Matches 201 - 250 out of 301 < 1 2 3 4 5 6 7 >
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5254595 Aryloxypropanolaminotetralins, a process for their preparation and pharmaceutical compositions containing them  
Aryloxypropanolaminotetralins with beta-antagonist activity of the formula ##STR1## wherein R is hydrogen, hydroxy or methoxy and Ar is an optionally substituted aromatic or heteroaromatic group,...
5223517 Heterocyclically substituted cycloalkano[b]-indolesulphonamides  
Heterocyclically substituted cycloalkano[b]-indolesulphonamides can be prepared by reaction of appropriate N-unsubstituted indoles with acrylonitrile, followed by hydrolysis, esterification or...
5221686 Spiro[1,2-benzisothiazole-3(2H),5'-oxazolidine]-2',4'-dione 1,1-dioxides as antihyperglycemic agents  
This invention relates to novel spiro[1,2-benzisothiazole-3(2H),5'-oxazolidine]-2',4'-dione 1,1-dioxides characterized by the general formula (I), ##STR1## wherein R is lower alkyl containing 1 to...
5219842 Method of improving intestinal floras  
A β-glucooligosaccharide-containing composition comprising at least one material selected from food, drink and medicine, and at least one selected from a glucooligosaccharide comprising at least...
5219875 Antimicrobial compositions comprising iodopropargyl butylcarbamate and 1,2-benzisothiazolin-3-one and methods of controlling microbes  
A synergistic antimicrobial composition comprising 1,2-benzisothiazolin-3-one and iodopropargyl butylcarbamate in a ratio to each other which exhibits synergism is disclosed.
5187173 2-saccharinylmethyl and 4,5,6,7-tetrahydro-2-saccharinylmethyl phosphates, phosphonates and phosphinates useful as proteolytic enzyme inhibitors and compositions and method of use thereof  
4-R 1 -R 2 -R 3 -2-Saccharinylmethyl, 4-R 4 -4-R 5 -6-R 6 -4,5,6,7-tetrahydro-2-saccharinylmethyl and 4,7-C-4,5,6,7-tetrahydro-2-saccharinylmethyl phosphates, phosphonates and phosphinates of...
5185356 Three component biocidal isothiazolinone composition  
A particulate composition comprising an isothiazolinone or isothiazolothione or a salt or complex thereof and a water soluble metal salt. The salt is typically a metal salt, for example the sodium...
5160526 Alkene stabilizers for 3-isothiazolone compounds  
A method of stabilizing a 3-isothiazolone compound against chemical decomposition comprising introducing a sufficient amount of an alkene to stabilize said 3-isothiazolone compound and a...
5153189 Sulfimidoperoxycarboxylic acids  
Sulfimidoperoxycarboxylic acids of the formula ##STR1## in which A is a group of the formula ##STR2## n is the number 0, 1 or 2, R 1 is hydrogen, fluorine, chlorine, bromine, C 1 -C 20 - alkyl,...
5145501 Bromate stabilizers for 3-isothiazolones  
A composition comprising (a) a 3-isothiazolone compound of the formula ##STR1## wherein R and R 1 are independently selected from hydrogen, halogen or R is a (C 1 -C 4 ) alkyl group and R 1 ...
5128339 Proteolytic enzyme inhibition method  
4-R 4 -R 5 -2-Saccharinylmethyl aryl carboxylates, useful in the treatment of degenerative diseases, are prepared by reacting a 4-R 4 -R 5 -2-halomethylsaccharin with an arylcarboxylic acid in...
5114960 Substituted isoxazole derivatives  
Compounds of the formula ##STR1## wherein A taken together with the two carbon atoms denoted as α and β is a group of the formula ##STR2## and the dotted line is the double bond present in...
5036082 Insectidical nitro-substituted heterocyclic compounds  
Nitro-substituted heterocyclic compounds of the formula (I) ##STR1## wherein R is hydrogen or alkyl, Z is an optionally substituted aryl or optionally substituted heterocyclic group containing at...
5021438 1,3,4,5-tetrahydrobenz(c,d)indoles  
Novel compounds having an affinity for 5-hydroxytryptamine receptors of the formula ##STR1## in which R 1 stands for H, alkyl, aralkyl or heteroarylalkyl, X stands for H, OCH 3 , OH, SCH 3 ,...
5001115 Prodrugs of biologically active hydroxyaromatic compounds  
Prodrugs of bio-active hydroxyaromatic drugs having the structural formula: A pharmaceutically acceptable prodrug of a biologically active, therapeutically effective hydroxyaromatic drug, said...
4987146 N-hetaryl imidazole derivatives  
N-hetaryl imidazole derivatives of general Formula I ##STR1## are disclosed in which Het represents an optionally substituted monocyclic or bicyclic heteroaromate, R 3 represents hydrogen, a...
