|
Match
|
Document |
Document Title |
|
|
7625948 |
Ester compound and medicinal use thereof
A novel therapeutic agent for hyperlipidemia, which is an ester compound represented by the formula (1″)
(wherein
R 1 and R 2 are each hydrogen atom or optionally substituted aryl,...
|
|
|
7576127 |
Aromatic prodrugs of propofol, compositions and uses thereof
Prodrugs of propofol, methods of making prodrugs of propofol, pharmaceutical compositions of prodrugs of propofol and methods of using prodrugs of propofol and pharmaceutical compositions thereof...
|
|
|
7538140 |
Ester compound and medicinal use thereof
A novel therapeutic agent for hyperlipidemia, which is an ester compound represented by the formula (1″)
(wherein
R 1 and R 2 are each hydrogen atom or optionally substituted aryl,...
|
|
|
7468360 |
Therapeutic amides and related compounds
Disclosed herein is a compound having a structure:
Therapeutic methods, compositions, and medicaments relating thereto are also disclosed.
|
|
|
7432392 |
Ester derivatives and medical use thereof
A therapeutic agent for hyperlipidemia which has no side effects on the liver unlike conventional MTP inhibitors and has excellent MTP inhibitory activity. Also, provided is an ester compound...
|
|
|
7427406 |
Aerosols
Cosmetic and/or pharmaceutical preparations comprising (a) a carbonate of the formula (I):
wherein R 1 is a linear alkyl and/or alkenyl group having from 6 to 22 carbon atoms, a 2-ethylhexyl,...
|
|
|
7241807 |
Prodrugs of propofol, compositions and uses thereof
The present invention provides propofol prodrugs, methods of making propofol prodrugs, pharmaceutical compositions of propofol prodrugs and methods of using propofol prodrugs and pharmaceutical...
|
|
|
7204994 |
Juvenile hormone compositions and methods for making same
The present invention relates to hormone coating layers having desirable hormone delivery characteristics and product lifetime. In one embodiment, the invention is a hormone composition including a...
|
|
|
7119246 |
Method of treating acne
This invention relates to a method for the treatment of acne that comprises applying a fluid comprising a polyalkylene carbonate over the area affected by acne and penetrating pores within the...
|
|
|
6875764 |
Urea and thiourea compounds useful for treatment of coccidiosis
The present invention relates to novel compounds, pharmaceutical compositions containing the same as well as a method for treatment of parasitic disorders, wherein said compounds are administered....
|
|
|
6864285 |
Covalent derivatives of alkanolamides of monocarboxylic and dicarboxylic acids functionally active on the CB2 cannabinoid receptor
The present invention relates to novel covalent derivatives of alkanolamides of monocarboxylic and dicarboxylic acids with aminoalcohols of general formula (I) which can usefully be used as...
|
|
|
6861448 |
NAD synthetase inhibitors and uses thereof
Disclosed are compounds that inhibit the microbial NAD synthetase enzyme. For example, disclosed are compounds of the formula Ar 1 —X—Ar 2 —Y—L—Z—Q, wherein Q is Q 1 Ar 3 or Ar 3 Q 1 ;...
|
|
|
6797504 |
Inhibitors of serine protease activity of matriptase or MTSP1
The present invention provides compounds which inhibit serine protease activity of matriptase or MTSP1. Also provided are pharmaceutical compositions comprising those compounds and methods of using...
|
|
|
6794384 |
Hydroxylation activated drug release
The present invention concerns prodrugs whose aromatic oxidation, particularly their enzymatic aromatic hydroxylation, results in their activation by the release of a drug moiety. It particularly...
|
|
|
6720306 |
Tetrapartate prodrugs
A compound of Formula I, providing tetrapartate prodrugs is provided wherein: L 1 is a bifunctional linking moiety; D is a moiety that is a leaving group, or a residue of a compound to be...
|
|
|
6683112 |
Gabapentin prodrugs and formulations
The present invention relates to novel prodrugs of gabapentin and to pharmaceutical formulations and sustained release formulations containing the prodrugs.
|
|
|
6667340 |
Inhibitors of phosphatidyl myo-inositol cycle
The present invention relates to the preparation and biological activity of 3-deoxy-Dmyo-inositol ether lipid analogs as inhibitors of phosphatidylinositol-3-kinase signaling and cancer cell...
