Matches 301 - 350 out of 409 < 1 2 3 4 5 6 7 8 9 >
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5276037 Heterocyclic 5-lipoxygenase inhibitors  
The invention concerns an aryl derivative of the formula I, ##STR1## wherein Ar 1 is optionally substituted phenyl, naphthyl or a heterocyclic moiety, and X 1 is oxy, thio, sulphinyl, sulphonyl,...
5270043 Arthropodicidal composition comprising thiodicarb and a phenylpyrazole  
The invention provides arthropodicidal compositions comprising an arthropodicidally effective amount of (A) 5-amino-3-cyano-1-(2,6-dichloro-4-trifluoromethylphenyl)-4-t rifluoromethyl...
5256670 N-aryl-3-aryl-4-substituted- 2,3,4,5-tetrahydro-1H-pyrazole-1-carboxamides, insecticidal compositions containing such compounds and methods of controlling insects such compounds  
This invention relates to N-aryl-3-aryl-4-substituted-2,3,4,5-tetrahydro-1H-pyrazole-1 -carboxamide compounds which are useful as pesticides, compositions containing those compounds, methods of...
5252596 Phenoxyalkylamine derivative and method for controlling noxious organisms containing the same  
Disclosed are a novel phenoxyalkylamine compound represented by the following formula: ##STR1## wherein R 1 represents a lower alkyl group or a lower haloalkyl group; R 2 represents hydrogen atom...
5250561 Tetrahydroindazole, tetrahydrocyclopentapyrazole, and hexahydrocycloheptapyrazole compounds and their use as HMG-COA reductase inhibitors  
Compounds of the general formula I: ##STR1## are disclosed as useful in the treatment or prevention of hypercholesterolemia, hyperlipoproteinemia and atherosclerosis. Novel intermediate compounds...
5240947 2,3,4,5-substituted furo[2,3-c]pyrazole derivatives  
The present invention provides a novel series of 2,3,4,5-substituted furo[2,3-c]pyrazole compounds. These compounds are found potent in inhibiting thrombocyte aggregation and antiallergy effect.
5225432 Control of micro-organisms on plants with 1-hydroxymethylpyrazoles  
A method of protecting plants and seeds thereof which are susceptible to attack by microorganisms. To the plant or seed is applied a compound having the formula ##STR1## wherein R and R' are...
5223510 Alkylaminoalkyl derivatives of benzofuran, benzothiophene, indole and indolizine, process for their preparation and compositions containing them  
The subject of the invention is benzofuran, benzothiophene, indole or indolizine compounds of general formula: ##STR1## in which: Het represents one of the groups: ##STR2## in which T,T' and...
5218123 Didehydrotryptophan derivatives and pharmaceutical use thereof  
Novel didehydrotryptophan derivatives useful as agents in the reduction of gastric acid secretion and in the treatment of anxiety, psychoses, and the symptoms of cognitive decline are disclosed....
5208251 Styryl pyrazoles, isoxazoles and analogs thereof having activity as 5-lipoxygenase inhibitors, pharmaceutical compositions and methods of use therefor  
The present invention is 3,5-substituted, isoxazoles, pyrazoles, isothiazoles, and analogs thereof having 5-lipoxygenase or cyclooxygenase inhibiting activity or as a sunscreen.
5206258 Use of heteroaryl-3-oxo-propanenitrile derivatives in treating clinical wherein myelopoiesis suppression occurs  
Heteroaryl-3-oxo-propanenitrile derivatives of formula (I) ##STR1## wherein X represents an oxygen atom or a --CH(R 4 )--, --O--CH(R 4 )--,--S(O) n --, --S(O) n --CH(R 4 )--, --CH(R 4 )--O--,...
5196546 Selective pyrazoline insecticides and fungicides  
Certain pyrazolines have been found to be useful as aphicides and fungicides.
5196408 N-sulfenylated pyrazolines, compositions and use  
N-sulfenylated and N-acrylated pyrazoline arthropodicides, compositions containing them and methods for controlling arthropods by applying compounds of the invention to them or to their...
5189065 Use of derivatives of 9,10-dihydrophenanthrene for the preparation of an anti-tumor medicament  
The use of products of formula (I) is described, wherein X and Y represent hydrogen, hydroxy or alkoxy; and R 1 and R 2 represent H, alkyl, alkenyl or alkynyl, arylalkyl, acyl or R 1 and R 2 ...
5177072 Treatment of autoimmune inflammatory, and psoriatic diseases with heterocyclic aminoalkyl esters of mycophenolic acid and derivatives  
Heterocyclic aminoalkyl esters of mycophenolic acid, and the derivatives and pharmaceutically acceptable salts thereof, are useful as immunosuppressive agents, anti-inflammatory agents, anti-tumor...