4960781 Fungicidal disazolyl-hydroxyalkyl derivatives  
Fungicidal bisazolyl-hydroxyalkyl derivatives of the formula ##STR1## in which Ar stands for optionally substituted aryl, X stands for a grouping --CH 2 CH 2 --, --OCH 2 --, --SCH 2 -- or...
4957931 Certain 1,2-benzisoxazole and 1,2-benzisothiazole derivatives  
Disclosed are 1,2-benzisoxazole and 1,2-benzisothiazole derivatives represented by formula I ##STR1## wherein X represents oxygen or sulfur; Z represents carbon (CH) so as to complete the...
4943307 Plant-protective pesticidal composition  
The invention relates to a plant-protective solution containing 2.5 to 40 % by weight of one or more water-insoluble plant-protective ingredient(s) 20 to 71.5 % by weight of dimethylformamide...
4923887 Liquid formulations of 1,2-benzisothiazolin-3-one, their preparation and their use  
Antimicrobially active liquid composition formulation which comprises 1,2-benzisothiazolin-3-one and at least one amine-oxyethylate of the formula ##STR1## wherein R is alkyl or alkenyl each having...
4915943 Compositions containing biosynthetic pesticide products, processes for their production and their use  
The compositions contain a biosynthetic pesticide product, preferably originating from microorganisms of the genus Bacillus, in suspension in a liquid and at least one substance of general formula:...
4900739 Novel spirosuccinimides as aldose reductase inhibitors and antihyperglycemic agents  
This invention relates to novel spirosuccinimide derivatives, to the processes for their preparation, to methods for using the compounds, and to pharmaceutical preparations thereof. The compounds...
4880802 Substituted basic 2-aminotetralin useful as cardiotonic agents  
For treatment of disorders of the central nervous system, the cardiovascular system or the intestinal tract, the new substituted basic 2-aminotetralins of the formula ##STR1## in which R 1 ...
4871754 Aqueous formulation of 1,2-benzisothiazolin-3-one  
Aqueous solutions are protected from infestation by micro-organisms by use of a biocide which is an aqueous formulation of the lithium salt of 1,2-benzisothiazolin-3-one.
4866081 Microbicidal preservative composition  
A composition comprising 2-(thiocyanomethylthio)benzothiazole and 3-iodo-2-propinyl-N-butylcarbamate. The composition can be useful as a microbicidal preservative to prevent deterioration of raw...
4855311 Benzoisothiazole oximes which are plant protection agents for control of fungi and bacteria  
Derivatives of benzoisothiazole oxime which exhibit marked effect when used in plant protection agents for control of fungi and bacteria. They are of particular utility for the prevention of rice...
4849438 1,2-benzoisothiazol-3(2H)-one 1,1-dioxide, ion(1-),2-hydroxy-N,N,N-trimethyl-ethanaminium which is plant protection agent for control of fungi and bacteria  
1,2-benzoisothiazol-3(2H)-one, 1,1-dioxide, ion(1-),2-hydroxy-N,N,N-trimethyl-ethanaminium represented by the following formula (I): ##STR1## is found to have great utility as an effective...
4845098 Saccharine salts of substituted hydroxypropylamines, compositions and use  
Fungicidal saccharine salts of substituted hydroxypropylamines of the formula ##STR1## in which R 1 is optionally substituted phenyl, phenoxy, phenylthio, phenylalkyl, phenoxyalkyl, or...
4831033 Use of amodiaquin in treatment of nervous system degeneration  
A procedure for the treatment of degenerative diseases of the central nervous system, including Alzheimer's disease, multiple sclerosis and the like, by the administration of amodiaquin and related...
4829063 Saccharine salts of substituted amines  
Fungicidally active novel saccharine salts of substituted amines of the formula ##STR1## in which A represents in each case optionally substituted 2-decahydronaphthyl or β-naphthyl and R 1 and...
4826836 Saccharine salts of aminomethyl heterocyclic compounds, compositions and use  
Fungicidally active novel saccharine salts of aminomethyl heterocyclic compounds of the formula ##STR1## in which R represents optionally substituted cycloalkyl, optionally substituted aryl or...
4824844 Saccharine salts of substituted amines, fungicidal compositions and use  
Fungicidally active saccharine salts of substituted amines of the formula ##STR1## in which A represents in each case optionally substituted cyclohexyl, cyclohexenyl or phenyl, R 1 represents...
4808605 Tetrahydronaphthalene derivatives as calcium antagonists  
Compounds of the formula ##STR1## wherein R is lower-alkyl, R 1 is halogen, R 2 is C 1 -C 12 -alkyl, R 3 is hydroxy, lower-alkoxy, lower-alkyl-carbonyloxy,...
4801591 2-alkenylene-thieno-1,2-thiazole derivatives with lipid-lowering activity  
The invention relates to new thieno-1,2-thiazole derivatives of the formula ##STR1## wherein A, with the two carbon atoms of the thiazole ring, forms a group of the formula ##STR2## and the broken...
