Matches 151 - 200 out of 222 < 1 2 3 4 5 >
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4443456 Pyridyl alkylene amidinoureas  
This invention relates to a novel class of amidinourea and amidinothiourea compounds wherein the urea nitrogen atom is substituted by a heterocyclic alkylene group, and their use in pharmaceutical...
4351833 9-Amino-1-hydroxyoctahydrobenzo[c]quinolines and derivatives thereof as analgesics and anti-emetics  
9-Amino-1-hydroxyoctahydrobenzo[c]quinoline derivatives of formula ##STR1## and pharmaceutically acceptable acid addition salts thereof wherein R is hydrogen, COR 7 or SO 2 R 8 where R 7 is...
4347244 Ganglioside containing compositions for treating diarrhea  
The invention is concerned with a medium onto which is fixed a ganglioside or ganglioside derivative having an affinity for the toxins produced by the bacteria responsible for diarrheas and in...
4344952 Method of treating diarrhoea with gamma-piperidino-butyrophenones  
A method of treating diarrhoea and promoting weight gain in mammals by administration of an effective amount of a compound selected from the group consisting of...
4332814 Treatment of diarrhoea  
Vasoconstrictor α-adrenergic agonists of formula (I) A--B--C (I) wherein, A is a 2-imidazoline group or a guanidine group; B is a chemical bond...
4331602 Pharmacologically active 4-[2-hydroxy-4-(substituted]phenyl)naphthalen-2(1H)-ones and 2-ols, derivatives thereof and intermediates therefor  
Compounds having the formula ##STR1## wherein ##STR2## R 1 is hydrogen, benzyl or alkanoyl, X is C 2 -4 alkylene; and Z-W is alkyl, phenylalkyl or pyridylalkyl which can have an oxygen atom as...
4326074 Amidinoureas  
A new class of chemical compounds and their process of preparation is described. These compounds have valuable properties as anti-diarrheal agents.
4309545 Oximino-1-hydroxyoctahydrobenzo[c]quinolines and derivatives thereof  
9-Amino-1-hydroxyoctahydrobenzo[c]quinoline derivatives of formula ##STR1## and pharmaceutically acceptable acid addition salts thereof wherein R is hydrogen, COR 7 or SO 2 R 8 where R 7 is...
4285867 Pharmacologically active 4-[2-hydroxy-4-(substituted)phenyl]naphthalen-2(1H)-ones and 2-ols, derivatives thereof and intermediates therefor  
Compounds having the formula ##STR1## wherein ##STR2## R 1 is hydrogen, benzyl or alkanoyl, X is C 2 -4 alkylene; and Z-W is alkyl, phenylalkyl or pyridylalkyl which can have an oxygen atom as...
4277605 Chemical compounds  
3-Hydroxy-7-oxomorphinans and 3-hydroxy-7-oxoisomorphinans, optionally substituted on the 17-nitrogen atom, are potent, orally active antidiarrheal agents.
4261981 Medical compound produced from ragweed  
A composition made from ragweed for the treatment of diarrhea, intestinal disorders, ulcers, and hemorrhoids is disclosed. A composition which effectively reduces swelling and pain in the...
4242340 Method for the treatment of diarrheal disease conditions and symptoms in mammals  
A new class of chemical compounds and their process of preparation is described. These compounds have valuable properties as anti-secretory, anti-spasmodic, anti-ulcerogenic and anti-diarrheal agents.
4242339 Method for treatment of gastrointestinal spasmodic disease conditions or symptoms in mammals  
A new class of chemical compounds and their process of preparation is described. These compounds have valuable properties as anti-secretory, anti-spasmodic, anti-ulcerogenic and anti-diarrheal agents.
4242338 Method for treatment of gastrointestinal secretory and ulcerogenic disease conditions or symptoms in mammals  
A new class of chemical compounds and their process of preparation is described. These compounds have valuable properties as anti-secretory, anti-spasmodic, anti-ulcerogenic and anti-diarrheal agents.
4242337 Method for treatment of diarrheal disease conditions or symptons in mammals  
A new class of chemical compounds and their process of preparation is described. These compounds have valuable properties as anti-secretory, anti-spasmodic, anti-ulcerogenic and anti-diarrheal agents.
4218450 Method for treatment of gastrointestinal spasmodic disease conditions or symptoms in mammals  
A new class of chemical compounds and their process of preparation is described. These compounds have valuable properties as anti-secretory, anti-spasmodic, anti-ulcerogenic and anti-diarrheal agents.
4208427 Preventing enteropooling induced diarrhea by prostacyclin or 11-oxo-prostaglandin administration  
The present invention relates to a method for the prophylaxis and treatment of the diarrheogenic effects of enteropooling inducers by administration of an anti-enteropooling dose of an...