|
|
|
6645978 |
Lipoxin A4 and its analogs for the treatment of dry eye
Ophthalmic compositions containing Lipoxin A 4 and its analogs and methods of their use for treating dry eve are disclosed.
|
|
|
6583175 |
Alkylxanthates and use of alkylxanthates in the integrated pest management
This invention relates to novel alkylxanthates of formulae 1 to 3 and use of alkylxanthates of formulae 1 to 6 in the integrated pest management, more specifically alkyl xanthates are used as...
|
|
|
6495152 |
Sulfur containing polyhydroxyalkanoate compositions and method of production
A class of biopolymer including sulfur in the form of a thioester in the polymer backbone or a thioether in the polymer side chains has been developed. These are preferably produced by fermentation...
|
|
|
6369103 |
Method for preventing or reducing risk of onset of cardiovascular events employing an HMG CoA reductase inhibitor
A method is provided for preventing or reducing the risk of onset of a cardiovascular event by administering an HMG CoA reductase inhibitor such as pravastatin, to a patient which has one or more...
|
|
|
6350724 |
Lice removing composition
The present invention provides a composition, and a method of use thereof, that is pesticide-free and yet is capable of cleansing an individual of a pest infestation. The composition of the present...
|
|
|
6335022 |
Nanoemulsion based on oxyethylenated or non-oxyethylenated sorbitan fatty esters, and its uses in the cosmetics, dermatological and/or ophthalmological fields
The present invention relates to a nanoemulsion, the oil globules of which have an average size of less than 100 nm, comprising (1) a surfactant which is solid at a temperature of less than or...
|
|
|
6262084 |
Compounds that inhibit the binding of integrins to their receptors
A method for the inhibition of the binding of α 4 β 1 integrin to its receptors, for example VCAM-1 (vascular cell adhesion molecule-1) and fibronectin; compounds that inhibit this binding;...
|
|
|
6251833 |
2-arylcyclopentan-1,3-diones
The present invention relates to novel 2-aryl-3-hydroxy-Δ 2 -cyclopentene-1-one derivatives of the formula (I) ##STR1## in which A, B, D 1 , D 2 , G, W, X, Y and Z are each as defined in the...
|
|
|
6248782 |
Method of treating viral diseases
A therapeutic process for treating disease in mammals caused by retroviruses in which the infected mammal is treated with a ribonucleotide reductase inhibitor such as a polyhydroxy benzoic,...
|
|
|
6201017 |
Ectoparasite controlling agent for animals
An ectoparasite-controlling agent for animals comprising 0.1 to 20% by weight of the neonocotinoid compounds defined in the specification and 10 to 95% by weight of a glycol or glycol monoalkyl...
|
|
|
6180095 |
Polymeric prodrugs of amino- and hydroxyl-containing bioactive agents
The present invention is directed to double prodrugs containing polymeric-based transport forms. These polymeric prodrugs are preferably of the formula: ##STR1## wherein: L 1 is a bifunctional...
|
|
|
6159988 |
Arylcycloalkyl derivatives, their production and their use
Compounds of formula I, ##STR1## and the physiologically tolerable salts thereof, wherein the substituents R 1 -R 4 have the meanings given in the specifications and show an activity against...
|
|
|
6124352 |
Antifungal agents
A method of treating fungal diseases as well as pharmaceutical, veterinary and agricultural compositions useful in such treatment. The method includes administering an effective antifungal amount...
|
|
|
6096773 |
Compounds that inhibit the binding of integrins to their receptors
A method for the inhibition of the binding of α 4 β 1 integrin to its receptors, for example VCAM-1 (vascular cell adhesion molecule-1) and fibronectin; compounds that inhibit this binding;...
|
|
|
6080784 |
Protein kinase C modulators N
Compositions with protein kinase C-modulatory, anti-inflammatory and other activities are disclosed.
|
|
|
6077866 |
Benzophenone hydrazone derivatives as insecticides
Novel benzophenonehydrazone derivatives represented by the formula (I): ##STR1## wherein, R 1 is halogen; R 2 is hydrogen or C 1 -4 alkyl; R 3 is cyano, optically substituted C 1 -4 alkyl, C 2...
