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5164381 |
Pharmacologically active 1,5-diaryl-3-substituted pyrazoles and method for synthesizing the same
1,5-Diaryl-3-substituted pyrazoles, a method of their preparation, compositions containing the same and methods of their use are disclosed. The pyrazoles are useful in alleviating inflammatory and...
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5157025 |
Method for lowering serum cholesterol employing a phosphorus containing ACE inhibitor alone or in combination with a cholesterol lowering drug
A method is provided for lowering serum cholesterol and thereby inhibiting fatty streak lesions of atherosclerosis by administering to a patient a phosphorus-containing ACE inhibitor, such as...
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5155100 |
Phosphono/biaryl substituted dipeptide derivatives
The invention relates to the N-phosphonomethyl-biaryl substituted dipeptide derivatives of formula I ##STR1## wherein A represents a direct bond, lower alkylene, phenylene or cyclohexylene; m...
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5153179 |
Medicament with improved penetration of the tissue membrane
A composition useful as a medicament with improved penetration of cell membranes comprising an active material and a compound of general formula: ##STR1## wherein either residue R 1 or R 2 is an...
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5147865 |
Phosphonopyrrolidine- and piperidine-containing pseudopeptides of the statin type, a process for their preparation and their use as medicaments against retroviruses
The invention relates to new phosphonopyrrolidine- and piperidine-containing pseudopeptides, to a process for their preparation and to their use as medicaments, in particular as antiviral agents in...
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5128330 |
Oxazinone substituted phosphines
A new class of phosphines in which the phosphorous atom is bonded directly to the carbon of an oxazinone: ##STR1## In addition to their anti-inflammatory activity, these phosphines are useful as...
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5002937 |
Diphosphonic acid compounds and use for calcium metabolism disorders
The present invention provides compounds of the formula: ##STR1## The present invention also provides processes for the preparation of these compounds and pharmaceutical compositions containing...
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4997822 |
Heterocyclic compounds having a 2-(2-(N,N-bis(2-chloroethyl)-diamidophosphoryloxy) ethyl) radical
There are disclosed compounds of the formula ##STR1## The compounds have antitumour and AIDS treatment activity.
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4971957 |
Carboxamide compounds, processes for preparing the same and a pharmaceutical composition containing the same
Novel carboxamide compounds represented by the general formula (I) possess excellent activities for lowering lipids and thus they are useful as agents for treating and preventing various diseases...
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4940706 |
2,4-disubstituted 1,3-dioxolanes and pharmaceutical use
The present invention describes novel 2,4-disubstituted 1,3-dioxolanes having the formula I ##STR1## wherein R 1 represents a long chain alkyl group; X is a covalent single bond, a carbonyl group,...
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4937237 |
Phosphinic acid substituted aromatic steroids as inhibitors of steroid 5-60 -reductase
Invented are phosphinic acid substituted analogues of steroidal synthetic compounds, pharamaceutical compositions containing these compounds, and methods of using these compounds to inhibit steroid...
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4908356 |
Aldophosphamide derivatives useful as antitumor agents
A compound of the formula ##STR1## wherein R 1 and R 2 may be the same of different and are each independently hydrogen or lower alkyl which may be unsubstituted or monosubstituted with halogen,...
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4891362 |
Substituted amidophosphonates and amidophosphates
Novel substituted N-alkyl-N-alkoxyamidophosphonates or -thiophosphonates and N-alkyl-N-alkoxyamidophosphates or -thiophosphates of formula ##STR1## wherein R is C 1 -C 4 alkyl or C 1 -C 4 ...
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4882319 |
Phosphonic acid substituted aromatic steroids as inhibitors of steroid 5-α-reductase
Invented are phosphonic acid substituted analogues of steroidal synthetic compounds, pharmaceutical compositions containing these compounds, and methods of using these compounds to inhibit steroid...
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4870065 |
N-alkyl or N-alkylene substituted glycin amides as insecticides or fungicides
The present invention relates to novel compounds of the formula (I) ##STR1## wherein R 1 and R 2 are the same or different and stand for alkyl having 1 to 4 carbon atoms optionally substituted by...
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4849414 |
Substituted aminoalkanoylaminoalkyl phosphonate angiotensin converting enzyme inhibitors
Compounds of the formula ##STR1## wherein X is various amino or imino acids and esters are disclosed. These compounds are useful as anti-hypertensive agents due to their angiotensin converting...
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4804654 |
Certain N-(R-sulfonyl) phosphonamidothioates and dithioates
Compounds of the formula ##STR1## wherein the symbols have assigned meanings, and their use as insecticides and/or miticides.