4203985 Antidiarrheal triazinones  
New compositions containing as the principle active ingredient a 1,4-disubstituted-1,2-dihydro-1,3,5-triazin-2-one are used for remedial or prophylactic treatment of diarrhea and organic...
4203920 Amidinoureas  
A new class of chemical compounds and their process of preparation is described. These compounds have valuable properties as anti-diarrheal agents.
4198409 Triazinones for veterinary use  
New compositions containing as the principle active ingredient a 1,4-disubstituted-1,2-dihydro-1,3,5-triazin-2-one are used for remedial or prophylactic treatment of diarrhea and organic...
4194045 1-(3,3-Diaryl-3-oxadiazolalkyl)-4-phenyl-4-piperidinomethanols and related compounds  
This invention encompasses novel 1-(3,3-diaryl-3-oxadiazolalkyl)-4-phenyl-4-piperidinomethano ls and related compounds. These compounds are useful anti-diarrheal agents which possess little or no...
4192886 Methods for treating gastrointestinal disease  
There is described a method for the prophylactic or curative treatment of a disease condition of the gastrointestinal tract, which condition has an allergic basis, in cattle or pigs, which...
4181728 Spiro-polycyclicimidazolidinedione derivatives  
Novel spiro-polycyclicimidazolidinedione derivatives useful as aldose reductase inhibitors and as therapeutic agents for the treatment of chronic diabetic complications are disclosed. The...
4164568 Oral scour formulations with citrate  
A veterinary composition comprising 40 to 80% of an actively absorbed monosaccharide, 7.5 to 30% of an actively absorbed naturally occurring amino acid, and 0.5 to 10% of an agent which is citric...
4125531 2-Substituted-1-azabicyclo[2.2.2]octanes  
This invention encompasses novel 2-(2,2-diphenyl-4-pentenyl-1-azabicyclo[2.2.2]octane and related compounds. These compounds are useful anti-diarrheal agents which possess little if any analgesic...
4120952 Method for the treatment of diarrhea in monogastric animals  
Monogastric animals such as pigs, humans and equines are given an oral dosage of pregelatinized starch in paste form or in a liquid mixture upon the occurrance of diarrhea.
4116963 3,3,3-Triarylalkyl-4-phenylalkyl-4-hydroxy piperidines and related compounds  
The present invention encompasses compounds of the formula ##STR1## AND THE PHARMACEUTICALLY ACCEPTABLE ACID ADDITION SALTS THEREOF WHEREIN R represents hydrogen, alkanoyl having 1 to 7 carbon...
4115564 Treatment of diarrhea with amidinoureas  
A new class of chemical compounds and their process of preparation is described. These compounds have valuable properties as anti-diarrheal agents.
4072686 1-(3,3,3-Triarylalkyl)-4-phenyl-piperidinealkanols  
The present invention encompasses compounds of the formula ##STR1## and pharmaceutically acceptable acid addition salts thereof wherein the Alk is straight or branched chain alkylene containing 2-4...
4066654 1-Triarylalkyl-4-phenyl-4-piperidine carboxylic acids and derivatives  
The present invention encompasses compounds of the formula ##STR1## wherein the Alk is straight or branched chain alkylene containing 2-4 carbon atoms; Ar and Ar' are phenyl, Alkyl substituted...
4057549 Triarylpropyl-azabicyclooctanes  
The present invention comprehends a method for treating diarrhea comprising administering to an animal in need of anti-diarrheal treatment an effective antidiarrheal amount of a compound of the...
4053477 5-(1,1-Diphenyl-3-(4-phenylpiperidino)propyl)-2-methyl-1,3,4-oxadiazole and related compounds  
This invention encompasses novel 5-[1,1-diphenyl-3-(4-phenylpiperidino)propyl]-2-methyl-1,3,4 -oxadiazoles and structurally related compounds. These compounds are useful anti-diarrheal agents which...
4045442 1-(Substituted amino)alkanoyl-2-(dibenzoxazepine-10-carbonyl)hydrazines and derivatives thereof  
The reaction of 1-(halo/cyano/sulfonyloxy)alkanoyl-2-(dibenzoxazepine-10-car bonyl)hydrazin es with an amine affords the corresponding 1-(substituted...
4029815 Anti-diarrheal anthranilic acids  
This invention relates to compositions of matter useful as anti-diarrheal agents and to the method of controlling and treating diarrhea in warm blooded animals. The active anti-diarrheal agents are...
4028364 2-Azabicyclo[2.2.2.]octan-2-yl-diphenyl-alkanones and related compounds  
This invention encompasses novel 2-azabicyclo[2.2.2]-octan-2-yl-diphenyl-alkanones and related compounds. These compounds are useful as anti-diarrheal agents.
