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4511581 |
Fungicidal indanylbenzamide
A fungicidal indanylbenzamide derivative of the formula: ##STR1## wherein X is a lower alkyl, nitro, or trifluoromethyl group or a halogen atom, and R 1 , R 2 and R 3 , which are same or...
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4508735 |
Anti-arrhythmic N-alkanoylaminoalkyl fluorenes
9-(N-alkanoylaminoalkyl)-fluorenes are anti-arrhythmic agents.
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4499303 |
Antihyperlipidemic N-benzoylsulfamates, N-benzylsulfamates and benzylsulfonamides
This invention relates to novel N-benzoylsulfamates, N-benzylsulfamates and benzylsulfonamides and pharmacologically acceptable salts thereof, a method for lowering serum levels in mammals by...
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4478836 |
1-Aryl 2-aminomethyl cyclopropane carboxyamide (Z) derivatives and their use as useful drugs in the treatment of disturbances of the central nervous system
The present invention concerns new derivatives of 1-aryl 2-aminomethyl cyclopropane carboxamides (Z) of general formula I: ##STR1## in which: R represents a hydrogen or halogen atom, a lower alkyl...
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4477467 |
Insect repellent
An insect repellent is disclosed which comprises, as essential ingredients, N,N-diethyltoluamide as a repellent component, and an aromatic proton donor in which the aromatic rings are substituted...
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4456618 |
Naphthenic and heterocyclic retinoic acid analogues
Naphthenic and heterocyclic retinoic acid analogues such as (E)-6-[2-(2,6,6-trimethyl-1-cyclohexen-1-yl)ethenyl]-2-napht
haldehyde, methyl...
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4454339 |
9-Fluoroprostaglandin derivatives, and use as medicinal agents
9-Fluoroprostane derivatives of Formula I ##STR1## wherein R 1 is CH 2 OH or ##STR2## wherein R 2 is hydrogen, alkyl, cycloalkyl, aryl, or a heterocyclic residue; or R 1 is the residue ##STR3##...
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4435425 |
Fluorinated diaminobutane derivatives
Fluorinated diaminobutane compounds in vivo are inhibitors of gamma-aminobutyric acid transaminase and have the following formula: ##STR1## wherein: R 1 represents hydrogen, C 1 -C 6 alkyl, or...
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4427700 |
Repellent for black fly
A significant enhancement of repellency toward the black fly (Simulium venustum Say, and Prosimulium hirtipes Fries) of N,N-diethyl-m-toluamide has been obtained by the addition, or conjunctive...
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4425357 |
Acyl anilines exerting a fungicidal action
Acyl anilines are disclosed having the formula ##STR1## wherein R and R 1 (like or unlike each other)=H; CH 3 ; C 2 H 5 ; n.C 3 H 7 ; --CH 2 --CHCH 2 ; --CHCH--CH 3 ; R 3 and R 4...
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4424205 |
Hydroxyphenylacetamides having analgesic and anti-irritant activity
A compound, or pharmaceutically acceptable salt thereof, having the formula: ##STR1## wherein R is a linear or branched C 3 -C 11 alkyl, alkynyl or aralkyl group, a linear or branched C 3 -C 22 ...
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4423040 |
Vehicle composition containing 1-substituted azacyclohexan-2-ones
Compositions useful for carrying physiologically active agents such as therapeutic agents through skin and other body membranes comprising the agent and an effective, non-toxic amount of a compound...
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4410519 |
Tetraline derivatives, their production and pharmaceutical compositions containing them
An optically active or racemic 2-amino-5-hydroxy-1,2,3,4-tetrahydronaphthalene wherein the nitrogen atom of the amino group carrier two alkyl groups, one of which is unsubstituted and the other is...
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4404226 |
Use of guanfacine in treating schizophrenia
This invention provides a new neuroleptic use of a guanidine derivative and novel pharmaceutical compositions for such use.
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4404215 |
Piperidyl phenyl trifluoroethanols
This invention relates to novel arylethanol and to process for producing the said compounds. The arylethanols of the invention have valuable pharmacological properties and find a use in human or...
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4402975 |
Aminocarboxylic acids, amino alcohols, or the derivatives thereof, processes for production thereof, and pharmaceutical uses thereof
A compound represented by the following formula ##STR1## wherein R 1 represents a hydrogen atom, an acyl group or an alkoxycarbonyl group; X 1 represents an alkylene group having 3 to 6 carbon...
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4401665 |
Sleep-aid composition containing an analgesic and diphenhydramine dihydrogencitrate, and method of use
An analgesic and sleep-aid composition containing an analgesic (e.g. aspirin, APAP or combinations thereof) and diphenhydramine dihydrogencitrate. Discloses several dosage forms including a two...
