Matches 301 - 350 out of 443 < 1 2 3 4 5 6 7 8 9 >
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4876265 Process and compositions for controlling mites parasitizing on honey bees  
A process for controlling parasitic honeybee mites, such as Varroa jacobsoni, Acarapis woodi and Tropilaelaps clareae, by the use of 2-(2,4-dimethylphenylimino)-3-methylthiazoline or an acid...
4861789 Dihydro-indene-amine-dihydrooxazoles  
A compound of formula (I): ##STR1## or a pharmaceutically acceptable acid addition salt and/or a pharmaceutically acceptable solvate thereof, wherein A represents a residue of a benzene ring...
4859684 (1H-imidazol-1-ylmethyl) substituted benzimidazole derivatives and use thereof in treating androgen dependent disorders  
Novel (1H-imidazol-1-ylmethyl) substituted benzimidazole derivatives, compositions containing the same, and methods of treating androgen dependent disorders in mammals.
4857328 Skin therapeutic mixture containing aloe vera extract  
According to the present invention, a skin therapeutic mixture is useful for the alleviation of certain skin disorders such as acne, psoriasis, burns, pimples, blackheads, and open sores, and such...
4851406 Heterocyclic-substituted indoles and pharmaceutical compositions containing them  
The present invention provides indole derivatives of the general formula: ##STR1## wherein R 1 is a hydrogen atom or an alkyl, alkenyl, cycloalkyl, cycloalkenyl, carboxyl, cyano, alkylcarbonyl,...
4851422 Antibiotic 2-(3-oxo-2-isoxazolidinyl)-5-oxo-2-tetrahydrofuran-carboxylates  
The compound represented by the formula: ##STR1## where R 1 stands for amino or an organic residue bonded through nitrogen; R 2 stands for carboxyl or a group derivable therefrom; R 3 , R 4 , R 5...
4837242 Thiazoles and pyrazoles as fungicides  
Heterocyclic derivatives represented by the following formula have excellent preventive, curative and systemic controlliing effects on various plant microbes. ##STR1## wherein R 1 represents a...
4831032 Cardiotonic benzimidazoles  
The present invention provides benzimidazoles of the general formula: ##STR1## wherein R 1 , X, A, and R 2 are as defined in the specification. The present invention also provides processes for...
4826861 Novel heterocyclic compounds substituted with an amino group, their processes of manufacture and the pharmaceutical compositions containing them  
This invention relates to 2-aminothiazoles and to their process of manufacture. These compounds are endowed with potent antimicrobial and antifungic properties. They are useful in antibacterial and...
4814341 2-guanidino-4-(2-furyl) thiazoles as antiulcer agents  
A series of novel thiazole compounds, having a guanidino or substituted guanidino group at the 2-position and a 5-(N,N-disubstituted aminomethyl)-2-furyl group at the 4-position. The compounds of...
4810719 Anti-inflammator 1,n-diarylpyrazol-3-amines  
There are described compounds of formula I, ##STR1## in which either R 2 represents hydrogen, alkyl or Ar 2 , and R 3 represents hydrogen, alkyl or alkyl substituted by Ar 3 ; or R 2 and...
4808588 Heterocyclic ureas and carbonates useful as pharmaceuticals  
Compounds of formula (I), or a pharmaceutically acceptable salt thereof: ##STR1## wherein: Het is monocyclic heteroaryl having two adjacent carbon atoms, a and b, depicted in formula (I); p1 R 1 ...
4798838 Certain pyridinyl or imidazolinyl-4-thiazolyl-phenoxy alkanoic acid derivatives having lipid lowering activity  
The present invention relates to novel phenoxy derivatives represented by the formula (I): ##STR1## wherein: A is an imidazolyl group, a pyridyl group, a pyridyloxy group, an oxo-substituted...
4795755 Heterocyclic derivatives  
This invention relates to heterocyclic derivatives which are histamine H-2 antagonists and which inhibit gastric acid secretion. According to the invention there is provided a guanidine derivative...
4788209 Antifungal 2-anilinothiazolines  
Fungal infections of the skin and mucous membranes may be controlled by topical administration of a pharmaceutical composition comprising a N-(3- or 4-alkylphenyl)4,5-dihydro-2-thiazolamine.
4786639 Method for the treatment of reversible airways obstruction and asthma  
A method for the treatment and/or prophylaxis of reversible airways obstruction and asthma in mammals, which method comprises administering to the mammal in need of said treatment an effective...
4785008 N-substituted 2-amino-thiazoles, process for their preparation and their therapeutic application  
The subject of the invention is N-substituted 2-aminothiazoles of formula ##STR1## in which: X is a C--H group or a nitrogen atom, R 1 and R 2 are, independently of each other, a hydrogen...
