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4532136 |
4,4,4-Trichloro-1-pyridyl-but-2-ene-1-ones and fungicides made therewith
4,4,4-trichloro-(x-pyridyl)-but-2-ene-1-one, wherein x is 2, 3 and 4, and a process for making the same. The compounds are effective fungicides used singly or in combination.
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4529598 |
Insect repellent compounds
Compounds having the formula ##STR1## in which R is C 3 -C 5 alkyl or C 3 -C 5 alkenyl and n is an integer from 1 to 3, are effective to repel insects.
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4529728 |
1H,3H-pyrrolo[1,2-c]thiazole derivatives having anti-allergic and anti-inflammatory activity
New compounds of the formula ##STR1## in which R 1 and R 2 =H or alkyl and (a) R=CN or alkylcarbonyl, or (b) R=CON(R 3 )R 4 , in which R 3 =H and R 4 =NH 2 , alkylamino, dialkylamino,...
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4525360 |
Anti-psychotic phenylindene derivatives and acid addition salts thereof
The present invention relates to novel phenylindene derivatives having interesting pharmacodynamic properties which make them useful as psychopharmacologicals in the treatment especially of...
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4521428 |
Anorexigenic trifluoromethylphenyltetrahydropyridines and pharmaceutical compositions containing them
Novel 4-(3-trifluoromethylphenyl)-1,2,3,6-tetrahydropyridines of formula ##STR1## wherein R is an unsubstituted or by an alkyl group of from 1 to 4 carbon atoms substituted pyridyl, pyridyl 1-oxide...
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4512995 |
Phenoxyalkenylpyridine derivatives and fungicidal methods of use
3-[2-aryloxy-3-hydroxy-3-phenyl or 3-t-butylprop-1-enyl]pyridine and derivatives thereof are disclosed. These compounds are useful as fungicides, especially agricultural fungicides.
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4500535 |
Method of regulating the immune response with pyridine derivatives
A series of 4-(2-carboxymethylthiomethyl)pyridines and related compounds, and their pharmaceutically acceptable salts, are disclosed as having immunoregulatory activity. Preferred compounds include...
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4497830 |
Carbacyclins, their preparation and pharmacological use
Compounds of Formula I ##STR1## wherein X is oxygen or CH 2 ; A is CH 2 --CH 2 , trans-CHCH or C.tbd.C; W is free or functionally modified hydroxymethylene or free or functionally...
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4496559 |
2-Selenopyridine-N-oxide derivatives and their use as fungicides and bactericides
Disclosed are selected derivatives of 2-selenopyridine-N-oxide and their use as fungicides and bactericides.
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4478836 |
1-Aryl 2-aminomethyl cyclopropane carboxyamide (Z) derivatives and their use as useful drugs in the treatment of disturbances of the central nervous system
The present invention concerns new derivatives of 1-aryl 2-aminomethyl cyclopropane carboxamides (Z) of general formula I: ##STR1## in which: R represents a hydrogen or halogen atom, a lower alkyl...
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4474789 |
(Trichloromethyl)pyridine compounds useful for promoting growth and/or improving feed utilization efficiency in ruminants
(Trichloromethyl)pyridine compounds improve growth rate and feed utilization efficiency when orally administered to ruminants in amounts sufficient to cause any one or more of the following...
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4472408 |
Substituted trifluoromethylphenyltetrahydropyridines having an anorectic activity
The invention relates to 4-(3-trifluoromethylphenyl)-1,2,3,6-tetrahydropyridines of formula ##STR1## in which R represents a cyano, acetyl or cycloalkyl group of from 3 to 7 carbon atoms and Alk...
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RE31624 |
Method of treating inflammation
A method of treating inflammation and inhibiting prostaglandin synthesis employing substituted 2-(arylmethoxy)phenol compounds.
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4443449 |
Arylcyclobutylalkylamines and anti-depression composition and methods using same
Compounds of formula I ##STR1## in which R 1 is H or C 1 -3 alkyl; R 2 is H or C 1 -3 alkyl; R 3 and/or R 4 are H, C 1 -3 alkyl, C 3 -6 alkenyl, C 3 -6 alkynyl, C 3 -7 cycloalkyl or R 3 and R...
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4438122 |
Combating fungi with 1-phenoxy-2-pyridinyl-alkanols
1-Phenoxy-2-pyridinyl(pyrimidinyl)-alkanols of the formula ##STR1## in which R represents alkyl, optionally substituted aryl or optionally substituted aralkyl, X represents a nitrogen atom or...
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4431650 |
Esters of benzofuranyl acids
This invention relates to novel esters of benzofuranyl acids, novel intermediates therefor, synthesis thereof, and the control of pests.
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4427682 |
Pyridine alkyl benzoic and thenoic acid compounds and their pharmaceutical compositions
The pyridine derivatives of the general formula: ##STR1## [wherein A represents an alkylene group containing from 1 to 5 carbon atoms unsubstituted or substituted by a hydroxy group, B represents a...
