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6887864 Azepane derivatives  
This invention provides novel azepane derivatives or pharmaceutically acceptable salts thereof, according to the general formula (I) wherein the symbols are defined in the specification, as well as...
6803370 Alpha amino acid derivatives—inhibitors of leukocyte adhesion mediated by VLA-4  
Disclosed are certain alpha amino acid compounds which bind VLA-4. Certain of these compounds also inhibit leukocyte adhesion and, in particular, leukocyte adhesion mediated by VLA-4. Such...
6093823 Process for the continuous production of basic cyclic optically active α- amino acids  
The invention pertains to a process for the continuous production of basic cyclic optically active α-amino acids of general formula (I) by continuous racemate splitting via diastereomeric salt ...
5856318 Nitrogen-containing cyclohetero cyclo-heteroaminoaryl derivatives for CNS disorders  
Certain nitrogen-containing cyclohetero cycloalkylaminoaryl compounds are described for treatment of CNS disorders such as cerebral ischemia, psychoses and convulsions. Compounds of particular...
5674864 N-substituted derivatives of α-mercapto alkylamines, their preparation process and the intermediates obtained, their use as medicaments and the compositions containing them  
Novel α-mercapto-alkylamines in all possible racemic, enantiomeric and diastereoisomeric forms of the formula ##STR1## wherein the substituents are as defined in the specification.
5423998 Peroxy carboxylic amino-derivatives  
Amino-derivative (poly)peroxycarboxylic acids which have the formula: ##STR1## wherein the symbols have the following meanings: R, R1, and R2, which may be equal to or different from one another,...
5192498 Elimination of sulfide odor in thiocarbamate herbicides  
It has now been discovered that the undesirable odor in thiocarbamate compounds can be suppressed or mostly eliminated by the process of this invention. Generally, the process of this invention...
5147572 Flotation composition using a mixture of collectors  
The present invention relates to improved flotation composition comprising a mixture of (A) at least one metal salt of a phosphorus acid represented by the Formula: ##STR1## wherein each R1 is...
5120843 Pharmaceutically active amines  
The aromatic amines (I), alkyl amines (II), bicyclic amines (III). ##STR1## cycloalkyl amines (IV), aromatic bicyclic amines (V), hydroquinone amines (VI), quinone amines (VII), amino-ethers (VIII)...
5089471 Peptidyl beta-aminoacyl aminodiol carbamates as anti-hypertensive agents  
Non-peptidyl compounds characterized generally as β-aminoacyl aminodiol carbamates are useful as renin inhibitors for the treatment of hypertension.
5041545 2-hydroxybenzophenone hydrazides and derivatives thereof  
Hydrazide functionalized 2-hydroxybenzophenone ultraviolet light and heat stabilizers and derivatives are disclosed having the general formula: ##STR1## wherein R1, R2, R3, R4, R5, R6, X, Y, Z, all...
5025005 Lipid derivatives, their production and use  
Novel lipid derivatives of the formula ##STR1## [wherein R1 is alkyl or alkylcarbamoyl; R2 is hydrogen, hydroxy which may be substituted, amino which may be substituted or cyclic amino; R3 is a...
5008261 Agents for repelling insects and mites  
It has been found that the substituted α,ω-amino-alcohol derivatives, some of which are known, of the formula I ##STR1## in which X represents hydrogen, COR11, COOR12 or R13, R1 represents o...
4977141 Peptidyl α-aminoacyl aminodiol carbamates as anti-hypertensive agents  
Non-peptidyl compounds characterized generally as aminoacyl aminodiol carbamates are useful as renin inhibitors for the treatment of hypertension.
4900834 Substituted α,ω-aminoalcohol derivatives  
It has been found that the substituted α,ω-amino-alcohol derivatives, some of which are known, of the formula I ##STR1## in which X represents hydrogen, COR11, COOR12 or R13, R1 represents o...
4725680 Process for the preparation of carbamates, thiocarbamates and ureas  
The invention relates to a process for preparing carbamic acid derivatives of formula: ##STR1## in which R1 or R2 denotes a hydrogen atom or a substituted or unsubstituted, saturated or unsaturated...
4686220 Substituted 2-[b-substituted-amino)-ethylamino]-1,4-naphthalenediones for treating asthma, allergic diseases and inflammation in warm-blooded animals  
This disclosure describes certain substituted piperazine-1,4-naphthalenediones useful as anti-asthmatic agents.
