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7572461 |
Borer-resistant wood, wood products, and wooden structures and methods
The invention provides methods for suppressing the degradation of wood, wood products, and wooden structures due to infestation by wood-boring organisms, by use of a polyurea composition. The...
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7511074 |
Tetrafluorobenzyl derivatives and pharmaceutical composition for preventing and treating acute and chronic neurodegenerative diseases in central nervous system containing the same
The present invention relates to a tetrafluorobenzyl derivative and a pharmaceutical composition for prevention and treatment of acute and chronic neurodegenerative disease in central nervous...
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7510722 |
Apparatus for dispensing a bird haze product from a can
An aerosol tiny mist hazer apparatus. The apparatus has an aerosol can that contains about 10% by weight Methyl Anthranilate oil and about 90% by weight of an isobutane and propane propellant...
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7459585 |
Benzene derivatives and pharmaceutical use thereof
The present invention provides an AP-1 activation inhibitor, NF-kappa B activation inhibitor, inflammatory cytokine production inhibitor, matrix metalloprotease production inhibitor, inflammatory...
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7273887 |
Topical anesthetic formulation
The topical anesthetic formulation of the present invention is typically a solution that preferably includes lidocaine, USP as the active anesthetic ingredient with benzyl alcohol and isopropyl...
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7247654 |
3,4-disubstituted benzamidines and benzylamines, and analogues thereof, useful as serine protease inhibitors
The present invention relates generally to compounds that inhibit serine proteases. In particular it is directed to novel 3,4-disubstituted benzamidines and benzylamines, or a stereoisomer or...
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7153869 |
Substituted amino acids as erythropoietin mimetics
This invention relates to a series of substitituted amino acids of Formula I
pharmaceutical compositions containing them and intermediates used in their manufacture. The compounds of the...
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7074820 |
Amidino derivatives and their use as thrombin inhibitors
There is provided compounds of formula I,
wherein R 1 , R 2 , R 3 , Y, n and B have meanings given in the description which are useful as competitive inhibitors of trypsin-like proteases, such...
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7034015 |
Aminobenzoephenones
The invention relates to a novel class of aminobenzophenones derivatives, to pharmaceutical preparations comprising said compounds, to dosage units of such preparations, to methods of treating...
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6964982 |
Compounds, compositions and methods for preventing neurodegeneration in acute and chronic injuries in the central nervous system
The present invention provides compositions and methods for prevention and prophylaxis of neurological diseases accompanied by neuronal death. The invention includes synthesis of 5-benzylamino...
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6964782 |
Stable hydrogen peroxide compositions, products and methods of use
Disclosed are several preferred embodiments of hydrogen peroxide which are packaged with ease of use and extended shelf-life in mind. The embodiments include foam, mist, gel, and disposable...
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6958146 |
Compounds to affect insect behavior and to enhance insecticides
Various exemplary compounds, compositions and methods are disclosed. An exemplary composition includes an insecticide comprising a formula weight greater than approximately 220 and a compound...
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6951844 |
Phenyl naphthol ligands for thyroid hormone receptor
New thyroid receptor ligands are provided which have the general formula I
wherein R 1 is halogen, trifluoromethyl, substituted or unsubstituted aryl, substituted or unsubstituted C 1-6 ...
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6949585 |
Cyclooctanone derivatives and cyclodecanone derivative, and use thereof
The present invention provides a compound which has cytokine production inhibitory activity and is useful for the treatment of diseases which is associated with cytokine. The compound is...
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6949575 |
Method of inhibiting amyloid protein aggregation and imaging amyloid deposits using aminoindane derivatives
The present invention provides compounds of Formula (I) and a method of treating Alzheimer's disease using a compound of Formula (I), wherein: R 1 and R 2 include alkyl and phenylalkyl; R 3 is...
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6946474 |
Nitrogen-containing compounds and their use as glycine transport inhibitors
The present invention provides trichloroethyl-sulfonylurea-containing compounds that inhibit glycing transporters, pharmaceutical compositions comprising such compounds, methods for using such...
