|
Match
|
Document |
Document Title |
|
|
4959390 |
Polyhydroxybenzyloxypropanolamines
Compounds of the present invention, are represented by the general formula ##STR1## wherein R 1 group which may be alkyl of from 1 to about 6 carbon atoms, alkenyl of from 2 to about 6 carbon...
|
|
|
4943591 |
Dichloroaniline derivatives
The invention provides compounds of the general formula (I) ##STR1## wherein X represents a C 1 -6 alkylene, C 2 -6 alkenylene or C 2 -6 alkynylene chain and Y represents a bond, or a C 1 -4...
|
|
|
4940585 |
Method for the treatment of nicotine withdrawal syndrome
A therapeutic method for treatment of nicotine withdrawal syndrome symptoms of a patient in need thereof by administering to the patient a therapeutic composition of a pharmaceutically acceptable...
|
|
|
4937268 |
Chemical compounds
This invention relates to compounds of the general formula (I) and physiologically acceptable salts and solvates thereof wherein Ar represents ##STR1## where R 3 is a bond or a straight or...
|
|
|
4931474 |
Ether derivative and an acaricidal or insecticidal composition comprising said derivative
An ether derivative compound of the formula: ##STR1## wherein R 1 is hydrogen, chloro, methyl or (C 1 -C 3 )-alkoxy, R 2 is (C 1 -C 6 )-alkyl, R 3 is hydrogen, chloro, bromo, fluoro, --CF 3 ,...
|
|
|
4919937 |
Percutaneous administration of tamoxifen
Anti-estrogen drug of which the active product is comprised of 1 (p-dimethylaminoethoxyphenyl) trans-1-(p-hy-droxyphenyl)-2-phenylbut-1-ene, and present as a gel of the hydroalcoholic type which is...
|
|
|
4913891 |
Positron emitter labeled enzyme inhibitors
This invention involves a new strategy for imaging and mapping enzyme activity in the living human and animal body using positron emitter-labeled suicide enzyme inactivators or inhibitors which...
|
|
|
4914126 |
Aromatic amines
|
|
|
4908386 |
Ethanolamine derivatives
The present invention provides compounds of general formula (I) ##STR1## wherein Ar represents an unsubstituted or substituted phenyl gorup; R 1 and R 2 each represents a hydrogen atom or a C...
|
|
|
4898729 |
Treatment of hypertension, compounds and compositions for antihypertension and diuresis
Antihypertension action is achieved without diuresis by administration of a thiazide diuretic in an amount which while being sufficient to achieve antihypertension is insufficient to achieve...
|
|
|
4895845 |
Method of assisting weight loss
A method of assisting weight loss involving the combined administration of a rauwolfia alkaloid and at least one antidepressant, selected from the groups consisting of aminoazoles,...
|
|
|
4895715 |
Method of treating gynecomastia
A method of treating gynecomastia in noncastrated patients being treated with an antiandrogen for androgen-dependent diseases such as benign prostatic hypertrophy, who are in need of such treating...
|
|
|
4883804 |
Aromatic compounds
There are described compounds of formula I, ##STR1## in which X represents a C2 to 8 alkylene chain optionally interrupted by a double bond or by S(O) n , wherein n is 0, 1 or 2; Y represents O...
|
|
|
4880834 |
Method for administering ethanolamine derivatives to livestock
A method for treating livestock to decrease birth mortality rate and to increase post-natal survival rate by administering ethanolamine derivatives is disclosed.
|
|
|
4880841 |
Process of producing phenethylamine derivatives
Phenethylamine derivatives shown by the general formula ##STR1## wherein Ro represents a lower alkyl group; R 1 represents a lower alkyl group or a lower alkoxy group; R 2 represents hydrogen...
|
|
|
4871775 |
Substituted phenoxyalkanolamies and phenoxyalkanol-cycloalkylamines in pharmaceutical formulations and use thereof
New substituted phenoxyalkanolamines and phenoxyalkanol-cycloalkylamines of the general formula I ##STR1## in which R 1 and R 2 , which can be identical or different, denote alkyl groups with in...
|
|
|
4853381 |
Ethanolamine compounds
The invention provides compounds of the general formula (I) ##STR1## wherein Ar represents a phenyl group optionally substituted by one or more substituents selected from halogen atoms, or the...
|
|
|
4839155 |
Iodotamoxifen derivatives and use for estrogen receptor-positive breast cancer detection and therapy
Iodotamoxifen derivatives which are compounds of formula (3) ##STR1## wherein X represents 3- or 4- iodo and R 1 and R 2 , which may be the same or different, represent C 1 -3 alkyl, especially...
