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4670443 |
Benzo(f)isoquinoline compounds useful as calcium entry blockers
Benzo(f)isoquinoline compounds, particularly, penta- and tetrahydrobenzo(f)isoquinoline dicarboxylic acid compounds, their preparation and their use as calcium entry blockers are disclosed.
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4659716 |
Antihistaminic 8-(halo)-substituted 6,11-dihydro-11-(4-piperidylidene)-5H-benzo[5,6]cyclohepta[1,2-b]pyridin es
Disclosed are 7- and/or 8-(halo or trifluoromethyl)-substituted-6,11-dihydro-11-(4-piperidylide
ne)-5H-benzo[5 ,6]cyclohepta[1,2-b]pyridines and the pharmaceutically acceptable salts thereof, which...
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4639457 |
Benzocycloheptapyridone compounds for treating congestive heart failure
Novel benzocycloheptapyridone compounds are disclosed. The compounds exhibit inotropic potencies and are adaptable to being utilized as cardiotonic agents in the chemotherapeutic treatment of...
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4624954 |
6,7,8,9-tetrahydro-10-methylpyrido[1,2-a]indol-9-amines and derivatives thereof, useful for the treatment of cognitive impairments
Herein is disclosed 6,7,8,9-tetrahydro-10-methylpyrido[1,2-a]indol-9-amines and derivatives, therapeutically acceptable acid addition salts thereof, processes for their preparation, methods of...
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4605660 |
Indeno[2,1-c]pyridine compounds, and their use as calcium channel blockers
Indeno[2,1-c]pyridine compounds, particularly cyano substituted tetrahydroindeno[2,1-c]pyridine dicarboxylic acid ester compounds, their preparation and their use as calcium entry blockers are...
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4593033 |
Substituted indeno[2,1-c] pyridines useful as calcium channel blockers
Novel substituted indeno[2,1-c] pyridine compounds useful as calcium channel blockers, pharmaceutical compositions thereof, and methods of treatment are disclosed.
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4565818 |
Pharmaceutically active 1,2,3,4,4a,5,10,10a-octahydro-benzo[g]quinoline derivatives
A 6- and/or 7-oxy-trans-1,2,3,4,4a,5,10,10a-octahydro-benzo[g]quinoline in which the 3-position is substituted by an optionally amidated carboxy group, an optionally etherified hydroxymethyl group,...
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4550113 |
9-Amino-2,3,5,6,7,8-hexahydro-1H-cyclopenta(b)quinoline monohydrate hydrochloride as stimulant of neuro-muscular transmission of smooth muscles
A novel compound and composition are disclosed which stimulate neuro-muscular transmission of smooth muscles and cause excitation of conductance in the peripheral and central nervous systems,...
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4546099 |
N-Aminomethyl-3-phenyl-4-cyanopyrrole derivatives, compositions and use thereof as microbicides
The invention relates to novel N-aminomethyl-3-phenyl-4-cyanopyrrole derivatives of the formula I ##STR1## wherein R 1 and R 2 are each independently hydrogen, halogen, methoxy or methylthio, ...
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4543354 |
Anti-hypertensive 9-aminomethyl-benzo[f]quinoline-3,10-dione derivatives
Benzo[f]quinoline derivatives which are useful as antihypertensive agents and are represented by the formula: ##STR1## wherein R 1 is hydrogen or lower alkyl, R 2 is hydrogen, lower alkyl,...
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4542138 |
Dioxobenzocyclo-hepta-pyridine compounds, process and use as antihypertensives
6H-3,11b-Dihydrocarbalkoxy-5,7-dioxobenzo[6,7]cyclohepta[1,2
-c]pyridine compounds represented by the formula: ##STR1## wherein G is lower alkyl or halogen; R is lower alkyl, R' is hydrogen, lower...
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4535085 |
Perfluorotricyclic amines as oxygen carriers
A perfluorotricyclic amine compound which is usable as an oxygen carrier in an artificial blood, represented by the general formula ##STR1## wherein R denotes a perfluoroalkyl group having 1-4...
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4532248 |
Method of combatting coronary and vascular diseases
1,4-Dihydropyridines of the formula ##STR1## in which n is 0,1 or 2, and R 1 to R 7 can have a wide variety of meanings, which possess inotropic action, and many of which are new, are useful...
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4521423 |
7,8,9,10-Tetrahydrobenzo[h]quinolin-9-amine derivatives and compositions and methods for treating depression employing them
7,8,9,10-Tetrahydrobenzo[h]quinolin-9-amine derivatives of the formula ##STR1## in which R 1 and R 2 each independently is hydrogen or lower alkyl, or R 1 and R 2 together form a chain of the...
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4511569 |
Tricyclic lactams and derivatives useful in increasing cardiac contractility
Disclosed are 5,6-dihydro benzo[f]quinolines and derivatives which are effective in increasing cardiac contractility. These compounds are useful in the treatment of congestive heart failure.
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4466980 |
Thiaprostaglandin E.sub.1 derivatives, process for production thereof, and pharmaceutical use thereof
A novel compound selected from the group consisting of 7-(or 6- or 4-)thiaprostaglandin E 1 derivatives of the formula (I). ##STR1## wherein A represents --CH 2 -- or ##STR2## in which n is 0, 1...
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4405626 |
9-Hydroxyoctahydrobenzo(c)quinolines analgesic compositions containing them and processes for producing analgesic with them
1,9-Dihydroxyoctahydrobenzo[c]quinolines (I), 1-hydroxyhexahydrobenzo[c]quinoline-9(8H)-ones (II), and 1-hydroxy-tetrahydrobenzo[c]quinolines (IV) useful as CNS agents, especially as analgesics and...
