Patents in Class 514/487

Matches 1 - 50 out of 68

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Match	Document	Document Title
1	7829564	α- and β-amino acid hydroxyethylamino sulfonamides useful as retroviral protease inhibitors α-and β-amino acid hydroxyethylamino sulfonamide compounds are effective as retroviral protease inhibitors, and in particular as inhibitors of HIV protease.
2	7560483	Methods for synthesis of prodrugs from 1-acyl-alkyl derivatives and compositions thereof The present invention provides a method for synthesizing 1-(acyloxy)-alkyl derivatives from 1-acyl-alkyl derivatives, which typically proceeds stereospecifically, in high yield, does not require...
3	7262209	Carbonyloxy-cyanomethyl compounds as antiparasitic agents The invention relates to compounds of the general formula wherein Ar1, Ar2, R4, R5, R6, R7, R8, W, X, a and b have the significances given in the specification, and optionally the enantiomers...
4	6900213	Bisaryl derivatives having FSH modulatory activity The invention relates to bisaryl derivatives of the formula I, wherein (R,R) is selected from (H,H), O, (H,CH3), (H,OH) and (H,CN); Ar is substituted phenyl and A is a group of formula II, III, IV...
5	6852738	Acyl sulfamides for treatment of obesity, diabetes and lipid disorders A class of acyl sulfamides comprises compounds that are potent ligands for PPAR gamma and generally have antagonist or partial agonist activity. The compounds may be useful in the treatment,...
6	6726919	Injectable dispersion of propofol A sterile, injectable homogenized dispersion of micromatrices or microdroplets having a mean diameter from about 50 nm to about 1000 nm comprising about 1% to about 7.5% of propofol, about 1% to...
7	6696488	(Hydroxyethyl)ureas as inhibitors of alzheimer's β-amyloid production Novel (hydroxyethyl)ureas are described. These compounds are effective inhibitors of certain aspartyl proteases, notably secretases involved in the enzymatic cleavage of amyloid precursor protein...
8	6696497	Fungicidal mixtures A fungicidal composition comprises an acceptable carrier and/or surface active agent and a synergistically effective amount of (a) at least one benzophenone of formula I wherein R1, R2, R3, R4, R5,...
9	6573284	Method of treating melanoma Novel pro-drugs and assay reagents are provided which are useful as therapeutic agents especially for delivery and targetting therapeutically active agents to melanoma cells. The pro-drugs and...
10	6465457	Carbonate, carbamate, thiocarbonate dithiocarbonate and thiocarbomate derivatives useful as fungicides Fungicidal compounds of formula (I): wherein W is CH3O.CH═CCO2CH3, CH3ON═CCONR3R4 or CH3ON═CCO2CH3 and stereoisomers thereof; n is 0 or 1; X is oxygen or sulphur; Z is NR1; R1 is hydrogen or alkyl...
11	6416789	Synergistic combination of fungicides to protect wood and wood-based products from fungal decay, mold and mildew damage A wood treatment material having a synergistic combination of fungicides including boron-containing compounds, organo-iodine compounds and amine-oxides is provided. This combination is shown to be...
12	6143788	Bis-amino acid hydroxyethlamino sulfonamide retroviral protease inhibitors Selected bis-amino acid hydroxyethylamino sulfonamide compounds are effective as retroviral protease inhibitors, and in particular as inhibitors of HIV protease. The present invention relates to...
13	6114325	1,2-di-substituted benzene-carboxamide derivative, hair growth promoter and external composition for skin using the same A 1,2-di-substituted benzene-carboxamide derivative or a salt thereof expressed by the following Formula (I); ##STR1## wherein each of A and B is R1 or --(CH2)n-NR2 R3, wherein when A is R1, B is...
14	6077866	Benzophenone hydrazone derivatives as insecticides Novel benzophenonehydrazone derivatives represented by the formula (I): ##STR1## wherein, R1 is halogen; R2 is hydrogen or C1-4 alkyl; R3 is cyano, optically substituted C1-4 alkyl, C2-4 alkenyl,...
15	5811456	Monoamine oxidase B inhibitors, processes for their preparation and use thereof Novel monoamine oxidase B inhibitors of formula (I), wherein R1 H, an optionally substituted benzyloxy or phenylethoxy group; p=0-3; R3 H, a CN, OH, CCH group, a C1 -C3 alkoxy-carbonyl group, or ...
