|
Match
|
Document |
Document Title |
|
|
6936624 |
Agents for preserving technical materials against insects
The use of the compounds of the formula (I)
as agents for preserving technical materials against insects.
|
|
|
6916839 |
Pyrazolylarylalkines
The present invention relates to pyrazolylarylalkines and to their use, to a process for preparing pyrazolylarylalkines and also to intermediates.
|
|
|
6911462 |
Benzimidazole compounds for regulating IgE
This invention relates to a family of phenylbenzimidazole analogs, which are inhibitors of the IgE response to allergens. These compounds are useful in the treatment of allergy and/or asthma or any...
|
|
|
6906089 |
Triarylimidazole derivatives as cytokine inhibitors
Compounds of formula (I) or a pharmaceutically acceptable salt thereof:
wherein R 1 , R 2 and R 3 are various substituent groups; and one of X 1 and X 2 is N or CR″, and the other...
|
|
|
6900230 |
Heterocyclo-alkylsulfonyl pyrazoles as anti-inflammatory/analgesic agents
The present invention relates to compounds of the formula
wherein R 1 , R 3 , R 5 , R 6 , and A are defined as in the specification, to pharmaceutical compositions containing them and to their...
|
|
|
6897226 |
NK-1 receptor active amine oxide prodrugs
Compounds of the invention are amine oxide prodrugs showing activity on the NK1 receptor.
|
|
|
6897227 |
Prodrugs of proton pump inhibitors
Prodrugs of proton pump inhibitors of Formulas 1 through 4,
where the symbols are as defined in the specification, and the R group includes at least one acidic group or its pharmaceutically...
|
|
|
6893651 |
Active ingredient combinations having insecticidal and acaricidal properties
The invention relates to insecticidal and acaricidal mixtures comprising certain cyclic ketoenols and agonists or antagonists of nicotinic acetylcholine receptors for protecting plants against...
|
|
|
6878729 |
Medicinal uses of dihydropyrazoles
Compounds having a structure according to Formula (I):
are effective in a method of increasing erythropoietin and vascularization of tissue in a subject in need thereof.
|
|
|
6878726 |
Pyrazole ether derivatives as anti-inflammatory/analgesic agents
The present invention relates to compounds of the formula:
wherein R 1 , R 2 , R 3 , R 4 , R 5 , R 6 , R 7 , R 8 , A, X and Y are defined as in the specification, to pharmaceutical...
|
|
|
6875778 |
Alkylene-tethered bis-nitroiminoimidazolidines, process for preparing the same, and insecticides containing the same
The present invention provides a novel alkylene-tethered bis-nitroiminoimidazolidine compound having superior insecticidal activity. The nitroimino imidazolidine compound is a...
|
|
|
6864252 |
Hydrazinyl and nitrogen oxide pyrazoles
The present invention relates to hydrazinyl and nitrogen oxide pyrazoles of the formula I:
wherein the ring of the formula (R 5 )-A-(SO m R 4 ), m, X, R 1 through R 5 are as defined in the...
|
|
|
6852740 |
Pyrazole derivatives as p38 kinase inhibitors
A class of pyrazole derivatives is described for use in treating p38 kinase mediated disorders. Compounds of particular interest are defined by Formula I
wherein Q, R 1 , R 2 , R 3 and R 4 ...
|
|
|
6849639 |
Integrin inhibitors and their methods of use
The invention comprises novel compounds that are effective in the prophylaxis and treatment of diseases, such as integrin receptors mediated diseases, in particular, diseases or conditions mediated...
|
|
|
6838458 |
5-(alkylidene-cycloalkyl)-and 5-(alkylidene-heterocyclyl)-pyrazoles
The present invention relates to 5-(alkylidene-cycloalkyl)-pyrazoles and 5-(alkylidene-heterocyclyl)-pyrazoles of the formula I:
wherein the ring of the formula (R 5 )-A-(SO m R 4 ), m, B,...
|
|
|
6835743 |
Pesticidal pyrazoles and derivatives
Process for the protection of a building that has already been built or is going to be built, whereby an effective amount of an insecticidally active compound is spread around or under the said...
|
|
|
6831083 |
Pyrazoline derivative or tetrahydropyridazine derivative and medicinal use thereof
Using a compound selected from compounds represented by the following formula (1) (which include 3-phenyl-2-pyrazoline derivatives and 3-phenyl-tetrahydropyridazine derivatives) and...
