Match Document Document Title
5639824 Separating agent containing a support and a cyclodextrin derivative  
Chemically bonded bodies comprising a support and a cyclic oligosaccharide derivative, at least one of the 2-, 3- and 6-position hydroxyl groups of which is chemically bonded to the support through...
5639734 Disaccharide inflammation inhibitors and uses thereof  
The present invention provides a composition of matter comprising a biosynthetic anti-inflammatory oligosaccharide, comprising the structure of: sugar - sugar - X - R; wherein said sugar is...
5639732 Phosphorous-containing cysteine and serine protease inhibitors  
The present invention is directed to novel phosphorous-containing inhibitors of cysteine or serine proteases. Methods for the use of the protease inhibitors are also described.
5637569 Ganglioside analogs  
Ganglioside lactam analogue derivatives of general formula (I) in which A is a sialic acid residue of formula (II) which is bound via the dashed line in the 2-position; and in which Z 1 is --OH or...
5637681 Aminosaccharide biguanides  
Novel aminosaccharide biguanides are prepared by either reacting a aminosaccharide with a mono- or multi-functional cyanoguanidine or by reacting a monocyano-guanidine of an aminosaccharide with a...
5635609 Particles prepared by transacylation reaction between an esterified polysaccharide and a polyamine, methods of preparation therefor and compositions containing same  
Particles, preparation methods therefor, and compositions containing same. The particles include at least one esterified polysaccharide and at least one polyamine, as well as at least one gellable...
5631374 Reagents for detection of primary amines  
The present invention is directed to derivatives of aroyl-2-quinoline-carboxaldehyde and their use in detection and quantification of minute amounts of primary amines.
5627273 Method for preparing hydrophobically-terminated polysaccharide polymers and detergent compositions comprising the polysaccharide polymers  
The present invention is directed to methods of preparing hydrophobically-terminated polysaccharide polymers. The methods utilized to prepare the hydrophobically-terminated polysaccharide polymers...
5624906 Oral hygiene compositions comprising heteroatom containing alkyl aldonamide compounds  
The present invention is related to new oral hygiene compositions that have improved foam, viscosity, clarity and good taste due to the inclusion of a new type of alkyl aldonamide compound,...
5623049 Nucleic acid-binding oligomers possessing N-branching for therapy and diagnostics  
The invention relates to nucleic acid-binding oligomers possessing N-branching of the general formula (I), ##STR1## and their monomers, where the individual radicals have the meaning given in the...
5622945 Rubyrin macrocycles  
The present invention is directed to the synthesis and use of novel macrocyclic compounds, based upon a new class of expanded porphyrins, termed rubyrins. Disclosed herein is the structure and...
5620902 Sialic acid glycosides, antigens, immunoadsorbents, and methods for their preparation  
The stereochemistry of sialylation of an acceptor saccharide to obtain an α (2-3) or α (2-6) linkage is controlled to favor the α anomer by use of an aromatic ester of the sialyl reagent. The...
5621088 Process for derivatizing polyglucosamines  
Processes for the preparation of polyglucosamine derivatives, e.g., hydroxypropyl chitosan and carboxymethyl chitosan, are disclosed. The polyglucosamine derivatives can be prepared in a covalently...
5616568 Functionalized derivatives of hyaluronic acid  
Hyaluronate functionalized with dihydrazide is provided and may be cross-linked. A method for producing hyaluronate functionalized with dihydrazide includes mixing hyaluronate and dihydrazide in...
5614616 Process for the production of polysaccharides  
Polysaccharides corresponding to formula (I) ##STR1## in which S is a recurrent monosaccharide unit and B is a group of formula (Ia) attached to the monosaccharide unit S by an O atom ##STR2##...
5604206 Complexes containing S(+) phenyl alkane acids and amino sugars  
New complexes of S(+)-ibuprofen and amino sugars are described. These complexes are particularly suitable for the treatment of inflammations and pains.
5601799 Partially delipidated D25 polysaccaride composition for imaging and diagnosis  
The present invention relates to a D 25 polysaccharide compound whose lipid has been partially removed and to its derivatives, wherein at least 85% by weight, preferably 90% of the compound, exists...