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4681874 |
Thiazinephosphonic acid derivatives
Novel thiazinephosphonic acid derivatives (I): ##STR1## wherein R 1 and R 2 each is lower alkoxy, lower alkynyloxy, lower alkylthio, arylthio (e.g., monocyclic aromatic group), or lower...
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4656163 |
Compositions and methods of combating pests employing sulphenic acid amides in combination with known nematicides or insecticides
The present invention relates to the use of the sulphenic acid amides of the general formula (I) ##STR1## in which X represents identical or different halogen atoms, Y 1 and Y 2 are identical...
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4650791 |
Certain 3-alkoxy-2-cyclic-imido-propyl-phosphate-ethyl-cyclic ammonium hydroxide inner salts which inhibit activities of platelet activating factor
A novel phospholipid of the formula: ##STR1## wherein R 1 is an alkyl group of 10 to 24 carbon atoms, R 2 is a cyclic imide group and A + is a cyclic ammonio group and a salt thereof have...
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4624695 |
O-diaminophosphinyl derivatives of oximes as urease inhibitors
The invention relates to novel urease inhibited fertilizer compositions containing urea and a urease inhibiting amount of one or more o-diaminophosphinyl derivatives of oximes, and methods and...
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4617295 |
Pesticidal oxime N-alkyl-N-α-(alkylthio-phosphorothio)acyl carbamates
Oxime N-alkyl-N-α-(alkylthio-phosphorothio)acyl carbamates represented the structure: ##STR1## wherein the R represents various imino radicals, Q is oxygen or sulfur and the numbered R groups...
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4608367 |
γ-Pyrone phosphoric ester derivatives and insecticidal and miticidal compositions thereof
γ-Pyrone phosphoric ester derivative represented by the general formula below is useful as an effective component of an insecticidal or miticidal composition for agricultural and horticultural...
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4605647 |
Oxaazaphosphorine compounds and pharmaceutical compositions
New oxaazaphosphorine compounds corresponding to the formula: ##STR1## in which R is alkyl, cycloalkyl or alkoxy, phenyl, phenylalkyl, phenoxy or thiophenoxy in which the phenyl ring may be...
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4576933 |
Method of use of 1-(alkyl for alkylcarbanoyl)-2-carbamoylglycerol derivatives
Glycerol derivatives, inclusive of salts thereof, of the formula ##STR1## wherein R 1 is alkyl or alkylcarbamoyl containing 10 to 30 carbon atoms, R 2 and R 3 are independently hydrogen, C 1 -6...
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4562185 |
Five-membered nitrogen-containing hetero-cyclic compounds and their use as pest-combating agents
The present invention relates to combating pests with five-membered nitrogen-containing heterocyclic compounds of the formula (I) ##STR1## in which R 1 , R 2 , R 3 , X and Y have the meaning given...
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4494977 |
Quaternary ammonium salts of α-1,4-thiazine alkanephosphonic acids
This invention relates to quaternary ammonium salts of α-1,4-thiazine alkanephosphonic acids; and to the preparation and uses thereof.
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4368196 |
Phosphoric acid esters, and their use for combating pests
Novel phosphoric acid esters of the formula ##STR1## where R 1 is alkoxy of a maximum of 4 carbon atoms or phenyl, R 2 is alkyl of a maximum of 3 carbon atoms, alkoxy or alkylthio of a maximum of...
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4342584 |
Microbiocidal process using di-quaternary ammonium salts of α-1,4-thiazine alkanephosphonic acids
This invention relates to novel di-quaternary ammonium salts of α-1,4-thiazine alkanephosphonic acids; the preparation thereof; and uses thereof.
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4339443 |
Compounds and compositions
There are described pesticidal compositions comprising one or more compounds of the formula I, ##STR1## in which Ra is a group R 2 or --OR 2 , E is oxygen or sulphur, Rm is --O .crclbar . M...
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4339444 |
Novel oxime-phosphate compounds
Novel acyclic and heterocyclic oxime phosphate compounds have been found to exhibit insecticidal, miticidal and nematocidal activity.
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4322413 |
1,2,3,5-Thiatriazolidin-4(2H)-one-1,1-dioxide phosphoric acid derivatives and their use for combating pests
Heterocyclic phosphoric acid derivatives of the formula ##STR1## where R, R 1 , R 2 , R 3 , X and Y have the meanings given in the disclosure. The compounds are suitable for combating pests from...
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4316896 |
Aminoacid derivatives as antihypertensives
The invention relates to new phosphoryl aminoacid derivatives and related compounds which are useful as antihypertensives.
