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7498311 |
Treatment of migraine
A method for treating migraine in non-epileptic subjects which involves administering to subjects an effective amount of a pharmaceutical composition comprising a sulfamate of the following formula:
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7479507 |
Anti-inflammatory substituted phenols and elastomeric compositions for oral delivery of drugs
3,5-di-substituted-4-hydroxybenzylidene phosphonates and sulfonates useful in treating inflammatory disease, particularly osteoarthritis, and elastomeric particles for oral delivery of drugs are...
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7459585 |
Benzene derivatives and pharmaceutical use thereof
The present invention provides an AP-1 activation inhibitor, NF-kappa B activation inhibitor, inflammatory cytokine production inhibitor, matrix metalloprotease production inhibitor, inflammatory...
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7351695 |
Topiramate salts and compositions comprising and methods of making and using the same
The invention encompasses novel salts of topiramate, and pharmaceutically acceptable polymorphs, solvates, hydrates, dehydrates, co-crystals, anhydrous, or amorphous forms thereof, as well as...
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7351427 |
Pharmaceutical composition, a method of preparing it and a method of treatment by use thereof
Pharmaceutically acceptable liposome-encapsulated busulphan formulations for parenteral administration are provided, as well as such formulations furthermore comprising glutathione and/or at least...
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7268152 |
Glucocorticoid mimetics, methods of making them, pharmaceutical compositions, and uses thereof
Compounds of Formula (IA) and Formula (IB)
wherein R 1 , R 2 , R 3 , R 4 , R 5 , and R 6 are as defined herein for Formula (IA) or Formula (IB), or a tautomer, prodrug, solvate, or salt...
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7244762 |
Antitumoral d-homoestra-1,3,5 (10)-trien-3-yl 2-substituted sulfamates
This invention relates to 2-substituted D-homo-estra-1,3,5(10)-trien-3-yl sulfamates of general formula I (I), in which R3 means a C1-C5-alkyl or C1-C5-alkyloxy group as well as their use for the...
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7235590 |
Use of treosulfan and derivatives thereof for treating multiple sclerosis
The invention relates to the use of treosulfan and/or derivatives thereof for producing a pharmaceutical composition used in the treatment of multiple sclerosis.
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7199081 |
Aqueous compositions for seed treatment
An aqueous composition suitable for applying fungicides to plant propagation materials is provided, comprising water and a blend of the following components, by weight:
a) 2–10% of a...
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7183317 |
Compounds and methods to increase plasma HDL cholesterol levels and improve HDL functionality
It has been discovered that certain selected ethers of probucol, and their pharmaceutically acceptable salts or prodrugs, are useful for increasing circulating HDL cholesterol. These compounds may...
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7176192 |
Method for treating patients for radiation exposure
This invention relates to a method of treating a patient suffering from ionizing radiation exposure, or of treating a patient about to undergo ionizing radiation therapy. The method includes...
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7173019 |
Linked cyclitols and their polysulfated derivatives
The invention relates to compounds of the following formula (I). In these compounds, R 1 , R 2 , R 3 and R 4 are each independently a substituted or unsubstituted cyclitol with a ring comprising...
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7153877 |
Method and composition for preventing or reducing the symptoms of insulin resistance syndrome
A method for preventing and or reducing the symptoms of insulin resistance and a related syndrome in persons comprises identifying persons having or at risk for having such symptoms, and...
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7119110 |
Method and composition for preventing or reducing the symptoms of insulin resistance syndrome
A method for preventing and or reducing the symptoms of insulin resistance and a related syndrome in persons comprises identifying persons having or at risk for having such symptoms, and...
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7112608 |
Hydroxyphenylundecane, a process for their production and their use
The present invention relates to novel hydroxyphenylundecane derivatives of the formula (I),
a method for the preparation of said compounds by cultivation of the fungus Cryphonectria...
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7109174 |
Anticonvulsant derivatives useful for preventing the development of type II diabetes mellitus and syndrome X
Anticonvulsant derivatives useful for preventing the development of Type II diabetes mellitus and Syndrome X are disclosed.
