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8071650 |
Thiourea derivatives and the pharmaceutical compositions containing the same
The present invention relates to novel thiourea derivatives as a modulator for vanilloid receptor (VR) and the pharmaceutical compositions containing the same. As diseases associated with the...
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8052985 |
Storage-stable compositions containing hydrogen cyanamide and propionic acid
An aqueous storage-stable composition comprises from about 10 to about 35% by weight hydrogen cyanamide, from about 3 to about 25% by weight propionic acid, potassium propionate or ammonium...
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8021648 |
Hydrogen cyanamide pesticide formulations
Agricultural crops are protected from the growth of undesirable vegetation as well as nematode and insect infestations, by the application of hydrogen cyanamide in combination with a short-chain,...
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7968108 |
Hydrogen cyanamide pesticide formulations
Agricultural crops are protected from the growth of undesirable vegetation as well as nematode and insect infestations, by the application of hydrogen cyanamide in combination with a short-chain,...
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7572460 |
Hydrogen cyanamide pesticide formulations
Agricultural crops are protected from the growth of undesirable vegetation as well as nematode and insect infestations, by the application of hydrogen cyanamide in combination with a short-chain,...
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7365098 |
N'-cyano-N-methyl-imidamide derivatives
The present invention relates to novel N′-cyano-N-methylimidamide derivatives of the general formula (I) in whichn represents 2, 3, 4 or 5,R represents optionally halogen-substituted C1-C4-alkyl, a...
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7214714 |
20-hydroxyeicosatetraenoic acid production inhibitors
A hydroxyformamidine compound represented by the following formula or a pharmaceutically acceptable salt thereof [wherein R1 represents a substituted morpholino group, a substituted piperidino...
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7048925 |
Acid-sensitive polyacetals and methods
Polyacetals comprising a recurring units represented by a formula selected from the group consisting of formula (I) and (II): wherein A comprises at least one acetal group; B is selected from the...
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7045315 |
Methods for modulating expression of exogenous genes in mammalian systems
In accordance with the present invention, there are provided various methods for modulating the expression of an exogenous gene in an isolated cell and in a mammalian subject employing modified...
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6946485 |
Treatment of post-angioplasty restenosis and atherosclerosis with Ras antagonists
Disclosed are methods for inhibiting Ras activity such as cell proliferation associated with vascular injury such as post-angioplasty restenosis and atherosclerosis. Preferred Ras antagonists are...
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6878374 |
Biodegradable polyacetals
A polymer comprising recurring units represented by formula (I): wherein X is selected from the group consisting of C(O)OR1, C(O)SR1, C(O)NR1R2, and VZ, where R1 and R2 are each individually...
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6878706 |
Cyanamides useful as reversible inhibitors of cysteine proteases
Compounds according to the following formula (I): wherein the variables Q and R1 to R6 are as described herein, which reversibly inhibit the cysteine proteases, such as cathepsins K, S, F, L and B;...
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6806292 |
Substituted imide derivatives
The present invention relates to novel substituted imide derivatives of the general formula (I) in whichR1 represents optionally substituted cycloalkyl,R2 represents optionally substituted alkyl or...
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6706761 |
Dyed compositions containing insecticides
The invention relates to insecticide-comprising polymer-based compositions which, in order to recognize the point in time when the insecticide is exhausted, comprise at least one dye which, after...
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6638979 |
Imidamide derivatives
The present invention relates to novel imidamide derivatives of the formula (I) in whichR, R1, R2 and R3 are each as defined in the description, to a process for their preparation and to their use...
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6599920 |
Naphthalene compounds, intermediates, formulations, and methods
This invention relates to the field of pharmaceutical and organic chemistry and provides naphthalene compounds, intermediates, formulations, and methods.
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6555138 |
Polyethylene glycol matrix pellets for greasy, oily or sticky drug substances
A drug delivery system for oral administration in solid dry form of greasy/oily/sticky substance(s) and pharmaceutically active substance(s) or pharmaceutically active substance(s) which...
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6423748 |
Amido polybiguanides and the use thereof as antimicrobial agents
Amido polybiguanides and their use as antimicrobial agents in pharmaceutical compositions are disclosed. A method of synthesis of amido polybiguanides is also disclosed. The amido polybiguanides...