5166169 Treating agent for peripheral circulatory disturbances  
A preventing and treating agent for peripheral circulatory disturbances containing a compound represented by formula (I): ##STR1## wherein R represents an imidazolyl group, a thiazolyl group, or a...
5153226 Acat inhibitors for treating hypocholesterolemia  
The present invention are novel amino acid amide compounds of the following general formula which inhibit the enzyme acylcoenzyme A:cholesterol acyltransferase: ##STR1## wherein R is phenyl or 1-...
5116850 Heterocyclic pyrazoline carboxanilides  
Heterocyclic pyrazoline carboxanilide insecticides including all geometric and stereoisomers thereof, as well as agricultural compositions containing them.
5109014 N-aryl-3-aryl-4-substituted-2,3,4,5-tetrahydro-1H-pyrazole-1-carboxamides  
This invention relates to novel N-aryl-3-aryl-4-substituted-2,3,4,5-tetrahydro-1H-pyrazole-1 -carboxamide compounds which are useful as pesticides, compositions containing those compounds, methods...
5108991 Vehicle composition containing 1-substituted azacycloalkan-2-ones  
Compositions useful for carrying physiologically active agents such as therapeutic agents through skin and other body membranes comprising the agent and an effective, non-toxic amount of a compound...
5106843 Heterocyclic compounds useful as 5-HT.sub.3 antagonists  
Aryl ureas and carbamic acid derivatives of formula A--NHCW--Y--B and pharmaceutically acceptable salts thereof wherein A is a specified aromatic radical including 3,5-dichlorophenyl W is O...
5095029 Fungicidal 1,3,5-triaryl-2-pyrazolines  
Combating fungi with 1,3,5-triaryl-2-pyrazolines of the formula ##STR1## in which R 1 , R 2 and R 3 are optionally substituted phenyl. Those compounds in which R 2 is phenyl, R 3 is...
5091405 Insecticidal pyrazolines  
Pyrazolines and their intermediates, including all geometric and stereoisomers of the pyrazolines and intermediates, agricultural compositions containing the pyrazolines, and methods for use as...
5070098 Substituted pyrazoline derivatives, pesticidal compositions and use  
This invention relates to novel substituted pyrazoline derivatives of the general formula ##STR1## processes for their preparation and their use as pesticides.
5068241 Pesticidal substituted pyrazoline derivatives, compositions and use  
Pesticidal substituted pyrazoline derivatives of the formula ##STR1## in which R 1 represents optionally substituted phenyl or optionally substituted alkyl, R 2 represents hydrogen, optionally...
5037815 Non-steroidal anti-inflammatory compositions protected against gastrointestinal injury with a combination of certain H.sub.1 - and H.sub.2 -receptor blockers  
A pharmaceutical composition and process for administering non-steroidal drugs which are protected againsts injury to the gastrointestinal tract by a combination of certain H 1 - and H 2 ...
5032591 Pharmaceutical preparations  
A pharmaceutical product comprising a potassium channel activator antihypertensive agent and a β-blocker antihypertensive agent as a combined preparation for simultaneous, separate or sequential...
5006548 Acrylamidobenzoic acid derivatives and their use  
Compounds of the general formula: ##STR1## wherein R 1 is heterocyclic group other than pyridyl and which is unsubstituted or substituted with lower alkyl or lower alkoxycarbonyl, R 2 is...
4999368 Selective pyrazoline insecticides and fungicides, compositions and use  
A pyrazoline having the formula: ##STR1## wherein: R 1 and R 2 are selected independently from a group consisting of hydrogen with the proviso that only one of R 1 and R 2 can be hydrogen,...
4999367 Ethers of 1-benzyl-3-hydroxymethyl-indazole with aliphatic 2-hydroxyacids, compositions and use  
Compunds of the formula A--CH 2 --O--CRR'--COOR'" (I) wherein A, R, R' and R'" have the meanings mentioned in the description, ts thereof with pharmaceutically...
4999359 Heterocyclic ethylene diamine compounds and their pharmaceutical compositions and methods  
A compound, or a solvate or salt thereof, of formula I: ##STR1## in which: R.CO-- is an acyl group containing a substituted or unsubstituted carbocyclic aromatic or heterocyclic aromatic group; ...
4997844 Indazole compounds, pharmaceutical compositions and use  
The invention provides a series of novel heterocyclic amides of the formula I in which the group A CRa can be --CRbCRa--, --CHRb--CHRa-- or --NCRa--, the amidic group Re.L can be Re.X.CO.NH,...
4977153 3-aminopropyloxyphenyl derivatives, pharmaceutical compositions containing them and method for the therapy of diseases  
Compounds of formula (I), ##STR1## characterized in that R signifies optionally substituted heteroaryl-, heteroarylakyl or heteroarylalkenyl, R 1 signifies hydrogen or a substituent, R 2 is...
