Matches 351 - 400 out of 621 < 1 2 3 4 5 6 7 8 9 10 11 12 13 >
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5462912 Agricultural chemical composition enhancer comprising quaternary di(polyoxyalkylene) ammonium alkyl sulfates  
An agricultural chemical composition which can be safely applied to crops without causing any chemical damage; comprising a mixture, which exerts excellent potentiating effects on various...
5457083 Synergistic antimicrobial combination of polyether phosphonates and non-oxidizing biocides  
Synergistic antimicrobial combinations of polyether polyamino methylene phosphonates and one or more members selected from the group consisting essentially of the following non-oxidizing biocides: ...
5451564 Antimicrobial composition comprising N-hydroxy heterocyclic thiones  
A composition comprising (a) a metal salt or complex with an organic compound of the general formula ##STR1## and (b) an oxy-phosphorus compound where W may be --SH or an optionally substituted...
5447712 Method of reducing cyclophosphamide induced hemorrhagic cystitis  
A method is provided for reducing side effects caused by chemotherapeutic agents by administering to a patient in need thereof a therapeutically effective amount of a composition including...
5436257 Oxazolidine derivatives having anti-diabetic and anti-obesity properties, their preparation and their therapeutic uses  
Compounds of formula (I): ##STR1## wherein: R is an alkyl group; X is oxygen or sulfur; Y is hydrogen atom or --A--COOH, in which A is an alkylene group; Ar is aryl or substituted aryl group; and...
5432189 Bis-aryl amide and urea antagonists of platelet activating factor  
Bis-aryl amide and urea compounds of the general formula: ##STR1## wherein X is a divalent amide or urea substituent and Y is a nitrogen containing heterocycle, which compounds are inhibitors of...
5430045 Method of reducing or preventing bone marrow hypoplasia  
The present invention provides a method for reducing, or preventing, bone marrow hypoplasia in a patient at risk of, or having, same. To this end, when a glutathione intracellular stimulator is...
5424320 Heteroaryl coumarins as inhibitors of leukotriene biosynthesis  
Compounds having the formula I: ##STR1## are inhibitors of leukotriene biosynthesis. These compounds are useful as anti-asthmatic, anti-allergic, anti-inflammatory, and cytoprotective agents. They...
5418235 Aminoalkyl-substituted 5-mercaptothiazoles, the preparation and use thereof  
Aminoalkyl-substituted 5-mercaptothiazoles of the formula ##STR1## where R 1 , n and A have the meanings stated in the description, and the preparation thereof are described. The compounds are...
5418249 Thiazolidinyl-terminated non-peptidyl α-succinamidoacyl aminodiols as anti-hypertensive agents  
Non-peptidyl compounds characterized generally as α-succinamidoacyl aminodiols having a thiazolidinyl-type group at the N-terminus are useful as renin inhibitors for the treatment of hypertension.
5413997 Triphenylmethane derivatives  
A triphenylmethane derivative represented by the following general formula: ##STR1## exhibits bone absorption inhibiting effects and is useful as a medicament for treating osteoporosis.
5411975 Thiazolidinyl terminated alkylamino ethynyl alanine amino diol compounds for treatment of hypertension  
Compounds characterized generally as thiazolidinyl-terminated alkylamino ethynyl alanine amino diol derivatives are useful as renin inhibitors for the treatment of hypertension. Compounds of...
5409944 Alkanesulfonamido-1-indanone derivatives as inhibitors of cyclooxygenase  
Disclosed are compounds of Formula I useful in the treatment of cyclooxygenase mediated diseases such as pain, fever and inflammation of a variety of conditions including rheumatic fever, symptoms...
5401761 Thiazolidinedione hypoglycemic agents  
Compounds of the formula ##STR1## where R is alkyl, cycloalkyl, phenyl or substituted phenyl are useful as hypoglycemic agents.
5401762 Aminoalkyl-substituted thiazolin-2-ones, the preparation and use thereof  
Aminoalkyl-substituted thiazolin-2-one derivatives of the formula ##STR1## where n and A have the meanings stated in the description, and the preparation thereof are described. The compounds are...
5399576 Thiazoles  
Novel thiazoles of formula I ##STR1## wherein R 1 and R 4 are lower alkyl, lower alk-2-en-1-yl or lower alk-2-yn-1-yl, R 2 and R 3 are each independently of the other hydrogen or lower alkyl...
5395845 Pyrethrinoid esters of thiazole alcohols  
In all possible stereoisomer forms and mixtures thereof of the formula ##STR1## wherein one of R 1 , R 2 or R 3 is: ##STR2##
5393754 Organophosphorus compounds, and insecticides, acaricides and nematocides containing same  
Insecticidal, acaricidal or nematocidal compositions which comprise a series of organophosphorus compounds represented by the following representative structural formulae: ##STR1## show excellent...