5599915 Sialyl Lewis X mimetics  
Sialyl Lewis x mimetic compounds are disclosed that are free of sialyl groups and glycosidically-linked fucosyl groups. These compounds exhibit about the same inhibition of selectin-medicated...
5599914 Glycosphingolipids with a group capable of coupling in the sphingoid portion, the preparation and use thereof  
The invention relates to the chemical modification of the sphingoid portions of glycosphingolipids. It has been possible by a series of reactions to introduce an amino group in the position of the...
5597811 Oxirane carboxylic acid derivatives of polyglucosamines  
Polyglucosamine derivatives, e.g., chitosan, substituted with oxirane carboxylic acids, e.g., epoxysuccinic acid, are disclosed. The polyglucosamine derivatives can be prepared in a covalently...
5597573 Lipid-A analogs: new monosaccharide and disaccharide intermediates for eliciting therapeutic antibodies and for antitumor and antiviral activities  
The present invention relates to novel amidine components of formula (II): ##STR1## A method for eliciting antibodies in an animal which bind to Lipid A or LPS comprising administering to the...
5593969 Lipid-A analogs: monosaccharide and dissaccharide compounds for inhibiting binding of lipid A receptors to lipid A receptors  
A compound of the formula: ##STR1## wherein: each of R 1 , R 1 ', R 2 and R 2 ' independent of each other is a substituted or unsubstituted, branched or linear C 1 -12 alkyl, alkene or alkyne...
5585473 Compounds and methods for monosaccharide analysis  
Compounds and methods are provided for use in monosaccharide analysis. The present invention discloses hydrazino monosaccharide derivatives. Methods for preparing and using hydrazino monosaccharide...
5580553 Cosmetic composition containing alkenylsuccinic acid ester of saccharide  
There is disclosed a cosmetic composition containing as an essential ingredient an alkenylsuccinic acid half ester of a saccharide which can be obtained by reacting the sugar with an...
5576426 Aldolase catalyzed stereoselective synthesis of arabinohexulose, xyloheptulose, threohexulose and xylohexulose  
The present invention relates to aldolase catalyzed stereo-selective synthesis of sugars and compositions of matter comprising arabinohexulose, xyloheptulose, threohexulose, and xylohexulose.
5567683 Substituted lactose and lactosamine derivatives as cell adhesion inhibitors  
Simple lactose or lactosamine related compounds which behave as ligands for the ELAM-1 and related receptors are described. These compounds are useful in the treatment of conditions characterized...
5563250 Cleavable conjugates for the delivery and release of agents in native form  
The present invention provides cleavable conjugates whose linkers contain a labile bond that is cleavable under a variety of mild conditions, including weakly acidic. Since the agent may be bonded...
5563252 Polymerizable saccharide monomers which contain a single, polymerizable, α-methyl styryl moiety  
Polymerizable, saccharide-derived monomers are prepared in processes which utilize water as the reaction solvent and which preferably do not utilize a cosolvent. The saccharide monomers are...
5552387 Polycyclic ether antibiotics  
An antibiotic of the formula ##STR1## wherein R is hydrogen or a pharmaceutically acceptable cation and Me is methyl.
5543506 Polysaccharide derivative and separating agent  
The present invention provides a novel polysaccharide derivative in which part or all of the hydroxyl groups or the amino groups contained in a polysaccharide are replaced by two or more kinds of...
5539090 Release and isolation of N-glycans and O-glycans  
N- and O-glycans are released from a glycoconjugate with a substantially anhydrous hydrazine reagent, the glycoconjugate being substantially salt-free and substantially anhydrous. Released N- and...
5529986 Conjugate, its preparation and use and a substrate prepared with the conjugate  
The present invention relates to a water-soluble conjugate having antithrombin-binding activity comprising a substantially straight-chained organic polymer backbone having at least 30 molecules of...
5527675 Method for degradation and sequencing of polymers which sequentially eliminate terminal residues  
A method and apparatus for sequentially degrading at least a portion of a polymer of backbone repeating units, the polymer having a terminal repeating unit comprised of a nucleophile and a backbone...