16	5773469	Diaryl antimicrobial agents The invention relates to diaryl antimicrobial compounds of the general formula: ##STR1## where G, E L, J, q, m, X, Ar, W, p, n and A are as described herein, pharmaceutical compositions containing...
17	5762963	Method and compositions for controlling oral and pharyngeal pain using capsaicinoids Methods and compositions are provided for the oral delivery of temporally increasing concentrations of capsaicin, its derivatives, and analogs (collectively, "capsaicinoids"), to provide oral or...
18	5763474	Substituted N-arylmethylamino derivatives of cyclobutene-3,4-diones The compounds of the formula: ##STR1## wherein R1 is straight chain alkyl, branched chain alkyl cycloalkyl, hydroxyalkyl, fluoroalkyl or polyfluoroalkyl; R2 and R3 are, independently, hydrogen or...
19	5744481	β-amino acid hydroxyethylamino sulfonamides useful as retroviral protease inhibitors α- and β-amino acid hydroxyethylamino sulfonamide compounds are effective as retroviral protease inhibitors, and in particular as inhibitors of HIV protease.
20	5728729	3-methoxy-2-phenylacrylic acid esters used as pest-control agents, especially as fungicides 3-Methoxy-2-phenyl-acrylic esters of the formula ##STR1## in which R represents optionally substituted alkyl, cycloalkyl or aryl and n represents a number 0 or 1,a process for their preparation and...
21	5709890	Polyaspartic acid and its analogues in combination with insecticides An insecticide composition is enhanced from the standpoint of its ability to be absorbed by insects, such as red fire ants, particularly dithiophosphate ester pesticides by the addition of a small...
22	5684018	Acyloxyisopropyl carbamates as prodrugs for amine drugs This invention relates to novel acyloxyisopropyl carbamates as bioreversible prodrug moieties for amino drugs and to methods of synthesizng these compounds.
23	5523325	Amidrazones and their use as pesticides This invention relates to amidrazones, insecticidal amidrazone compositions, and methods of using such compositions.
24	5482972	Substituted amino acid amides There are described new amino acid amides of the formula (I) ##STR1## in which n, R1, R2, R4, R5, R6, R7, X1, X 2 and X3 having the meaning given in the description, and a process for their...
25	5416117	Cyclopropenone derivatives A novel cyclopropenone derivative (I) which possesses a potent inhibitory activity against thiol protease such as papain, cathepsin B, cathepsin H, cathepsin L, calpain or the like with excellent...
26	5364850	Substituted tyrosyl diamide compounds The present invention provides substituted tyrosyl diamide compounds of general Formula I: ##STR1## and the pharmaceutically-acceptable salts thereof, which are useful for inducing analgesia in...
27	5360783	Water-based pesticidal composition A water-based pesticidal composition contains 100 weight parts of substantially water-insoluble pesticide and 1.7-200 weight parts of a surface active agent. The surface active agent contains...
28	5356931	Use of α-arylacrylic derivatives for controlling pests Alpha-Arylacrylic acid derivatives of the general formula I ##STR1## where X is ethylene or ethenylene; n is 0 or 1; m is 0, 1, 2, 3 or 4; R1 is cyano, cyanato, thiocyanato, nitro, hydroxyl,...
29	5331006	Amino acid analogs as CCK antagonists Novel unnatural dipeptoids useful as agents in the treatment of obesity, hypersecretion of gastric acid in the gut, gastrin-dependent tumors, or as antipsychotics are disclosed. Further, the...
30	5217994	Method of inhibiting osteoclast-mediated bone resorption by administration of aminoalkyl-substituted phenyl derivatives Compounds of the general formula ##STR1## and the pharmaceutically acceptable salts thereof wherein n is an integer of from 0 to 6; Y is CH2, O, SO2, --CONH--, --NHCO--, or ##STR2## R1 and R2 are...
31	5214061	Method of using p-acylaminophenoxycarbamates and derivatives as analgesics This invention relates to p-acylaminophenoxycarbamates having the formula ##STR1## where R1 and R2 are each independently hydrogen, loweralkyl, aryl and arylloweralkyl; R3 is hydrogen, loweralkyl,...
32	5180420	Water dispersible granules The water dispersible granule of the present invention contains (a) a pesticidal active ingredient which is solid at room temperature, (b) an anionic surface active agent, and (c) a kaolin series...
33	5141956	Pesticidal composition Ethyl 2-[4-(3-chlorophenoxy)phenoxy]ethylcarbamate is suitable controlling phytophagous cicadas in rice crops and fruit pests such as leaf rollers, citrus fruit pests such as scale insects, and...
