Patents in Class 544/2

Matches 1 - 50 out of 109

1 2 3 >

Match	Document	Document Title
1	7608658	Amine-functionalized liquid polyisoprene This invention discloses a process for manufacturing an elastomeric article by liquid injection molding, said process comprising the steps of: (I) heating a curable composition comprised of (1) a...
2	7531668	2-arylcarboxamide-nitrogenous heterocycle compound A compound represented by the formula [I]: [wherein R 1 and R 2 are the same or different and each represents C 1-6 alkyl, C 3-8 cycloalkyl, et al; R 3a , R 3b , and R 4 are the same or...
3	7507730	Substituted pyrazolo[1,5-a]pyrimidines as potassium channel activators Novel heterocyclic dihydropyrimidine compounds useful as inhibitors of potassium channel function (especially inhibitors of the K v 1 subfamily of voltage gated K + channels, especially inhibitors...
4	7504499	Methods of attaching biological compounds to solid supports using triazine Disclosed are methods of attaching biologically active compounds to a solid surface, comprising modifying the solid surface using triazine chloride and attaching the biologically active compound to...
5	7408059	Method for producing 3, 4-dihydro-1,2,3-oxathiazin-4-one-2,2-dioxide compound or salt thereof A method produces a 3,4-dihydro-1,2,3-oxathiazin-4-one-2,2-dioxide compound of following formula (2): wherein R 1 and R 2 are the same as or different from each other and are each hydrogen...
6	7294650	Benzothiophen and thiochrone containing phenethanolamine derivatives for the treatment of respiratory disorders Compounds of formula (I): and salts, solvates, and physiologically functional derivatives thereof, useful for the prophylaxis or treatment of a clinical condition for which a selective β 2...
7	7259258	Methods of attaching biological compounds to solid supports using triazine Disclosed are methods of attaching biologically active compounds to a solid surface, comprising modifying the solid surface using triazine chloride and attaching the biologically active compound to...
8	7196108	Bicyclic heterocycles for the treatment of diabetes and other diseases The invention relates to certain bicyclic heterocycles havng the structure shown below which are useful in the treatment of diseases related to lipid and carbohydrate metabolism, such as type 2...
9	7141562	Substituted benzoxazinones and uses thereof Compound of the Formula: and pharmaceutically acceptable salts or prodrugs thereof, wherein: X is CH or N, Y is C or S, Z is —SO 2 — or —(CR a R b ) r —, n is 1 or 2, R 2 is aryl or...
10	7105660	Intramolecular amidation of sulfamates catalyzed by metalloporphyrins An intramolecular amidation processes for substrates such as sulfamates using chiral and non-chiral metalloporphyrin complexes which can maximize catalytic activity, enhance efficiency,...
11	7053109	Aminediols for the treatment of Alzheimer's disease The present invention relates to compounds of formula (I): useful in treating Alzheimer's disease and other similar diseases. These compounds include inhibitors of the beta-secretase enzyme...
12	6852885	Production method of high purity organic compound There is provided a method for obtaining a target organic compound such as an alkyladamantyl ester efficiently by purifying a crude organic compound which contains, as impurities, sublimable...
13	6849623	Xanthine and phenazone-acesulfame-H complexes having improved taste, process for their preparation and their use Complex compounds or adducts of xanthine derivatives, for example propentofylline or pentoxyfylline, or phenazone derivatives, for example phenazone, propylphenazone and aminophenazone, and...
14	6797522	Synthetic receptors The invention is directed to synthetic receptor(s) which comprises a polyfunctional organic template covalently linked to two or more oligomers which may independently be the same or different and...
15	6759544	Antimicrobially active acesulfame complexes, process for their preparation and their use Complex compounds containing acesulfame have good antimicrobial action, in particular antibacterial action, and are distinguished by the fact that they are complex compounds of metallic elements...
16	6734304	Method for producing asymmetrical 4,6-bis(aryloxy)pyrimidine derivatives The invention relates to a novel process for preparing known asymmetrical 4,6-bis(aryloxy)pyrimidine derivatives.
