Matches 151 - 200 out of 460 < 1 2 3 4 5 6 7 8 9 10 >
Match Document Document Title
6200997 Heterocyclyl-substituted phenyl compounds, processes and intermediates for their preparation and their use for controlling harmful fungi and animal pests  
The present invention relates to heterocyclyl-substituted phenyl compounds of the formula I, ##STR1## where the substituents have the following meanings: Y is halogen, C 1 -C 4 -alkyl, C 1 -C...
6200998 Arylthiazolidinedione derivitives  
Substituted 5-aryl-2,4-thiazolidinediones are potent agonists of PPAR, and are therefore useful in the treatment, control or prevention of diabetes, hyperglycemia, hyperlipidemia (including...
6194441 Oxazolidinone derivatives and their use as antibacterial agents  
The invention concerns a compound of formula (I) wherein for example R 1 is of the formula --NHC(O)R a wherein R a is hydrogen, or (1-4C)alkyl; R 2 and R 3 are independently hydrogen or...
6150371 Method for preventing and for treating autoimmune disease  
A method for preventing or treating autoimmune diseases (excluding type I diabetes) by administering an insulin resistance improving substance as an active ingredient.
6143772 Compounds derived from 3-(benzofuran-5-yl)oxazolidin-2-one, preparation method therefor and therapeutical use thereof  
Compounds derived from 3-(benzofuran-5-yl) oxazolidin-2-one, of general formula (I) ##STR1## in which: R 1 represents a phenyl group, a phenylmethyl group, an alkyl group or a fluoroalkyl group,...
6139858 Termite-controlling agent  
A termite-controlling agent comprising 5-tert-butyl-2-[2-(2,6-difluorophenyl)-4,5-dihydrooxazol-4-y l]phenetole as an active ingredient and cellulose, which can be a sheet formulation or a powdery...
6136832 5,5-disubstituted-3,4-dihydroxy-2(5H)-furanones and methods of use therefor  
The present invention relates to synthetic methods for the production of both optically active and racemic 5,5-disubstituted-3,4-dihydroxy-2(5H)-furanones;...
6127422 Anti-viral method  
A method of inhibiting an envelope virus selected from the group consisting of influenza bovine diarrheal, hepatitis C and tick borne encephalitis virus that udergoes hemagglutinin-mediated fusion...
6124334 Hetero-aromatic ring substituted phenyloxazolidinone antimicrobials  
A hetero-aromatic (Q) substituted phenyloxazolidinone antimicrobial of Formula I ##STR1## wherein Q is a 5-member hetero-aromatic having from one to four nitrogen atoms or alternatively a...
6117895 Pharmaceutical preparations for TNF inhibition  
Compounds of formula I ##STR1## are useful for treating TNF-mediated diseases.
6103768 Fatty acid based compositions and methods for the control of plant infections and pests  
The invention described here concerns the unique utility of fatty acids and their derivatives to eradicate existing fungal and bacterial infections in plants. Also, described herein are combination...
6096771 Isoxazole derivatives  
An isoxazole compound having the following formula: ##STR1## wherein R 1 represents hydrogen, halogen, alkyl, alkoxy, hydroxyl, alkylthio, amino, alkanoyl, alkanoylamino, alkanoyloxy,...
6090820 Spirocyclic and bicyclic diazinyl and carbazinyl oxazolidinones  
A compound of structural Formula I or II which is useful for treating microbial infections in humans or other warm-blooded animals, or pharmaceultically acceptable salts thereof as defined herein....
6087385 Flavonoid derivatives  
The present invention provides thiazolidinediones which are useful as antiproliferative, antiinflammatory and antiinfective agents. These compounds are useful for the treatment of certain endocrine...
6086905 Topical compositions useful as skin penetration barriers  
Methods for preventing the penetration of toxic chemicals through the stratum corneum of the skin of a mammal are disclosed which employ, as a penetration prevention agent, at least one compound...
6083967 S-oxide and S,S-dioxide tetrahydrothiopyran phenyloxazolidinones  
The present invention provides compounds of formula I and formula II useful as antimicrobial agents wherein R 1 is methyl, ethyl, cyclopropyl, or dichloromethyl; R 2 and R 3 are independently...