|
|
|
4831051 |
Aromatic derivatives comprising an aminoalkoxy chain, the salts thereof, the process for preparing these derivatives and salts and the application thereof in therapeutics
New aromatic derivatives having an activity antagonistic to calcium and corresponding to formula: ##STR1## in which: A represents a chain having any one of the following structures: ##STR2## Ar...
|
|
|
4824868 |
Propylamine derivatives useful for the treatment of dementia
Disclosed are e.g. certain novel 2-benzyl-3-(substituted)-phenoxypropylamines, their methods of synthesis and pharmaceutical compositions. Said compounds are useful as potent and centrally active...
|
|
|
4820736 |
Use of clomiphene to predict fertility in a human female
The invention relates to the use of clomiphene and its citrate salt in predicting fertility in a human female.
|
|
|
4820737 |
Lacrimal secretion stimulant (lss)
Ophthalmic compositions useful as tear stimulants when topically applied to the eye for effective treatment of dry eye syndrome.
|
|
|
4818772 |
Derivatives of 4-aminoethoxy-5-isopropyl-2-methylbenzenes: methods of synthesis and utilization as medicines
A compound with alpha 1-blocking activity having the formula: ##STR1## wherein R 1 is --H, --CH 3 or --COCH 3 ; R 2 is --H or CH 3 ; and R 3 is ##STR2## wherein Σ is --H or one or more...
|
|
|
4803225 |
Dihydroxy-phenethylamino compounds useful as pharmaceuticals
There are provided compounds of formula I, ##STR1## and pharmaceutically acceptable derivatives thereof. There are also described the use of the compounds of formula I as pharmaceuticals, methods...
|
|
|
4803227 |
Aminoalkyl ethers of phenols as anticancer agents for the breast and colon
The use of (a) N,N-dialkyl-2-[(4-phenylmethyl)phenoxy]ethanamine and N-morpholino-2-[(4-phenylmethyl)phenoxy]ethanamine compounds and their salts, as anticancer agents, is described. These...
|
|
|
4792551 |
9-anthryloxyaminoalkanes and related compounds as anti-inflammatory and analgetic agents
Compounds useful for treating inflammation, pain and swelling, represented by the formula: ##STR1## and the pharmaceutically acceptable acid addition salts thereof, wherein: Y and Z are each...
|
|
|
4792570 |
3- and 4-biphenyloxyaminoalkanes and related compounds as anti-inflammatory and analgetic agents
Compounds useful for treating inflammation, swelling and associated pain, represented by the formula: ##STR1## and the pharmaceutically acceptable acid addition salts thereof, wherein: a is an...
|
|
|
4764533 |
Erythro-1,2-1-pentanones
Erythro-1,2,3-triphenyl-1-pentanones of Formula 1 ##STR1## wherein R 1 may be a dimethylamino, diethylamino, piperidin-1-yl- or pyrrolidin-1-yl group and R 2 represents a hydrogen atom, a methoxy...
|
|
|
4762855 |
Novel pharmaceutical compositions improving oxygenation of the brain and a process for their production
2,2-Bisphenoxy-dimethyl-aminoethane to improve brain disfunction.
|
|
|
4749700 |
Novel methods of administering antihistamines, antinausea and antiemetic pharmaceutical agents and novel dosage forms containing same
Invention relates to nasal administration of physiologically active therapeutic agents and dosage forms useful for such administration.
|
|
|
4699928 |
Fluoroallylamine derivatives
Fluoroallylamine derivatives of the following Formula I are novel MAO-inhibitors and at low dose levels selectively inhibit MAO-B: ##STR1## wherein: R 1 and R 2 independently represent hydrogen,...
|
|
|
4692469 |
Propylamine derivatives
Disclosed are e.g. certain novel 2-benzyl-3-(substituted)-phenoxypropylamines, their methods of synthesis and pharmaceutical compositions. Said compounds are useful as potent and centrally active...
|
|
|
4692465 |
2-phenylethylamine derivatives
Compounds of formula (I): ##STR1## or a pharmaceutically acceptable salt, ester or amide thereof, wherein: Ar is benzofuran-2-yl, or phenyl optionally substituted by groups R 1 and/or R 2 wherein...