17	6727359	Composition comprising 6-methyl-3,4dihydro-1,2,3-oxathiazin-4-one-2,2-dioxide, its salts, preparation thereof and uses therefor Acesulfame-K is a widely used sweetener in food and beverage. It is prepared by using the substituted sodium phenoxide or substituted phenol as the starting substance to synthesize the following...
18	6528648	Detecting reagent for double-stranded nucleic acid and double-stranded nucleic acid detecting method The present invention provides a novel detecting reagent for double-stranded nucleic acid, and a method of using it to detect double-stranded nucleic acid formed by hybridization with a probe, with...
19	6436927	IL-8 receptor antagonists The present invention involves certain 8-ureido and 8-thioureido, 1,2-benzothiazines, 1,2,4-benzothioxazines and 1,2,4-benzothiodiazines useful in the treatment of disease states mediated by the...
20	6407097	Methoximinomethyloxathiazines The invention relates to novel methoximinomethyloxathiazines, to two processes for their preparation and to their use as pesticides.
21	6268311	1-Amino-3-benzyluracils 1-Amino-3-benzyluracils I ##STR1## (X=oxygen, sulfur; R 1 =C 1 -C 4 -haloalkyl; R 2 =H, halogen; R 3 , R 7 =H, CN, SCN, halogen, C 1 -C 4 -haloalkyl, C 1 -C 4 -haloalkoxy, C 1 -C 4 ...
22	6265398	Substituted pyridines/pyrimidines, their preparation and their use as pesticides The present invention relates to novel substituted pyridines/pyrimidines of the formula I ##STR1## where A is CH or N; X is NH, O or S(O) q where q is 0, 1 or 2; Y 1 , Y 2 and Y 3 ...
23	6245934	Method for preparing salts of aspartame from N-protected aspartame Method for preparing a salt of aspartylphenylalanine methyl ester from N-protected aspartylphenylalanine methyl ester involving cleaving off the protective group by treatment with an acid, in the...
24	6020335	(N-(pyridinylmethyl)-heterocyclic)ylideneamine compounds as nicotinic acetylcholine receptor binding agents An (N-(pyridinylmethyl)-heterocyclic)ylideneamine compound of the formula ##STR1## wherein R 3 , A, and B are as described below, and its pharmaceutically acceptable salts and prodrugs. Compounds...
25	5962437	Lipid analogs for treating viral infections A method of treating viral infections, and in particular HIV-1, hepatitis B virus and herpes viruses, is disclosed. The method comprising administering to a subject in need of such treatment an...
26	5922113	Antibacterial and antifouling oxathiazines and their oxides Use of 3-aryl-5,6-dihydro-1,4,2-oxathiazines and their oxides having the formula ##STR1## wherein n is 0, 1 or 2; R 1 is hydrogen, C 1 -4 alkyl or benzyl; and R represents (a) phenyl; phenyl...
27	5914351	Anti-viral aromatic hydrazones Compounds of the formula ##STR1## wherein Q is a hydrazone derivative; R 1 is hydrogen, halogen, alkyl or alkoxy; R 2 is hydrogen, halogen, alkyl, alkoxy, alkenoxy, alkynyloxy, halomethyl,...
28	5874382	Cyclic sulfonamide herbicides Compounds of Formula I and II, and their agriculturally-suitable salts, are disclosed which are useful for controlling undesired vegetation ##STR1## wherein X is a direct bond; O; S; NH; N(C 1 -C...
29	5824677	Substituted amino alcohol compounds Disclosed are compounds having a straight or branched aliphatic hydrocarbon structure of formula I: ##STR1## In formula I, n is an integer from one to four and m is an integer from four to twenty....
30	5780465	4-substituted 5-polycyclylpyrimidine herbicides 4-Substituted 5-polycyclylpyrimidine compounds in which the 5-substituent is polycyclic and is attached to the pyrimidine moiety through an aliphatic carbon atom, such as...
31	5744010	Process for the preparation of the non-toxic salts of 6-methyl-3,4-dihydro-1,2,3-oxathiazin-4-one 2,2-dioxide and arrangement for carrying out this process The invention relates to a process for the preparation of acesulfam salts by reaction of salts of amidosulfonic acid with diketene to give a salt of acetoacetamidosulfonic acid (I), ring closure by...
32	5688809	5-heteroarylindole derivatives The present invention relates to compounds of the formula ##STR1## The present invention also relates to intermediates for the preparation of compounds of the formula I, pharmaceutical compositions...
33	5624981	Polyalkylpiperidine containing acetic acid and 3-amino-acrylic acid derivatives Polyalkylpiperidine-containing acetic acid and 3-aminoacrylic acid derivatives I ##STR1## where R 1 is hydrogen, C 1 - to C 6 -alkyl, formyl, C 2 - to C 6 -alkanoyl, C 1 - to C 12 -alkoxy, C...
