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5021448 |
Method of reducing serum uric acid and/or increasing renal uric acid clearance with thromboxane synthetase inhibitor inhibitor and/or thromboxane receptor antagonist
A method of reducing serum uric acid and/or increasing renal clearance of uric acid in a mammal in need thereof comprising administering to such mammal a uricosuric effective amount of a...
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4987130 |
Substituted amine derivatives, their production and use
Substituted amino derivatives represented by the formula: ##STR1## wherein R 1 and R 2 each stand for an acyclic hydrocarbon residue or an alicyclic hydrocarbon residue; R 3 and R 4 each stand...
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4973474 |
2,4-diaminopyrimidine 3-oxide derivatives and their use for the treatment and prevention of hair loss
New 2,4-diaminopyrimidine 3-oxide derivatives and their use for the treatment and the prevention of hair loss. The compounds correspond to the formula: ##STR1## in which: R 1 and R 2 denote...
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4971979 |
Alkadiene derivatives, and pharmaceutical compositions containing them
Substituted alkadienes of formula: ##STR1## in which R 1 is hydroxy or acetoxy, R 2 is hydrogen, carboxy, alkoxycarbonyl, phenyl or benzoyl, and R 3 is alkylthio or alkoxy and R 4 is...
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4960790 |
Derivatives of taxol, pharmaceutical compositions thereof and methods for the preparation thereof
Derivatives of taxol represented by the formula ##STR1## wherein R and R' are each H or the residue of an amino acid selected from the group consisting of alanine, leucine, isoleucine, saline,...
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4946852 |
4(R)-substituted 6(S)-phenoxymethyl-, 6(S)-β-phenylethyl- and 6(S)-β-styryl-tetrahydropyran-2-ones, a highly stereoselective process for their preparation, pharmaceutical products based on these compounds, and their use
4(R)-Substituted 6(S)-phenyloxymethyl-, 6(S)-β-phenylethyl- and 6(S)-β-styryl-tetrahydropyran-2-ones of the general formula V ##STR1## in which R 7 , R 8 and A have the meanings given, and the...
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4942184 |
Water soluble, antineoplastic derivatives of taxol
Antineoplastic, water soluble, taxol derivatives and methods for preparing the same are described.
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4935409 |
Aminophenylethylamine yield promoters
Animal growth promoters of the formula ##STR1## The intermediates of the formula ##STR2## are also new.
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4920109 |
Antifungal compositions and method of controlling mycotic infections
Method of potentiating antifungal agents with 25-azasterol compound to produce superior antifungal compositions and use of the compositions to control mycotic infections is disclosed.
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4920113 |
Fungicidal compositions and methods utilizing 25-azasterol and HMG-CoA synthase inhibitors
Novel fungicidal compositions comprising a 25-azasterol compound and a HMG-CoA synthase inhibitor compound are disclosed.
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4873260 |
Treatment of diabetic ketoacidosis
There is disclosed the use of β-lactone alkylene carboxylic acids and derivatives thereof, which are known compounds, for the use of treating diabetic ketoacidosis. The compounds are administered...
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4847271 |
Antihypercholesterolemic β-lactones
The compounds of the following general structural formula (I) ##STR1## are 3-hydroxy-3-methylglutaryl-coenzyme A (HMG-CoA) synthase inhibitors and useful as antihypercholesterolemic agents for the...
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4816477 |
Antihypercholesterolemic β-lactones
The compounds of the following structural formula (I) ##STR1## ar 3-hydroxy-3-methylglutaryl-coenzyme A (HMG-CoA) synthase inhibitors and useful as antihypercholesterolemic agents for the treatment...
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4814470 |
Taxol derivatives, their preparation and pharmaceutical compositions containing them
Taxol derivatives of formula ##STR1## in which R represents hydrogen or acetyl, one of R 1 or R 2 represents hydroxy and the other represents tert-butoxycarbonylamino and their isomers are useful...
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4806564 |
Antihypercholesterolemic beta-lactones
The compounds of the following structural formula (I) ##STR1## are 3-hydroxy-3-methylglutaryl-coenzyme A (HMG-CoA) synthase inhibitors and useful as antihypercholesterolemic agents for the treatmet...