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4390549 |
N-Tetrachloroethylthio benzoyl anilides useful as acaricides and to control mosquitoes
N-tetrachloroethylthio benzoyl anilide compounds having the formula ##STR1## in which R is chlorine, hydrogen, or trifluoromethyl and X is hydrogen or fluorine, useful as acaricides and to control...
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4376783 |
Acylated guanidines and medicaments containing them
The novel acylated guanidines, ureas and substituted ureas correspond to the general formula: ##STR1## in which R 1 repesents a substituted or unsubstituted aromatic ring, R 2 represents an...
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4355045 |
Anti-inflammatory 1-phenylethanolamine derivatives pharmaceutical compositions thereof and processes for their manufacture
The invention relates to topically anti-inflammatory 1-phenylethanolamine derivatives of the general formula I: ##STR1## or acid-addition salts thereof, to pharmaceutical compositions thereof, and...
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4346101 |
Benzamide derivative analgesics
Benzamide derivative analgesic compounds of the formula ##STR1## wherein P, Q, R 1 , R 2 , X and Y are as defined in the specification, e.g.,...
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4320142 |
N-[(phenyl(oxy or amino))thioacetyl]-1,2-diamine anthropodicides
Compounds of formula (I) are pesticides active against arthropods. ##STR1## wherein R 1 , R 2 , and R 3 are H, alkyl, alkoxy, halo, CN or CF 3 or two are linked to form a 3 or 4 carbon atom...
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4313956 |
Novel sypathomimetic amine prodrugs
Novel, transient prodrug forms of the phenolic dihydroxy sympathomimetic amines have (i) the structural formula (I): ##STR1## wherein X is O, S or NR 5 ; n is 1 or 2; R 1 is the...
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4311706 |
Novel dopa/dopamine prodrugs
Novel, transient prodrug forms of dopa and dopamine have (i) the structural formula (I): ##STR1## wherein each R is independently selected from the group consisting of hydrogen, R 3 -CO- and...
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4309444 |
Biologically active amides
Cinnamamides of formula (I), ##STR1## wherein X is fluoro, chloro, bromo, iodo or trifluoromethyl and R is branched alkyl, have anticonvulsant properties.
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4272550 |
Omega-[4-(polyfluoro-2-hydroxy-2-propyl)-2,3,6-substituted-phenoxy and phenylthio]alkanoic acids and compounds related thereto
Omega-[4-(polyfluoro-2-hydroxy-2-propyl)-2,3,6-substituted-p
henoxy and phenylthio]alkanoic acids and compounds related thereto having antihypertensive activity are preparable by reaction of the...
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4271193 |
N1-Benzoyl-N2-phenyldiaminopropanols and pharmaceutical compositions thereof, and processes for their preparation
N 1 -benzoyl-N 2 -phenyl-1,3-diaminopropan-2-ols are disclosed which exhibit a stabilizing effect on the gastric mucosa and enhance the stability and resistance of the gastic mucosa against...
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4228185 |
N-4-(2',2'-Dichlorocyclopropropyl)phenyl 2"-iodobenzamide
This invention relates to the novel compound N-4-(2',2'-dichlorocyclopropyl)phenyl 2"-iodobenzamide, having the formula ##STR1## which has been found useful as a fungicide.
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4212878 |
Phenylacetamide derivative analgesics
N-[(1-Amino-4-(mono or di-oxygen-group-substituted)cyclohex-1-yl)methyl]phenylaceta
mide derivatives of the formula 1 ##STR1## wherein R, R 1 , R 2 , R 3 , P, Q, X and Y are defined in the...
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4209532 |
Biocidal 2-aryl-1,3-cyclohexane dione compounds and alkali metal and ammonium salts thereof
2-Aryl-1,3-cyclohexanedione compounds and their alkali metal and ammonium salts exhibit outstanding herbicidal, miticidal and mite ovicidal activity.
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4197308 |
Analgesic N-(2-heterocyclic-amino cycloaliphatic) benzamides
Cis- and trans-N-(2-aminocycloaliphatic)benzamide compounds of the formula ##STR1## e.g., N-methyl-N-[2-(N-pyrrolidinyl)cyclohexyl]-3,4- dichlorobenzamide, and their pharmaceutically acceptable...
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4197316 |
Treatment of dry skin
Preventive as well as therapeutic treatment to alleviate the symptoms of disorders characterized by cracking, flaking or scaling of the skin consisting of the topical application of a lotion, cream...
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4193931 |
Polyene compounds
Novel 7-(substituted indanyl or naphthyl)-3-methyl-octa-2,4,6-triene derivatives useful as anti-tumor agents are disclosed.