6075023 Method for combatting fish mycoses and one-celled ectoparasites  
6060501 Combined treatment of multiple sclerosis  
A pharmaceutically composition for treating MS comprising an effective amount of a combination of a PDE IV inhibitor and an anti-inflammatory and immunomodulatory drug in a pharmaceutically...
6057351 Compounds of the 3-aryl 2,4 dioxo oxazolidine family and use thereof in cosmetic and pharmaceuticals  
6051590 Immunosuppressant tricyclic compounds  
The compounds of Formula I are useful as immunosuppressive agents.
6040306 Method of treating psoriasis, arthritis and reducing the toxicity of cancer chemotherapy  
The present invention is a method of treating a person who has psoriasis or arthritis or reducing the toxicity of cancer chemotherapy which comprises administering to the patient an anti-psoriasis...
6040317 Sulfonamide fibrinogen receptor antagonists  
A series of non-peptide derivatives that are antagonists of the fibrinogen IIb/IIIa receptor and thus are platelet anti-aggregation compounds useful in the prevention and treatment of diseases...
6040328 Aromatic diselenides and selenosulfides, their preparation and their uses, more particularly their therapeutical use  
The objects of the present invention are: novel organoselenium compounds: aromatic diselenides and selenosulphides; the use of said novel compounds as antioxidant agents; pharmaceutical...
6034081 Potentiation of biocide activity using an N-alkyl heterocyclic compound  
A method for increasing the effectiveness of a microbicide is described, wherein a microbicide and an N-alkyl heterocyclic compound are applied to a substrate or aqueous system subject to the...
6034101 ***WITHDRAWN PATENT AS PER THE LATEST USPTO WITHDRAWN LIST***
Dosage form and method for administering drug  
A dosage form and a method are disclosed and claimed for administering a drug in a sustained and constantly ascending rate per unit time to provide an intended therapeutic effect while...
6028090 Adhesion receptor antagonists III  
Novel oxazolidinone derivatives of the formula I ##STR1## in which R 1 is a phenyl radical which is unsubstituted or is monosubstituted by CN, H 2 N--CH 2 --, A 2 N--CH 2 --, H 2 ...
6025374 Azetidine, pyrrolidine and piperidine derivatives as 5HT1 receptor agonists  
A class of substituted azetidine, pyrrolidine and piperidine derivatives are selective agonists of 5-HT 1 -like receptors, being potent agonists of the human 5-HT 1D α receptor subtype whilst...
6025376 Chiral methylphenyloxazolidinones  
This invention relates to (R)-(-)-methylphenyloxazolidinone derivatives, a process for their production and their use as pharmaceutical agents.
6008237 Arylthiazolidinedione derivatives  
Substituted 5-aryl-2,4-thiazolidinediones are potent agonists of PPAR, and are therefore useful in the treatment, control or prevention of diabetes, hyperglycemia, hyperlipidemia (including...
5998453 Oxazolidinone compounds and pharmaceutical preparation containing them  
Pharmaceutical preparations for the local treatment of inflammations are claimed herein, characterized in that they contain as the active ingredient one or two compounds of general Formula I...
5990135 Retroviral protease inhibiting compounds  
A retroviral protease inhibiting compound of the formula: ##STR1## is disclosed.
5981559 Azole derivative with leukotriene (LTs) antagonizing activity and thromboxane (TX) A.sub.2 antagonizing activity  
An azole derivative represented by general formula (I) or a pharmaceutically acceptable salt thereof, having both of a leukotriene antagonistic effect and a thromboxane A2 antagonistic effect and...
5968958 5-Methanesulfonamido-3H-isobenzofuran-1-ones as inhibitors of cyclooxygenase-2  
The invention encompasses the novel compound of Formula I as well as a method of treating cyclooxygenase-2 mediated diseases comprising administration to a patient in need of such treatment of a...
5962486 Indole derivatives as prodrugs of 5-HT.sub.1 -like receptor agonists  
A compound of formula (I), wherein A is C 1 -6 alkyl, --O--C 1 -6 alkyl, --O--phenyl or phenyl, optionally substituted by C 1 -3 alkyl or halogen; n is an integer of from 0 to 3; W is a group of...