4782083 3,4-dihydro-2H-1-benzopyrans useful as anti-hypertensive agents  
Compounds of formula (I) and pharmaceutically acceptable salts thereof: ##STR1## wherein: one of R 1 and R 2 is hydrogen or C 1 -4 alkyl and the other is C 1 -4 alkyl or R 1 and R 2 together...
4772603 Method for treating congestive heart failure, angina, occlusive peripheral vascular disease or cerebral vascular disease in mammals  
A method for the treatment and/or prophylaxis of congestive heart failure, angina, occlusive peripheral vascular disease or cerebral vascular disease in mammals, such as humans, which method...
4771062 Diaryl sulphide derivatives  
A diaryl sulphide derivative of the formula ##STR1## in which R 1 represents a thiazolamino radical of the formulae ##STR2## wherein R 5 represents hydrogen, alkyl, aralkyl or acyl, R 6 and R...
4761422 (2-amino-4-aryl-thiazole-5-yl)ethanols and their derivatives having diuretic activity and methods for preparing the same  
This invention relates to a series of thiazole derivatives having the general formula ##STR1## The compounds of the invention have an interesting diuretic activity and low toxicity.
4738963 Method for the treatment of incontinence in mammals  
A method for the treatment and/or prophylaxis of incontinence in mammals, which method comprises administering to the mammal in need of said treatment an effective amount of a compound of formula...
4735957 Thiazole derivatives, processes for the preparation thereof and pharmaceutical composition comprising the same  
New thiazole derivatives of the formula: ##STR1## wherein R 1 is lower alkyl, carboxy, a drivative of carboxy, hydroxymethyl, halomethyl, lower alkylthiomethyl, hydroxyiminomethyl or alkenyl which...
4720493 Thienylthiazole compounds  
Thienylthiazole compounds of the formula: ##STR1## and pharmaceutically acceptable acid addition salts thereof, wherein: R is amino, guanidino, alkylamino, alkenylamino, unsubstituted or optionally...
4698357 2,4-dichloro-5-nitro-thiazole  
The compound 2,4-dichloro-5-nitro-thiazole of the formula ##STR1## is microbicidally active.
4695567 Pyrrolobenzimidazoles, pharmaceutical compositions containing them and method of using them to treat certain heart and circulatory diseases  
The present invention provided pyrrolobenzimidazoles or tautomer thereof, of the general formula: ##STR1## wherein R 1 is hydrogen, C 1 -C 6 alkyl, C 2 -C 6 alkenyl or C 3 -C 7 cycloalkyl; ...
4684664 Derivatives of β-(4-isocyano-1,2,3,4-diepoxycyclopentyl) acrylic acid  
Disclosed herein are derivatives of β-(4-isocyano-1,2,3,4-diepoxycyclopentyl)acrylic acid, the derivatives showing an antibacterial activity, an antifungal activity and an antimycoplasmal activity.
4683228 Guanidinopyrazolylamides, guanidimoimidazolylamides, compositions containing them, and method of using them to inhibit gastric acid secretion  
A guanidine derivative of the formula I: ##STR1## in which R 1 , R 2 , R 3 , R 4 , ring X and D are a variety of radicals defined in the specification and A is a 3-8C alkylene chain which is...
4681883 Histamine H.sub.2 -antagonist oxazole and thiazole derivatives and compositions therefor  
This invention relates to aminoalkylphenoxyalkyl substituted heterocycles. These compounds antagonize the action of histamine on histamine H 2 -receptors in the brain. A compound of the invention...
4680300 Anti-inflammatory guanidines  
A compound having the formula ##STR1## where Ar=naphthyl, biphenyl, or quinolinyl; X=oxygen or NH; Y=2 to 8; R 1 =phenyl, substituted phenyl, hydrogen, lower alkyl; and R 2 is the...
4678775 Method of controlling pests  
A method of controlling a pest which comprises bringing into contact with the pest a pest-controlling amount of an agent selected from the group consisting of (1) a non-formamidine -p-octopamine...
4665083 Iminothiazolidine derivatives  
The invention relates to novel iminothiazolidine derivatives of the formula (I), ##STR1## wherein R 1 and R 3 represent, independently from each other, hydrogen or lower alkyl group, R 3 is...
4663341 Insecticidal n-aryl-3-aryl-4,5-dihydro-1h-pyrazole-1-carboxamides  
This invention relates to N-aryl-3-aryl-4,5-dihydro-1H-pyrazole-1-carboxamide compounds which are useful as pesticides, compositions containing those compounds, methods of controlling pests and...
4659727 Ethene derivatives  
Ethene derivatives of the formula: [R 5 (R 1 CR 4 CR 2 R 3 ) m ] n I wherein R 5 represents optionally substituted heterocyclyl or a group --CR 4 CR 2 R 3 , or optionally...
