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6713461 |
Pharmaceutical complex
This invention relates to a complex of eletriptan and a sulphobutylether-beta-cyclodextrin, or a pharmaceutically acceptable salt thereof, and to processes for the preparation of, pharmaceutical...
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6699847 |
Antiparasitic formulation
Long-acting antiparasitic formulations of doramectin, suitable for injection, are described herein.
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6699848 |
Bioadhesive anti-inflammatory pharmaceutical compositions
Disclosed are compounds having the formula wherein R 2 is hydrogen, a monomeric glycoside or an oligomeric glycoside, R 3 is hydrogen, a monomeric glycoside, an oligomeric glycoside, or a...
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6696081 |
Carbohydrate based lipid compositions and supramolecular structures comprising same
Novel lipid compounds and compositions comprising carbohydrate backbones are used to make supramolecular structures such as vesicles, liposomes (single lamellar, multilamellar, and giant),...
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6680304 |
Disaccharides with anti-arthrosic properties
The invention relates to novel disaccharides of formula (I), wherein R 1 is selected from the group consisting of hydrogen, linear or branched (C 1 -C 4 ) alkyl, phenylalkyl with less than ten...
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6677309 |
Anti-cancer drug aldehyde conjugate drugs with enhanced cytotoxicity compounds, compositions and methods
Monomeric and dimeric anti-cancer drug aldehyde conjugate compounds and pharmaceutically acceptable salts thereof. Specifically, monomeric and dimeric aldehyde conjugates of 1-2,...
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6673357 |
Alkaloid glycoside for use as a medicament
The invention concerns an alkaloid glycoside for use in medicine. In a preferred aspect, the alkaloid glycoside is used for the stimulation of a class I-restricted immune response and/or a class...
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6670330 |
Cancer chemotherapy with 2-deoxy-D-glucose
A class of glycolytic inhibitors is useful in the treatment of solid tumors by attacking anaerobic cells at the center on the tumor. 2-deoxyglucose, oxamate and various analogs thereof are...
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6670338 |
Pentasaccharides processes for their preparation and pharmaceutical compositions containing them
Pentasaccharides in acidic form and their pharmaceutically acceptable salts, the anionic form thereof having the formula: wherein: R represents hydrogen or an —SO 3 − , (C 1 -C 3 )alkyl or...
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6664243 |
Benzyllactobionamides as inhibitors of smooth muscle cell proliferation
This invention provides smooth muscle cell proliferation inhibitors of formula I having the structure wherein R 1 -R 13 are as defined herein.
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6664235 |
Medicaments comprising sialic acid derivatives as active ingredients
A medicament for treatment of a viral infection which comprises as an active ingredient a compound represented by the following formula (I) or its Pharmaceutically acceptable salt, or a hydrate...
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6663886 |
Inhibition of cell-cell binding by lipid assemblies
This invention relates generally to the field of therapeutic compounds designed to interfere between the binding of ligands and their receptors on cell surface. More specifically, it provides...
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6656913 |
Inhibition of exoprotein production from gram positive bacteria
A method of inhibiting the production of exoproteins from Gram positive bacteria, such as harmful proteins produced by Staphylococcus species, is described. The method is particularly useful for...
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6649594 |
Compositions for metabolic protection and repair of lips
An effective barrier function for the lips is restored and maintained by the topical administration of various formulations, including mixtures of ceramides and essential and nonessential free...
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6649172 |
Amphipathic aldehydes and their uses as adjuvants and immunoeffectors
This invention relates to novel aldehyde containing compounds and their uses as adjuvants and immunoeffectors.
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6646000 |
Method to control plant pests, improve plant productivity and other purposes
A method of treating plant and animal systems and inanimate surfaces for the purposes of controlling plant pests, introducing pesticides and nutrients into plants, mitigating frost damage to...
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6645940 |
Oligosaccharide derivatives and process for producing the same
An oligosaccharide derivative, at higher homogeneity than fucose polysaccharide and rhamnose polysaccharide and with greater antiulcer effects, which is represented by the following general...