4975444 Cycloalkyl-substituted glutaramide antihypertensive agents  
Compounds of the formula ##STR1## wherein A is a carbocyclic, saturated or unsaturated ring; R 1 is hydrogen or alkyl; R and R 4 are each alkyl, cycloalkyl, benzyl or a readily hydrolyzable ester...
4968676 Fungicidal cyclohexylamines  
Cyclohexylamines of the formula ##STR1## where X is a single bond or an alkylene chain, Y is hydrogen or an aryl, cyclohexyl, 4-cyclohexylcyclohexyl, perhydro-1- or 2-naphthyl or piperidyl radical,...
4960784 Insecticidal substituted indazoles  
Certain substituted indazoles, including all geometric and stereoisomers thereof, agricultural compositions containing the indazoles and use of the indazoles as insecticides.
4956378 4,5-dihydro pyrazole compounds  
There are described compounds of formula I, ##STR1## in which Ar 1 and Ar 2 , which may be the same or different, each independently represent phenyl or pyridinyl, the phenyl or the pyridinyl each...
4943585 N-substituted azoles and insecticide, arachnicide, and nematocide compositions thereof  
4897427 Method of combatting pruning wound diseases  
The invention relates to a method of combatting pruning wound diseases in plants employing a compound of the formula ##STR1## wherein X is H or Cl and R is butyl, 1-cyclopropyl-ethyl or...
4888340 Insecticides pyrazolines, compositions and use  
Compounds of formula I ##STR1## in which X, Y and Z have various meanings, are described, as well as processes for their preparation and their use as insecticides and acaricides.
4874778 1-carbamoyl-2-pyrazolines, composition containing them, and insecticidal and acaricidal method of using them  
The invention relates to 1-carbamoyl-3-phenyl-4-benzyl-Δ 2 -pyrazolines of the formula ##STR1## wherein R 1 and R 2 are each independently hydrogen, methyl halogen, trifluoromethyl, C 1 -C 4 ...
4871737 3-Amino-5-methyl-1H-pyrazole-4-carboxylic acids and esters thereof as anticonvulsants muscle relaxants and anxiolytics  
A novel method of controlling epilepsy, muscle tension, muscular spasticity, and anxiety in living animal bodies by administering compounds of the formula: ##STR1## wherein: R 1 is hydrogen,...
4867979 Antidiarrheal compositions and use thereof  
Antidiarrheal compositions showing enhanced antidiarrheal activity comprise a non-steroidal anti-inflammatory drug compound and a polymeric hydroabsorptive agent. A patient in need of remedial or...
4863947 N-aryl-3-aryl-4,5-dihydro-1H-pyrazole-1-carboxamides and methods of their production  
This invention relates to novel N-aryl-3-aryl-4,5-dihydro-1H-pyrazole-1-carboxamide compounds which are useful as pesticides, compositions containing those compounds, methods of controlling pests...
4861776 Heterocyclic aminoalkyl esters of mycophenolic acid and derivatives thereof, compositions and use  
Heterocyclic aminoalkyl esters of mycophenolic acid, and the derivatives and pharmaceutically acceptable salts thereof, are useful as immunosuppressive agents, anti-inflammatory agents, anti-tumor...
4851406 Heterocyclic-substituted indoles and pharmaceutical compositions containing them  
The present invention provides indole derivatives of the general formula: ##STR1## wherein R 1 is a hydrogen atom or an alkyl, alkenyl, cycloalkyl, cycloalkenyl, carboxyl, cyano, alkylcarbonyl,...
4837220 Insecticidal 3-substituted 4-fluorophenyl-1-(fluoroalkoxyphenylcarbamoyl)-pyrazolines  
Pyrazolines of general formula I ##STR1## wherein R 1 and R 2 are the same or different and are hydrogen or fluorine, are described, as well as processes for their preparation and their use as...
4833143 Antidepressant amines  
Compounds of formula I ##STR1## in which R 1 is a heterocyclic ring containing one or more heteroatoms selected from N, O and S; in which R 2 is H, a straight or branched chain alkyl group...
4826847 Beta-blocking oxindole derivatives  
The present invention provides oxindole derivatives of the formula: ##STR1## wherein the various substituents are defined hereinbelow. The above compounds display nitrate-like as well as...
4824859 Pyrazoline compounds compositions and use  
There are described compounds of formula I, ##STR1## in which Ar 1 and Ar 2 , which may be the same or different, each independently represent phenyl or pyridinyl, the phenyl or the pyridinyl each...
Matches 301 - 350 out of 409 < 1 2 3 4 5 6 7 8 9 >