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6262122 |
Enantiomers of 4-[[(cyanoimino) [(1,2,2-trimethylpropyl)amino]methyl]amino]benzonitrile
The (R)-enantiomer of 4-[[(cyanoimino)-[(1,2,2-trimethylpropyl)amino]methyl]amino]
-benzonitrile as well as the corresponding (S)-enantiomer are useful for promoting hair growth such as in male...
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6194464 |
Imidic acid derivatives and their use as pesticides
The present invention relates to new imidic acid derivatives of the formula (I) ##STR1##to a plurality of processes for their preparation, and to their use as pesticides.
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6147098 |
Substituted guanidines and diaminonitroethenes, their preparation and use
Guanidine and diaminonitroethene derivatives represented by the formula ##STR1## wherein X, R1, R2, R3 and R4 are defined in the description, compositions thereof and methods for preparing the...
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6054411 |
Cyanamide aqueous solution
Addition of a dicarboxylic acid such as adipic acid to a cyanamide aqueous solution brings about improvement in storage stability of the cyanamide aqueous solution.
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5998442 |
Benzo [B] thiophene compounds, and compositions for treating bone loss, and hyperlipidemia
The invention provides benzo[b]thiophene compounds, formulations, and methods of inhibiting bone loss or bone resorption, particularly osteoporosis, and cardiovascular-related pathological...
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5922693 |
Cleaning compositions containing biostatic agent
The present invention relates to an aqueous cleaning composition containing (a) 1 to 10 weight % of at least one surfactant selected from the group consisting of anionic surfactants and ethoxylated...
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5594033 |
Secoaporphine compound on arrhythmia
Novel secoaporphine compounds having the formula I ##STR1## wherein a) R1, R2 and R3, R4 are each methyl group; or b) R1, R2, and R4 are each methyl group; R3 is benzyl, ethyl or allyl; or c) R1,...
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5430059 |
Butenoic acid derivatives
A butenoic acid compound of the following formula: ##STR1## in which Z is O, S, vinylene or azomethyne, A is an alkylene group and J is phenyl group, is a useful in treating heart disease.
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5262419 |
Method for the prophylaxis and/or treatment of ulcerative gastrointestinal conditions using a potassium channel activator
Ulcerative conditions of the gastro-intestinal tract, e.g., antiinflammatory-drug-induced ulcers, are treated or prevented by the administration of a potassium channel activator. Methods and...
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5087640 |
Novel cyanoguanidine derivatives
Compounds of the formula: ##STR1## wherein R1 and R2 are independently fluorine, chlorine or bromine atom, and R3 is a C4 -C7 alkyl having at least a branch at the C1 position, exhibit K+ channel...
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5021429 |
Pharmacologically active aminoalkylphenyl compounds and their use
Compounds of the general formula: ##STR1## and physiologically acceptable salts, and hydrates, N-oxides and bioprecursors of such compounds and such salts in which R1 and R2, which may be the same...
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5011837 |
Aryl cyanoguanidines: potassium channel activators and method of making same
Novel compounds of the formula ##STR1## and tautomers thereof, wherein at least one of R2, R3 and R4 is a strong electron withdrawing group, are disclosed. These compounds possess potassium channel...
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5006523 |
Antiarrhythmic agents: aryl cyanoguanidine potassium channel blockers
Novel compounds of the formula ##STR1## and tautomers thereof are disclosed. These compounds possess potassium channel blocking activity and, as such, are useful as antiarrhythmic agents.
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4943307 |
Plant-protective pesticidal composition
The invention relates to a plant-protective solution containing 2.5 to 40 % by weight of one or more water-insoluble plant-protective ingredient(s) 20 to 71.5 % by weight of dimethylformamide...
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4871756 |
Leukotriene antagonists
Compounds having the formula: ##STR1## are antagonists of leukotrienes of C4, D4, E4 and the slow reacting substance of anaphylaxis.As such, these compounds will be useful as anti-asthmatic,...
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4870056 |
Acylated cyanamide composition
Acylated cyanamide compounds useful for ethanol deterrence of the formula RCONHCN, wherein R is a lipophilic acyl group or is derived from an (N-substituted)-alpha-aminoacyl group.
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4857550 |
Novel insecticidal dibenzoyl-tert-butylcarbazonitrile compounds and method for the preparation thereof
The present invention provides novel insecticidal dibenzoyl-tert-butylcarbazonitrile compounds and a method for the preparation thereof. It also provides methods for controlling insects with said...