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4302451 |
Pesticidal phosphorus sulfenamides
[(N,N-diarylamino)thio]phosphoramide compounds such as N-[N-[2-chloro-5-(trifluoromethyl)phenyl]-N-[2,4-dinitro-6-(
trifluoromethy l)phenyl]amino thio]-N-(1-methylethyl)phosphoramidic acid, diethyl...
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4288451 |
Combating arthropods with ferrocene-containing synergistic compositions
An arthropodicidal composition containing, as active ingredients, an arthropodicidally effective amount of (1) at least one ferrocene derivative of the formula ##STR1## in which R and R 1 each...
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4247546 |
Phosphonylureidobenzene derivatives and their medicinal use
The invention includes phosphonylureidobenzene compounds of the general formula ##STR1## or pharmaceutically acceptable salts in which R 1 and R 2 are identical or different and represent an...
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4159324 |
Combating insects, acarids and nematodes with O-(1-fluoro-2-halo-ethyl)(thiono)phosphoric(phosphonic) acid ester-amides
O-(1-Fluoro-2-halo-ethyl)(thiono)phosphoric(phosphonic) acid ester-amides of the formula ##STR1## in which R and R 1 independently represent hydrogen, alkyl, haloalkyl or cyanoalkyl, or R and R...
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4155996 |
3-(Phosphoryloxy) and (phosphonyloxy)-thiophenes
Novel 3-(phosphoryloxy) or (phosphonyloxy)-thiophenes of the formula ##STR1## wherein R is alkyl of 1 to 4 carbon atoms, R 1 is selected from the group consisting of alkyl of 1 to 4 carbon atoms,...
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4140774 |
Method of combating nematodes using S-(amidocarbonyl)-methyl-O-alkyl-mono(di)thiophosphoric acid ester amides
Compounds of the formula ##STR1## in which R represents halogen, C 1 -C 6 -alkyl, C 1 -C 3 -haloalkyl, C 1 -C 2 alkoxy, NO 2 or S-CH 3 , R 1 represents hydrogen or C 1 -C 6 -alkyl, R 2 ...
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4018917 |
Isourea acetylphosphate insecticides
Compounds are described herein which are useful as insecticides, and which are defined by the following formula ##STR1## wherein R is lower alkoxy, R 1 is lower alkyl or lower alkoxy, R 2 is...
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3996353 |
Phosphonated N,N-disubstituted fatty morpholines as bacterial and fungicidal agents
Phosphonated N,N-disubstituted fatty acid morpholine derivatives were prepared by the free radical addition of dialkyl phosphites to terminal and nonterminal double bonds of N,N-disubstituted fatty...
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3979512 |
S-(amidocarbonyl)-methyl-O-alkyl-monothiophosphoric acid ester amides
S-(amidocarbonyl)-methyl-O-alkyl monothiophosphoric acid ester amides of the formula ##EQU1## in which R and R' each independently is alkyl of 1 to 6 carbon atoms, R" is alkyl or alkenyl of 1 to...
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3966921 |
Certain pesticidal phosphorus containing amidines
Compounds of the formula ##EQU1## wherein R 1 represents phenyl, or phenyl mono- to trisubstituted by halogen, mono- or disubstituted by C 1 -C 4 -alkyl, C 1 -C 4 -alkylthio, nitro, cyano or...
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3880998 |
Pesticidal utility of certain phosphorus-containing imino perhydrooxazines
Method for controlling pests employing compounds corresponding to the formula ##SPC1## Wherein X is oxygen or sulfur, R 1 is lower alkoxy; R 2 is lower alkoxy or lower alkylthio; R 3 is lower...
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3794730 |
CONTROL OF INSECTS WITH CERTAIN PHOSPHORUS-CONTAINING THIOMORPHOLINONES
Organophosphorus compounds containing the thiomorpholinone moiety have been found to be highly active both as contact and systemic insecticides and miticides. These compounds also possess excellent...
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3679796 |
METHODS OF CONTROLLING RODENTS AND LEPORINE ANIMALS
Methods of selectively combating and controlling rodents and leporine animals using certain phosphorus acid esters, i.e. phosphoric, phosphonic, thionophosphoric and thionophosphonic acid esters,...
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3466369 |
SATURATED HYDROCARBON IMIDAZOLYL PHOSPHORUS COMPOUNDS AS FUNGICIDES
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3356568 |
Method for control of arthropods
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3323990 |
Fungicidal methods and compositions
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3269894 |
Synergistic organo-phosphate insecticides
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