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4791139 |
Diphenyl ether derivatives and their use as insecticides
A compound of formula: ##STR1## wherein W represents one or more substituents selected from halo, alkyl, alkoxy, alkoxyalkyl, haloalkyl and haloalkoxy or W represents a bidentate group linking...
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4756909 |
Method for relieving pain or producing analgesia with n-butanol
A method for treating a host for inducing relief of pain or anesthesia which comprises administering hydrolyzed epichlorohydrin, magnesium thiosulfate, or a butanol at the site of the painful area.
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4719226 |
Percutaneous absorption type preparation and process for preparing the same
A percutaneous absorption type preparation and a process for preparing the same, where the preparation comprises a backing readily conformable to the skin or mucosa and substantially impermeable to...
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4714710 |
Insecticidal and acaricidal oxetane and thietane derivatives, compositions, and method of use therefor
There are described new compounds of general formula I ##STR1## in which R 1 is aryl or aryl substituted by C 1 -4 -alkyl, halo-C 1 -4 -alkyl, phenyl-C 1 -4 -alkyl, C 2 -4 -alkenyl, halo-C 2 -4...
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4668694 |
1-arylalkoxyphenyl-pyrazolines, ketones or enoles as anti-inflammatory or anti-allergic agents
This disclosure describes novel pharmaceutical compositions of matter which possess useful anti-inflammatory and anti-allergic properties, the active ingredients of said compositions of matter...
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4608385 |
Fungicidal N-phenylcarbamates
Use of an N-phenylcarbamate of the formula: ##STR1## as a fungicidal agent against phytopathogenic fungi, particularly their strains resistant to benzimidazole thiophanate fungicides and/or cyclic...
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4598089 |
Leucine derivatives
Novel compounds of the formula ##STR1## wherein A signifies the group ##STR2## or --(CH 2 ) 5 --, which inhibit pancreas lipase and can be used for the control or prevention of obesity and...
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4555522 |
Antithrombotic and/or antihypertensive compositions
Hypertension and thrombotic conditions in mammals are treated by administration of sulphite, bisulphite or cyclic sulphite ester of a monohydric or polyhydric alcohol.
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4542155 |
Tetrahydrofuranyl substituted prostaglandin analogs
Tetrahydrofuranyl substituted prostaglandin analogs are provided having the structural formula ##STR1## and including all stereoisomers thereof. The compounds are cardiovascular agents useful, for...
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4470984 |
Combating pests with novel oxime-carbamates
An N-sulphenylated oxime-carbamate of the formula ##STR1## in which R 1 is optionally substituted alkyl, cycloalkyl, aryl or aralkyl, R 2 is alkyl, alkenyl or alkynyl, or R 1 and R 2 ...
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4468397 |
Combating pests with novel imino ethers
Hydroxamic acid esters of the formula ##STR1## in which R 1 is an optionally substituted alkyl, cycloalkyl, aryl or aralkyl radical and R 2 is an alkyl, alkenyl or alkinyl radical, or R 1 ...
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4463013 |
Oxygen substituted amino-cyclohexyl-benzeneacetamides and -benzamides as water diuretic drugs
Conditions of inappropriate hyperhydration in warm blooded animals can be treated with an essentially water only diuretic drug compound selected from the group ##STR1## wherein m, n, p, A, E, R, R...
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4438112 |
Prostanoid compounds and pharmaceutical formulations
Prostanoids are described of the formulae ##STR1## (and the salts thereof) in which: X is cis or trans --CHCH-- or CH 2 CH 2 --; R 1 is C 1 -7 alkyl terminated by --COOR 10 where R 10 is...
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4370323 |
2-Cyanoaziridinyl-(1)-2-substituted-aziridinyl-(1)-methanes
A 2-cyanoaziridinyl-(1)-2-substituted-aziridinyl-(1)-methane ##STR1## wherein R is a nitrile or carbamoyl group, and R 1 and R 2 each independently is a hydrogen atom, an aliphatic hydrocarbon...
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4366168 |
Anticoccidial combinations
Combinations of a polyether antibiotic and a 2,4-dinitro-N-[4-(fluoroalkoxy)phenyl]-6-(trifluoromethyl)be
nzenamine are synergistic in controlling coccidiosis in animals.
