Matches 351 - 400 out of 408 < 1 2 3 4 5 6 7 8 9 >
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4786639 Method for the treatment of reversible airways obstruction and asthma  
A method for the treatment and/or prophylaxis of reversible airways obstruction and asthma in mammals, which method comprises administering to the mammal in need of said treatment an effective...
4778511 Fluorine-containing N-sulphenylated indazoles for use as bactericides and fungicides  
Novel fluorine-containing N-sulfenylated indazoles are prepared by reacting the corresponding indazoles with sulfenyl halides in the presence of a solvent and/or diluent and in the presence of an...
4772603 Method for treating congestive heart failure, angina, occlusive peripheral vascular disease or cerebral vascular disease in mammals  
A method for the treatment and/or prophylaxis of congestive heart failure, angina, occlusive peripheral vascular disease or cerebral vascular disease in mammals, such as humans, which method...
4767779 Pyrazoline-1-carboxamides, composition containing them, and insecticidal method of using them  
Pyrazolines of the following formula are insecticides: ##STR1## wherein R A , R B and R C are aromatic groups; R N is hydrogen or lower alkyl; and W is oxygen or sulfur.
4738963 Method for the treatment of incontinence in mammals  
A method for the treatment and/or prophylaxis of incontinence in mammals, which method comprises administering to the mammal in need of said treatment an effective amount of a compound of formula...
4692444 1,4-Dihydro[1]benzothiopyrano[4,3-c]pyrazole derivatives, compositions containing them, and pharmacological methods of using them  
This invention provides a benzene-fused heterocyclic compound of the formula: ##STR1## wherein R 1 is halogen, nitro, amino, hydroxy, lower alkyl, lower alkoxy or acylamino, X is --S--,...
4677210 1-arylalkoxy- and 1-arylalkylthioaryl-2-pyrazolines as anti-inflammatory or anti-allergic agents  
4663341 Insecticidal n-aryl-3-aryl-4,5-dihydro-1h-pyrazole-1-carboxamides  
This invention relates to N-aryl-3-aryl-4,5-dihydro-1H-pyrazole-1-carboxamide compounds which are useful as pesticides, compositions containing those compounds, methods of controlling pests and...
4624961 Method for enhancing memory or correcting memory deficiency with arylamidopyrazolidines and arylamidodiazabicycloalkanes  
A pharmaceutical method for improving memory or correcting memory deficiency is disclosed, utilizing compounds having the formula: ##STR1## wherein m and n are zero and one and when m is zero, the...
4608383 Cardioactive pyrazole and imidazole aryloxypropanolamines  
The present invention provides aryloxypropanolamines of the general formula: ##STR1## wherein R 1 , R 2 , R 3 and R 4 , which may be the same or different, are hydrogen or halogen atoms or lower...
4572914 Insecticidal 4-substituted-3-chlorophenyl-1-(fluoroalkoxyphenylcarbamoyl)pyrazolines  
The invention relates to new pyrazoline derivatives and to insecticidal compositions on the basis of the compounds. The compositions can be used for controlling insects in a dosage from 0.01 to 1...
4572913 Use of 3-(arylmethyleneamino)-1-aryl-2-pyrazolines in the prophylaxis and treatment of inflammation, pain, pyresis, and asthma  
Compounds of formula (I) ##STR1## inhibit both the cyclo-oxygenase and lipoxygenase pathways of arachidonic acid oxygenation and are useful in medicine as, e.g., anti-inflammatory and...
4568688 Antihypotensive tetrahydro-1H-pyrazolo[5,1-a]isoindoles  
New substituted tetrahydro-1H-pyrazolo[5,1-a]isoindoles of the formula I ##STR1## in which R 1 denotes a hydrogen or halogen atom or an alkoxy group having 1 to 4 carbon atoms, R 2 , R 3 and R 4...
4556654 Antimicrobial substituted anthra[1,9-cd]pyrazol-6(2H)-ones  
Substituted anthra[1,9-cd]pyrazol-6(2H-ones have antimicrobial activity. Methods for their preparation, use and pharmaceutical compositions are disclosed.
4547518 Antiemetic N-(1-substituted-4,5-dihydro-1H-pyrazol-4-yl)benzamides  
N-(1-Substituted-4,5-dihydro-1H-pyrazol-4-yl)benzamides having the general formula: ##STR1## wherein R is loweralkyl, cycloalkyl or phenylloweralkyl and R 1 is selected from hydroxy, cyano, nitro,...
4540706 Insecticidal 1-N-phenylcarbamoyl-3-(4-difluoromethoxyphenyl)-4-phenyl-2-pyrazoline derivatives  
Pyrazoline derivatives useful as insecticides having the formula ##STR1## wherein X represents a hydrogen atom or a halogen atom; Y represents a halogen atom, a trifluoromethyl group or --A--R'; R...