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6943191 |
Disubstituted lavendustin A analogs and pharmaceutical composition comprising the analogs
Disubstituted lavendustin A analogs that are PTK inhibitors having antiproliferative activity are described. Preferred compounds of the disclosure, without limitation, satisfy either Formula 1 or...
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6921539 |
Antimicrobial therapeutic compositions and method of use
The invention provides therapeutic antimicrobial compositions and methods for their use based on natural organic phenolic compounds combined with pharmacological agents. The antimicrobial...
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6916837 |
Amidino derivatives and anticoagulants and thrombosis therapeutic agents containing them
Amidino derivatives represented by the following general formula (I):
{where X is a group represented by R 1 SO 2 NR 2 — (wherein R 1 represents optionally substituted C 6-14 aryl, etc....
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6897236 |
Aminobenzophenones as inhibitors of IL-1β and TNF-α
The present invention relates to compounds of formula (I) wherein R 1 , R 2 and R 3 independently represent one or more, same or different substituents selected from the group consisting of...
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6881756 |
Method for treating skin disorders
The present invention relates to a method for reducing inflammation in the skin and/or treating inflammatory skin disorders, pain, or pruritis by topically applying a composition comprising totarol...
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6861449 |
Method of treating neutrophil-related diseases with topical anesthetics
A therapeutic method is provided to treat neutrophil-associated pulmonary diseases, such as chronic obstructive pulmonary disease, by locally administering to a mammal in need of such treatment, an...
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6844003 |
Compounds derived from benzoic acid esters, composition containing said compounds and use thereof
The invention relates to novel compounds of formula (I) wherein R 1 represents a polymer, aryl or alkyl group, R 2 presents a hydrogen atom, a halogen atom, a radical CN, CF 3 , OH, OCF 3 , COOH,...
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6838472 |
Substituted urea retinoid agonists
The current invention provide novel compounds, methods of treating or preventing emphysema, cancer and dermatological disorders, pharmaceutical compositions suitable for the treatment or prevention...
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6790866 |
Sulfonamide and carboxamide derivatives and drugs containing the same as the active ingredient
The sulfonamide or carboamide derivatives of the formula (I) and a pharmaceutical composition which comprise them as an active ingredient: (wherein A ring, B ring is carbocyclic ring,...
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6787562 |
Substituted aryl and heteroaryl compounds as E-type prostaglandin antagonists
Compounds of the formula I; useful for the treatment of pain wherein A, Z, B, R 1 , X and D are as defined in the specification, methods of making such compounds, methods of using such compounds...
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6759434 |
Anti-infective compositions, methods and systems for treating disordered tissue
The present invention relates to the treatment of disordered epithelial tissues such as cold sores and other complications resulting from disorders such as herpes, and the like. The invention...
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6734212 |
Methods and compositions for treating or preventing bacterial infection
The invention relates to compositions and methods for treating or preventing disease or disorders caused by or associated with certain bacterial infection, especially Escherichia coli ( E. coli )...
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6730329 |
Zinc containing compositions for anti-viral use
One aspect of the invention relates to anti-viral composition containing at least one zinc compound and at least one phenolic antioxidant (and optionally other ingredients such as at least one...
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6713511 |
Fatty acid derivatives
The invention relates to a novel acylate which is the reaction product of (a) a substance which is selected from the group consisting of naturally occuring alpha-aminocarboxylic acids,...
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6699904 |
PPAR agonists
PPAR alpha activators, pharmaceutical compositions containing such compounds and the use of such compounds to elevate certain plasma lipid levels, including high density lipoprotein-cholesterol and...
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6696440 |
Treatment of asthma with MEK inhibitors
This invention provides a method of preventing or treating asthma by administering to a patient in need of treatment an effective amount of a selective MEK inhibitor, especially a phenyl amine of...
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6673788 |
Electrophilic ketones for the treatment of herpesvirus infections
A class of compounds is described which can be used for the treatment of viral infections. Compounds of particular interest are defined by Formula II: wherein each of R 1 , R 2 , and R 3 is...