|
|
|
4683235 |
Analgesic method
This invention provides a method of producing analgesia in mammals which comprises administering codeine and fluoxetine or norfluoxetine. Pharmaceutical formulations useful in this method are also...
|
|
|
4649160 |
Substituted phenoxy-aminopropanols
Substituted phenoxy-aminopropanols of the formula ##STR1## wherein R is a branched-chain alkyl of 3 or 4 carbon atoms, R 1 is hydrogen, halogen or lower alkyl and R 2 and R 3 , independently, are...
|
|
|
4647590 |
Pharmaceutical compositions and their use in the treatment of glaucoma
1-moprolol is instilled locally in the form of an opthalmic pharmaceutical composition to treat glaucoma.
|
|
|
4647591 |
Method for improving memory
Fluoxetine can be employed to improve memory in mammals and to treat amnesia.
|
|
|
4629727 |
Therapeutic agents
Compounds of formula I ##STR1## in which n=0 or 1; in which, when n=0, R 1 is H, an alkyl, a cycloalkyl, a cycloalkylmethyl, an alkenyl or, an alkynyl group a heterocyclic ring or an optionally...
|
|
|
4626549 |
Treatment of obesity with aryloxyphenylpropylamines
3-Aryloxy-3-phenylpropylamines and acid addition salts thereof are useful in blocking uptake of monoamines by brain neurons, and are thus effective in treating disorders of sleep, sexual...
|
|
|
4605673 |
7H-dibenzo(a,c,)cyclohepten-5-one-(7) derivatives
The invention is concerned with 7H-dibenzo(a,c)-cyclohepten-5-one-(7) derivatives of general formula I ##STR1## wherein R 1 and R 2 can be the same or different, a hydrogen atom, an alkyl radical...
|
|
|
4588719 |
Bicyclic benzenoid aminoalkylene ethers and thioethers, pharmaceutical compositions and use
A class of bicyclic benzenoid aminoalkylene ether and thioether compounds exhibiting pharmacological activity, including anti-secretory and anti-ulcerogenic activity, pharmaceutical compositions...
|
|
|
4584404 |
Substituted phenoxyphenylproply dimethylamines
Selective biogenic amine uptake inhibitors, 3-substituted phenyloxy-3-phenylpropyldimethylamines.
|
|
|
4562211 |
Pharmaceutically active 2-substituted-1-(omega-aminoalkoxy)benzenes
2-Substituted-1-(omega-aminoalkoxy)benzenes are prepared and found useful as pharmaceutical agents, particularly as antidepressants.
|
|
|
4556677 |
Alkane and alkene derivatives and their use
The invention provides novel compounds of the formula ##STR1## wherein R 1 is hydrogen, hydroxy, alkoxy of 1 to 4 carbon atoms, benzyloxy, allyloxy, 2,3-epoxypropoxy, methoxymethoxy,...
|
|
|
4536503 |
Naphthoxyalkylamines and related compounds as antiinflammatory agents
Compounds of the formula: ##STR1## and the pharmaceutically acceptable acid addition salts thereof, wherein; Y is halo, alkoxy, alkyl, or dialkylamino; a is 0, 1 or 2; b is an integer from...
|
|
|
4513010 |
Method of treating navicular disease in horses
A method of treating navicular disease in horses comprising the administration of Isoxsuprine over an extended period and an injectable paste composition including isoxsuprine hydrochloride and...
|
|
|
4460605 |
2-[2'-Hydroxy-3'-(1,1-dimethylpropylamino)-propoxy ]-β-phenylpropiophenone, its physiologically acceptable acid addition salts, and pharmaceutical compositions
The 2-[2'-hydroxy-3'-(1,1-dimethylpropylamino)-propoxy]-β-pheny
lpropiophe none of formula I ##STR1## and its acid addition salts are described. Moreover, the preparation of this compound and of...
|
|
|
4443441 |
Fixation of intraocular lenses
The fixation of an intraocular lens is aided by instilling into an eye having an intraocular lens about one drop of an ophthalmic solution containing an α-adrenergic blocking agent, such as...
|
|
|
4424216 |
Method for the reduction of mucin viscosity
A method for reducing mucin viscosity which comprises administering an effective dose of a compound having protected sulfhydryl groups which metabolize in vivo to produce free sulfhydryl groups.
|
|
|
4419354 |
9,10-Bis(aminoalkoxy)anthracenes
This disclosure describes certain substituted 9,10-bis(2-aminoethoxy)anthracenes which are useful as modulators of the immune response system in warm-blooded animals and for inducing the regression...
|