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3867389 ALPHA-(N-BENZOYLOXY AND PHENYLAMINO ALKYL-PIPERAZINO)-BETA-BENZOYL-PROPIONIC ACID DERIVATIVES  
The present invention relates to new pharmacologically valuable ketone derivatives exhibiting a distinct dilatory action on the cerebral vessels and which have the general formula ##SPC1## And...
3865842 Beta-[benzo(b) thienyl-3]-alpha-allyl-propionic acid esters  
β-[Benzo(b)thienyl-3] propionic acid derivatives in the form of their amino esters (and salts thereof) are prepared. These compounds have spasmolytic, vasodilatatric, antiserotonic and local...
3864344 3-(Benzoyl)-2-(4'-anilino carbonyl or benzoxy-alkyl piperazino)-propionitriles  
The present invention relates to new pharmacologically valuable ketone derivatives exhibiting a distinct dilatory action on the cerebral vessels and which have the general formula ##SPC1## And...
3862176 DERIVATIVES OF 5-CINNAMOYL BENZOFURAN  
Compounds of the formula ##SPC1## In which ##SPC2## Is dimethylamino, diethylamino, diisopropylamino, pyrrolidino, piperidino, morpholino or perhydroazepino; n is 2 or 3; and R3, r4 and R5, which...
3862162 CERTAIN-2-AMINO-1,4-DIHYDRO-4-PHENYL-6-LOWER ALKYL (OR PHENYL)-3-PYRIDINECARBOXYLATES  
2-Amino-1,4 dihydropyridines bearing an ester carbonyl function in the 3-position, being optionally substituted by lower alkyl in the 5-position, and being substituted in the 4- and 6-positions by...
3862177 NOVEL 1-(2'-BENZOYL ETH-1'-YL)-2-(4"-CINNAMYL PIPERAZIN-1"-YL METHYL) BENZIMIDAZOLES, THEIR PROCESS OF PREPARATION AND THEIR THERAPEUTIC APPLICATION  
Compounds of the formula ##SPC1## In which Ar is phenyl optionally substituted by a halogen atom, by one or two methyl groups or by 1-4 carbon alkoxy groups are provided as novel therapeutic...
3856798 BICYCLIC DERIVATIVES OF 1, 4- DIHYDROPYRIDINE  
1,4-Dihydropyridines bearing carbonyl functions in the 3- and 5-positions, being optionally substituted by lower alkyl in the 6-position, being substituted in the 4-position by lower alkyl,...
3853875 ESTERS OF 2-ALKYL THIAZOLE 5-CARBOXYLIC ACID  
New esters of 2-alkyl thiazole 5-carboxylic acid of formula I: ##SPC1## wherein n represents the whole numbers 0, 1, 2, 3, 4 or 5, n' represents the whole numbers 1, 2, 3, 4 or 5, m represents the...
3852284 NOVEL SUBSTITUTED OXAZINO(5,6,E)INDOLES  
Compounds of the formula Wherein R is alkyl having 2 or 3 carbon atoms, alkyl having 2 or 3 carbon atoms substituted by one or more hydroxyl and dialkylamino wherein the latter alkyl has 1 to 4...
3852312 PREPARATION OF MANNICH BASES  
Steroidal Mannich bases are prepared by reaction of a steroid bearing an ethynyl and a hydroxy function at any of positions 3 and 17 (or 17a) with an N,N-dialkyl substituted-amino-methanol in the...
3846470 DERIVATIVES OF 3-BENZOYL-2-(β-HYDROXYPHENETHYLAMINO)-PROPIONITRILE  
The present invention relates to new pharmacologically valuable ketone derivatives exhibiting a distinct dilatory action on the cerebral vessels and which have the general formula ##SPC1## And...
3843725 4[2-(α-METHYL-PHENETHYLAMINO)-ETHOXY]-BENZENES  
This invention relates to phenoxyalkylamines having the formula: ##SPC1## In which R1 is hydrogen, halogen, an alkyl or an alkoxy group, A is an alkyl, alkylaryl, cycloalkyl, alkenyl, cycloalkenyl...
