Matches 301 - 344 out of 344 < 1 2 3 4 5 6 7
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4442102 1,5-Diphenylpyrazolin-3-one compounds, process and intermediates for preparation thereof and pharmaceutical compositions containing same  
New 1,5-diphenylpyrazolin-3-one compounds and a method of preparing them are described. The compounds have the general formula I ##STR1## where R 1 is a hydrogen or halogen atom, or a lower alkyl,...
4440774 3-Amino-2-hydroxypropoxyaryl imidazole derivatives  
Novel substituted imidazoles of the formula ##STR1## and methods for their preparation are disclosed. These imidazoles, and their salts, exhibit pharmacological activity which includes...
4435399 2-Aryl-1-(imidazol-1-yl)-8-(4-piperazin-1-ylphenoxy) octan-2-ol antifungal agents  
A series of novel 2-aryl-1-(imidazol-1-yl)-8-(4-piperazin-1-ylphenoxy)octan-2- ol derivatives has been prepared, including their pharmaceutically acceptable acid addition salts. These particular...
4428950 (Hetarylphenoxy)-(phenylpiperazinyl)-propanols, their preparation and drugs containing these compounds  
Novel (hetarylphenoxy)-(phenylpiperazinyl)-propanols of the formula ##STR1## where R 1 is hydrogen, amino or alkyl of 1 to 4 carbon atoms, R 2 is hydrogen, halogen, alkyl of 1 to 4 carbon atoms...
4421753 1-(5-Amino-4H-1,2,4-triazol-3-yl)-4-substituted-piperazines  
This disclosure describes novel 1-(5-amino-4H-1,2,4-triazol-3-yl)-4-substituted-piperazines which are useful as hypotensive agents in mammals.
4410525 Alkoxy pyrazole derivatives and compositions  
The invention relates to 3-aryl-5-alkoxy-pyrazoles, represented by general formula (I): ##STR1## wherein Ar represents an aryl group which may be substituted; R represents a hydrogen atom or an...
4410540 Cardiotonic 4-aroylimidazolidin-2-ones  
This invention relates to aroyl-2-imidazolidinones of the following general structure which are useful as cardiotonics and antihypertensive agents ##STR1## wherein Ar is furanyl, thienyl,...
4405635 4-Aroylimidazol-2-ones and their use as pharmaceuticals  
Novel 4-aroylimidazol-2-ones of the following general structure which are useful as antihypertensives, cardiotonics, antithrombotics, bronchodilators and uterospasmolytics ##STR1## wherein Ar is...
4386091 2-Phenoxyalkyl-1,2,4-triazol-3-one antidepressants  
Phenoxyalkyl substituted-1,2,4-triazolones having antidepressant properties typified by 4-[3-[4-(3-chlorophenyl)-1-piperazinyl]propyl]-5-ethyl-2,4-d ihydro-2-(2-ph...
4382934 Isatin derivatives, processes for the preparation thereof and pharmaceutical composition comprising the same  
A compound of the general formula: ##STR1## wherein R 1 and R 2 are hydrogen, halogen, lower alkyl, lower alkoxy, halo (lower) alkyl, lower alkanoylamino, lower alkoxyalylamino, or a 5 to 6...
4338317 Phenoxyethyl-1,2,4,-triazol-3-one antidepressants  
Phenoxyethyl substituted-1,2,4,-triazolones having antidepressant properties typified by 2-[3-[4-(3-chlorophenyl)-1-piperazinyl]propyl]-5-ethyl-4-(2- phenoxyethyl)- 2H-1,2,4-triazol-3(4H)-one are...
4330544 Amino-alkoxy pyrazoles and pharmaceutical compositions  
An aminoalkoxypyrazole of the general formula (I) ##STR1## wherein Ar is a phenyl, benzyl or naphthyl group, or a phenyl group substituted by one or more halogen atoms, or by one or more alkyl,...
4328227 Novel O-propyloximes  
Compounds of general formula ##STR1## wherein R 1 represents a radical selected from the group consisting of (a) hydrogen, carboxyl; (b) alkyl, alkenyl each having up to 6 carbon atoms and...