4025524 2-{3-[4-Azatricyclo(4.3.1.1.sup.3,8) undecan-4-yl]-1,1-diphenylpropyl}-5-methyl-1,3,4-oxadiazole and congeners  
Preparation and the valuable antispasmodic, antiarrhythmic, antidiarrheal, and antiviral properties of 2-{3-[4-azatricyclo(4.3.1.1 3 ,8)undecan-4-yl]-1,1-diphenylpropyl}-5-me thyl-1,3,4-oxadiazole...
4024279 Treatment of dysmenorrhea and migraine symptoms  
A pharmaceutical composition for the treatment of, or for the alleviation of primary dysmenorrhea, for the treatment of acute migraine and for attaining the relaxation of smooth muscle, and a...
4022778 10-Aryl-1,2,3,4-tetrahydropyrazino(1,2-α)indole and derivatives thereof  
Novel 10-aryl-1,2,3,4-tetrahydropyrazino(1,2-α)indole and derivatives and intermediates for their preparation are described, the products having anticonvulsant and central nervous system...
4017491 1,1-Diaryl-1H-tetrazole amines  
The present invention relates to compounds of the following formula ##STR1## wherein Y is straight or branched chain alkylene containing 1-4 carbon atoms; X is hydrogen, halo such as fluoro,...
4013668 5-(1,1-Diphenyl-3-(5- or 6-hydroxy-2-azabicyclo(2.2.2)oct-2-yl)propyl)-2-alkyl-1,3,4-oxadiazoles and related compounds  
This invention encompasses novel 5-[1,1-diphenyl-3-(5-or 6-hydroxy-2-azabicyclo[2.2.2]oct-2-yl)propyl]-2-alkyl-1,3,4- oxadiazoles and their lower O-alkanoyl derivatives. These compounds are useful...
4013667 2,2-Diaryl-3-(1-azabicyclo[2.2.2]oct-2-yl)propionamides and intermediates thereto  
This invention encompasses novel 2,2-diaryl-3-(1-azabicyclo[2.2.2]oct-2-yl)propionamides and intermediates thereto. These compounds are useful anti-diarrheal agents which possess little or no...
4012393 2-[5-(CYCLIC AMINO) ETHYL-10,11-DIHYDRO-5H-dibenzo[a,d]-cyclohepten-5- yl]- 5  
This invention encompasses novel 2-[5-(cyclic amino)ethyl-10,11-dihydro-5H-dibenzo[a,d] cyclohepten-5-yl]-5-alkyl-1,3,4-oxadiazoles and congeners, useful as anti-diarrheal agents.
4010262 Method for reducing the incidence of scours in monogastric animals and for the treatment of scours  
Monogastric animals such as pigs are fed a daily ration of pregelatinized starch in a paste form during the first 5 - 7 days after they are weaned.
4003904 Anti-diarrheal oxadiazoles  
The present invention encompasses a compound of the formula ##STR1## and the pharmaceutically acceptable acid addition salts thereof wherein Y is alkylene having 1-4 carbon atoms; R 1 and R 2...
4002618 2,2-Diphenyl-5-(4-substituted-piperidino)-3-trans-pentenenitriles  
This invention encompasses novel 2,2-diphenyl-5-(4-substituted-piperidino)-3-trans-pentenenit riles. These compounds are useful anti-diarrheal agents and also possess analgesic activity.
3998832 Anti-diarrheal compounds  
The present invention comprehends a method for treating diarrhea comprising administering to an animal in need of anti-diarrheal treatment an effective antidiarrheal amount of a compound of the...
3989719 Dibenzoxazepine N-carboxylic acid hydrazides and derivatives  
Derivatives of the dibenzoxazepine N-carboxylic acid hydrazides are acylated to yield N,N'-diacyl hydrazines which are useful pharmacological agents as is evidenced by their acetylcholine...
3978225 Heterocyclic homoprostanoidal derivatives  
Heterocyclic homoprostanoidal derivatives are prepared. These compounds have valuable antiprostaglandin activity specifically inhibiting prostaglandin synthesis and antagonizing diarrhea induced by...
3959275 Fused ring N-[1-(3-cyano-3,3-diphenylpropyl)-4-phenylpiperidine-4-carbonyloxy]imide s  
Preparation of the subject compounds by reaction of 1-(3-cyano-3,3-diphenylpropyl)-4-phenylpiperidine-4-carboxyl ic acid with an N-hydroxy compound of the type HO--N Q wherein ##EQU1## represents...
3928574 Method and composition for treating diarrhea in mammals  
This invention relates to a composition for the treatment of diarrhea in bovine animals which, in addition to the fluid and electrolyte losses sustained by the patient, contains up to as much as...
Matches 151 - 200 out of 222 < 1 2 3 4 5 >