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4380542 |
9-Hydroxyoctahydrobenzo[c]quinolines and their pharmaceutical compositions and method of use
1,9-Dihydroxyoctahydrobenzo[c]quinolines (I), 1-hydroxyhexahydrobenzo[c]quinoline-9(8H)-ones (II), and 1-hydroxy-tetrahydrobenzo[c]quinolines (IV) useful as CNS agents, especially as analgesics and...
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4341786 |
Pharmaceutical compositions and method of producing central alpha.sub.1 agonist activity utilizing octahydrobenzo[f]quinoline compounds
Octahydrobenzo[f]quinoline compounds having 7- and 10-substituents are centrally acting alpha 1 agonists.
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4282233 |
Antihistaminic 11-(4-piperidylidene)-5H-benzo-[5,6]-cyclohepta-[1,2-b]-pyridines
11-(4-Piperidylidene)-5H-benzo-[5,6]-cyclohepta-[1,2-b]-pyri
dines and their 5,6-dihydro derivatives are disclosed. The compounds are useful as antihistamines with little or no sedative effects.
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4169893 |
4-Hydroxy-naphthpyridine-2(1H)-one-3-carboxylic acids and esters
Anti-allergic 4-hydroxy-naphthpyridine-2(1H)-one-3-carboxylic acids and esters are prepared by reacting a 1,3-dioxo-1-naphth[4,5-b]oxazine with an alkali metal salt of a malonic ester (and...
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4150136 |
Benz[g]isoquinolines and use thereof
The present invention provides novel compounds of the formula, ##STR1## wherein R 1 is hydrogen, halogen, alkyl or alkoxy; R 2 may, for example, be hydrogen, alkyl, alkenyl, alkinyl or...
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4118497 |
Antidepressantly active 5-(4-aminophenyl)-hexahydro-1H-indeno-(1,2-b)pyridine
The invention relates to hexahydro-1H-indeno/1,2-b/pyridines and a process for their manufacture. These compounds and the physiologically tolerable salts thereof are useful as agents for the...
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4103014 |
Use of 4aRS,5SR,9bRS-2-ethyl-1,3,4,4a,5,9b-hexahydro-7-methyl-5-p-tolyl-2H-inde no[1,2-c]pyridines in inhibiting spermatogenesis
The present invention relates to the use of the known compound of formula ##STR1## for an agent for inhibiting spermatogenesis in male animals.
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4085215 |
Certain 5,6,7,8-tetrahydroquinoline-8-thiocarboxamides
The invention relates to novel pyridine derivatives which have a fused 5,6, or 7-membered saturated hydrocarbon ring adjacent to the nitrogen of the pyridine ring, and a group X situated on said...
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4081543 |
5-Substituted-1,2,3,4-tetrahydrobenzo[g]isoquinolines
This invention provides new compounds of formula I, ##STR1## wherein R 1 is hydrogen, halogen of an atomic number from 9 to 35, or alkyl or alkoxy of 1 to 4 carbon atoms, R 2 is hydrogen,...
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4049811 |
Compositions using cycloalkano-quinolone derivatives and their method of use
Cycloalkano-quinolone derivatives having anti-microbial activity characterized by the formula: ##STR1## wherein one of R 1 and R 2 designates hydrogen, halogen, nitro, amino, hydroxyl, acylamino,...
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4046895 |
Phenanthridine derivatives and related compounds
The invention provides a compound of formula I ##STR1## wherein R 1 and R 2 are the same or different and represent hydrogen or alkyl of 1-6 carbon atoms, R 3 represents hydrogen, alkyl of 1-6...
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4034095 |
Benzo[5,6]cyclohepta[1,2-c]pyridines
Novel benzo[5,6]cyclohepta[1,2-c]pyridines useful as anti-depressant and anti-cholinergic agents.
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4034096 |
Nitrogen containing derivatives of cyclopenteno-quinolone compounds and bacteriostatic compositions
New cyclopenteno-quinolone derivatives of the formula ##STR1## wherein R is a saturated or unsaturated aliphatic hydrocarbyl, e.g., alkyl and alkenyl, X is hydrogen or alkyl, and Y is...
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3998960 |
Pharmaceutical compositions containing a 2-(heteroaryl-methyl)-5,9β-dialkyl-6,7-benzomorphan and method of use
Pharmaceutical compositions containing as an active ingredient a compound of the formula ##STR1## wherein R is hydrogen, methyl or acetyl, R 1 and R 2 , which may be identical to or different...
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3995040 |
Cyclopenteno-3-carboxyl-4-quinolone derivatives and their bacteriostatic compositions
New cyclopenteno-quinolone derivatives of the formula ##SPC1## Wherein R is a saturated or unsaturated aliphatic hydrocarbyl, e.g., alkyl and alkenyl, X is hydrogen or alkyl, and Y is...
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3988460 |
Cyclopentenoquinolone compounds for treating bacterial infections
Certain novel cyclopentenoquinolone derivatives of the formula: ##SPC1## Wherein R and X, which may be the same or different, are hydrogen or lower saturated or unsaturated aliphatic...
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3962445 |
Anti-allergenic carbostyril derivatives
A class of 4-hydroxy-3-nitroearbostyril derivatives are useful in the inhibition of certain types of antigen antibody reactions.
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3900564 |
Ocotea alkaloid for relief of anxiety
Crystalline glaziovine having the formula: ##SPC1## And its acid addition salts have psychotropic properties useful in therapeutic compositions for the relief of anxiety. The alkaloid is obtained...
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3324003 |
Method of controlling growth of bacteria using 4-methyl-1-benzo[f]quinolone-2-carboxylic acid
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3212970 |
Treatment of psoriasis
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3179564 |
Antirigor thioxanthenes
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3110650 |
Synergistic analgesic compositions
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3737544 |
Title is not available
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