4327108 Methods useful in the treatment of cardiac arrhythmia using 4-substituted-2-iminoimidazolidine compounds  
This invention provides a novel class of 2-iminoimidazolidines which include 4-substituted derivatives such as 4-(2-chloroethyl)-1-methyl-2-methylimino-3-phenyl imidazolidine fumarate: ##STR1##...
4327107 Method useful in the treatment of sugar cataracts using 4-substituted-2-iminoimidazolidine compounds  
This invention provides a novel class of 2-iminoimidazolidines which include 4-substituted derivatives such as 4-(2-chloroethyl)-1-methyl-2-methylimino-3-phenyl imidazolidine fumarate: ##STR1##...
4327098 Pharmaceutical compositions useful in the treatment of cardiovascular hypertension and containing 4-substituted-2-iminoimadazolidine compounds  
This invention provides a novel class of 2-iminoimidazolidines which include 4-substituted derivatives such as 4-(2-chloroethyl)-1-methyl-2-methylimino-3-phenyl imidazolidine fumarate: ##STR1##...
4288447 Antihyperglycemic 4-substituted 2-iminoimidazolidine compositions  
This invention provides a novel class of 2-iminoimidazolidines which include 4-substituted derivatives such as 4-(2-chloroethyl)-1-methyl-2-methylimino-3-phenyl imidazolidine fumarate: ##STR1##...
4272538 5-Nitro-imidazole with antiprotozoic activity  
5-nitro-imidazole derivatives of the formula ##STR1## in which R 1 is hydrogen, methyl, ethyl or phenyl, n is 2 or 3, and R 2 is methyl, ethyl, carboxymethyl or carboxyethyl, and the...
4258047 Pyrazole derivatives, pharmaceutical formulations thereof  
Pyrazole derivatives of the formula ##STR1## wherein R 1 is H or Cl; R 2 is 1-methyl-4-piperidyloxy-carbonyl, 2-(4-phenylpiperazino)-ethoxycarbonyl, benzoxazol-2-yl, benzthiazol-2-yl,...
4241060 Nitroimidazoles and compositions thereof  
Nitroimidazoles of the formula ##STR1## wherein R 1 and R 2 are as hereinafter set forth, are described. The nitroimidazoles are useful as hypoxic-cell radiosensitizers, as well as being useful...
4237131 Prostaglandin analogues  
A compound of the formula (I): ##STR1## wherein: X is O or S; Y is --CH 2 --CH 2 --, --CHCH-- or --C.tbd.C--; n is 1 to 5; R 1 is hydrogen or CO 2 R 1 represents an ester group in...
4235899 Substituted O-(2-hydroxypropyl)-aldoximes  
Compounds of general formula ##STR1## wherein X represents a methine group and Y is an oxygen atom, or X represents a nitrogen atom and Y the group NR 3 in which R 3 represents a radical selected...
4209516 Triazole derivatives  
The present invention relates to new triazole derivatives of the formula ##STR1## wherein R 1 represents hydrogen, lower alkyl, optionally esterified or etherified hydroxymethyl, formyl,...
4199580 3-Amino-2-or-propoxy-tetrahydronaphthyl or indanyl-substituted imidazoles and use  
Novel 3-amino-2-OR-propoxy-tetrahydronaphthyl or indanyl substituted imidazoles and methods for their preparation are disclosed. These imidazoles, and their salts, exhibit pharmacological activity...
4174393 1,3,4-Substituted pyrazoline derivatives  
The invention relates to novel 1,3,4-substituted-Δ 2 -pyrazolines having an insecticidal activity. The compounds are particularly active against larvae of insects for example larvae of Colorado...
4132791 Use of etoperidone in parkinsonism and in other extrapyramidal syndromes characterized by tremors  
Treatment of tremors in Parkinsonism and in other extrapyramidal syndromes by administering an amount of trazodone of the formula ##STR1## AND OF ETOPERIDONE OF THE FORMULA: ##STR2## IN THE RANGE...