34	5614626	1,2,3-Oxathiazin-4(3F)-one 2,2-dioxides, a process for their preparation and their use as electrophilic fluorinating agents The invention relates to compounds of the formula (I) ##STR1## which R is hydrogen or (C 1 -C 4 )-alkyl, to a process for their preparation and to their use as electrophilic fluorinating agents.
35	5532228	Side-chain homologous vitamin D derivatives, process for their production, pharmaceutical preparations containing these derivatives and their use as pharmaceutical agents The invention discloses side-chain homologous vitamin D derivatives of formula I ##STR1## in which R 1 , R 2 , R 3 , R 4 , R 5 , R 6 , B, and D have the meanings defined in the specification and...
36	5525729	Benz-1,2,3-oxathiazin-4(3F)-one-2,2-dioxides, a process for their preparation and their use as electrophilic fluorinating agents The invention relates to compounds of the formula (I) ##STR1## where R 1 , R 2 , R 3 and R 4 are, independently of one another, hydrogen, CF 3 , NO 2 , CN, halogen, --S(NSO 2 CF 3 )CF 3 , (C 1 ...
37	5463052	Method for producing benzylidene derivatives A selective and high-yield method is described for producing stereoisomeric benzylidene derivatives of the formula III: ##STR1## wherein R 1 and R 2 each independently is lower alkyl, lower...
38	5418230	Benzylidene derivatives Benzylidene derivatives having anti-inflammatory activities, are shown by the following formula I: ##STR1## wherein A is -CH 2 - or -CH 2 CH 2 -; B is a bond or -CH 2 -, -CHOH-, -CO-, -O-, or A...
39	5356862	Herbicidal sulfonylureas The invention relates to herbicidal sulfonylurea compounds, agriculturally suitable compositions thereof and a method for their use as general or selective preemergent or postemergent herbicides or...
40	5330987	Substituted pyridopyrimidinones and related heterocycles as angiotensin II antagonists Novel substituted pyridopyrimidinones of formula (I), which are useful as angiotensin II antagonists, are disclosed. ##STR1##
41	5283355	Benzoquinone compounds Compounds of the Formula (5) and processes for their preparation and use, particularly in the manufacture of unsymmetrical triphenodioxazine dyes: ##STR1## wherein: Y is H, alkyl, substituted...
42	5281614	Substituted 1,2,4-triazoles bearing acidic functional groups as angiotensin II antagonists Novel substituted triazolinone, triazolinethione, and triazolinimine compounds of the formula I are useful as angiotensin II antagonists. ##STR1##
43	5260285	Substituted imidazopyridazines as angiotensin II antagonists Novel substituted imidazopyridazines of formula (I) which are useful as angiotensin II antagonists, are disclosed. ##STR1##
44	5250521	Substituted pyrazolopyrimidines as angiotensin II antagonists Novel substituted pyrazolopyrimidines of formula (I) which are useful as angiotensin II antagonists, are disclosed. ##STR1##
45	5223501	Substituted pyrimidinones bearing acidic functional groups as angiotensin II antagonists Novel substituted fused pyrimidinones of formula (I) are useful as angiotensin II antagonists. ##STR1##
46	5212301	Substituted fluorobenzenes Introduction of a fluoro substituent into an aromatic ring adjacent an electron donating group is difficult producing mixed isomers and low yields of desired products. A process for the...
47	5162340	Substituted 1-(2H)-isoquinolinones bearing acidic functional groups as angiotensin II antagonists Substituted 1-(2H)-isoquinolinones of the structural formula: ##STR1## are angiotensin II antagonists which are useful in the treatment of hypertension and congestive heart failure.
48	5158959	Decahydroisoquinoline carboxylic acids What are disclosed are aminoacid compounds of the formula ##STR1## wherein n is 0 or 1, and salts thereof, said compounds and salts having hypotensive properties; methods for making the compounds;...
49	5106840	Method of preparing n-oxo-tetrahydro-beta-carbolines The invention relates to a method of preparing N-oxo-tetrahydro-β-carbolines having formula 1. ##STR1## wherein R 1 is lower alkyl or alkoxy, halogen, trifluoromethyl, lower alkylthio, hydroxy,...
50	5097027	Heterocyclic compounds Heterocyclic compounds of the formula ##STR1## are used as pigments for surface coatings and for coloring and pigmenting high molecular weight organic material.

Matches 1 - 50 out of 109

1 2 3 >