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7053071 |
Induction of apoptosis in cancer cells
The present invention provides compounds that are inducers or inhibitors of apoptosis or apoptosis preceded by cell-cycle arrest. In addition, the present invention provides pharmaceutical...
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7044624 |
Vehicle light with movable reflector portion and shutter portion for selectively switching an illuminated area of light incident on a predetermined portion of the vehicle light during driving
A vehicle light can include a light source, a major reflecting surface, a projection lens, and a shutter. A first reflecting surface of an ellipse group reflecting surface preferably has a first...
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7018983 |
Treatment of migraine
A method for treating migraine in non-epileptic subjects which involves administering to subjects an effective amount of a pharmaceutical composition comprising a sulfamate of the following formula:
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6955812 |
Health food and preparation having an anti-obesity effect
The present invention discloses an anti-obesity agent comprising:
D-cysteinolic acid represented by Formula I, as an active ingredient: Formula I:
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6921774 |
Compounds and their use as glycine transport inhibitors
The invention provides novel compounds of the formula I below:
wherein the meaning of each substituent is defined in the application. The compounds are useful as inhibitors of the glycine...
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6858649 |
Selective potentiation of serotonin receptor subtypes
The selective potentiation and/or inhibition of the 5-HT 2A and/or 5-HT 1A response to serotonin (5-HT) is achieved using analogs of oleamide. Selective potentiation and/or inhibition of the 5-HT...
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6852755 |
Nitrogen mustard compounds and prodrugs therefor
This invention pertains to nitrogen mustard compounds (Formula (II)) and prodrugs therefor (Formula (I)), methods for their preparation, pharmaceutical compositions comprising such compounds, and...
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6852701 |
Anticonvulsant derivatives useful for preventing the development of Type II diabetes mellitus and Syndrome X
Anticonvulsant derivatives useful for preventing the development of Type II diabetes mellitus and Syndrome X are disclosed.
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6750252 |
Tri-substituted phenyl derivatives and analogues
The present invention relates to certain tri-substituted phenyl derivatives and analogues of formula (I), to a process for preparing such compounds, having the utility in clinical conditions...
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6727279 |
Arylsulphonamides and analogues
The present invention relates to novel arylsulphonamides and analogues, to processes for their preparation and to their use for the prophylaxis and treatment of neurodegenerative disorders, in...
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6699840 |
Controlled- or delayed-release forms of topiramate
The invention encompasses novel salts of topiramate, and pharmaceutically acceptable polymorphs, solvates, hydrates, dehydrates, co-crystals, anhydrous, or amorphous forms thereof, as well as...
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6649621 |
Prevention or reversal of sensorineural hearing loss (SNHL) through biologic mechanisms
The invention presents methods for preventing and treating sensorineural hearing loss and is directed to the restoration or protection of hair cells in individuals experiencing a non-presbycusis...
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6649182 |
Planting method and biodegradable material for preventing pests
A planting method for preventing pests, especially snails, is disclosed. The method includes the steps of (a) providing a biodegradable material, (b) adding a pesticide into the biodegradable...
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6641830 |
Deer repellent
A deer repellent to deter deer from eating trees, shrubs and plants. The deer repellent is a mixture of milk, eggs, corn oil and sodium lauryl sulfate. The mixture is blended and applied to the...
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6630509 |
Phenalkyloxy-phenyl derivatives
The present invention relates to certain phenalkyloxy-phenyl derivatives of formula (I) and analogs, to a process for preparing such compounds, which compounds have utility in treating clinical...
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6627656 |
Method of treatment using phenyl and biaryl derivatives as prostaglandin E inhibitors and compounds useful therefore
This invention encompasses a method for the treatment or prevention of prostaglandin mediated diseases comprising administering to a mammalian patient a compound of formula I: in an amount that...