4613461 Process for preparing esters of thiolcarbamic acids  
The invention relates to a new process for preparing known thiolcarbamate esters of the general formula (I) ##STR1## wherein R1 and R2 stand independently for hydrogen or a straight or branched...
4521242 Substituted phenyl carbamates, herbicidal compositions containing the same as active ingredient and method of controlling weeds  
There are provided novel substituted phenyl (thiono)carbamates capable of effectively controlling broad-leaved annual weeds and annual weeds belonging to the families Gramineae and Cyperaceae such...
4497739 Synthesizing thiocarbamic acid esters  
A process for the synthesis of thiocarbamic acid esters by reacting amine compounds having a general formula ##STR1## wherein A is an arylene radical, simple or substituted by halogens hydrocarbon...
4491465 Substituted phenyl (thiono)carbamates, herbicidal compositions containing the same as active ingredient and method of controlling weeds  
There are provided novel substituted phenyl (thiono)carbamates capable of effectively controlling broad-leaved annual weeds and annual weeds belonging to the families Gramineae and Cyperaceae such...
4400512 Azaspiro compounds  
This invention relates to a method of using compounds selected from those of the following formula : ##STR1## wherein R1 is hydrogen, alkyl or alkenyl; R2 is hydrogen, alkyl, cycloalkyl or...
4400199 Thiolcarbamate compounds and their use as herbicides  
Chloroalkylthiolcarbamate compounds of the formula: ##STR1## wherein Z represents ##STR2## and when Z is ##STR3## n is an integer of 4 to 10, whereas when Z is ##STR4## n is an integer of 3 to 10....
4343737 Process for production of thiolcarbamates and the thiolcarbamates obtained by said process  
A process for producing a thiolcarbamate compound of the following formula ##STR1## wherein R1 represents a hydrogen atom, an alkyl group having 1 to 5 carbon atoms, an alkoxy group having 1 to 5...
4341702 Herbicidal active sulfoxide and sulfone compounds  
Herbicidal active sulfoxide and sulfone compounds and their method of use as described herein. The compounds have the following generic formula: ##STR1## wherein n is 1 or 2; R is selected from the...
4299765 Herbicidal active sulfoxide compounds  
Herbicidal active sulfoxide and sulfone compounds and their method of use as described herein. The compounds have the following generic formula: ##STR1## wherein n is 1 or 2; R is selected from the...
4298524 Preparation of thion- and thiol-carbamic esters  
Thion-carbamic esters are obtained reacting in a single stage an alkaline xanthogenate, an amine and an oxidizer, according to the reaction: ##STR1## wherein: R, R1, R2 each are an alkyl,...
4298740 Process for the production of thiolcarbamate compounds  
In the process for the production of a thiolcarbamate compound of the formula ##STR1## wherein R1 and R2 are as defined in claim, comprising reacting a tertiary halogen compound of the formula...
4264503 Polymerization process using a sodium carboxylactamate catalyst  
The polymerization of 2-pyrrolidone is achieved in high yield in the presence of a sodium-derived catalyst activator produced by the reaction of carbon dioxide with the sodium lactamate derived...
4252804 Therapeutically useful 3,4,5-trimethoxybenzene derivatives  
Compounds of the formula I ##STR1## wherein m and n are 0, 1 or 2, X represents oxygen, imino, benzylimino, or morpholinoethylimino, Y represents CO, CONH, COO or SO2, and NR1 R2 represents a...
4248779 Process for producing thiolcarbamates  
A thiolcarbamate having the formula ##STR1## wherein R1 and R2 are the same or different and respectively represent an alkyl, alkoxy, alkenyl, cycloalkyl, hydroxyalkyl, phenyl or benzyl group and...
4234484 Process for the preparation of cyclic enamides  
Special cyclic enamides are prepared by splitting off alcohols catalytically from the corresponding alkoxylated cyclic amides, in the presence of at least one tetraalkylammonium and/or alkali metal...
4222938 Preparation of thiolcarbamates  
Thiolcarbamates are prepared from carbamoyl halides and xanthates.
4222765 Thiolcarbamic acid esters  
Thiolcarbamic acid esters having the formula ##STR1## wherein X represents hydrogen or chlorine atom and n represents an integer of 2 to 3 are disclosed.
4163088 Antistatic polyamide compositions with polyalkyleneglycol ether having secondary terminal urethane groups  
The invention relates to antistatic polyamide compositions comprising a polyamide and as an antistatic agent from 0.1 to 20%, preferably from 1.5 to 15%, by weight based on the total weight of the...