3835141 QUINALYTHIOHYDROXIMIC ACIDS AND THEIR DERIVATIVES  
Thiohydroximic acid compounds of the formula: ##SPC1## Wherein Het is pyridyl, pyrazinyl, quinolyl, isoquinolyl, or these radicals substituted by halogen, lower alkyl or lower alkoxy, and R is...
3818015 1(POLYMETHOXYBENZYL) 6 HYDROXYL 1,2,3,4 TETRAHYDRO ISOQUINOLINES  
A tetrahydroisoquinoline compound of the formula: ##SPC1## Wherein R is a trimethoxyphenyl, dimethoxyphenyl or methylene-dioxyphenyl radical, and pharmaceutically acceptable acid addition salts...
3817981 N-(6)-ARALKYL-ADENOSINE COMPOUNDS  
Novel N(6)-Aralkyl-Adenosine Compounds of the formula ##SPC1## Wherein R1 is hydrogen, halogen or hydroxyl; R2 is hydrogen, halogen, hydroxyl, alkyl or alkoxy; R3 is hydroxyl, amino, alkoxy,...
3789120 SULFAMOYL AZIDE PROCESS AND COMPOSITION FOR LOWERING BLOOD PRESSURE  
This invention is concerned with a pharmaceutical process and pharmaceutical compositions for lowering blood pressure in mammals by the administration thereto sulfamoyl azides of the Formula R1 R2...
3759974 SUBSTITUTED 4-CYANO-4-PHENYL-AMINOCYCLOHEXANES  
Basically substituted 4-cyano-4-phenyl-aminocyclo-hexanes of the general formula ##SPC1## Wherein A, B, C, A', B', C' are each hydrogen, halogen, trifluoromethyl, lower alkyl or lower alkoxy; R is...
3725469 PROSTANOIC ACID DERIVATIVES  
This invention is a group of compounds of the formula: ##SPC1## Wherein R1 is hydrogen or a pharmacologically acceptable cation, essentially free of pyrogens, antigens, proteins, enzymes, cellular...
3714171 1-(2-CYCLOHEXYLETHYL) -6 OR 7 METHOXY-1,2,3,4-TETRAHYDROISOQUINOLINE AND ACID ADDITION SALTS THEREOF  
A 6- or a 7-methoxyisoquinoline compound having the formula ##SPC1## Wherein n is 1-3 and its pharmaceutically acceptable acid addition salts are cutaneous vasodilators. Compound (I) is produced...
3696112 SULPHUR-CONTAINING 1,4-DIHYDROPYRIDINE DERIVATIVES  
Sulphur-containing 1,4-dihydropyridine derivatives of the formula: ##SPC1## Wherein R is hydrogen, saturated or unsaturated, straight, branched or cyclic alkyl of one to six carbon atoms,...
3687965 NOVEL 5-(N-SUBSTITUTED AMINOMETHYL)-2-OXAZOLIDINONES AND THEIR PROCESS OF PREPARATION  
5-AMINOMETHYL-2-OXAZOLIDINONES OF THE GENERAL FORMULA: ##SPC1## In which: represents either a dialkylamino radical in which the alkyl portions have one to five carbon atoms, or a heterocyclic...
3681480 ADAMANTYL AND ADAMANTYLALKYL 2-AMINOETHYL PHOSPHATES, PHOSPHONATES AND PHOSPHINATES  
The compounds are adamantyl and adamantylalkyl 2-aminoethyl phosphates, phosphonates and phosphinates having renin inhibitory activity.
3676492 AMINO ACID AMIDES OF DISUBSTITUTED PHENETHYLAMINES  
Amino acid amides of disubstituted phenethylamines represented by the formula: ##SPC1## Wherein R is hydrogen, lower alkyl, hydroxymethyl, hydroxybenzyl, β-hydroxyethyl, mercaptomethyl,...
3673187 BIS-(DIHYDROXYPHENYL-ETHYLOL)-SUBSTITUTED ALKYLENEDIAMINES AND THE SALTS THEREOF  
Compounds of the formula wherein R1 is hydrogen or methyl, R2 is methyl, methoxy, ethoxy or chlorine and, if R1 is methyl, additionally hydrogen, and m is a whole number from 0 to 10, inclusive,...
