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5869522 |
Antiviral naphthoquinone compounds, compositions and uses thereof
The present invention provides novel antiviral naphthoquinone compounds, which may be isolated from plants of the genus Conospermum or synthesized chemically, in accordance with the present...
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5861430 |
Benzopyran phenol derivates for use as antibacterial, antiviral or immunostimulating agents
A method of inhibiting microorganisms, including bacteria, using benzopyran phenol derivates from propolis. Propolis is extracted with an alcohol, and the resulting compounds are effective as...
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5859027 |
Antimicrobial agent
The invention provides a method of treating a fungal infection comprising administering to an animal having a fungal infection a composition comprising an infection treating effective amount of a...
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5859045 |
Crystalline -! 3R 4R-trans-7 methoxy 2,2-dimethyl1-3-phenyl 1-4 4-12 pyrrolidin-1 -Y1!ethoxyl 1!chromane hydrogen fumarate
The present invention provides novel crystalline (-)-3R,4R-trans-7-methoxy-2,2-dimethyl-3-phenyl-4-{4- 2-(pyrrolidin-1-yl)e thoxy!phenyl}chromane, hydrogen fumarate useful for reducing or...
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5858371 |
Pharmaceutical composition for the control and treatment of anorectal and colonic diseases
A Novel composition and a method for treating anorectal diseases including hemorrhoids and colonic diseases with long term effectiveness and low prolapse rates is disclosed. The compositions are...
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5855892 |
Method for decreasing LDL-cholesterol concentration and increasing HDL-cholesterol concentration in the blood to reduce the risk of atherosclerosis and vascular disease
A method of altering the concentration of cholesterol constituents in human blood is provided. A daidzein material is administered to a human to increase the concentration of HDL-cholesterol and to...
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5856352 |
Abruquinone derivatives useful in the treatment of inflammation and allergic reactions
Disclosed are methods of providing antiinflammatory activity and inhibiting allergic reaction by administering Abruquinones A, B, D, E, or F to a subject in need thereof.
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5854280 |
Antifungal sordaridin derivatives
A compound of formula ##STR1## wherein Z is a tetrahydro-pyrano group selected from ##STR2## having antifungal activity processes for their preparation and their use in medicines.
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5851792 |
Aglucone isoflavone enriched vegetable protein whey whey protein material aglucone isoflavone material high genistein content material and high daidzein content material and process for producing the same from a vegetable protein whey
An aglucone isoflavone enriched vegetable protein whey, whey protein material, high genistein material, high daidzein material, and aglucone isoflavone material are provided, as well as a process...
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5849265 |
Pharmaceutical aerosol formulation comprising a medicament, a propellant and a fluorinated surfactant
A pharmaceutical aerosol formulation which comprises particulate medicament, a fluorocarbon of hydrogen-containing chlorofluorocarbon propellant and a surfactant of general formula (I), wherein n...
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5849798 |
Polyaromatic heterocyclic compounds and pharmaceutical/cosmetic compositions comprised thereof
Novel pharmaceutically/cosmetically-active polyaromatic heterocyclic compounds have the structural formula (I): ##STR1## in which Z is a divalent radical selected from among --O--, --S-- or --Nr'--...
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5849755 |
3-amidochromanylsulfonyl(thio)ureas, processes for their preparation, their use, and pharmaceutical preparations comprising them
3-amidochromanylsulfonyl(thio)ureas of the formula (I): ##STR1## which are valuable pharmaceutically active compounds for the treatment of disturbances of the cardiovascular system, in particular...
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5846988 |
Thiazolidine-4-carboxylic acid derivatives as cytoprotective agents
Compounds useful as cytoprotective agents are disclosed. The compounds possess dual activity, containing a phenolic portion selected to have antioxidant or free radical scavenging properties and a...
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5844061 |
Polyphenol derivative compositions and perparation thereof
Polyphenol derivative compositions including oligomer or polymer esters containing N+2 monomer moieties, whose monomer moieties correspond to the following formula ##STR1## in which N is a number...
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5843989 |
C.sub.4 -amide substituted compounds and their use as therapeutic agents
The invention provides certain 5 and/or 8 substituted benzopyran, pyranopyridine or tetrahydroquinaline compounds having C 4 -amide substituent and processes for making them. The compounds...