|
|
|
6787556 |
Benzoic acid derivatives for the treatment of diabetes mellitus
The present invention relates to the use of certain benzoic acid derivatives of formula (I), as disclosed in the specification, which act as peroxisome proliferator activated receptor (PPAR)...
|
|
|
6756384 |
Imidazole compounds
A novel class of imidazo heterocyclic compounds, pharmaceutical compositions comprising them and use thereof in the treatment and/or prevention of diseases and disorders related to the histamine H3...
|
|
|
6750230 |
Pyrazole derivatives
This invention relates to the use of pyrazole derivatives of the formula and pharmaceutically acceptable salts and solvates thereof, in the manufacture of a reverse transcriptase inhibitor or...
|
|
|
6734143 |
2-methoxyimino-2(pyridinyloxymethyl)phenyl acetamides useful as fungicides
The present invention provides 2-methoxyimino-2-(pyridinyloxymethyl) phenyl acetamides according to formula (I) as well as their use as fungicidal compounds.
|
|
|
6730635 |
Microcapsule suspensions
The invention relates to microcapsule suspensions containing (A) a particulate disperse phase of microcapsules comprising: (1) sleeves that are reaction products of mixtures of toluylene...
|
|
|
6716457 |
Effects of bactericide (peracetic acid-hydrogen peroxide-water combination) to agricultural chemicals in bacteria control when they are in contact with one another
The present invention relates to a process for inhibiting or eliminating the growth of microorganisms in pesticide suspensions. More particularly, the process of the present invention includes the...
|
|
|
6716881 |
Carbanilides used as pesticides
The present invention provides carbanilides of formula (I), wherein A, Q, R, X, Z and m are as defined herein. A plurality of processes for preparing these compounds is provided, along with...
|
|
|
6706739 |
Imidazolidinone compounds
A compound having the formula: in which R 1 , R 2 , R 3 , T, W, m, x, and y are defined as in the specification. Also disclosed is a method of treating enterovirus infection by using a compound...
|
|
|
6706743 |
β3 adrenergic receptor agonists and uses thereof
The instant invention provides β 3 adrenergic receptor agonists of structural Formula (I), the stereoisomers and prodrugs thereof, and the pharmaceutically acceptable salts of the compounds,...
|
|
|
6685954 |
Insecticidal combination to control mammal fleas, in particular fleas on cats and dogs
Process and composition, in particular for controlling fleas on small mammals, characterized in that the composition includes, on the one hand, at least one insecticide of 1-N-arylpyrazole type, in...
|
|
|
6683097 |
Imidazole derivatives
Novel imidazole derivatives are disclosed. These compounds have a good affinity to the NMDA (N-methyl-D-aspartate)-receptor subtype selective blockers, which have a key function in modulating...
|
|
|
6680065 |
Shaped bodies which release agrochemical active substances
The present invention relates to shaped articles which release agrochemical active compounds, are used for treatment of woody plants and are employed in a hollow preformed in the woody plant, are...
|
|
|
6677341 |
(R)-Chiral halogenated substituted heteroaryl benzyl aminoalcohol compounds useful for inhibiting cholesteryl ester transfer protein activity
The invention relates to substituted aryl and heteroaryl (R)-Chiral Halogenated 1-Substitutedamino-(n+1)-Alkanol compounds useful as inhibitors of cholesteryl ester transfer protein (CETP; plasma...
|
|
|
6670387 |
Thrombopoietin mimetics
Non-peptide TPO mimetics are disclosed, as well as a method of treating thrombocytopenia, in a mammal, including a human, in need thereof, which comprises administering to such mammal an effective...
|
|
|
6664277 |
Prenylation inhibitors containing dimethylcyclobutane and methods of their synthesis and use
The present invention is directed to compounds useful in the treatment of diseases associated with prenylation of proteins and pharmaceutically acceptable salts thereof, to pharmaceutical...
|
|
|
6660732 |
Compounds useful as anti-inflammatory agents
Disclosed are novel aromatic compounds which are useful for treating diseases or pathological conditions involving inflammation such as chronic inflammatory diseases. Also disclosed are...
|
|
|
6656933 |
Compounds useful as anti-inflammatory agents
Disclosed are novel aromatic compounds which are useful for treating diseases or pathological conditions involving inflammation such as chronic inflammatory diseases. Also disclosed are...
|
|
|
6649637 |
Inhibition of intracellular replication by pyridinylimidazoles
Substituted pyridinylimidazoles SB203580 and SB202190 strongly inhibit replication and cause stage conversion from active tachyzoites to relatively dormant bradyzoites of the medically important,...
