestuffs of the formula ##STR1## in which D is the residue of an organic dyestuff, R is hydrogen or a lower alkyl, R 1 is hydrogen or a substituent, R 2 is hydrogen, halogen,...
4051244 2,4-Diamino 5-bromo 6-chloro pyrimidines, process for their preparation and use as pharmaceuticals  
Compounds of the general formula ##STR1## wherein R 1 and R 3 represent hydrogen or alkyl containing 1 to 4 carbons; R 2 and R 4 represent hydrogen, alkyl containing 1 to 8 carbons,...
4027027 Pyridyloxyalkyleneamino-phenoxy-propanol-2-compounds  
Compounds of the formula ##STR1## WHEREIN Ar 1 and Ar 2 denote an optionally substituted aromatic hydrocarbon radical or a monocyclic, monoazacyclic or diazacyclic radical of aromatic character...
3996228 Pyrimidinoaminoethyl ergoline derivatives  
Pyrimidinoaminoethyl ergoline derivatives of the formula: ##STR1## wherein R is hydrogen or methyl; R 1 and R 2 are independently selected from the group consisting of hydrogen, alkyl having 1 to...
3984411 Pyrimidines  
Compounds having the formula ##SPC1## Process for the preparation of such compounds which comprises reacting a pound having the formula: ##SPC2## Medicaments containing a compound of formula (I) or...
3968214 5-Methylthio-pyrimidine vasodilators  
The compounds of the formula: ##SPC1## In which Y represents a chlorine atom or an alkoxy, dialkylaminoalkoxy, pyridylalkoxy group, R 1 and R 2 are identical or different substituents and...
3966732 Nitroimidazolyl pyrimidines  
Nitroimidazolyl pyrimidines of the formula ##SPC1## And physiologically acceptable acid addition salts thereon wherein X is alkyl of 1-4 carbon atoms, R 1 and R 2 each are a hydrogen atom, alkyl...
3957785 Bβ-Pyrimidino-aminomethyl-10α-ergoline and 10α-methoxyergoline derivatives  
Novel 8β-pyrimidino-aminomethyl-10α-ergoline and 10α-methoxyergoline derivatives which possess a high and prolonged adrenolytic activity and a low toxicity, and some of which also possess...
3941804 1-Heteroarylsulphonyl-2-imino-imidazolidines  
Compounds of the class of 1-heteroarylsulphonyl-2-imino-imidazolidines which are substituted in the 3-position by an aliphatic or cycloaliphatic hydrocarbon radical, especially a cycloalkyl...
3941786 Process for the production of 4-hydroxy-6-hydroxymethylpyrimidine  
Process for the production of 2-R 1 substituted-4- hydroxy-5-R 2 substituted -6-hydroxy methyl-pyrimidines having the following general formula: ##EQU1## wherein R 1 can be an alkyl group, a...
3926994 Heterocyclic compounds  
The disclosure relates to derivatives of tetrahydropyrimidine, imidazoline, tetrahydro-1H-1,3-diazepine and hexahydro-1,3-diazocine of the general formula ##SPC1## Or an acid addition salt thereof...
3927023 Imidazolyl benzofurans  
Imidazolyl and tetrahydropyrimidyl benzofurans of the formula: ##SPC1## Are disclosed. In the above structure A, B, and C are hydrogen or lower alkyl of 1 to 6 carbon atoms, halogen, lower alkoxy...
3920655 Nitroimidazolyl benzoquinazolines  
Nitroimidazolyl pyrimidines of the formula ##SPC1## And physiologically acceptable acid addition salts thereof wherein X is alkyl of 1-4 carbon atoms, R 1 and R 2 each are a hydrogen atom, alkyl...
3907797 5-(3-Iodinepropargyloxy)pyrimidines  
(Iodinepropargyloxy)-pyrimidines of the general formula ##EQU1## wherein R is selected from among hydrogen, alkyl, alkoxy, alkylthio, alkylsulfinyl and alkylsulfonyl radicals are described, and a...
3883529 NEW CELLULOSE REACTIVE DYESTUFFS  
Reactive dyestuffs of the triphenylmethane or xanthene series having the formula: ##SPC1## Wherein R 1 represents H or an alkyl group and R 2 represents an alkyl, aryl or substituted aryl group,...
3862190 5-(UNSUBSTITUTED AND SUBSTITUTED PHENOXY)-4-AMINO PYRIMIDINES  
The preparation of novel 5-(substituted phenoxy)-4-amino and substituted amino pyrimidines is described. These compounds, possessing anti-secretory an;d anti-ulcer activity, are effective...
3846428 NITROFURYLPYRIMIDINES  
Compounds of the formula Wherein R is saturated or unsaturated, straight-chain or branched hydrocarbon aliphatic group of 1-6 carbon atoms or cyclic alkyl of 3-7 carbon atoms, alkyl of 1-6 carbon...
3843656 2-METHYLAMINO-4'-METHYL-4-PIPERAZINYL-6-CHLORO-5-METHYLTHIO-PYRIMIDINE, SALTS THEREOF, AND PROCESS FOR THEIR PREPARATION  
The compound of the formula: ##SPC1## Salts of this compound and process for the preparation of the compound which comprises condensing one mole of 2,4,6-trichloro-5-methylthio-pyrimidine with 1...
3817998 2-AMINO AND SUBSTITUTED AMINO-4, 6-DIAMINO-5-PYRIMIDINESULFONAMIDES  
2-Amino and substituted amino-4,6-diamino-5-pyrimidinesulfonamides, e.g., 4,6-diamino-2-methylamino-5-pyrimidinesulfonamide, are prepared by treating...
3755312 6-SUBSTITUTED-1, 2,4-PYRIMIDO[4,5-E]THIADIAZINE-1,1-DIOXIDES  
Substituted 8-amino 1,2,4-pyrimido[4,5-e]-thiadiazines-1,1-dioxides, e.g., 8-amino-3-ethyl-6-methylthio-1,2,4-pyrimido[4,5-e]thiadiazin e-1,1-dioxide, are prepared from substituted...
3621022 ANTIBACTERIAL 5-NITROFURYL-PYRIMIDINES  
Novel 5-nitrofuran derivatives and the physiologically acceptable salts thereof having the formula: ##SPC1## Wherein R 1 and R 2 each represent hydrogen, hydroxyl, lower alkyl, alkoxy, amino or...
3549654 1,1'-ALKYLENE-BIS(3,3-DICHLORO-2-PYRROLIDINONES)  
3528967 N1-ACETYL-N1-(CYCLOPROPYL-4-PYRIMIDINYL)-SULPHANILAMIDES  
3511837 4-PYRIMIDYL-1,4-DIHYDROPYRIDINE DERIVATIVES AND THEIR PRODUCTION  
3464987 1,2-DIHYDRO-1-HYDROXY-2-IMINO-6-(LOWER ALKYL)PYRIMIDINES  
3457278 CYCLOPROPYL-4-SULFANILAMIDO-PYRIMIDINES  
3435035 PYRIMIDINE SULFONES  
3431263 CERTAIN 2-BENZENESULFONAMIDO-5-OXYPYRIMIDINES  
3422098 SULFANILAMIDO-PYRIMIDINES  
3382248 6-amino-4, 5-di(substituted amino)-1, 2-dihydro-1-hydroxy-2-iminopyrimidines  
3337543 Novel method of preparing 1, 3-diazaphenothiazines  
3331841 Certain derivatives of 2-amino-5-alkoxypyrimidine  
3322767 Tham salts  
3317536 4-benzenesulfonamido-pyrimidine derivatives