4515801 Fungicidally active pyrano-pyrazole derivatives  
Pyrano-pyrazole derivative of the formula ##STR1## in which R 1 represents hydrogen, alkyl, alkanoyl, alkoxycarbonyl, optionally substituted phenyl or optionally substituted phenylalkyl, R 2 ...
4490384 Benzisoxazole carboxylic acids  
Described are compounds of the formula ##STR1## wherein X is hydrogen, loweralkyl, halo, loweralkoxy or trifluoromethyl, and Z is hydrogen, loweralkyl, halo, hydroxy or alkoxy, or compounds of the...
4474797 Fungicidal 1-methyl-3,4-dihalo-5-substituted-sulfonylpyrazoles  
Compounds of the formula: ##STR1## wherein R 1 is vinyl, 2-haloethyl or the group --CH 2 CH 2 OS(O) 2 CH 3 ; and Y is chloro or bromo are fungicidal.
4465679 1,2-Diaza-3-one compounds, their use in treating hypertension and pharmaceutical compositions thereof  
Compounds of the formula ##STR1## and their pharmaceutically-acceptable salts, wherein the substituents are as defined herein, having antihypertensive activity.
4464386 Insecticidal 3-difluoromethoxyphenyl-1-phenylcarbamoyl-2-pyrazolines  
Pyrazoline derivatives useful as insecticides having the formula ##STR1## wherein R 1 represents hydrogen atom, a lower alkyl group, (CH 2 ) n CN group, (CH 2 ) n OR group, phenyl group or a...
4457930 Todopropargylsulphamides, microbicidal compositions and use  
3-Iodopropargyl-sulphamides of the formula ##STR1## in which R represents hydrogen, alkyl, optionally substituted cycloalkyl, optionally substituted phenylalkyl, optionally substituted...
4439440 1-Alkoxycarbonylphenylcarbamoyl-3-phenyl-4-cyanoalkyl-2-pyrazolines and use as insecticides  
The invention relates to new pyrazoline derivatives having insecticidal activity; the new compounds can be represented by the general formula ##STR1## wherein R is an alkoxycarbonyl group having 2...
4438128 Cardioactive aryloxypropanolamines  
The present invention provides aryloxypropanolamines of the general formula: ##STR1## wherein R 1 , R 2 , R 3 and R 4 , which may be the same or different, are hydrogen or halogen atoms or lower...
4421927 New cinnamoyl-cinnamic acid derivative, and its use as pharmaceutical  
The present invention relates to a new cinnamoyl-cinnamic acid derivative selected from the group constituted by: (i) the m-cinnamoyl-cinnamic acid derivatives of formula ##STR1## in which: X o...
4419363 Alkanolamine derivatives  
Novel 1-aryloxy-3-amidoamidoalkylamino-2-propanol derivatives, processes for their manufacture, pharmaceutical compositions containing them and methods of using them in the treatment of heart...
4409234 Pyrazoloindazole derivatives and bronchodilating composition  
Novel pyrazoloindazole derivatives of the formula ##STR1## wherein R 1 is a hydrogen atom, halogen atom, a hydroxyl group, a lower alkyl group, a lower alkoxyl group or benzyloxyl group; R 2 is a...
4407813 Insecticidal pyrazoline derivatives and composition  
Pyrazoline derivatives having the formula ##STR1## wherein R 1 represents hydrogen atom, a lower alkyl group, phenyl group or a halogen-substituted phenyl group; R 2 represents hydrogen atom or...
4407797 1,2-Dithiol-3-ylideneammonium derivatives, compositions and use  
New compounds of the formula: ##STR1## wherein X .crclbar . is an anion, R is (C 1 -7) alkyl [unsubstituted or substituted by hydroxy, carboxy, alkoxycarbonyl, cyano, dialkylamino, alkylcarbonyl,...
4397851 2,3-Dihalo-2,3-(disubstituted) propanoate antimicrobial compounds  
Antimicrobial compounds of the formula: ##STR1## wherein Hal is bromine or chlorine; R is C 1 -4 alkyl, straight or branched chain; and one of R 1 and R 2 is hydrogen and the other is selected...
4389403 1-Aroyl-2-phenylamino-2-imidazolines, drugs containing these compounds, and use thereof  
1-Aroyl-2-phenylamino-2-imidazolines of the general formula ##STR1## where R 1 and R 2 are identical or different and each is chlorine, bromine, fluorine, methyl, ethyl, methoxy, trifluoromethyl...
4382947 Combating pests with N-methyl-carbamic acid O-pyrazol-4-yl esters  
N-Methyl-carbamic acid O-pyrazol-4-yl esters of the formula ##STR1## in which R is optionally substituted alkyl, alkenyl, alkynyl, cycloalkyl or phenyl, which possess insecticidal, acaricidal and...
4371526 Phosphinylalkanoyl substituted 4,5-dihydropyrazole-5-carboxylic acid derivatives and hypotensive method and composition  
Compounds of the formula ##STR1## are disclosed. These compounds are useful as hypotensive agents due to their angiotensin converting enzyme inhibition activity.