4150022 Process for the production of ammonium salts of dithiocarbamic acid  
This invention relates to a new process for the production of ammonium salts of dithiocarbamic acid; the process comprising reacting bis-alkyl aminomethanes with sulphur.
4147715 Thiocarbamate preparation utilizing quaternary ammonium salt catalysts  
Thiocarbamates are prepared by a process comprising reacting an aqueous solution of a thiocarbamate salt with an organic halide in the presence of a catalytic amount of a quaternary ammonium salt...
4118500 Fungicidal alkoxy mono- and dialkoxy N-substituted cyclic amines  
Novel alkoxy derivatives of N-substituted cyclic amines of the formula ##STR1## where R1 is hydrogen, an alkyl group having from 1 to 8 carbon atoms, an aryl group having from 6 to 10 carbon atoms,...
4113767 Process for the preparation of alkali metal salts of 3,3-dimethyl-2-oxo-butyric acid  
6-Tert.-butyl-3-mercapto-4-amino-1,2,4-triazin-5(4H)-one is prepared by reacting pinacolone with a sulfur chloride at 0° to 80° C, optionally reacting the mixture with an aqueous amine solution, h...
4110319 Thiocarbamate additives for sulfur vulcanizable polymers  
Thiocarbamates such as N,N-oxydiethylenecarbamyl 1-dodecyl disulfide are used to affect the vulcanization characteristics of sulfur vulcanizable polymers by increasing the state of vulcanization...
4086226 Process for the synthesis of thiolcarbamates  
A new and improved process for synthesizing thiolcarbamates, which are known herbicides, is disclosed. The thiolcarbamates are obtained in good yields, and without involving the use of highly...
4029646 Benzyl N,N-hexamethylenethiolcarbamate compounds and herbicidal compositions  
Certain thiolcarbamate compounds of the general formula ##STR1## wherein X is alkyl, e.g., lower alkyl, e.g., of from 1 to 4 carbon atoms, lower alkoxy of from, e.g., 1 to 3 carbon atoms, or...
4005071 P-Chlorobenzyl N,N-hexamethylenethiolcarbamate  
Certain novel thiolcarbamate compounds of the general formula ##STR1## wherein X is alkyl, e.g., lower alkyl, e.g., of from 1 to 4 carbon atoms, lower alkoxy of from, e.g., 1 to 3 carbon atoms, or...
4003907 Δ1 -1-Azacycloalkene-2-carboxylic acids and their production  
A compound of the formula ##STR1## or a salt thereof, OR OF THE FORMULA ##STR2## OR A SALT THEREOF, WHEREIN R1 and R2 are the same or different and each is hydrogen, lower alkyl, cycloalkyl of 4 to...
4001217 Azetidinyl carbothiolates  
New and valuable carbothiolates of azetidines having a good herbicidal action, herbicides containing these compounds, and a process for controlling the growth of unwanted plants with these compounds.
3989684 Method of making R-S (o) C NR1 R2 compounds  
Intermediate compounds useful for manufacturing herbicidal active sulfoxide and sulfone compounds are described herein. The compounds have the following generic formula: ##EQU1## wherein R is...
3984419 Perhydrofluorenetetrol and perhydro-phenanthrenetetrol derivatives  
Compounds are provided having the structure ##SPC1##Wherein n is 1 or 2, n1 is 0, 1 or 2 and n2 is 0, 1, 2 or 3, R1, R2, R3 and R4 may be the same or different and can be hydrogen, lower alkyl,...
3954729 Process for preparing a thiolcarbamate  
Thiolcarbamates are prepared by reacting a secondary amine having the formula ##EQU1## wherein R1 and R2 are the same or different and each represent hydrogen, lower alkyl, alkoxy, alkenyl,...
3953427 Process for the preparation of substituted S-alkyl thio-carbamates  
The invention relates to a new and advantageous process for the preparation of substituted S-alkyl thiocarbamates having the general formula (I), ##EQU1## wherein R1 stands for a C1-4 alkyl group,...
3947511 1-Hydrocarbyl-3-mono- and -dithiocarbamoylureas  
Novel 1-hydrocarbyl-3-(thiocarbamoylthio)ureas and 1-hydrocarbyl-3-(carbamoylthio)ureas are prepared by reacting, in liquid phase, an appropriate isocyanate and S-thiocarbamoylhydrosulfamine or...
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