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4424202 |
Azelaaldehydates as psychotropic agents
A method for producing a psychotropic response, especially for alleviating the symptoms of alcohol withdrawal, comprises administering to a human or animal subject in need thereof a...
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4414217 |
3,5-Di(t-butyl)-4-hydroxyphenyl substituted pyridines
3,5-Di(t-butyl)-4-hydroxyphenyl and 3,5-di(t-butyl)-4-hydroxybenzoyl-substituted pyridines have pharmacological activity as antiinflammatory agents.
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4411886 |
Stabilized cosmetic compositions
Stabilized cosmetic compositions containing as an active ingredient a compound represented by the formula ##STR1## wherein R is sodium, potassium or ammonium and x is 1 or R is aluminum and x is 3....
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4409227 |
4-(((Heterocyclo)thio)methyl)benzoic acids, esters and amides and their pharmaceutical use
4-(((Heterocyclo)thio)methyl)benzoic acids, esters, amides and pharmaceutically-acceptable salts thereof having hypoglycemic activity in mammals, including a method of use and...
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4407807 |
Pyridylpropyl cycloalkanecarboxylates: insect repellents
Compounds having the formula ##STR1## in which R is C 3 -C 5 cycloalkyl, are insect repellents.
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4401673 |
Pesticidal 3-(buta-1',3'-dienyl)-cyclopropane-1-carboxylic acid esters
Novel 3-(buta-1',3'-dienyl)-cyclopropane-1-carboxylic acid compounds of the formula ##STR1## wherein X 1 and X 2 are individually a halogen and A is selected from the group consisting of (A)...
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4397851 |
2,3-Dihalo-2,3-(disubstituted) propanoate antimicrobial compounds
Antimicrobial compounds of the formula: ##STR1## wherein Hal is bromine or chlorine; R is C 1 -4 alkyl, straight or branched chain; and one of R 1 and R 2 is hydrogen and the other is selected...
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4393068 |
Pyridylalkyl thiocarbonates as insect repellents
Novel compounds having the formula ##STR1## in which R is alkyl, cycloalkyl, aralkyl, chlorophenyl or chlorobenzyl, R 1 is hydrogen or lower alkyl and n is 1, 2, or 3, are insect repellents.
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4391827 |
3-(2-Hydroxy-4-(substituted)phenyl)-cycloalkanone and cycloalkanol analgesic agents and intermediates therefor
Cycloalkanones, cycloalkanols and unsaturated analogs thereof, each of which has at the 3-position a 2-hydroxy-4-substituted phenyl group wherein the 4-position substituent is alkyl which can have...
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4390537 |
1-(Substituted-aminoalkoxyphenyl)-2-methylene-1-alkanones, compositions and use
1-(Substituted-aminoalkoxyphenyl)-2-methylene-1-alkanones, a class of compounds possessing anti-allergic properties for use in the treatment of allergic conditions, such as asthma prepared by...
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4389403 |
1-Aroyl-2-phenylamino-2-imidazolines, drugs containing these compounds, and use thereof
1-Aroyl-2-phenylamino-2-imidazolines of the general formula ##STR1## where R 1 and R 2 are identical or different and each is chlorine, bromine, fluorine, methyl, ethyl, methoxy, trifluoromethyl...
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4388326 |
Phenyl hydroxypropyl sulfoxide enzyme inhibitors
Organic sulfoxides having a latent allyl group bound to the sulfur are enzyme inhibitors of the suicide or K cat type.
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4383999 |
Inhibition of GABA uptake by N-substituted azaheterocyclic carboxylic acids and their esters
N-Substituted azaheterocyclic carboxylic acids and their esters, useful as inhibitors of GABA uptake, are prepared by reacting an appropriate N-alkylating derivative with an ester of an...
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4382942 |
3-(1,2,5,6-Tetrahydropyridin-3-yl)-phenols and their use in pharmaceutical compositions
Novel 3-(1,2,5,6-tetrahydropyridin-3-yl)-phenols of the formula ##STR1## wherein X is selected from the group consisting of hydrogen and an acyl of an organic carboxylic acid of 2 to 7 carbon...
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4376767 |
Pyridylmethyl esters of selected bio-affecting carboxylic acids
Novel pharmaceutically useful derivatives of selected known bio-affecting carboxylic acids are disclosed, said derivatives having the structural formula ##STR1## wherein R 1 and R 2 , which can be...
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4370342 |
S-Alkyl 3-alkylthiopropionothioate compounds, their production and their medicinal use
The invention relates to S-alkyl 3-alkylthiopropionothioates of Formula (I) as defined herein. Also included in the invention are methods for the manufacture of said S-alkylthiopropionothioates,...
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4358450 |
O-Alkylated oximes and pharmaceutical composition thereof
Compounds of general formula ##STR1## wherein R 1 represents a member selected from the group consisting of (a) an unsubstituted at most binuclear aryl group having from 6 to 10 carbon atoms, such...