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4191780 |
Bromhexine derivatives and process for making same
Bromhexine derivatives corresponding to the following general formula ##STR1## and antitussive compositions therefrom, as well as a process for making same are described.
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4190674 |
3-Fluoro-N-cyclopropylcinnamide
Cinnamamides of formula (I), ##STR1## wherein X is fluoro, chloro, bromo, iodo or trifluoromethyl and R is cycloalkyl or cycloalkyl alkyl, have anticonvulsant properties. The compound...
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4185124 |
2-(4-Biphenylyl)-N-(2-diethylamino alkyl)propionamide and salts thereof used as spasmolytic agents
New compounds useful as spasmolytic agents are provided with the following formula: ##STR1## wherein n is either 2 or 3. In addition, salts of these new compounds are provided and are suitable for...
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4179524 |
Biologically active amide
This application discloses the compound trans-3-fluoro-N-allylcinnamamide the use thereof as an anticonvulsant and a pharmaceutical preparation thereof which includes the compound or a...
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4179501 |
Analgesic N-(2-aminocycloaliphatic)azidobenzamides
Cis- and trans-N-(2-aminocycloaliphatic)benzamide compounds of the formula ##STR1## e.g., N-methyl-N-[2-(N-pyrrolidinyl)cyclohexyl]-3,4-dichlorobenzam
ide, and their pharmaceutically acceptable...
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4176196 |
Hypoglycemic arylcyclohexane acetic acids
Novel hypoglycemic agents comprising 3-hydroxy-3-arylcyclohexane-1-acetic acid, 3-arylcyclohexene-1-acetic acids and derivatives thereof are disclosed.
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4175135 |
Method of controlling acarina ectoparasites on warmblooded animals by orally administering to the animal an ectoparasitically effective amount of a 2-aryl-1,3-cyclohexanedione compound, and alkali metal salts, ammonium salts and enol esters thereof
A method of controlling acarina ectoparasites on warmblooded animals by orally administering to the animals an ectoparasitically effective amount of a 2-aryl-1,3-cyclohexanedione compound and...
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4173652 |
Pharmaceutical hydroxamic acid compositions and uses thereof
New and useful phenylalkylcarbohydroxamic acids are disclosed of the formula ##STR1## wherein: (a) R is selected from the group consisting of alkoxy of one to six carbon atoms, alkenyloxy of two to...
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4158063 |
Acylamino(alkyl)benzene derivatives and process for preparing them
The invention relates to acylamino(alkyl)benzene derivatives of the general formula ##STR1## in which W represents a group which can be converted into a carboxyl group, or an aldehyde group or an...
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4145435 |
2-Aminocycloaliphatic amide compounds
Cis- and trans-N-(2-aminocycloaliphatic)-2-arylacetamide derivative compounds of the formula ##STR1## e.g., N- 2-(N', N'-dimethylamino)cyclohexyl!-N-methyl-2-(4-bromophenyl)aceta
mide and...
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4141987 |
1-Aryloxy-3-thenamidoalkylamino-2-propanol derivatives
Novel 1-heterocyclyloxy- or 1-aryloxy-3-amidoalkylamino-2-propanol derivatives, processes for their manufacture, pharmaceutical compositions containing them and methods of using them in the...
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4139635 |
Cysteamine derivatives for oral treatment of seborrhea
A method for treating a scalp characterized by an excessive secretion of sebum, to improve the condition thereof by reducing said excessive secretion comprising orally administering to a human...
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4136198 |
Method for the control of trypanosomiasis
A composition comprising from 0.02 to 17 parts by weight of glycerol per part by weight of an iron chelating agent selected from the group consisting of salicyl hydroxyamic acid; 2,3- and...
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4128664 |
Substituted benzamides as anti-inflammatory agents
Compounds in which 2,6-di(t-butyl)phenol is substituted in the 4 position by an N-substituted carboxamido group have valuable pharmacological activity as anti-inflammatory agents.
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4123554 |
Fungicidal and germicidal benzanilides
The present invention relates to a compound having the following general formula (I): ##STR1## wherein X stands for a halogen atom or a methyl radical; and R stands for an alkyl or alkoxy radical...
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4122190 |
Treating acromegaly
α-Adrenoceptor agonists are useful in the treatment of acromegaly.
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4115582 |
N-1,1,2,2-tetrachloro-2-fluoroethylthio benzanilide and its use as fungicide and acaricide
N-1,1,2,2-tetrachloro-2-fluoroethylthio benzanilide which has the structural formula ##STR1## and its use as a fungicide and acaricide.
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