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6646013 |
Nutrient formulations for disease reduction
The instant invention provides a combination of multiple nutrients useful to reduce colon rectal cancer in a mannalian or human subject. Further, the combination provides synergistic ratios of the...
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6645935 |
Synthesis of glycoconjugates of the lewis Y epitope and uses thereof
The present invention provides a method of synthesizing an allyl pentasaccharide having the structure: as well as related oligosaccharide ceramides and other glycoconjugates useful as vaccines...
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6635622 |
Glycolipid derivative
The present invention is a compound of general formula (I) or a pharmaceutically acceptable salt of, wherein W represents carbon chain from 9 to 17 which containing double bond or hydroxy group...
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6632797 |
Method of treating angiogenesis
The present invention relates to a method of treating angiogenesis in tumor conditions in a mammal suffering therefrom which comprises administering to a mammal in need thereof an effective amount...
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6630135 |
Use of sustained release antibiotic compositions in ophthalmic surgical procedures
An improved method of sterilizing the field of surgery prior to an ophthalmic surgical procedure is described. The invention eliminates the need for painful and potentially traumatic injections of...
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6630452 |
Nutritional formulation containing prebiotic substances
A nutritional composition is provided which comprises oligofructose and sialyllactose.
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6627612 |
Surfactants based upon alkyl polyglycosides
The invention relates to a series of polyglycoside derivatives that contain water-soluble groups introduced into the molecule by reaction with the hydroxyl groups present in the starting...
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6620792 |
Pharmaceutical compositions containing monosialoganglioside GM1 or derivative thereof suitable for the treatment of parkinson's disease
The present invention refers to pharmaceutical compositions containing monosialoganglioside GM 1 or a derivative thereof, namely, the inner ester AGF 2 and the methyl ester AGF4, suitable for the...
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6620793 |
Therapeutic use of ganglioside GM1 in the treatment of spinal cord injury
The invention relates to a method for amelioration of neurological outcome in humans with spinal cord damage by administration of ganglioside GM 1 . Another object of the present invention is to...
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6610660 |
O2-arylated or O2-glycosylated 1-substituted diazen-1-ium-1,2-diolates and O2-substituted 1-&lsqb (2-carboxylato) pyrrolidin-1-yl&rsqb diazen-1-ium-1,2-diolates
Diazeniumdiolates, wherein the N 1 position is substituted by an inorganic or organic moiety and the O 2 -oxygen is bound to a substituted or unsubstituted aromatic group, are provided. Also...
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6610316 |
Disinfection by particle-bound and insolubilized detergents
A detergent such as nonionic, cationic or anionic detergents and preferably a “sugar detergent” such as octyl-glucopyranoside is rendered insoluble by being bound to an inert substrate. This...
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6608032 |
Medicinal compositions
Medicinal compositions for treating or preventing diabetes, rheumatoid, diseases wherein inflammation should be inhibited, diseases wherein α-glycosidase should be inhibited, diseases wherein the...
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6605596 |
Indolocarbazole anticancer agents and methods of using them
The present invention relates to anti-tumor compounds, compositions and methods. In particular, the invention relates to indolocarbazole analogues of the following general formulas that inhibit...
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6602899 |
β-D-5 thioxylose derivatives, preparation method and therapeutic use
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6596779 |
Stable emulsion, process for the preparation thereof and agent for this purpose
The present invention relates to emulsions which remain perfectly stable over time, prepared from an emulsifier comprising at least one polyglycoside, i.e. polypentoside with or without pohexoside,...
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6596694 |
Caloporoside derivatives, methods of their preparation and use
The present invention relates to novel caloporoside derivatives and method of their use. The caloporoside derivatives may be formed by fermentation of microorganisms, such as Gloeoporus dichrous ...
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6596702 |
Compositions for use in rehydration and nutrition during athletic exercise and methods of making same
The invention provides sports beverages which supply a readily metabolizable, natural carbohydrate, trehalose. The use of trehalose provides twice the concentration of glucose molecules for...