4131675 Use of combinations of L-DOPA with trazodone and L-DOPA with etoperidone in Parkinsonism  
A combination of trazodone or etoperidone with L-DOPA is used in the treatment of Parkinsonism by oral administration to a patient.
4117145 1-Substituted pyrazoles  
Pyrazoles of the formula ##STR1## wherein R is hydrogen, alkyl, trifluoromethyl, aryl, aralkyl or a heterocycle; R 1 is hydrogen, alkyl, aryl or aralkyl; R 3 is an unsubstituted or...
4081544 Certain 2-(alpha(2-pyridyl)-benzyl)imidazolines and derivatives thereof  
The present 2-substituted imidazolines and 2-substituted-3,4,5,6-tetrahydropyrimidines possess valuable anti-depressant and anti-inflammatory properties. The compounds are prepared by the...
4079136 Imidazolylacetic acid amides, their production, antimycotic compositions comprising said compounds and their use as antimycotic agents  
The invention relates to imidazolylcarboxylic acid amide antimycotic compositions and their use.
4057632 Method of treatment using tetrazole-5-carboxamide derivatives  
Anti-allergic agents of N-aromatic 1H-(or 2H) tetrazole-5-carboxamide derivation present the following formulae: ##STR1## in which R 1 is --CN or --CONH 2 ; R 2 is hydrogen, lower alkyl,...
4021555 Pharmaceutical preparation and method for treatment of parkinsonism  
Administration of mepiprazole during L-dopa therapy for parkinsonism reduces undesired side effects of L-dopa and enhances the desired effects of L-dopa.
4018924 Phenyl-imidazolyl-acetamide derivatives  
Cyclic amides of α-phenyl-α-imidazolyl acetic acid which are further substituted by an alkyl group or phenyl group on the α-carbon atom are antimycotic agents. A typical embodiment is diphenyl...
4006232 Therapeutic method of treating cardiac arrhythmias utilizing 3-substituted diphenylhydantoins  
3-substituted-5,5-diphenylhydantoin derivatives in which the 5,5-diphenylhydantoin moiety is attached at C 3 by a loweralkylene bridge to a 4-phenyl-1-piperidyl, 4-hydroxy-4-phenyl-1-piperidyl,...
3992537 Pharmaceutical compositions containing an N-phenyl-imidazolidine-2-one and method of use  
Pharmaceutical compositions containing as an active ingredient a compound of the formula ##SPC1## Wherein R' is in the m- or p-position and is selected from the group consisting of --CH 2 --A,...
3973019 Pharmaceutical compositions containing 1,4-bis-(5'-nitroimidazolyl-2'-methylene-imino) piperazine compounds for treating protozoal diseases and methods for treating such diseases  
1,4-BIS-5'-NITROIMIDAZOLYL-2'-METHYLENE-IMINO) PIPERAZINES OF THE FORMULA ##SPC1## In which R 1 is hydrogen, methyl, ethyl or 2-hydroxyethyl and R 2 is hydrogen or methyl, are prepared by...
3941881 Novel 3 or 5-aminopyrazolium salts and fungicidal use thereof  
There are provided certain novel 1,2-dimethyl pyrazolium compounds having nitrogen containing substituents in the 3 or 5 position, and to both a method for controlling plant pathogenic fungi with...
3890439 Imidazolidinone derivatives in the treatment of emesis and psychosomatic disturbances  
Compounds of the class of 1-[2-[4-[3-(p-fluoro-benzoyl)-alkyl]-1-piperazinyl]-ethyl]-3 -alkyl-2-imida zolidinone which may be substituted in the 4-position of the imidazolidinone ring by an alkyl...
3549756 ANTITRICHOMONAL COMPOSITIONS CONTAINING 1-SUBSTITUTED - 2 - MORPHOLINYL OR THIAMORPHOLINYL-5-NITROIMIDAZOLES  
3325358 Method of treating inflammation  
3301832 Nitrosopiperazinothioazoles  
3798325 Title is not available  
3814810 Title is not available  
3737547 Title is not available  
Matches 301 - 344 out of 344 < 1 2 3 4 5 6 7