3666762 2'β-ISOPROPYL-5'α-n-PROPYL-9,10-DIHYDRO-ERGOPEPTINES  
The invention concerns novel compounds of the formula: ##SPC1## Wherein R1 is hydrogen or methyl, and acid addition salts thereof. Processes and an intermediate employed for the production of the...
3624084 2,4,6-TRISUBSTITUTED DERIVATIVES OF PYRIMIDINE  
New 2,4,6-trisubstituted pyrimidine derivatives of the general formula ##SPC1## In which R1 is hydrogen, lower alkyl, aralkyl, R2 is hydrogen, halogen, lower alkyl, hydroxyalkylamino,...
3622587 CERTAIN 3-PYRIDYLMETHYL-2-(P-CHLORO PHENOXY)-2-METHYL PROPIONATE-N-OXIDES AND DERIVATIVES THEREOF  
Compounds represented by the formula: ##SPC1## Wherein A is a bivalent radical selected from the group consisting of --COOCH2 -- and --CH2 OOC--, and therapeutically acceptable salts thereof.
3544557 BENZHYDRYL ETHERS  
3542793 4-UNSUBSTITUTED-5-AMINO- OR 5-ACYLAMINO-PYRAZOLO(3,4-B)PYRIDINES  
3542870 1 - (3,5 - DIHALO - 4 - HYDROXY - PHENYL) - 2 - (2-ARYLOXY OR 2 - ARYLALKYL - ISOPROPYLAMINO)-PROPANOLS  
3541103 2-(4-BENZYLPIPERIDINO)ETHYLGUANIDINES  
3541097 PROCESS FOR THE PRODUCTION OF COUMARIN DERIVATIVES  
3535315 AMINOALKYL DERIVATIVES OF 6,11-DIHYDRODIBENZO-(B,E)-OXEPINE AND -THIEPINE  
3534041 POLYCYCLIC PIPERAZINES  
3532685 N,N' - ALKYLENE-N,N'-BIS((ALKOXY BENZOYLOXY)ALKYL)ALKYLENE DIIMINES  
3531488 DISULPHONAMIDES  
3530140 CERTAIN PYRIDYL-HYDRAZINO-2-YL-IMIDAZOLINES  
3523120 PIPERONYL-PIPERAZINE COMPOUNDS  
3520893 3-(GAMMA-AMINO-BETA-HYDROXYPROPYL)-4-METHYL-7-ALKOXYCARBONYLALKOXY COUMARINS  
3518268 SUBSTITUTED 5-CARBONYL- OR 5-THIOCARBONYL-DIBENZO(B,F)AZEPINES  
3515721 3-TERTIARY-AMINOETHYL-4-METHYL OR PHENYL-7-ETHOXYCARBONYLMETHOXY - HALO OR MONONITRO COUMARINS AND CONGENERS  
3514459 7-HYDROXY-3-AMINOALKYL-2-OXO-1,2-DIHYDROQUINOLINE ESTERS AND ETHERS  
3511839 SUBSTITUTED BENZOIC ACID ESTERS OF CERTAIN DIBENZ(B,F)AZEPINE DERIVATIVES  
3509194 1,3-DISILYL-1,3,2-DIAZASILACYCLOALKANES AND PROCESS OF PREPARING  
3509164 DERIVATIVES OF 1-(P-HYDROXYPHENYL)-2-(4-BENZYL-1-PIPERIDINO)-(ALKANOLS)  
3505334 PIPERAZINO-PHENYLETHANOL DERIVATIVES  
3493573 DIMETHYL XANTHINE DERIVATIVES AND PRODUCTION THEREOF  
3803236 PARA-AMINOPROPYL-2-HYDROXY-ETHERS OF PHENYLAMINOTROPONES AND THE SALTS THEREOF  
3790569 2-PROPANOL DERIVATIVES  
3804904 SUBSTITUTED PHENYL SULPHOXIDES AND SULPHONES AND THE USE THEREOF AS VASODILATORS