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7598294 |
3,4-methylenedioxy-substituted chalcones as therapeutic agents
The present invention pertains to the use of a compounds for the manufacture of a medicament for use in the treatment of a proliferative condition, wherein the compounds have the following formula:...
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7572831 |
Composition containing chalcone
The present invention provides an MMP-inhibitory composition comprising chalcone or its derivatives. They inhibit the MMPs in collagenase subfamily as well as those in gelatinase subfamily. The MMP...
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7364747 |
Process and product for inhibiting or preventing bacterial infections
The combination of a polymyxin composition and a hop composition produces unexpected and synergistic activity against gram positive bacteria.
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7348363 |
Method of controlling zoological and aquatic plant growth
A method of controlling target aquatic microorganism pest populations by exposing the target population to an effective amount of an aquacidal compound. The aquacidal compounds are selected from...
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7335384 |
Nutrient compositions for the treatment and prevention of inflammation and disorders associated therewith
The present disclosure describes a novel composition for the treatment and/or prevention of neurogenic inflammation. Such composition is also useful in the treatment and/or prevention of disease...
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7312243 |
Materials and methods for treatment of gastrointestinal disorders
The subject invention pertains to materials and methods for the prevention and treatment of gastrointestinal diseases, including inflammatory bowel diseases such as Crohn's disease and ulcerative...
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7064124 |
NF-κB inhibitor containing substituted benzoic acid derivative as active ingredient
A NF-κB inhibitor represented by the following formula (I) is provided:
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6949586 |
Synergistic composition of trans-tetracos-15-enoic acid and Apocynin and method of treatment for hepatotoxicity
The present invention relates to a synergistic hepatoprotective pharmaceutical composition comprising an effective amount of trans-tetracos-15-enoic acid (TCA) and Apocynin (APO), the present...
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6906076 |
Compounds and methods of use to treat infectious diseases
The present invention concerns alkyl aryl carbonyl compounds that possess anti-infective activity. The compounds of the invention can be used to target specific nuclear localization signal, thereby...
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6822002 |
Use of L-carnitine and its alkanoyl derivatives as osmotic agents in solutions for medical use
The use of L-carnitine and its alkanoyl devivatives, optionally in the form of a pharmaceutically acceptable salt, as osmotic agents in the preparation of solutions for medical use, particularly...
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6790463 |
Uses of targeted oxidative therapeutic formulation in arteriosclerosis
The use of a pharmaceutical formulation in treating coronary arteriosclerosis and a two-component pharmaceutical formulation. The pharmaceutical formulation contains peroxidic species or reaction...
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6677376 |
Non-peptidic cyclophilin binding compounds and their use
The invention relates to non-peptidic compounds that possess bioactive properties, such as the ability to protect neuronal cells from otherwise lethal treatments or the ability to promote the...
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6599530 |
Oral compacted composition comprising catechol derivatives
The present invention relates to an oral compacted composition comprising entacapone, nitecapone, or a pharmaceutically acceptable salt thereof and croscarmellose sodium. The composition is...
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6579903 |
Klainetins and their derivatives, method for their preparation and use thereof
The invention relates to compounds of formula I and of formula II in which R 1 , R 2 , R 3 , R 4 , R 5 , X 1 , X 2 , X 3 , X 4 , X 5 and Y are defined in the specification. The compounds of...
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6498195 |
Use of 1-propanone-1-(2,4-dihydroxyphenyl)-3-hydroxy-3-(4′-hydroxyphenyl) as an anticarcinogenic agent
Compositions and methods are provided for prevention and treatment of cancer. The compositions comprise pure hydroxylated chalcone compounds of licorice root ( Glycyrrhiza glabra ) including...
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6423740 |
Chalcones having antiproliferative activity
The invention relates to a novel class of compounds that have structures related to certain naturally occurring or synthetic chalcones. The invention also relates to pharmaceutical compositions...
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6417233 |
Ubiguinone-containing composition suitable for promoting enhanced intramitochondrial transportation of ubiguinones and methods of using same
Compositions containing as active ingredients a lipid-soluble benzoquinone, e.g. Coenzyme Q10 and at least one omega-3 polyunsaturated fatty acid selected from eicosapentaenoic acid (EPA),...