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5840735 |
Sex steroid activity inhibitors
Inhibitors of sex steroid activity, for example those having the general structure ##STR1## may be used as part of a pharmaceutical composition to provide antiestrogenic effects and/or to suppress...
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5837725 |
Bridged bicyclic aromatic compounds and their use in modulating gene expression of retinoid receptors
Bridged bicyclic aromatic compounds are provided having the structure ##STR1## wherein R 1 , R 2 , R 3 , R 4 , R 5 and n are as defined herein. The novel compounds are useful for modulating gene...
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5837702 |
4-arylamino-benzopyran and related compounds
Compounds having the formula ##STR1## and pharmaceutically acceptable salts thereof wherein X is alkyl, Y is a single bond, --CH 2 --, --C(O)--, --O--, --S-- or --N(R 8 )-- where R 8 is hydrogen,...
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5824702 |
Genistein as a preventive against ultraviolet induced skin photodamage and cancer
A method of inhibiting the harmful effect of UVR exposure to the human skin comprising topically applying a therapeutically effective amount of genistein to the skin at a time sufficiently close to...
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5814669 |
Amino acid derivatives and their use as pesticides
The invention relates to novel amino acid derivatives, to a process for their preparation and to their use as pesticides, in particular as fungicides, and as intermediates for preparing known...
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5811448 |
Substituted chromanysulfonyl (thio) ureas, processing for their preparation and pharmaceutical uses thereof
Substituted chromanylsulfonyl(thio)ureas, processes for their preparation, their use in pharmaceutical preparations, and pharmaceutical preparations comprising them Chromanylsulfonyl(thio)ureas of...
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5811083 |
Tocopherol derivatives for use in cosmetic compositions
Novel tocopherol derivatives useful for regulating skin aging and other skin disorders, as well as compositions containing the derivatives and methods for their use are described. The tocopherol...
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5807564 |
Method of strengthening antibacterial action of antibiotics
A method of increasing the activity of an antibiotic against methicillin resistant Staphylococcus aureus in a patient by administering to the patient the antibiotic in combination with a catechin...
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5807586 |
Method of dietary supplementation
The present invention relates to a method of supplementing the dietary needs of women whereby an effective amount of a life stage appropriate dietary supplement is administered to a woman at each...
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5804597 |
Agent for the prevention or treatment of cataracts
An agent for the prevention or treatment of cataracts comprising a proanthocyanidin oligomer is provided. The oral administration or application to the eyes of the agent of the invention produces a...
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5804567 |
Method of increasing the effectiveness of anti-metabolites
A method for treating cancer in a patient by administering to a patient an nti-cancer effective amount of an anti-metabolite selected from the group consisting of 1-β-arabinofuranosylcytosine and...
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5798381 |
Biologically active bistramides, process for their production and their applications in therapy
Bistramide derivatives with virtually no toxic effects, of formula (I) wherein --R 1 , X, Y and R 2 are a saturated or unsaturated hydrocarbonaceous chain having from 1 to 20 carbon atoms,...
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5795911 |
Composition for treating Condyloma acuminata
A composition for a treatment of HPV-infected Condyloma acuminata which comprises containing tea catechin as a main component. This medication has no danger of side-effects and may be easily...
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5795874 |
Water soluble antibiotics
The compound of the formula I ##STR1## wherein R 1 , R 2 , R 3 , R 4 , R 5 , R 6 , R 7 , and R 8 are as defined herein, are described. These compounds are antibacterial agents.
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5792448 |
Use of flavonoids for preserving and/or enhancing the mechanical properties of the hair and process for protecting the hair using these compounds
The use of flavonoids for preserving and/or enhancing the mechanical properties of hair, and a process for protecting the mechanical properties of hair are disclosed.
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5792789 |
Acids and esters of diosmetin
Acids and esters of diosmetin of formula: ##STR1## wherein R 1 , R 2 , R 3 , R 4 , R 5 , R 6 and R 7 are as defined in the description, and the physiologically tolerable salts thereof. The said...
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5780502 |
Use of 3,4-diphenyl chromans for the manufacture of a pharmaceutical composition for inhibiting one or more symptoms of premenstrual syndrome
The present invention provides novel uses of compounds of general formula I ##STR1## wherein R 1 , R 4 and R 5 are individually hydrogen, hydroxy, halogen, trifluoromethyl, C 1 -6 alkyl, C 1 -6...