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6670400 |
Phenoxyethylamine derivatives having high affinity for the 5-HT1A receptor, preparation thereof, use thereof as drugs, and pharmaceutical compositions containing said derivatives
Phenoxyethylamine derivatives of general formula (I) having high affinity for the 5-HT 1A receptor, methods for preparing same, pharmaceutical compositions containing said derivatives, and their...
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6649656 |
Anthranilic acid derivatives
The present invention relates to an anthranilic acid derivative expressed by the following formula (1) or the following formula (2), or its pharmacologically permissible salt or solvate.
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6646003 |
Method of treating ocular inflammatory and angiogenesis-related disorders of the posterior segment of the eye using an amide derivative of flurbiprofen or ketorolac
The topical use of certain flurbiprofen amide derivatives and ketorolac amide derivatives to treat ophthalmic angiogenesis-related and inflammatory disorders of the posterior segment of the eye is...
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6620852 |
Topical anesthetic
The present invention is directed to an improved flowable anesthetic composition that does not need to be applied by an applicator. The anesthetic composition of the present invention may be...
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6589986 |
Methods of treating anxiety disorders
This invention provides methods for treating, preventing or inhibiting anxiety, anxiety-related conditions and phobias in a mammal using compounds of the formula: wherein: R 1 is H, alkyl,...
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6569901 |
Alkynyl-substituted propionic acid derivatives, their preparation and use
The present invention relates to compounds of formula (I) The compounds are useful in the treatment and/or prevention of conditions mediated by nuclear receptors, in particular the Peroxisome...
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6562326 |
Topical composition for burn healing
A method of treating skin includes applying a topical composition to an affected area of skin, such as a burn, irritation, blister, rash or other similar skin condition. The topical composition has...
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6555578 |
Thyromimetic antiobesity agents
The invention relates to pharmaceutical compositions and methods useful in the treatment of obesity which methods comprise administering to animal, including a human or companion animal, in need of...
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6552083 |
Agents inhibiting chronic rejection reactions after organ transplantation
The present invention relates to an agent for inhibiting diseases associated with chronic rejection after organ transplantation, such as transplanted heart-accelerated coronary arteriosclerosis,...
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6545018 |
Oxamic acids and derivatives as thyroid receptor ligands
The present invention provides novel compounds of the Formula and prodrugs thereof, geometric and optical isomers thereof, and pharmaceutically acceptable salts of such compounds, prodrugs and...
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6534048 |
Topical clonidine preparation
An aqueous gel in unit dose form and suitable for topical delivery of clonidine and comprising clonidine, a water-gelling amount of a pharmaceutically acceptable gelling agent and having a pH value...
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6524623 |
Therapeutic compositions and methods of use thereof
A therapeutic composition and a method of using the composition are provided. The composition includes an osmotic agent and an active agent. The osmotic agent improves the delivery of the active...
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6506798 |
4-Arylamino, 4-aryloxy, and 4-arylthio diarylamines and derivatives thereof as selective MEK inhibitors
The invention provides compounds of formula (II), wherein Ar, R 3 , R 4 , R 5 , R 6 , R 7 , R 8 and W have the meanings given in the description. They are selective MEK inhibitors.
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6500838 |
Treatment of stereotypic, self-injurious and compulsive behaviors in man and animals using antagonists of NMDA receptors
NMDA receptor antagonists can be used in methods of treatment, for reducing the frequency of stereotypic behaviors in animals and for reducing the frequency of analogous compulsive behaviors in...
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6489365 |
Amidine derivatives, the preparation and use thereof as medicaments with Itb4 antagonistic effect
Compounds of the formula which is explained more fully in the specification, may be prepared by conventional methods and used therapeutically in conventional galenic preparations.
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6472390 |
Use of therapeutic dosages for nitric oxide donors which do not significantly lower blood pressure or pulmonary artery pressure
Patients with pathologic conditions involving constriction or proliferation of smooth muscle or disease associated with cysteine containing proteins, or who are at risk for such, are administered a...
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6465514 |
Methods and compositions for the promotion of hair growth
Compositions, medicaments, and methods for the promotion of hair growth are disclosed. These compositions and medicaments are comprised of either local anesthetics of the secondary or tertiary...
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