Matches 151 - 200 out of 312 < 1 2 3 4 5 6 7 >
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6114382 Methods for treating inflammatory bowel disease  
The present invention provides novel compositions and methods relating to the treatment of Inflammatory Bowel Disease ("IBD"), most notably, Ulcerative Colitis, Crohn's Disease, Colitis and...
6096784 Inhibitors of oleamide hydrolase  
Inhibitors of oleamide hydrolase, responsible for the hydrolysis of an endogenous sleep-inducing lipid (1, cis-9-octadecenamide) were designed and synthesized. The most potent inhibitors possess an...
6083987 Phenylenediamine derivative, radical scavenger, brain-infarction depressant, and brain-edema depressant  
A phenylenediamine derivative or a salt thereof in accordance with the present invention is expressed by the following formula 1: ##STR1## wherein A represents a group expressed by --CO--, --CH 2 ...
6075023 Method for combatting fish mycoses and one-celled ectoparasites  
6037361 Fluorinated butyric acids and their derivatives as inhibitors of matrix metalloproteinases  
Fluorinated butyric acid compounds and derivatives are described as well as acid methods for the preparation and pharmaceutical compositions of same, which are useful as inhibitors of matrix...
6028110 Succinyl hydroxamic acid, N-formyl-N-hydroxy amino carboxylic acid and succinic acid amide derivatives as metalloprotease inhibitors  
A pharmaceutical or veterinary composition comprising a compound of formula I ##STR1## wherein X is a --CO 2 H group and R 1 , R 2 , R 3 , R 4 , R 5 are as defined in the specification, or a...
6017906 Polyamine conjugates for treatment of infection  
The present invention relates to methods of preventing or treating an infection or disease caused by an infectious agent. The present invention also relates to the augmentation of the efficacy of...
6013673 Naphthyloxy acetic acid derivatives  
A naphthyloxyacetic acid derivative of the formula (I) ##STR1## wherein R 1 is H, alkyl, alkylene-(--COOR 10 , --OH, --CONR 4 R 5 , --CONR 6 -alkylene-OH, --NR 4 R 5 , -cyano or -tetrazolyl); A...
6004992 Aminocarboxylic acid fluorobutenyl esters  
The present invention relates to novel fluorobutenyl aminocarboxylates of the formula (I) R--CO--O--CH 2 --CH 2 --CXCF 2 (I) in which X represents hydrogen or halogen and R...
5994270 Fungicides for the control of take-all disease of plants  
Plant disease caused by soil-borne fungus Gaeumannonyces graminis (Gg) is controlled by applying to the seed or the soil a fungicide which has the following general formula: ##STR1##
5994405 Agent for contact lenses  
An agent for contact lenses, comprising chloroacetamide. According to the present invention, chloroacetamide, which is the bacteriocidal component to be contained, is scarcely adsorbed not only to...
5990170 Therapeutic use of mono and bicarboxylic acid amides active at the peripheral cannabinoid receptor  
The following description concerns a therapeutic method for the treatment of diseases connected with the modulation of the cannabinoid peripheral receptor, comprising administering amidic...
5985926 Method for inhibiting intracellular viral replication  
There is disclosed a method of preventing or delaying the occurrence of acquired immunodeficiency syndrome (AIDS) in human immunodeficiency virus (HIV) seropositive humans by administering an...
5985910 3- [4- (2- Phenyl-Indole-1-ylmethyl) Phenyl]- Acrylamides as estrogenic agents  
The present invention relates to new 3-[4-(2-Phenyl-Indole-1-ylmethyl)-Phenyl]-Acrylamide compounds which are useful as estrogenic agents, as well as pharmaceutical compositions and methods of...
5981580 Fatty acid analogs and prodrugs  
Novel derivatives of fatty acid analogs that have from one to three heteroatoms in the fatty acid moiety which can be oxygen, sulfur or nitrogen, are disclosed in which the carboxy-terminus has...
5976516 Hair cosmetic compositions  
Described is a hair cosmetic composition comprising an amide compound having a melting point of 0 to 50° C. The hair cosmetic composition according to the present invention can impart the hair...