5525710 Highly porous chitosan bodies  
There is provided a crosslinked, highly porous chitosan body, wherein the porous body is characterized in that it has an open-celled 3-dimensional lattice structure, a density of less than about...
5523212 Aryl N-alkylacridanthiocarboxylate derivatives useful for chemiluminescent detection  
Aryl N-alkylacridanthiocarboxylate compounds which produce chemiluminescence. The compounds produce light with peroxide and peroxidase. The compounds are used as a substrate in assays for various...
5521294 2,2-difluoro-3-carbamoyl ribose sulfonate compounds and process for the preparation of beta nucleosides  
This invention provides novel 1-alkylsulfonyl-2,2-difluoro-3-carbamoyl ribose intermediates and intermediate nucleosides derived therefrom. The compounds are particularly useful in the preparation...
5514547 Molecular genetic identification using probes that recognize polymorphic loci  
Polynucleotide sequences and cloned DNA fragments useful for visualizing DNA polymorphism and other genetic analyses are disclosed herein. Specifically, polynucleotide probes and methods are...
5508268 Parenteral elsamitrucin formulations  
Stable parenteral antitumor formulations contain elsamitrucin salt, a stabilizer and a buffer. The formations are optionally stored in sealed containers under air or nitrogen headspace.
5498707 Hydrogen sulfide converter  
A composition adapted to convert hydrogen sulfide and organic sulfides to nontoxic polymers. The compositions comprise amine resin solutions made by reacting sterically hindered amines such as...
5498604 Lewis-type sugar chain derivative  
The object of the present invention is to provide a new SLe-type sugar chain derivative represented by the following formula (I), which is useful as a pharmaceutical and which contains moranoline:...
5496937 Polysaccharide substances, process for producing them and use of them  
A polysaccharide substance having the following formula is provided: ##STR1## Also provided is a method of producing the polysaccharide substance in which an oligosaccharide having a degree of...
5496930 Unsaturatd sugar compounds  
A process for highly regioselective esterification and ester cleavage on unsaturated sugar compounds with the aid of lipases and esterases, and products which can be prepared by this process....
5491072 N-alkylacridan carboxyl derivatives useful for chemiluminescent detection  
N-alkylacridan carboxylic acid derivative compounds (I) are used to generate chemiluminescence by the action of a peroxidase enzyme and an oxidant. The compounds I are useful in assays of all types.
5489578 Sulfated ligands for l-selectin and methods of treating inflammation  
Sulfated oligosaccharides which bind to L-selectin receptors and act as agonists are formulated into pharmaceutical formulations and administered by injection to treat inflammation. Compounds which...
5476671 Synthetic ceramides and their use in cosmetic compostions  
A novel pseudoceramide which has improved dispersibility in aqueous solutions and which can be produced by an economical manufacturing process. The process for producing new pseudoceramides and...
5472860 Method for preparing N-acetylneuraminic acid by N-acetylneuraminic acid lysase at a pH of 10-12  
A method for preparing N-acetylneuraminic acid characterized in reacting N-acetylglucosamine with pyruvic acid at an alkaline pH in the presence of N-acetylneuraminic acid lyase.
5472582 Analysis of carbohydrates using 2-aminoacridone  
The present invention provides for the use of the fluorescent label 2-aminoacridone for use in separating carbohydrate mixtures and analyzing the structure of carbohydrates. Carbohydrates for...
5472951 Stabilizer for phospholipid vesicles  
An oligosaccharide lipid is provided which has 2 to 20 saccharide units, and has a hydrophobic group linked by an ether linkage to an anomer carbon on a reducing end group. A stabilizer for a...
5473059 Modified hydrophobic cationic thickening compositions  
Water soluble quaternary ammonium ethers of polysaccharides or polyols wherein the quaternary ammonium ether substituents correspond to the formula ##STR1## wherein R 1 is a monohydroxylated or...
5470965 Complexable heterogenous oligosaccharides and alpha-hydosanes having therapeutical activity, process for their preparation and related pharmaceutical compositions  
Complexable heterogeneous oligosaccharides and pure alpha-hydosanes, namely not contaminated from other macromolecules (mucopolysaccharides, proteins, nucleic acids, etc.) of a defined molecular...