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5776442 |
Reduction of hair growth
Mammalian hair growth is reduced by applying to the skin a dermatologically acceptable composition including a catechin compound.
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5776906 |
Method for promoting fat-degradation in fat cells
For the purpose of providing a composition having an ability of promoting degradation of accumulated cellular fats, a substance having such ability was developed from naturally-occurring safe...
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5773005 |
Purified flavonoid and diterpene 5α-reductase inhibitors from thuja orientalis for androgen-related diseases
Strong 5αa-reductase inhibitors are extracted and fractionated from Thuja orientalis and other similar crude drugs or they may be purified as diterpenes in isolated form. The inhibitors are used...
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5770593 |
Method of determining a pharmaceutical combination preparations for use in anti-neoplastic therapy
The present invention provides a pharmaceutical combination preparation, wherein it contains at least two active materials, the first active material being an inhibitor of protein kinase C and the...
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5766595 |
Method of improving quality of eggs by feeding tea polyphenol
Method of improving the quality of an egg from a female adult fowl comprising adding an effective egg improving amount of at least one tea polyphenol to a feed composition for the fowl and...
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5767132 |
Pyridyl chroman
Amino(thio)ether derivatives of formula I ##STR1## wherein R 0 , R 1 , R 2 , R 3 , R 6 , R 7 , R 8 , R 9 , X and Z are as defined herein, and their salts, are active on the central nervous system.
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5767109 |
Complexing urushiols
This invention relates to use of cyclodextrins to complex urushiols to protect against and to treat irritation arising from exposure to urushiols. cyclodextrins, particularly gamma-cyclodextrins,...
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5763470 |
Benzopyran compounds and methods for their use
The present invention relates to organic molecules capable of modulating tyrosine kinase signal transduction in order to regulate, modulate and/or inhibit abnormal cell proliferation.
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5763414 |
Hesperidin and hesperetin as 3-hydroxy-3-methylglutaryl CoA (HMG-CoA) reductase inhibitor
A method for inhibiting the activity of 3-hydroxy-3-methylglutaryl CoA(HMG-CoA) reductase in mammals comprises administering hesperidin or hesperetin thereto.
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5760074 |
Treatment
The invention relates to certain cis and trans benzopyrans having substituted benzamides at position C-4 and to their use in treating and/or preventing certain CNS disorders.
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5760006 |
Anticonvulsant derivatives useful in treating psoriasis
The use of compounds of the following formula I: ##STR1## for treating psoriasis is disclosed.
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5756539 |
3, 4-diphenyl chromans for inhibiting one or more psychiatric disorders
A method of inhibiting one or more psychiatric disorders is disclosed comprising administering a compound of formula I ##STR1## wherein R 1 , R 4 and R 5 are individually hydrogen, hydroxy,...
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5753693 |
Anticonvulsant derivatives useful in treating manic-depressive bipolar disorder
This application relates to the use of topiramate and related sulfonamides for the treatment of manic-depressive bipolar disorder.
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5753674 |
Adenosine diphosphoribose polymerase binding nitroso aromatic compounds useful as retroviral inactivating agents, anti-retroviral agents, anti-retroviral agents and anti-tumor agents
The subject invention provides for novel compounds for inactivating viruses. These compounds include 6-nitroso-1,2-benzopyrone, 3-nitrosobenzamide, 5-nitroso-1 (2H)-isoquinolinone,...
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5753694 |
Anticonvulsant derivatives useful in treating amyotrophic lateral sclerosis (ALS)
Disclosed herein is a method of treating amyotrophic lateral sclerosis with topiramate and related compounds.
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5753695 |
Flavilium compounds and method of using
The invention relates to a compound of formula (I) ##STR1## wherein X is a pharmacologically acceptable anion, R 1 and R 2 are independently of each other hydrogen, or an --OY group in which Y...
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5747528 |
Chroman derivatives as anti-oxidants
Chroman derivatives of Formula I or a pharmaceutically acceptable salt thereof are inhibitors of VCAM-1 and ICAM-1 and are thus useful in the treatment of inflammation, atherosclerosis, restenosis,...
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5733920 |
Inhibitors of cyclin dependent kinases
The invention provides novel inhibitors of cyclin-dependent kinases, in particular inhibitors of the CDK/cyclin complexes such as CDK4/cyclin D1. The novel compounds are analogs of chromones. These...
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