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7226948 |
Treatment of neurodegenerative conditions with nimesulide
The present invention relates to the use of nimesulide and structurally related compounds in the prevention and/or treatment of neurodegenerative conditions. It is based, at least in part, on the...
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7115624 |
Method of inhibiting protein tyrosine phosphatase 1B and/or T-cell protein tyrosine phosphatase 4 and/or other PTPases with an Asp residue at position 48
The present invention provides a method of inhibiting a member of a family of Protein Tyrosine Phosphatases (PTPases, PTPs) such as PTP1B, TC-PTP, CD45, SHP-1, SHP-2, PTPα, PTPε, PTPμ, PTPδ,...
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6476011 |
Methods for introducing an estrogenic compound
The invention pertains to methods for introducing an estrogenic compound into a subject in need thereof involving administering an effective amount of a ring system compound having the formula (II)...
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6436925 |
Substituted benzamides, their production and their use as cysteine protease inhibitors
Benzamides of the formula I and its tautomeric forms, possible enantiomeric and diastereomeric forms, E and Z forms, and possible physiologically tolerated salts, in which the variables have the...
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6432986 |
Compositions, kits, and methods for inhibiting cerebral neurovascular disorders and muscular headaches
Methods, kits, and compositions for inhibiting a cerebral neurovascular disorder or a muscular headache in a human patient are provided. The methods comprise intranasally administering to the...
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6391918 |
N-sulphonyl and N-sulphinyl phenylglycinamide
Novel α-amino acid amides of formula (I) as well as possible isomers and mixtures of isomers thereof, wherein the substituents are defined as follows: n is the number zero or one; R 1 is...
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6387954 |
Alkenyl sulphonamide derivatives
The present invention provides certain alkenyl sulphonamide derivatives useful for potentiating glutamate receptor function in a mammal and therefore, useful for treating a wide variety of...
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6057322 |
Basically-substituted benzoylguanidines, a process for preparing them, their use as a medicament or diagnostic agent, and a medicament containing them
Compounds of the formula I ##STR1## and the pharmaceutically tolerated salts thereof, are described. A process for their preparation and their use as medicaments in cardiovascular diseases are also...
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6031003 |
Calcium receptor-active molecules
The present invention relates to the different roles inorganic ion receptors have in cellular and body processes. The present invention features: (1) molecules which can modulate one or more...
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5756498 |
Sulfonylalkanoylamino hydroxyethylamino sulfonyl urea derivatives useful as retroviral protease inhibitors
Sulfonylalkanoylamino hydroxyethylamino sulfonyl urea derivative compounds are effective as retroviral protease inhibitors, and in particular as inhibitors of HIV protease. In accordance with the...
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5708034 |
Substituted sulfonimidamides, processes for their preparation, their use as a medicament or diagnostic, and medicament comprising them
Substituted sulfonimidamides, processes for their preparation, their use as a medicament or diagnostic, and medicament comprising them Sulfonimidamides of the formula I ##STR1## in which at least...
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5607931 |
1,2-disubstituted ethly amides as inhibitors of ACAT
Amides of the formula ##STR1## wherein: R 1 is A and R 2 is B; R 1 is B and R 2 is A; or R 1 and R 2 are independently selected from the group B; A is phenyl, substituted phenyl,...
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5470834 |
Sulfoximine and suldodiimine matrix metalloproteinase inhibitors
Novel sulfoximine and sulfodiimine matrix metalloproteinase inhibitors of the formula, ##STR1## wherein: R 1 is selected from the group consisting of lower-alkyl, hydroxy lower-alkyl, amino...
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5459149 |
Penta-2,4-dienamides and use as pesticides
The present Application discloses pesticidally active compounds of formula (I): Q(CH 2 ) a (O) b Q 1 CR 2 =CR 3 CR 4 =CR 5 CXNR 1 R x or a salt or propesticide thereof, wherein Q is an...
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5368867 |
Process for the accelerated production of stable solutions, in equilibrium, of peracetic acid in low concentrations
The production of dilute equilibrium, storage stable solutions of peracetic acid from mixtures of aqueous hydrogen peroxide and acetic acid, or by dilution of more concentrated peracetic acid...
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5270043 |
Arthropodicidal composition comprising thiodicarb and a phenylpyrazole
The invention provides arthropodicidal compositions comprising an arthropodicidally effective amount of (A) 5-amino-3-cyano-1-(2,6-dichloro-4-trifluoromethylphenyl)-4-t
rifluoromethyl...
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5258406 |
Sulfonimidamides
This invention provides certain sulfonimidamide compounds, formulations and method of use of these compounds in treating susceptible neoplasms.
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4402980 |
Sulphonic acid cycloalkylamides and their use as microbicides
A N-sulphenylated sulphonic acid cyclohexylamide of the formula ##STR1## wherein R 1 denotes lower alkyl, chloroalkyl or dialkylamino, R 2 denotes a cycloalkyl radical which is optionally...
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4309425 |
Miticidal, insecticidal, ovicidal and fungicidal N-(N',N'-diarylaminothio)sulfonamides
Sulfonamides, such as N-[N-(2-chloro-5-(trifluoromethyl)phenyl]-N-[2,4-dinitro-6-(
trifluoromethy l)phenyl]aminothio]-N,4-dimethylbenzenesulfonamide, are useful for control of arthropod pests of...
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4105795 |
Antispasmodic substituted sulphoximides
This invention provides compounds of the general formula I ##STR1## wherein R 1 and R 2 independently represent groups selected from the group consisting of straight chain alkyl groups; branched...
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4066765 |
Arthropodicidal formamidines
Novel pesticidal compounds of the formula: ##STR1## wherein R 1 is lower alkyl of from 1 to 4 carbon atoms; R 2 is hydrogen, halogen or lower alkyl of from 1 to 4 carbon atoms; R 3 and R 4 are...
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4020153 |
Cyclic sulphonamides and sulphinamides having a physiological cooling effect
Compositions are disclosed having a physiological cooling action on the skin. The compositions contain, as the active ingredient certain cyclic sulphonamides and sulphinamides.
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4004031 |
Bis-(O-1-alkylthio-ethylimino)-N-methyl-carbamic acid)-N,N'-sulphide insecticides
Compounds of the formula I ##STR1## wherein R represents a C 1 -C 5 -alkyl radical their manufacture and their use as pest control agents.
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3947591 |
Pesticidal N,N"-thio and dithio bis(substituted phenyl formamidines)
Novel pesticidal compounds of the formula: ##SPC1## Wherein R 1 and R 2 are the same or different and are selected from the group consisting of lower alkyl of from 1 to 4 carbon atoms; R 3 and R...
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3249497 |
Solubilization of water-insoluble quaternary ammonium benzosulfimides
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