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4309425 |
Miticidal, insecticidal, ovicidal and fungicidal N-(N',N'-diarylaminothio)sulfonamides
Sulfonamides, such as N-[N-(2-chloro-5-(trifluoromethyl)phenyl]-N-[2,4-dinitro-6-(
trifluoromethy l)phenyl]aminothio]-N,4-dimethylbenzenesulfonamide, are useful for control of arthropod pests of...
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4279919 |
Novel lactones of cyclopentanols
Novel lactones of the formula ##STR1## wherein the dotted line indicates the optional presence of a second bond, A is a single bond or --CH 2 --CH 2 --, R is selected from the group consisting of...
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4271193 |
N1-Benzoyl-N2-phenyldiaminopropanols and pharmaceutical compositions thereof, and processes for their preparation
N 1 -benzoyl-N 2 -phenyl-1,3-diaminopropan-2-ols are disclosed which exhibit a stabilizing effect on the gastric mucosa and enhance the stability and resistance of the gastic mucosa against...
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4259321 |
Compositions and methods for controlling coccidiosis
Compositions and methods for the control of coccidiosis using antibiotic K-41 and its non-toxic salts as the active anti-coccidial agent.
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4239759 |
Morpholino containing compounds, compositions and use thereof
Compounds of the formula R--A--Z wherein R is a 4-biphenylyl or 4-phenoxyphenyl or a corresponding group monosubstituted or polysubstituted by one or more of F, Cl, and Br; A is --CH(CH 3 )--CH 2...
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4221809 |
β-Lactones of 2-hydroxy-cyclopentanecarboxylic acid
Novel lactones of the formula ##STR1## wherein the dotted line indicates the optional presence of a second bond, A is a single bond or --CH 2 --CH 2 --, R is selected from the group consisting of...
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4212878 |
Phenylacetamide derivative analgesics
N-[(1-Amino-4-(mono or di-oxygen-group-substituted)cyclohex-1-yl)methyl]phenylaceta
mide derivatives of the formula 1 ##STR1## wherein R, R 1 , R 2 , R 3 , P, Q, X and Y are defined in the...
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4169145 |
ω-Nor-cycloalkyl-13,14-dehydro-prostaglandins
ω-NOR-CYCLOALKYL-13,14-DEHYDRO-PROSTAGLANDIN COMPOUNDS, SPECIFICALLY 13,14-DEHYDRO-17-CYCLOHEXYL-20,19,18-TRINOR-PGF 2 α having antiulcer and luteolytic activity, are disclosed.
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4130641 |
Induction of interferon production by modified nucleic acid complexes
The present invention relates to the induction of interferon production in the cells of living organisms, including human beings. According to the invention, nucleic acid complexes, such as the...
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3881030 |
2,2-Diphenyl-3,3-dimethyloxetone insecticides
The invention provides derivatives of 2,2-diphenyl-3,3-dimethyloxetane in which the phenyl groups are substituted with alkoxy, alkylthio and/or methylenedioxy groups, which have insecticidal...
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3764692 |
METHOD OF TREATING OBESITY
The inhibition of fatty acid synthesis is obtained in biological systems by utilizing a specific stereoisomer of hydroxycitric acid and derivatives thereof such as esters or lactones and the...
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3536808 |
USE OF TRIMETHYLENE OXIDE COMPOUNDS TO COMBAT BACTERIA
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3474164 |
NOVEL COMPOUNDS AND METHOD FOR COMBATING MICROORGANISMS
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3458636 |
METHOD FOR COMBATING MICRO-ORGANISMS
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3433662 |
PROCESS FOR PRODUCING A STERILIZED INSTRUMENT
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3275505 |
Process for preparing a biocidal composition comprising halogenated levulinic acid
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3251738 |
Anti-microbial potentiation with agents having plant hormone activity
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3157577 |
Antiserum and plasma for aleutian disease (hypergammaglobulinemia) in mink
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3076748 |
Poliomyelitis virus attenuation with ultraviolet light and beta propiolactone
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3050405 |
Food preserving process
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