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6589939 |
Camptothecin derivatives having antitumor activity
Camptothecin derivatives of camptothecin of formula (I): wherein the groups R 1 , R 2 and R 3 are as defined in the description are disclosed. The compounds of formula (I) are endowed with...
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6586438 |
Antidiabetic formulation and method
A low dose antidiabetic pharmaceutical formulation is provided, especially adapted for treating Type II diabetes in drug naive patients, which includes a combination of metformin (employed in a...
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6583118 |
Chondroprotective agents
A chondroprotective agent comprising a flavonoid compound of the general formula (I): wherein R 1 to R 9 are, independently, a hydrogen atom, hydroxyl group, or methoxyl group and X is a...
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6576266 |
Plant extract based on glycerides, a method for the preparation of this extract and a cosmetic composition containing the same
The present invention is concerned with a plant extract comprising a mixture of di-O-D-galactosyl-di-O-acylglyceride with phytosphingolipids and phospholipids, as well as with a method for the...
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6576251 |
Carbohydrate mixture
The invention relates to a carbohydrate mixture for dietetic foods administered by the enteral or parenteral route and pharmaceuticals, characterized in that said mixture consists of (a)...
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6573245 |
Modified polysaccharide adjuvant-protein antigen conjugates, the preparation thereof and the use thereof
The present invention is directed to chemical conjugates (herein referred to as polysaccharide adjuvant-antigen conjugates) that have a polysaccharide backbone capable of binding to the cell...
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6573246 |
Modified ether glyceroglycolipids
This invention provides lipids having: 1) a glycerol backbone; 2) a hydrocarbon chain, preferably saturated and containing 16 or 18 carbon atoms, attached to C-1 of the backbone by an ether...
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6569891 |
Antihypertensive compound from Caesalpinia brasiliensis
A compound isolated from an aqueous leachate of heartwood of “Palo de Brazil” Caesalpinia brasiliensis has antihypertensive activity. The compound was isolated by reversed-phase high pressure...
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6569835 |
Combinations with statin and aryl-substituted propanolamine derivatives, their preparation pharmaceuticals comprising them, and their use
Substituted propanolamine derivatives, their pharmaceutically tolerated salts and physiologically functional derivatives thereof are described. Also described are compounds of formula I in which...
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6566340 |
Aryl-substituted propanolamine derivatives, their preparation, pharmaceuticals comprising them, and their use
Substituted propanolamine derivatives, their pharmaceutically tolerated salts and physiologically functional derivatives thereof are described. Also described are compounds of formula I in which...
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6566341 |
Derivative of isoindigo, indigo and indirubin for the treatment of cancer
A compound called NATURA, which is a derivative of Isoindigo is useful in aiding the general health of a patient and specifically is beneficial in preventing or treating cancer. This compound and...
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6562792 |
Hygromycin derivatives
The present invention relates to compounds of the formula 1 and to pharmaceutically acceptable salts, prodrugs and solvates thereof, wherein X, Y, V, W 1 , W 2 , Z 1 and Z 2 are as defined...
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6558670 |
Vaccine adjuvants
The present invention relates to adjuvant compositions which are suitable to be used in vaccines. In particular, the adjuvant compositions of the present invention comprises a saponin and an...
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6555372 |
Composition for enhancing cellular immunogenicity comprising alpha-glycosylceramides
A composition for enhancing immunogenicity of tumor cells or pathogen-infected cells comprising a compound having an α-glycosylceramide structure or a salt or solvate thereof is provided. Tumor...
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6552089 |
Method of treating or preventing alopecia
The present application discloses a method of treating alopecia which is based on the use of a tellurium compound such as ammonium trichloro(dioxoethylene-O,O-tellurate).
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6552001 |
Method breeding and feeds
A method of rearing useful organisms such as cultured animals which is effective in preventing the organisms from diseases, treating the organisms for diseases or maintaining the health of the...
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