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6410602 |
Method of increasing the production and improving the quality of semen
A method of increasing the volume, the total sperm count and the reproductive performance of semen from human and animal males, is described. The method comprises administration of an effective...
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6410265 |
Gene encoding a putive efflux protein for solvents/antibiotics in Pseudomonas mendocina
This invention relates to the isolation of a novel putative efflux gene from Pseudomonas mendocina . The putative efflux gene is useful for probing an organism's efflux system to gain an...
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6335361 |
Method of treating benign forgetfulness
Disclosed herein are methods to treat cognition disorders, particularly those associated with aging. The method comprises administering a combination of a carnitine and an oxidant. Preferably the...
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6306913 |
Container for 4-allylanisole and analog scolytid pesticides
A projectile can be used to administer pesticides such as one or more from the group consisting of 4-allylanisole, anisole, allylbenzene, 4-isopropylanisole, p-anisaldehyde, ethylbenzene, cumene,...
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6133322 |
Quinone derivatives for treating or preventing diseases associated with iron overload
A method of treating or preventing a disorder resulting from a mitochondr dysfunction induced by an iron overload including Friedreich Ataxia, hypertrophic cardiomyopathy, Hallervorden-Spatz...
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6107276 |
Pharmaceutical compositions including a drug, a cross-linked polymeric substance, an oil, and a surface active agent
The pharmaceutical compositions including a slightly soluble drug incorporated in a water-swellable, but water-insoluble cross-linked polymer, a surface active agent, and an oil show much improved...
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6090851 |
Use of an NADPH-oxidase inhibitor in the treatment of reperfusion injury
The present invention is directed to a method for the prophylactic and therapeutic treatment of reperfusion injury or injury due to a distal reperfusion. The method involves the administration of...
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5973004 |
L-carnitine, acetyl-L-carnitine, and pantothenic acid or ubiquinone, combined for prevention and treatment of syndromes related to ineffective energy metabolism
A combination can be of L-carnitine and acetyl-L-carnitine, preferably with pantothenic acid or ubiquinone, is administered orally or as a parenteral injection in domesticated animals, especially...
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5902831 |
Prevention of atherosclerosis using NADPH oxidase inhibitors
A method for the prevention and treatment of atherosclerosis and its related diseases in mammals, in which an NADPH oxidase inhibitor is administered, is provided. The NADPH oxidase inhibitor...
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5654331 |
Diaromatic compounds derived from a salicylic unit and their use in human and veterinary medicine and in cosmetics
Diaromatic compounds, characterised in that they correspond to the following general formula: ##STR1## in which: R 1 is --CH 3 , --CH 2 OH, --COR 8 or --CH 2 OCOR 9 , R 8 is H, OH, --OR 10 ,...
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5637600 |
Phenylpyrrole derivatives and their use as dopamine D.sub.3 antagonists
The present invention relates to pyrrole compounds, processes for their preparation, pharmaceutical compositions containing them and their use in therapy, in particular as anti-psychotic agents.
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5489614 |
Catechol derivatives, their physiologically acceptable salts, esters and use
Known and new catechol derivates may be used as medicinal antioxidants in the prevention or treatment of tissue damage induced by lipid peroxidation. The conditions and diseases to be treated are...
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5476876 |
Di-tert-butylphenol compounds useful as anti-inflammatory agents
The subject invention relates to compounds having the structure: ##STR1## wherein (a) X is selected from hydroxy, C 1 to about C 2 alkanoxy, thiol, C 1 to about C 2 alkanylthiol, and halo; ...
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5466717 |
Halogenated 4'-methoxyacetophenones as microbicides and preservatives
Halogenated 4'-methoxyacetophenones of formula I: ##STR1## wherein X is a halogen; Y is a halogen; and n is 1 or 2 as microbicides for inhibiting the growth of microorganisms in aqueous systems and...
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5420160 |
1-alkoxyhexatriene-2-carboxylates
There are described new 1-alkoxyhexatriene-2-carboxylates of the formula (I) ##STR1## in which R represents substituted phenyl, and a plurality of processes for their preparation. The new...
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5405875 |
Method of inhibiting neoplasia and tumor promotion
The present invention provides a method of inhibiting neoplasia and tumor promotion. The method comprises administering to a mammal, particularly a human, in need thereof an effective amount of a...