4656184 2-(N-substituted hydrazone), thiazoles useful as anti-inflammatories  
This invention relates to therapeutic compositions comprising, as active ingredient, N-substituted hydrazones having the formula: ##STR1## in which Z is a 2-thienyl or phenyl radical. Said...
4652575 2-(ethylene-thio methyl furanyl)amino thiazole derivatives having acid secretion inhibiting activity  
Compound of formula (I) ##STR1## wherein R is an alkyl or an aromatic group, having pharmaceutical utility as an agent for treating a condition mediated through gastric acid secretion for reducing...
4649145 Thiazole derivatives  
New thiazole derivatives of the general formula I ##STR1## and their salts with physiologically acceptable acids are described as well as a process for their manufacture. The new compounds exhibit...
4647557 Novel heterocyclic derivatives bearing an amino radical, processes for their production and the pharmaceutical compositions containing them  
This invention relates to novel heterocyclic derivatives bearing an amino group and to processes for making said compounds. More particularly this invention provides novel heterocyclic compounds...
4636516 3,5-di-tert-butyl-4-hydroxyphenyl-substituted heterocyclic compounds  
Novel 3,5-di-tert-butyl-4-hydroxyphenyl-substituted heterocyclic compounds shown by the formula ##STR1## wherein .circle.Het -- represents a specific heterocyclic group and the salts thereof. The...
4622330 Antiprotozoal 3-amino or substituted amino pyrazoles  
Novel 3-amino or substituted amino pyrazoles are disclosed as having antiprotozoal and antiparasitic activity in particular anticoccidial activity and are useful for controlling cecal and or...
4616025 Thiazolidine derivatives, process for the preparation and pharmaceutical compositions thereof  
New thiazolidine compounds of the formula (I) having anti-ulcer activity are disclosed: ##STR1## wherein Ar is a 2-furyl or a phenyl, naphthyl or pyridyl group optionally substituted by one or more...
4598154 Thiazole intermediates for cephalosporin compounds  
A cephalosporin compound of the formula: ##STR1## wherein R 1 is hydrogen or lower alkyl; R 2 is acetoxy or (1-methyl-1H-tetrazol-5-yl)thio, and R 3 is carboxy; or R 2 is a group of...
4585781 Heterocyclic derivatives  
This invention relates to compounds of the general formula (I) ##STR1## and physiologically acceptable salts and hydrates thereof, in which R 1 represents a hydrogen atom or an alkyl, alkanoyl,...
4582842 Anti-asthmatic 6H-dibenz-[b,e] [1,4]oxathiepin derivatives, compositions, and method of use therefor  
Novel 6H-dibenz[b,e] [1,4]oxathiepin derivatives of the formula I and Ia are employed in the treatment and control of allergic conditions such as allergic asthma. ##STR1##
4581453 Guanidinothiazole derivatives containing alkylene bridges, and their use for influencing lipid metabolism  
The invention relates to guanidinothiazol derivatives of Formula (I) as defined herein, said compounds being useful for influencing lipid metabolism, as antithombotic agents and as antimycotic...
4578388 Unsymmetrical guanidino, thioureido, isothioureido and nitromethyleneamino derivatives  
The compounds are C 2 -C 8 straight chain alkanes terminally substituted, symmetrically or unsymmetrically, by N-(N'-substituted guanidino), N-(N',N"-disubstituted guanidino). N-(N'-substituted...
4578390 Hydroxybenzylamino derivatives as anti-inflammatory agents  
Hydroxybenzylamino derivatives have been prepared from an appropriate hydroxybenzaldehyde and an amine followed by reduction. These compounds are found to be active topical anti-inflammatory agents.
4575501 2-Arylhydrazino-2-thiazolines, acyl derivatives of these compounds, 2-arylazo-2-thiazolines, preparation processes, and their use for combating ectoparasites and endoparasites  
2-Arylhydrazino-2-thiazolines, acyl derivatives of these compounds and 2-arylazo-2-thiazolines, of the general formula ##STR1## and salts thereof, are new, are prepared as described and find use...
4572912 Thiazolidine derivatives, their preparation and compositions containing them  
The compounds of formula (I): ##STR1## [in which: R 1 and R 2 are the same or different and each represents hydrogen or C 1 -C 5 alkyl; R 3 represents hydrogen, an acyl group, a (C 1 -C 6 ...
4571406 Anti-hypertensive chromans and chromenes  
Compounds of formula (I): ##STR1## wherein: either one of R 1 and R 2 is hydrogen and the other is selected from the class of C 1 -6 alkylcarbonyl, C 1 -6 alkoxycarbonyl, C 1 -6 alkylcarbonyloxy,...
Matches 301 - 350 out of 443 < 1 2 3 4 5 6 7 8 9 >