5972892 Topical composition containing a substance P antagonist  
The invention relates to a therapeutic composition for topical application containing at least one product with an irritant side effect and a substance P antagonist for reducing or even eliminating...
5958439 Plant protection composition containing one or more water soluble active materials and one or more polyalkoxylated amidoamines  
A composition containing, as active ingredient, one or more water soluble plant protection active materials and further containing an effective amount of one or more polyalkoxylated amidoamines of...
5929119 Fungicidal composition  
A composition which is suitable for controlling fungal pests, comprising conventional additives and an effective amount of a p-hydroxyaniline derivative of the general formula I ##STR1## where the...
5925674 Cycloalkylcarboxanilides  
This invention relates to cycloalkylcarboxanilides of the formula ##STR1## which are used to combat pests.
5925367 Pest control with UV blockers and pheromones  
A composition for controlling harmful insects and representatives of the order Acarina, containing as biologically active components a) a substance that modifies the behavior of the pests and b) at...
5907049 Meadowfoam amine oxides  
The present invention deals with the composition of matter and the utilization of certain amine oxides of meadowfoam amido propyl dimethyl amine. These materials are useful in personal care...
5900432 Therapeutic N-(4-benzoyl-2-methyl-phenyl)-3,3,3-trifluoro-2-hydroxy-2-methyl-propana mides  
Compounds of formula I: ##STR1## wherein, ring C, A--B, R 1 , n, R 2 , and R 3 have any of the meanings given in the specification, and their pharmaceutically acceptable salts are useful in the...
5889058 Peptidyl derivatives  
Methods of use for compounds of formula (I) are described wherein R represent a --CONHOH, carboxyl (--CO 2 H) or esterified carboxyl group; R 1 represents a hydrogen atom or an optionally...
5877220 Amide-based oligomeric cationic lipids  
The present invention provides amide-based oligomeric cationic lipids. The present invention further provides compositions of these amide-based cationic lipids with anionic macromolecules, methods...
5874444 Poly (ADP-ribose) polymerase inhibitors to treat diseases associated with cellular senescence  
Inhibition of the enzyme poly (ADP-ribose) polymerase can delay the onset of senescence and inhibitors of the enzyme can be used to treat diseases caused or exacerbated by cellular senescence.
5869453 Cytotoxic T-cell epitopes  
The present invention provides cytotoxic Epstein-Barr virus T-cell epitopes. The epitopes are selected from the group consisting of QAKWRLQTL, RYSIFFDY, HLAAQGMAY, YPLHEQHGM, SVRDRLARL, AVLLHEESM,...
5861435 Method for preventing settlement of aquatic fouling organisms  
A method for preventing settlement of aquatic fouling organisms on surface of an aquatic structure without environmental hazard is provided. The method is based upon absolutely novel concept to...
5859054 Leukotriene B4 derivatives, process for their production and their use as pharmaceutical agents  
Pharmacologically active leukotriene-B 4 derivatives of general formula I, ##STR1## are described, in which R 1 represents CH 2 OH, CH 3 , CF 3 , COOR 4 , CONR 5 R 6 , or R 2 represents...
5849728 Desquamation compositions  
The subject invention relates to desquamation compositions comprising a combination of salicylic acid and certain zwitterionic surfactants. The subject invention further relates to methods of...
5834517 Meadowfoam sulfosuccinates in personal care applications  
The present invention deals with a process for cleaning and conditioning hair and skin which comprises the contacting of hair or skin woth an effective concentration of certain novel meadowfoam...
5830869 Thiadiazole amide MMP inhibitors  
The present invention provides novel thiadiazole amide derivatives represented by formula I ##STR1## The compounds of the present invention inhibit various enzymes from the matrix metalloproteinase...
5827891 HIV protease inhibtors  
HIV protease inhibitors, obtainable by chemical synthesis, inhibit or block the biological activity of the HIV protease enzyme, causing the replication of the HIV virus to terminate. These...
5827852 Coated pharmaceutical compositions  
Pharmaceutical composition suitable for coating comprising a composition for oral administration in unit dosage form wherein said composition has been coated with from about 0.01% to about 10% by...
5824650 Topical composition containing a substance P antagoinst  
The invention relates to a therapeutic composition for topical application containing at least one product with an irritant side effect and a substance P antagonist for reducing or even eliminating...