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6620819 |
Anticonvulsant derivatives useful in treating psychosis
The anticonvulsant derivative topiramate useful in treating dementia and/or behavioral and psychotic disturbances in dementia is disclosed.
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6596320 |
Method for treating cancer having greater efficacy and reduced adverse effects
A method of treating patients with cancer that involves administration of a combination regimen of a platinum agent, a taxane agent, and a formula I toxicity-reducing agent. The preferred order of...
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6593364 |
Triterpene derivatives and remedies for liver diseases
A triterpene derivative useful for the treatment of hepatic disorders is disclosed. This compound comprises as an active ingredient a triterpene derivative represented by the following formula (I)...
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6552000 |
Anticonvulsant derivatives useful in treating autism
Anticonvulsant derivatives useful in treating autism.
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6525091 |
Substituted diarylureas as stimulators for Fas-mediated apoptosis
Substituted diarylureas, pharmaceutical compositions containing them, and their use for stimulating Fas-mediated apoptosis. The compounds, as single stereoisomers or mixtures of stereoisomers,...
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6525037 |
Method of treating atherosclerosis and complications resulting therefrom
This invention relates to a method of treating patients afflicted with atherosclerosis or to prevent the development of atherosclerosis in patients assessed to be high risk of developing the...
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6503884 |
Migraine treatment method using topiramate and related compounds
A method for treating migraine in non-epileptic subjects which involves administering to subjects an effective amount of a pharmaceutical composition comprising a sulfamate of the following formula:
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6495595 |
Pesticide formulations containing alkoxylated tristyrylphenol hemi-sulfate ester neutralized alkoxylated amine surfactants
The present invention relates to a surfactant for general use in agricultural compositions, including, but not limited to herbicidal, fungicidal and insecticidal formulations comprised of two...
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6489359 |
Sulphoxybenzamides
The present invention relates to new sulphoxybenzamides of general formula I, processes for preparing them as well as their use as medicaments.
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6486198 |
Compounds and methods for the treatment of post traumatic stress disorder
The application relates to the use of topiramate and related sulfamates for the treatment and/or prophylaxis of post traumatic stress disorder (PTSD).
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6486129 |
Antithrombotic compounds
The present invention relates to compounds of formula (1), wherein R 1 is phenyl, naphthyl, 1,2,3,4-tetrahydronaphthyl, (iso)quinolinyl, tetrahydro(iso)quinolinyl, 3,4-dihydro-1H-isoquinolinyl,...
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6472370 |
Anticonvulsant derivatives useful in treating post traumatic stress disorder
Anticonvulsant derivatives useful in treating post traumatic stress disorder, are disclosed.
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6468993 |
Method for reducing development of osteoporosis
This invention relates to a method of treating patients afflicted with osteoporosis. The method includes administering to a patient in need of treatment an effective amount of a thiol or reducible...
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6465020 |
Use of garlic extract as both preventive and therapeutic agents for human prostate and bladder cancers
This invention is concerned with the clinical investigation of the therapeutic effects of garlic extracts containing allicin, diallyl disulfide, and diallyl trisulfide. The intake of garlic or...
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6455573 |
Glycosidase inhibitors and methods of synthesizing same
A method for synthesizing Salacinol, its stereoisomers, and non-naturally occurring selenium and nitrogen analogues thereof having the general formula (I): The compounds are potentially useful...
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6440938 |
Prevention and/or treatment of allergic conditions
The present invention relates to the use of an inhibitor of cysteine proteinase activity in conjunction with an inhibitor of any serine proteinase activity other than trypsin for the manufacture of...
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6429223 |
Modified forms of pharmacologically active agents and uses therefor
In accordance with the present invention, there are provided modified forms of nonsteroidal anti-inflammatory drugs (NSAIDs). Modified NSAIDs according to the invention provide a new class of...
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6414020 |
Amidino protease inhibitors
Amidino and benzamidino compounds, including compounds of the formula: wherein R 1 -R 4 , R 6 -R 9 , Y, Z, n and m are set forth in the specification, as well as hydrates, solvates or...
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