5389657 Method for treating infertility  
The present invention provides a method of treating infertility comprising administering to a female mammal having fertility problems a therapeutically effective amount of the glutathione...
5387596 Benzylidenethiazolidine derivatives and their use for the inhibition lipid peroxides  
Benzylidenethiazolidine compounds of formula (I): ##STR1## [in which R 1 , R 2 and R 5 are each hydrogen or alkyl; R 3 and R 4 are each hydrogen, alkyl, formyl, alkylcarbonyl, arylcarbonyl,...
5378719 Imidazoles  
Novel imidazoles of formula I ##STR1## wherein R 1 and R 4 are lower alkyl, lower alk-2-en-1-yl or lower alk-2-yn-1-yl, R 2 and R 3 are each independently of the other hydrogen or lower...
5369107 Thiazole derivatives, processes for production thereof and pharmaceutical compositions comprising the same  
Compounds of the formula: ##STR1## wherein A is S, SO, or SO 2 , R 1 is H or acyl, R 2 is H, alkyl, hydroxyalkyl, halogen or carboxy, and R 3 is pyridyl are claimed. The compounds are useful as...
5366985 Method for preparation of an aqueous suspension  
A stable aqueous suspension, which is particularly suitable for eyedrops for the treatment of keratopathy and other diseases, containing 5-(3-ethoxy-4-n-pentyloxyphenyl)thiazolidine-2,4-dione can...
5358957 Butyric acid derivatives  
Compounds of the formula ##STR1## wherein A is a substituted or unsubstituted, aromatic or non-aromatic, monocyclic or bicyclic, heterocyclic radical that is bonded by way of a carbon atom to X;...
5350759 Bis-aryl amide antagonists of platelet activating factor  
Bis-aryl amide and urea compounds of the general formula: ##STR1## wherein X is a divalent amide or urea substituent and Y is a nitrogen containing heterocycle, which compounds are inhibitors of...
5344842 Thiosemicarbazone derivatives  
The invention relates to novel thiosemicarbazones of formula I ##STR1## wherein R 1 is lower alkyl, lower alk-2-en-1-yl or lower alk-2-yn-1-yl, R 2 and R 3 independently of one another are...
5342850 Thiazolidine-2,4-dione derivatives, their salts and their preparation processes  
The present invention provides novel thiazolidine-2,4-dione derivatives possessing blood sugar-lowering action and aldose reductase-inhibitory action, their salts, their preparative processes and...
5338746 Thiosemicarbazonic acid esters  
The invention relates to novel thiosemicarbazonic acid esters of formula I ##STR1## wherein R 1 and R 5 are lower alkyl, lower alk-2-en-1-yl or lower alk-2-yn-l-yl, R 2 and R 3 independently...
5334605 Thiazolylpyrroles having a fungicidal activity  
Compounds based on 2-thiazole-2-ylpyrrole, with a fungicidal activity, having the general formula (I): ##STR1##
5334606 Oxazolidindione substituted indole derivatives  
Compounds of formula (I): ##STR1## wherein Q 1 represents a phenyl group substituted by one or more halo; naphthyl; indolyl; benzthiophenyl; benzofuranyl; benzyl; or fluorenyl; R 1 is H, C 1...
5334614 Hydroxylamine derivatives  
The invention concerns hydroxylamine derivatives of the formula I ##STR1## wherein R 4 is hydrogen, carbamoyl, (1-4C)alkyl, cyclopentyl, cyclohexyl, tetrahydrofuran-3-yl, tetrahydropyran-4-yl,...
5330998 Thiazolidinedione derivatives as hypoglycemic agents  
Hypoglycemic thiazolidine-2,4-dione derivatives of the formula ##STR1## wherein the dotted line represents a bond or no bond; V is --CHCH--, --NCH--, --CHN--, S, O or NR; W is S, SO,...
5330999 2,4-thiazolidinedione compounds  
Compounds of formula (I): ##STR1## in which: R represents any one of the groups defined in the description. Medicinal products.
5328916 Heterocyclic compounds useful for inhibition of renin  
New heterocyclic compounds of the formula X--W--CR 1 R 2 --CO--Y--NR 3 --CHR 4 --CR 5 --CH 2 --(CR 6 R 7 ) r --Z--Het I in which R 1 to R 7 , W, X, Y, Z, r and Het...