5783593 Inhibitors of squalene synthetase and protein farnesyltransferase  
The present invention provides a compound of the formula ##STR1## which inhibit squalene synthetase and cholesterol biosynthesis and are useful in the treatment of e.g., hyperlipidaemia,...
5760085 Topical aromatic releasing compositions  
The present invention relates to topical aromatic releasing compositions containing one or more volatile aromatic compounds selected from the group consisting of 3-1-menthoxy propane-1,2-diol,...
5756547 Method for the treatment of preserving organs or tissue for transplantation  
Bucillamine and N-2,2-dimethyl-3-mercaptopropionyl)-L-cysteine or related compounds can be used to prevent damage to living tissue from the formation or presence of reactive oxygen species. These...
5753704 Therapeutic compositions comprising unsaturated dioic acids or derivatives thereof  
Disclosed are certain novel polyunsaturated dioic acids having between 8 and 16 carbon atoms (inclusive), excluding those compounds in the group consisting of: 2,5 octadienedioic acid; 1,7...
5750559 Potentiation of the antireactive-antiasthmatic effect of inhaled loop diuretics by inhaled non-steroidal anti-inflammatory drugs  
The antireactive-antiasthmatic effect of inhaled loop diuretics is potentiated by the use of a combination of a loop diuretic and a non-steroidal anti-inflammatory drug as an inhalant for combating...
5703129 5-amino-6-cyclohexyl-4-hydroxy-hexanamide derivatives as inhibitors of β-amyloid protein production  
A series of 5-amino-6-cyclohexyl-4-hydroxy-hexanamide derivatives of Formula I have been synthesized. ##STR1## As inhibitors of the production of β-amyloid protein from β-amyloid precursor...
5693630 Phenylethyl and phenylpropylamines  
Compounds of the general formula ##STR1## or pharmaceutically acceptable salts thereof, wherein Z is a saturated or unsaturated 3 to 6 carbon chain, m is 2 or 3, R 1 is a hydrogen atom, or a...
5684049 HIV-inhibiting benzeneacetamide derivatives  
A compound for use as a medicine having the formula ##STR1## a pharmaceutically acceptable acid addition salt form or a stereochemically isomeric form thereof, wherein R 1 and R 2 each...
5672597 Acetamide derivative  
An acetamide derivative having the general formula (I): ##STR1## or a pharmacologically acceptable salt thereof; a synthetic intermediate of the above-mentioned acetamide derivative; a treating...
5670545 Method for the treatment of ischemic disease and reperfusion injury and the prevention of the adverse effects of reactive oxygen species  
Bucillamine and N-2,2-dimethyl-3-mercaptopropionyl)-L-cysteine or related compounds can be used to prevent damage to living tissue from the formation or presence of reactive oxygen species. These...
5652250 N-substituted β-aryl- and β-heteroaryl-α-cyanoacrylamide derivatives and process for their preparation  
The present invention relates to new compounds of formula ##STR1## wherein A is a bicyclic ring chosen from naphthalene, tetrahydronaphthalene, quinoline, isoquinoline and indole. B is a R 2 ...
5652228 Topical desquamation compositions  
The subject invention relates to desquamation compositions comprising a combination of salicylic acid and certain zwitterionic surfactants. The subject invention further relates to methods of...
5650397 Antioccidial method  
The present invention is directed to anticoccidial methods, animal feed premixes, and animal feeds, employing a specified o-phenylenediamine or benzimidazole. The present invention is also directed...
5622916 Substituted 2-cylcohexen-1-yl-amine fungicidal and herbicidal agents  
A method of combating pests which comprises applying to such pests or to a pest habitat a pesticidally effective amount of a substituted 2-cyclohexen-1-yl-amine derivative of the formula ##STR1##...
5607978 Non-acidic cyclopentane heptanoic acid, 2-cycloalkyl or arylalkyl derivatives as therapeutic agents  
The present invention provides cyclopentane heptanoic acid, 2-cycloalkyl or arylalkyl derivatives, substituted in the 1-position with halo, methyl, hydroxyl, nitro, amino, amido, azido, oxime,...
Matches 151 - 200 out of 312 < 1 2 3 4 5 6 7 >