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4810725 |
1-aryloxy-3-(substituted aminoalkylamino)-2-propanols, pharmaceutical compositions and use
1-Aryloxy-3-(substituted aminoalkylamino)-2-propanols and pharmaceutically acceptable salts thereof have β-adrenergic blocking activity with some cardioselectivity and hence are useful as ...
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4782073 |
Amides of [(5,6-dichloro-3-oxo-9-alpha-substituted-2,3,9,9-alpha-tetrahydrofluoren -7-yl-oxyl]acetic acids, and pharmaceutical compositions thereof
The invention relates to novel amides of [(5,6-dichloro-3-oxo-9a-substituted-2,3,9,9a-tetrahydrofluor
en-7-yl)oxy]ac etic acids, their derivatives, and their salts. The compounds are useful for the...
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4726941 |
Acylated cyanamide composition for treating ethanol ingestion
Acylated cyanamide compounds useful for ethanol deterrence of the formula RCONHCN, wherein R is a lipophilic acyl group or is derived from an (N-substituted)-alpha-aminoacyl group.
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4692467 |
N'-cyano-n-tetrahydrownaphthyl-s-methyisothiourea as a growth promoting agent
This invention relates to novel cyanoguanidine compounds and the intermediate N'-cyano-N-(1,2,3,4-tetrahydro-1-naphthyl)-S-methylisothiour
ea. These novel compounds are useful as animal growth...
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4689348 |
Cyanoguanidines useful as animal growth promoting agents
This invention relates to novel cyanoguanidine compounds and the intermediate N'-cyano-N-(1,2,3,4-tetrahydro-1-naphthyl)-S-methylisothiour
ea. These novel compounds are useful as animal growth...
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4661520 |
Cyanoguanidine useful as an animal growth promoting agent
This invention relates to a novel cyanoguanidine compound, N'-cyano-N-(1,2,3,4-tetrahydro-1-naphthyl)guanidine, which is useful as an animal growth promoting agent.
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4659721 |
Alkanol derivatives, and pharmaceutical preparation containing these compounds
Alkanol derivatives corresponding to the general formula I R1 R2 N--(CH2)m --Q--CH2 X--CH2 --Y--(CH2)n --NHR3 (I)which have a highly selective action on histamine-H2 receptors are described. Due to...
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4568694 |
Growth-enhancing cystamine derivatives
Cystamine derivatives of the formula: ##STR1## [wherein n represents 2 or 3, R1 and R2 each represents a hydrogen atom, or an alkyl group optionally substituted by a hydroxy, amino, alkylamino or...
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4543352 |
Naphthalene aminoalkylene ethers and thioethers, and their pharmaceutical uses
A class of naphthalene aminoalkylene ether and thioether compounds exhibiting pharmacological activity including anti-secretory and anti-ulcerogenic activity, pharmaceutical compositions comprising...
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4524152 |
1-Cyano-3-(fluoroalkyl)guanidines for lowering blood pressure
1-Cyano-3-(fluoroalkyl)guanidines of the formula: ##STR1## in which R1, R2 and R3 are the same or different members of the class of hydrogen, fluorine, lower alkyl or lower alkenyl provided that at...
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4407816 |
3-Substituted-2-propenimidamides and method of manufacturing the same
New derivatives of 3-furyl-, 3-thienyl- and 3-phenyl-2-propenimidamides are disclosed, which are useful as anti-ulcer agents. These new compounds are synthesized by reacting an imino ether derived...
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4366164 |
Amine derivatives
The invention provides compounds of general formula ##STR1## and physiologically acceptable salts, hydrates and bioprecursors thereof, in which Y and Z, which may be the same or different, each...
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4332822 |
Guanidine derivatives
Novel cyanoguanidine derivatives having the formula ##STR1## wherein Ar is a phenyl or pyrrol-1-yl group substituted by one or more substituents selected from halogen, trifluoromethyl, lower alkyl,...
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4279911 |
Amine derivatives and pharmaceutical compositions containing them
The invention relates to compounds of the general formula (I) ##STR1## and physiologically acceptable salts, N-oxides, hydrates and bioprecursors thereof, in which Y represents O, S, CHNO2 or N...
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4202903 |
Acyl cyanoguanidines for treating rheumatoid arthritis
Certain novel acyl cyanoguanidines, their preparation, pharmaceutical compositions and novel methods of treating inflammation and autoimmune diseases such as rheumatoid arthritis are disclosed.
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