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4357336 |
Certain 2,2-dimethyl-3-(ethenyl or propenyl)-cyclopropane carboxylic acid esters of the pyridyl-lower alkyl series having insect repelling properties
Compounds having the formula ##STR1## in which R is hydrogen or C 1 -C 4 alkyl; X and Y are independently halogen or methyl; and n is an integer from 1 to 3, are effective insect repellents.
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4355034 |
Ethenyl derivatives of mercaptoalkylpyridines as anti-inflammatory agents
Mercaptoalkylpyridines carrying an ethenyl or ethynyl substituent are prepared from known pyridine compounds, principally pyridoxine, by known chemical procedures, and are useful in the treatment...
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4351838 |
Indane derivatives, process for their preparation, their use as pharmaceuticals and pharmaceutical compositions containing said derivatives
The invention provides compounds of formula ##STR1## wherein R 1 and R 2 are alkyl, R 3 is hydrogen, alkyl, alkenyl, phenylalkyl or a group --(CH 2 --CH 2 --O) n --R 4 in which n is 1 to 3...
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4348400 |
Pyridylpropyl alkyl-substituted benzoates and their use as insect repellents
Compounds having the formula ##STR1## in which R is C 1 -C 4 alkyl, are effective insect repellents.
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4337258 |
2,4-Dioxo-4-substituted-1-butanoic acid derivatives useful in treating urinary tract calcium oxalate lithiasis
2,4-Dioxo-4-substituted-1-butanoic acid derivatives of the formula: ##STR1## where R is hydrogen or C 1 -4 alkyl; and L is a lipophilic group consisting essentially of (1) ##STR2## where R'...
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4330551 |
Therapeutic method
Disclosed are therapeutic compositions that comprise an aqueous emulsion constituted by a pharmacologically acceptable cationic surfactant, a pharmacologically acceptable non-ionic surfactant, and...
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4327102 |
Certain 2-(phenyl sulfinylmethyl or ethyl) pyridine derivatives, composition containing same and method of using same
The invention provides a compound of formula I ##STR1## wherein R represents hydrogen, lower alkyl, phenyl, halophenyl, loweralkylphenyl, loweralkoxyphenyl or aralkyl of 7 to 12 carbon atoms, R 1 ...
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4324784 |
Process for preventing growth of marine organisms on a substance using hydrogen peroxide
A process for preventing growth of marine animals, i.e. shellfish, Polyzoa, and Hydrozoa on a surface, characterized by supplying hydrogen peroxide and/or a hydrogen peroxide-generating agent into...
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4322442 |
Combating fungi with 1-halo-1-propyn-3-ols
1-Halo-1-propyn-3-ols of the formula ##STR1## in which R is optionally substituted phenyl, pyridyl, furyl, thienyl or pyrazolyl, R' is optionally substituted phenyl, and X is halogen, which...
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4317828 |
Pyridine derivatives
The pyridine derivatives of the general formula: ##STR1## [wherein A represents an alkylene group containing from 1 to 5 carbon atoms unsubstituted or substituted by a hydroxy group, B represents a...
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4311703 |
Antidepressant and tranquilizing (α-phenyl-2-tolyl)-azacycloalkenes
Novel azacycloalkanes, azacycloalkenes and derivatives thereof and methods of preparing same are described. These compounds are useful as antidepressants, anticonvulsants, tranquilizers and...
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4307112 |
9-Deoxy-9A-methylene isosteres of PGI.sub.2 and process for their preparation
9-deoxy-9A-methylene-isosteres of PGI 2 , including processes for their preparation and pharmaceutical and veterinary compositions containing same, are disclosed. The compounds are useful as...
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4302462 |
4(or 3)-(3,4-Dihydroxyphenyl)pyridines, their cardiotonic use and cardiotonic use of their methyl ethers
4(or 3)-(3,4-Dihydroxyphenyl)pyridine, a cardiotonic agent, is prepared by demethylating 4(or 3)-(3,4-dimethoxyphenyl)pyridine, preferably by heating with aqueous hydrogen bromide....
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4267183 |
Tetrahydropyridine derivative
The invention concerns the novel amine 1-(2-chlorobenzyl)-1,2,3,6-tetrahydropyridine of the formula: ##STR1## and its pharmaceutically acceptable acid-addition salts, which have useful properties...
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4262000 |
Combating fungi with 3-substituted pyridine derivatives
3-Substituted pyridine derivatives of the formula ##STR1## in which A is --CO-- or --CH(OH)--, R is alkyl or optionally substituted phenyl, X each independently is halogen, alkyl, cycloalkyl,...
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4252804 |
Therapeutically useful 3,4,5-trimethoxybenzene derivatives
Compounds of the formula I ##STR1## wherein m and n are 0, 1 or 2, X represents oxygen, imino, benzylimino, or morpholinoethylimino, Y represents CO, CONH, COO or SO 2 , and NR 1 R 2 represents a...
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