5326770 Monoamine oxidase-B (MAO-B) inhibitory 5-substituted 2,4-thiazolidinediones useful in treating memory disorders of mammals  
This invention relates to monoamine oxidase-B (MAO-B) inhibitory 5-substituted 2,4-thiazolidinediones, such as Formula I, to pharmaceutical compositions thereof, process of preparation, and methods...
5324723 Oxazoles and thiazoles for the treatment of senile dementia  
1,3-Oxazole and 1,3-thiazole compounds of formula I, and their pharmaceutically acceptable salts and prodrugs: ##STR1## wherein X represents oxygen or sulphur; R 1 represents a non-aromatic...
5314891 Benzenesulphonamide derivatives  
The invention concerns benzenesulphonamide derivatives of the formula I ##STR1## wherein R 1 is (1-4C)alkyl, (3-4C)alkenyl or (3-4C)alkynyl; R 2 and R 3 together form --A 2 --X 2 --A 3 --...
5306724 Method for preventing and treating atherosclerosis  
The present invention provides a method for treating atherosclerosis. The method includes the step of administering to a patient having atherosclerosis, a noncysteine, non-thiol composition that...
5298516 Thiazolidone compounds and method of using the same as a vasodilator  
Compounds of formula (I): ##STR1## wherein W represents a sulfur atom and X represents a group of formula --N(R 1 )--, or W represents a group of formula --N(R 1 )-- and X represents a sulfur atom;...
5288743 Indole carboxylate derivatives which inhibit leukotriene biosynthesis  
Compounds of the structure ##STR1## where A is straight or branched divalent alkylene or divalent cycloalkylene, R 1 is selected from hydrogen; alkylthio; optionally substituted phenylthio;...
5273993 Compounds having one or more aminosulfonyloxy radicals useful as pharmaceuticals  
Methods of treating chronic arthritis and osteoporosis which utilize both known and novel compounds which would fall under the general formula: (HO)p--A--[--OS(O) 2 NR 1 R 2 ] z wherein A...
5258395 Thiazole compounds as inhibitors of SRS-A  
Novel heterocyclic compounds shown by the general formula ##STR1## or the pharmaceutically acceptable salts thereof useful as medicament in particular as antagonist of slow reacting substance of...
5256682 Isoxazolylimidazole derivatives, process for their production and their use in pharmaceutical agents  
4-Isoxazolyl-imidazole derivatives of formula I ##STR1## in which R 1 , R 2 , R 3 and R 4 have the meanings indicated, as well as their production and use in pharmaceutical agents, are described.
5246927 Benzazole derivatives, processes for their preparation containing such compounds and the use thereof  
The invention relates to new benzazole derivatives of the formula I ##STR1## wherein X is oxygen or sulphur, R 1 is lower alkyl, lower alkenyl or cycloalkyl, R 2 and R 3 independently of one...
5242939 Anilide derivatives with angiotensin II antagonist properties  
This invention relates to anilide derivatives of Formula I ##STR1## which antagonize the binding of angiotensin II to its receptors. The compounds are useful in the treatment of hypertension, heart...
5236941 5-(2-hydroxy-1-arylethylidene)- and 5-(2-oxo-1-arylethylidene)-2,4-thiazolidinediones and derivatives thereof  
5-(2-Hydroxy-1-phenyl (or-1-naphthalenyl)ethylidene) and 5-(2-oxo-1-phenyl (or 1-naphthalenyl)ethylidene)-2,4-thiazolidinediones and derivatives thereof are useful in lowering blood glucose levels...
5234917 Substituted 5-(alkyl)carboxamide imidazoles  
Angiotensin II receptor antagonists having the formula: ##STR1## which are useful in regulating hypertension and in the treatment of congestive heart failure, renal failure, and glaucoma...
5229405 Use of 2-iminothiazolidin-4-one derivatives as novel pharmaceutical active ingredients  
Compounds of the formula I ##STR1## in which R 1 is lower alk-2-en-1-yl, lower alk-3-en-2-yl, lower alk-2-yn-1-yl or lower alkyl substituted in the 2,3-position by radicals which can be eliminated...
5225426 Thiazolidine-2,4-dione compound and method of treatment of diabetic complications  
A novel compound is proposed which is effective in curing various complications as with catarat, retinopathy, neurotic disorder, and renal disorder. The thiazolidine-2,4-dione compound represented...
5223522 Thiazolidinedione hypoglycemic agents  
Hypoglycemic thiazolidine-2,4-dione derivatives of the formula ##STR1## wherein the dotted line represents a bond or no bond; A and B are each independently CH; X is S, SO, SO 2 , CH 2 , CHOH or...
Matches 351 - 400 out of 621 < 1 2 3 4 5 6 7 8 9 10 11 12 13 >