|
|
|
6649636 |
Heteroaryl phenyl pyrazole compounds as anti-inflammatory/analgesic agents
This invention relates to a compound of the formula: or a pharmaceutically acceptable salt thereof, wherein A and R 1 are each an optionally substituted 5 to 6-membered heteroaryl, wherein the...
|
|
|
6642234 |
Acrylonitrile compounds
The present invention relates to acrylonitrile compounds of formula (1): [wherein, R is a C 1 -C 6 alkyl, a C 3 -C 7 cycloalkyl optionally substituted by a C 1 -C 4 alkyl, a naphthyl, etc., R...
|
|
|
6638956 |
Pesticidal 1-arylpyrazoles
The invention relates to novel 1-arylpyrazole oxime derivatives, of general formula (I) or (I bis) These compounds are found to be generally safe systemic insecticides for control of arthropod,...
|
|
|
6632828 |
Substituted imidazole neuropeptide Y Y5 receptor antagonists
Compounds of the formula I or a pharmaceutically acceptable salt, solvate or N-oxide thereof, wherein X is ═CH— or ═N—; Y is H, halogen, trihaloalkyl, alkyl, alkenyl, cycloalkyl,...
|
|
|
6630473 |
Anti-inflammatory agents and inhibitors against increase in ocular tension caused by irradiation with lasers, containing 1,4-dihydropyridine derivatives
The present invention provides an anti-inflammatory medicament and an inhibitor of intraocular pressure rise due to laser irradiation, which contains 1,4-dihydropyridine derivative of the formula...
|
|
|
6624176 |
Heteroaromatic substituted amides with antagonistic activity to neurokinin 1 receptors
The present invention is a heteroaromatic substituted amide showing antagonist activity to neurokinin 1 (NK-1, substance P) receptors.
|
|
|
6620825 |
Adenosine A3 receptor antagonists
A pharmaceutical composition for antagonizing adenosine at adenosine A 3 receptors which comprises a 1,3-azole compound substituted on the 4- or 5-position, or both, by a pyridyl which may be...
|
|
|
6620826 |
Endothelin receptor antagonists
Novel N-phenyl imidazole derivatives, pharmaceutical compositions containing these compounds and their use as endothelin receptor antagonists are described.
|
|
|
6617314 |
Injectable formulations of avermectins and milbemycins
The present application relates to injection formulations of avermectins and milbemycins based on a solvent mixture comprising sesame oil, medium-chain triglycerides, glycol esters or fatty acid...
|
|
|
6596739 |
N-(1-phenylethyl)-5-phenyl-imidazole-2-amine compounds, their compositions and uses
The subject invention involves compounds having structure (I): wherein each R1 is independently alkyl, aryl, or heterocycle; each R2, R4, R7, and R8 is independently hydrogen or other substituent;...
|
|
|
6596728 |
Substituted 1,3-diaryl-2-pyrid-2-yl-3-(pyrid-2-ylamino)propanol derivatives, process for their preparation, pharmaceuticals comprising these compounds and their use
Substituted 1,3-diaryl-2-pyridin-2-yl-3-(pyridin-2-ylamino)propanol derivatives of the formula (I), and salts thereof, in which the radicals have the meanings given in the specification, and...
|
|
|
6579873 |
3 (5)-heteroaryl substituted pyrazoles as p38 kinase inhibitors
A class of pyrazole derivatives is described for use in treating p38 kinase mediated disorders. Compounds of particular interest are defined by Formula I wherein R 1 , R 2 , Ar 1 and HetAr 2 ...
|
|
|
6569873 |
Azolidines as beta-3 adrenergic receptor agonists
This invention provides compounds of Formula I having the structure wherein, A, X, Y, Z, W, R 1 , R 2 , R 3 , R 4 , R 5 , and R 6 are as defined hereinbefore or a pharmaceutically acceptable...
|
|
|
6569860 |
Alkoxycarbonylamino heteroaryl carboxylic acid derivatives as IP antagonists
This invention relates to compounds which are IP receptor antagonists and which are represented by Formula (I): wherein G 2 is a heteroaryl group containing one or two nitrogen atoms...
|
|
|
6562845 |
Materials and methods for the control of tephritidae fruit flies
The subject invention provides materials and methods for the effective control of fruit flies. Specifically, the subject invention pertains to the use of imidacloprid compounds to control fruit...
|