|
|
|
6051590 |
Immunosuppressant tricyclic compounds
The compounds of Formula I are useful as immunosuppressive agents.
|
|
|
5994414 |
Water-thin emulsion formed by high pressure homogenization process
A stable, water-thin emulsion is formed by processing a crude emulsion through a high pressure homogenizer at a pressure of about 900 to about 1100 bar. This emulsion contains low levels of...
|
|
|
5981580 |
Fatty acid analogs and prodrugs
Novel derivatives of fatty acid analogs that have from one to three heteroatoms in the fatty acid moiety which can be oxygen, sulfur or nitrogen, are disclosed in which the carboxy-terminus has...
|
|
|
5972636 |
ATP-dependent protease and use of inhibitors for same in the treatment of cachexia and muscle wasting
The ATP-ubiquitin-dependent process has been shown to be responsible for the excessive protein degradation which occurs in conditions or disease states in which there is severe loss of body mass...
|
|
|
5968976 |
Pharmaceutical composition containing selected lanthanum carbonate hydrates
Selected lanthanum carbonate hydrates may be administered into the gastrointestinal tract, to treat hyperphosphataemia in patients with renal failure.
|
|
|
5955483 |
Stabilization of biocidal activity in air drying alkyds
This invention is directed towards stabilizing the biocidal activity of an alkyd composition containing a halopropargyl compound and a transition metal drier by use of a chelating agent.
|
|
|
5945449 |
Sterile bicarbonate concentrate
A sterile bicarbonate concentrate for use in the present invention relates to a sterile calcium-free bicarbonate concentrate for use in peritoneal dialysis, hemofiltration, cardiac bypass surgery...
|
|
|
5939455 |
Therapeutic augmentation of oxyalkylene diesters and butyric acid derivatives
This invention provides a method of augmenting the therapeutic activity of an oxyalkylene-containing compound, butyric acid, a butyric acid salt or butyric acid derivative by administering an...
|
|
|
5927283 |
Allosteric modifiers of hemoglobin
A family of compounds has been found to be useful for right-shifting hemoglobin towards a low oxygen affinity state. The effect has particular application in a wide variety of treatments including...
|
|
|
5925674 |
Cycloalkylcarboxanilides
This invention relates to cycloalkylcarboxanilides of the formula ##STR1## which are used to combat pests.
|
|
|
RE36253 |
Nail oil composition
A nail oil composition is disclosed consisting essentially of a cosmetic oil containing at least 5% by weight jojoba oil, said cosmetic oil having at least 1% by weight tolnaftate dissolved...
|
|
|
5902595 |
Pesticidal composition and method of use
The present invention provides a pesticidal composition with an extraordinarily lethal effectiveness that can also be used to remove and repel parasites, such as lice. The pesticidal composition...
|
|
|
5855903 |
Use of dimethyl substituted oxymethyl cyclohexane derivatives for their insect repellency properties
Described is a method of repelling Musca domestica L.(Diptera:Muscidae), Aedes aegypti, Culex nigripalpus, Aedes atlanticus, Culex salinarius, Aedes vexans, Culex spp., Simulium spp., Psoroferia...
|
|
|
5840658 |
Process for the controlled fixing of scale inhibitor in a subterranean formation
A process for fixing of a scale inhibitor in a subterranean formation, which comprises: a) injecting into the formation a solution comprising a polymeric scale inhibitor, a metal cation, a...
|
|
|
5827881 |
Diesters of carbonic acid endowed with antiviral and anti-inflammatory activity
Diesters of carbonic acid disubstituted with primary, secondary or tertiary amine groups, pharmaceutically acceptable salts thereof, and their use as antiviral and inti-inflammatory agents.
|
|
|
5798385 |
Insect repellent composition and method of using same to repel insects
Described is a composition which is both an insect repellent and a perfume containing: Para-isopropylcyclohexanol; 3,7-dimethyl-2,6-octadien-1-al; 5,9-dimethyl-4,8-decadienal; ...
|
|
|
5767141 |
Substituted propane derivatives, a process for their preparation and the use of the compounds for treating diseases
Substituted propane derivatives, a process for their preparation and the use of the compounds for treating diseases Propane derivatives of the formula I ##STR1## in which the radicals have the...
|