4800202 Aminomethyltetrahydrofurans, fungicidal compositions and use  
Fungicidally active aminomethyltetrahydrofurans of the formula ##STR1## in which A represents a divalent alkylene or alkenylene chain which is in each case optionally substituted and R 1 and R...
4786650 3-acylaminobenzisothiazole-S,S-dioxide and insecticidal compositions and methods  
The invention relates to a novel 3-acylaminobenzisothiazole-S,S-dioxide of formula I ##STR1## to the preparation thereof, to insecticidal compositions containing said compound and to the use...
4777168 Bicyclic benzo-oxy heterocyclic ethers and thioethers, pharmaceutical compositions and use  
A class of bicyclic benzo-oxy heterocyclic ether and thioether compounds exhibiting parmacological activity, including anti-secretory and anti-ulcerogenic activity, pharaceutical compositions...
4764527 Hydroxypyrazole derivatives, composition containing them and their use against microorganisms  
1-Hydroxypyrazoles of the formula ##STR1## where R 1 , R 2 and R 3 independently of one another are each hydrogen or halogen, and microbicides containing these compounds.
4760076 Benzisothiazole derivatives and their use as insecticides  
The invention relates to the use of 3-acylaminobenzisothiazole-S,S-dioxides of the formula I ##STR1## wherein R 1 is C 1 -C 10 alkyl, phenyl, or C 1 -C 10 alkyl which is substituted by halogen...
4748164 Bicyclic benzonoid alkylene amino thieno [3,4-D] isothiazole ethers and thioethethers, pharmaceutical compositions and use  
A class of bicyclic benzenoid aminoalkylene ether and thioether compounds exhibiting pharmacological activity, including anti-secretory and anti-ulcero-genic activity, pharmaceutical compositions...
4728662 1,2-benzisoxazoloxyacetic acids and related compounds  
Novel 1,2-benzisoxazoloxyacetic acids and related compounds, methods for preparing same and methods of treatment by administering compositions containing such a compound are described. These...
4725612 Synergistic microbiocidal compositions containing a mixture of a bicyclic polyoxymethylene oxazolidine and a 1,2-benzisothiazolin-3-one  
A synergistic microbiocidal composition for inhibiting bacterial growth comprising Component (1) having the formula: ##STR1## in which R represents hydrogen or a halogen atom, and alkali ammonium...
4713389 Fungicidally and bactericidally active acylated saccharin derivatives  
Fungicidally and bactericidally active novel acylated saccharins of the formula ##STR1## in which X is oxygen or sulphur and R is --CO--R 1 or --SO 2 --OR 2 , R 1 is alkyl, halogenalkyl,...
4708959 4,5-trimethylene-4-isothiazoline-3-ones and their use as a bactericide and fungicide agent  
A 4,5-trimethylene-4-isothiazoline-3-one of the formula ##STR1## wherein R 1 represents (i) hydrogen, (ii) alkyl having 1-12 carbon atoms, (iii) alkyl having 2 or 3 carbon atoms and substituted by...
4703044 Imidazoquinolines containing other heterocyclic groups, useful as anti-ulcer or anti-secretory agents  
The invention provides novel imidazoquinolines, processes for their preparation and pharmaceutical compositions containing them. The compounds have Formula I ##STR1## wherein A is a C 1 -C 4 ...
4699906 Bicyclic benzenoid alkylene amino thieno[3,4-d]isothiazole ethers and thioethers, pharmaceutical compositions and use  
A class of bicyclic benzenoid aminoalkylene ether and thioether compounds exhibiting pharmacological activity, including anti-secretory and anti-ulcerogenic activity, pharmaceutical compositions...
4698358 Use of 3-acylaminobenzisothiazoles for controlling pests  
The use in pest control of 3-acrylaminobenzisothiazoles of the formula I ##STR1## wherein R 1 is unsubstituted or substituted alkyl or phenyl, R 2 , R 3 , R 4 and R 5 independently of one...
4683233 Salts of 2-keto-2H, 3H-1,2-benzisothiazole 1,1-dioxide as microbicides  
A method of combating fungi and bacteria which comprises applying to such fungi, bacteria or a habitat thereof, a fungicidally or bactericidally effective amount of at least one salt of 3-keto-2-,...
4666930 3-hydrazono-benzisothiazole 1,1-dioxide fungicides  
Compounds of the formula ##STR1## in which R 1 is alkyl, cycloalkyl, aryl or hydrogen, R 2 is --CO--R 3 , R 3 is alkyl, alkenyl or cycloalkyl, or is phenyl which is optionally substituted,...
4661504 Denatonium saccharide compositions and method of use  
A composition consisting essentially of an effective amount of denatonium saccharide which has a vile, bitter taste, a solvent which provides the composition with the capability of penetrating the...
Matches 201 - 250 out of 301 < 1 2 3 4 5 6 7 >