34	5112859	Biphenyl amide cholesterol ester hydrolase inhibitors The compounds of the formula: ##STR1## in which R1 is hydrogen or alkyl; R2 is alkyl, cycloalkyl, cycloalkylalkyl, phenylalkyl or alkylphenylalkyl; or R1 and R2 taken together complete a...
35	5091414	Pesticidal compounds A compound of Formula (I): (I) R1 (CACA1)x --C(X)NR2 R3where R1 is alkyl optionally substituted by a group selected from alkoxy, alkenyl, alkynyl, alkenyloxy, alkynyloxy, aryl, aryloxy, ary...
36	5064827	Polyhydroxybenzyloxpropanolamines Compounds of the present invention, are represented by the general formula ##STR1## wherein R1 group which may be alkyl of from 1 to about 6 carbon atoms, alkenyl of from 2 to about 6 carbon atoms,...
37	5021453	3-keto HMG-CoA reductase inhibitors Compounds of formula (I) and (II): ##STR1## are HMG-CoA reductase inhibitors.
38	4966914	Oculoselective beta-blockers as antiglaucoma agents In accordance with the present invention, disclosed herein are compounds of the formula ##STR1## wherein R is hydrogen, straight or branched loweralkyl, cycloalkyl, amino, loweralkoxy or acylamino,...
39	4948807	Phenyl carbamates Phenyl carbamates of the general formula ##STR1## wherein R1 to R5 are as defined in the claims, are useful as pharmaceuticals.
40	4908386	Ethanolamine derivatives The present invention provides compounds of general formula (I) ##STR1## wherein Ar represents an unsubstituted or substituted phenyl gorup; R1 and R2 each represents a hydrogen atom or a C1-3...
41	4897417	Prodrugs of 3,4-hydroxy benzoyloxypropanolamines In accordance with the present invention, disclosed herein are compounds of the formula ##STR1## wherein R is straight or branched loweralkyl, R1 is hydrogen, straight or branched loweralkyl,...
42	4853382	Aminophenol derivatives The invention provides compounds of the general formula (I) ##STR1## wherein Ar represents a phenyl group optionally substituted by one or more substituents selected from halogen atoms, or the...
43	4735959	Carboxylic acid amides and pharmaceutical compositions containing them There are described novel carboxylic acid derivatives of the formula ##STR1## and derivatives of the formula ##STR2## and the addition salts thereof, which exhibit an effect on the intermediary...
44	4728670	Biphenyl hydroxamic acids Biphenyl hydroxamic acids are provided having the structure ##STR1## wherein m is 1 to 7, X is S, O or NH, R is H, lower alkyl, aryl, aralkyl or cycloalkyl and R1 is H, lower alkyl, aryl, aralkyl,...
45	4717736	Antagonists of slow reacting substances of anaphylaxis Compounds having the formula: ##STR1## are antagonists of leukotrienes of C4, D4 and E4, the slow reacting substance of anaphylaxis. These compounds are useful as anti-asthmatic, anti-allergic,...
46	4639468	Derivatives of glycinamide, their preparation and their use A glycinamide derivative of the general formula I: ##STR1## wherein: R is a linear or ramified alkyl group C5 -C18, a linear or ramified alkenyl group C5, C6, C7, C8, C9, C10, C11, C12, C13, C14,...
47	4618623	Carbazic acid derivatives, process for their preparation and compositions containing the same The invention relates to new carbazic acid derivatives, a process for the preparation thereof and compositions--particularly feed additives and animal feeds--containing the same. The new compounds...
48	4618624	3-amino-4-hydroxy(or alkoxy)phenethanolamine derivatives and pharmacologically-acceptable acid addition salts thereof for increasing the growth rate and/or improving the lean meat to fat ratio of warm-blooded animals A method for increasing the growth rate and/or improving the lean meat to fat ratio in farm and domestic animals. An effective amount of a 3-amino-4-hydroxy(or alkoxy)phenethanolamine derivative,...
49	4582855	Aromatic and esters of hydroxypropylamines Novel compounds of the general formula ##STR1## wherein Ar represents a substituted or unsubstituted aromatic or heterocyclic group; W represents alkylene of from 1 to about 10 carbon atoms; and B...
50	4554290	Oxamic acid derivatives There are disclosed novel oxamic acid esters substituted on the nitrogen atom and corresponding to the formula I ##STR1## the production thereof, their use for controlling pests, and pesticidal...

Matches 1 - 50 out of 68

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