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5393776 |
Tocotrienol analogs in the treatment of hypercholesterolemia and hyperlipidemia
This invention relates to structurally novel acyclic tocotrienol analogs, which are useful for cholesterol/lipid lowering in cases of hypercholesterolemia and hyperlipidemia, and for...
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5189066 |
Pharmaceutical compositions of tebufelone
The subject invention involves compositions, consisting essentially of the drug active 1-3,5-bis(1,1-dimethylethyl)-4-hydroxyphenyl-5-hexyn-1-one (tebufelone) at a concentration of at least about...
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5110801 |
Treatment of acne
Acne is treated by administering to the subject a substance which is effective in blocking glucose entry into sebaceous cells, thereby inhibiting the production of sebum by these cells. Typically,...
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5081155 |
Hydroxy aromatic ketones
Novel hydroxy-aryl ketones are disclosed having a branched hydrocarbon chain on the aromatic nucleus ortho to the hydroxy group. The compounds were found to possess anti-microbial properties and...
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4933165 |
Coenzyme Q.sub.10 with HMG-CoA reductase inhibitors
A pharmaceutical composition and method of counteracting HMG-CoA reductase inhibitor-associated myopathy is disclosed. The method comprises the adjunct administration of an effective amount of a...
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4847303 |
Tert-butylphenyl compounds useful as anti-inflammatory agents
The present invention involves compounds having the structure: ##STR1## wherein: (a) --A 1 is selected from the group consisting of --OH, --H, and --O 2 CR; (b) --A 2 is selected from the...
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4708966 |
Novel anti-inflammatory agents, pharmaceutical compositions and methods for reducing inflammation
The present invention relates to novel specifically-substituted phenyl compounds, especially substituted di-tert-butyl phenol derivatives, which are effective as anti-inflammatory, analgesic and/or...
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4621098 |
Thioethers and pharmaceutical compositions containing them
The present invention provides thioethers of the general formula: ##STR1## wherein Ar is a phenyl radical which is optionally substituted one, two or three times by alkyl, alkenyl, alkoxy,...
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4617187 |
Therapeutic method for treating radiation ulcers
Cutaneous administration of ubidecarenone, for example, application of ubidecarenone in the form of an ointment has been proven to be effective for treatment of various skin disorders caused by...
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4613611 |
Method of treating diabetes mellitus using arylglyoxals
A method of treating diabetes mellitus using arylglyoxals which are known compounds.
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4525361 |
Aralkyl carboxylic acid compounds in compositions for potentiating immuno activity
Novel compounds of the formulae ##STR1## wherein R represents lower alkyl or lower alkoxy, A represents --CH 2 --, --CO-- or ##STR2## n represents an integer of 1 to 8, X represents hydrogen or...
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4514420 |
Antifibrotic agent
Compounds of the formula ##STR1## wherein A is methylene or carbonyl, n is an integer of 2 to 21, inclusive, and R is hydrogen or lower alkyl, are effective for the prophylaxis or treatment of...
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4474810 |
Arylglyoxals and their pharmaceutical use
Arylglyoxals which are new compounds, active as hypoglycemic agents.
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4436753 |
Method for therapy of ischemic disease
A mammal suffering from ischemic disease such as cerebral apoplexy, cardiac insufficiency, renal insufficiency due to vascular changes, etc. is remedied by administering to said mammal an effective...
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4390537 |
1-(Substituted-aminoalkoxyphenyl)-2-methylene-1-alkanones, compositions and use
1-(Substituted-aminoalkoxyphenyl)-2-methylene-1-alkanones, a class of compounds possessing anti-allergic properties for use in the treatment of allergic conditions, such as asthma prepared by...
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4333952 |
Growth promotors for ruminants
Compounds of formula (I): ##STR1## wherein: R 1 is hydrogen, halogen or C 1 -4 alkoxy; X is oxygen; NR 3 in which R 3 is hydrogen, C 1 -4 alkyl, or -Y-R 2 ; --CO; or --CHOH; Y is --CH...
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4243683 |
Tertiary alcohols
Tertiary alcohols of the formula: ##STR1## wherein Y 1 represents a carbonyl or hydroxymethylene group, and either (i) A 1 represents a direct bond and R 1 represents a phenyl group which may...
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