5948805 Fungicidal mixtures  
Advantageous combinations of an oxazolidinone and cymoxanil (or their agriculturally suitable salts) and their use to control fungus disease in plants are disclosed, the oxazolidinone having the...
5942535 a!-Annelated pyrrole derivatives and pharmaceutical use thereof  
The present invention relates to heterocyclic compounds of the formula ##STR1## in which R 1 -R 7 , B, a and X have the meanings recited in the specification. These compounds are usable in the...
5935973 Heterocyclcarboxamide derivatives and their use as therapeutic agents  
Compounds of formula I ##STR1## and pharmaceutically acceptable salts thereof in which A is methylene or O; B is methylene or O; g is 0,1,2,3 or 4; R 1 is an optional substituent; U is an alkylene...
5925662 Compounds derived from oxazolidin-2-one and preparation and therapeutical use thereof  
Derivatives of oxazolidin-2-one of general formula (I) ##STR1## in which: n is equal to 0 or 1, R 1 represents a cyano group, an alkyl group or a fluoroalkyl group, R 2 represents a...
5919809 3-substituted-2-oxindole derivatives  
This invention relates to novel 3-substituted-2-oxindole derivatives of the formula ##STR1## and the pharmaceutically-acceptable salts thereof which are inhibitors of prostaglandin H 2 synthase,...
5906832 Method for treating epilepsies  
A dosage form is disclosed for delivering an antiepileptic drug, which dosage form comprises for maintaining the integrity of the dosage form and of the antiepileptic drug.
5905072 Adjuvants for systemic fungicides, fungicidal compositions which contain them and their use  
Adjuvants for systemic fungicides in the form of a stable microemulsion comprise water, a mixture of methyl esters of fatty acids obtained by the transesterification of vegetable oils, an anionic...
5900427 N-heteroarenesulfonyl-protected amino acid reagents for peptide synthesis  
This invention relates to the use of heteroarenesulfonyl groups as protecting groups for amino groups, particularly the amino groups of amino acids, and specifically to nitrogen-protected...
5891898 Method for treating or preventing ulcerative diseases by administering thia- or oxazolidinone compounds  
A method for the treatment or prevention of an ulcerative disease comprising administering to a patient an effective amount of an active compound in admixture with a pharmacologically acceptable...
5889025 Antidiabetic compounds having hypolipidaemic, antihypertensive properties, process for their preparation and pharmaceutical compositions containing them  
Novel antidiabetic compounds, their tautomeric forms, their derivatives, their steroisomers, their polymorphs, their pharmaceutically acceptable salts, their pharmaceutically acceptable solvates...
5886014 Benzimidazole derivatives, their preparation and their therapeutic use  
Compounds of formula (I): ##STR1## wherein: X represents an optionally substituted benzimidazole group; Y represents an oxygen or sulfur atom; Z represents a 2,4-dioxothiazolidin-5-ylidenylmethyl,...
5883093 Phenyloxazolidinone antimicrobials  
The present invention relates to antimicrobial phenyloxazolidinone compounds having a pyrrolidinyl or azetidinyl moiety.
5866582 Fungicidal combination of a dicarboximide compound and cyprodinil  
Fungicidal combination comprising a compound A which is iprodione, vinclozoline or procymidone, and a compound B which is cyprodinil, also known as 2-phenylamino-4-cyclopropyl-6-methylpyrimidine,...
5866596 3,4-diaryloxazolone derivatives, their methods of preparation and their uses in therapeutics  
The present invention relates to the derivatives of formula: ##STR1## and to their use in therapeutics, especially as drugs with anti-inflammatory and analgesic properties.
5861424 Composition and method for treating cancer  
A pharmaceutical composition for treatment of cancer in a mammal comprising: (A) a therapeutically effective amount of at least one compound selected from the group consisting of compounds...
5861429 13-substituted milbemycin 5-oxime derivatives, their preparation and their use against insects and other pests  
Compounds of formula (I): ##STR1## wherein: R 1 is methyl, ethyl, isopropyl or sec-butyl; X is carbonyl or methylene; Z is C(R 2 ) 2 or C(CH 2 ) m , in which R 2 is alkyl, and m is...
Matches 151 - 200 out of 460 < 1 2 3 4 5 6 7 8 9 10 >