4357339 Control of pine beetles with 1,5-dimethyl-6,7-diazabicyclo[3.2.1]oct-6-ene  
1,5-Dimethyl-6,7-dioxabicyclo[3.2.1]-octane and 1,5-dimethyl-6,7-diazabicyclo[3.2.1]-oct-6-ene are synthesized. They are analogs of the western and southern pine beetle natural-pheromone,...
4352813 [(1-Benzyl-1H-indazol-3-yl)oxy] acetic acid salt with L. lysine  
A new salt of [(1-benzyl-1H-indazol-3-yl)oxy] acetic acid (or bendazac) with L. lysine. Following oral administrations of this compound in man, the concentrations of bendazac found in the blood are...
4333929 Carboxamidine derivatives and hypoglycemical use  
A compound of formula (II) or a pharmaceutically acceptable acid addition salt thereof ##STR1## wherein R 1 , R 2 , R 3 and R 4 are the same or different and each represents C 1 -6 alkyl; R 5 ...
4285972 Method of treating scours  
Scours in animals, particularly new-born calves, lambs, piglets and foals are treated with a compound containing an effective amount of an antidiarrheal amidinourea.
4284632 3-Pyrrolin-2-one derivatives and compositions  
New 3-cyclicaminoalkoxy-4-phenyl-3-pyrrolin-2-ones are disclosed. These compounds exhibit anti-hypertensive and vasodilatory action.
4281014 Stabilized compositions containing N-aminosulfenylated derivatives of carbofuran  
Insecticidal compositions containing N-aminosulfenyl derivatives of carbofuran are stabilized against spontaneous decomposition by incorporating an epoxide compound therein.
4279905 1-Benzoxepin-5 (2H)-one derivatives and pharmaceutical compositions  
Novel, 3-amino-1-benzoxepin-5 (2H)-one derivatives and methods for their production are disclosed. These derivatives correspond to the Formula I: ##STR1## wherein: R 1 and R 2 independently of...
4279902 Anti-arrhythmia agents  
Acetamide derivatives are provided having the structure ##STR1## wherein X is a single bond, --CH 2 -- or --O--, R 1 and R 2 may be the same or different and are lower alkyl, phenyl-lower...
4250185 1-(3,5-Dichlorobenzoyl)-3-phenylpyrazolines and their use as mildewicides  
Certain 1-(3,5-dichlorobenzoyl)-3-phenylpyrazolines which have the structural formula ##STR1## where R is hydrogen, alkyl, alkoxy or halo and their uses as a mildewicide.
4232035 Carbamate pesticidal compounds compositions and methods of use  
Novel N-dithioalkyl and N-dithioaryl substituted cyclic carbamoyloximes exhibit exceptional pesticidal activity.
4218436 Compounds and methods  
A method for the radioimmunoassay of PGE 1 -type and PGE 2 -type compounds and PGX is disclosed which utilizes antibodies formed against a prostaglandin mimic. Conjugates are disclosed which are...
4207327 N-(4-Pyrazolidinyl)benzamides and their amino precursors  
N-(4-Pyrazolidinyl)benzamides having the formula ##STR1## and their amino precursors are disclosed wherein R is lower alkyl, lower cycloalkyl or phenyllower-alkyl; R 1 is lower alkyl, lower...
4178379 Substituted pyrano[4,3-c]pyrazoles, compositions containing same, and method of use  
2,4,6,7-Tetrahydropyrano[4,3-c]pyrazoles are provided having the formula ##STR1## wherein Z is O, S, SO or SO 2 ; R is H, halo, lower alkyl, lower alkoxy, lower alkanoyl, aroyl, cyano or CF 3 ;...
4174393 1,3,4-Substituted pyrazoline derivatives  
The invention relates to novel 1,3,4-substituted-Δ 2 -pyrazolines having an insecticidal activity. The compounds are particularly active against larvae of insects for example larvae of Colorado...
4156007 Pyrazoline compounds  
The invention relates to new 1,3,4-substituted Δ 2 -pyrazolines having an insecticidal activity. The compounds are active in particular against larvae of insects such as larvae of colorado...
4140792 Combating arthropods with 1-(substituted-phenylcarbamoyl)-3-halophenyl-2-pyrazolines  
1-(Substituted-phenylcarbamoyl)-3-halophenyl-2-pyrazolines of the forumla ##STR1## in which R represents hydrogen or alkyl, R 1 represents hydrogen or halogenophenyl, R 2 represents...
4140787 Combating arthropods with 1-[haloalkyl-phenyl)-carbamoyl]-3-(4-halophenyl)-2-pyrazolines  
1-[(Haloalkyl-phenyl)-carbamoyl]-3-(4-halophenyl)-2-pyrazoli nes of the formula ##STR1## in which R is halogen, R 1 is hydrogen or alkyl, R 2 is hydrogen or halogen, and R 3 is...
Matches 351 - 400 out of 408 < 1 2 3 4 5 6 7 8 9 >