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4550106 |
4-Phenyl-4,5,6,7-tetrahydro-thieno[2,3-c]pyridines and salts thereof, compositions and use
Compounds of the formula ##STR1## wherein R 1 is amino, acetylamino, hydroxymethyl, methoxymethyl or ##STR2## R 2 and R 3 , which may be identical to or different from each other, are each...
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4550118 |
Heterocyclic compounds
Compounds of Formula I are described ##STR1## in which X and Y are independently --NH--, --O-- or --S--; Z may be a pyrimidine, triazine, triazole, thiazole, thiadiazole ring. The methods of...
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4548935 |
Dihydropyridine anti-ischaemic and anti-hypertensive agents, compositions and use
Dihydropyridine anti-ischaemic and anti-hypertensive agents of the formula: ##STR1## and their pharmaceutically acceptable salts; wherein R is aryl or heteroaryl; R 1 and R 2 are each...
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4539316 |
Pyridine derivatives of 1,2-diaminocyclobutene-3,4-diones
Compounds of the formula ##STR1## wherein R 12 is a leaving group, Z is S, O or CH 2 and A is a phenyl, furyl, thienyl or pyridyl ring substituted by a ##STR2## moiety, in which R 8 and R 9 are...
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4539322 |
Dihydropyridine derivatives and their use in treating heart conditions and hypertension
1,4-Dihydropyridine derivatives of the formula: ##STR1## and their pharmaceutically acceptable acid addition salts; where R is aryl or heteroaryl; R 1 and R 2 are each independently C 1 -C 4 ...
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4529596 |
Thieno [3,2-c] pyridine derivatives and their therapeutic application
This invention relates to new thieno [3,2-c] pyridine derivatives having the formula: ##STR1## in which: Y represents the OH group or an OR group in which R is a straight or branched lower alkyl...
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4528286 |
Method of using certain aryl-mercapto-lower-alkanamides as antiseborrheic agents
Aryl-mercapto-lower-alkanamides having the following formula ##STR1## wherein R 1 is selected from the group consisting of phenyl, C 1 -4 -alkylphenyl, halophenyl, hydroxyphenyl, C 1 -4...
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4517184 |
Benzodioxole derivatives
The invention relates to novel benzodioxole derivatives of the formula I ##STR1## in which R 1 represents an unsubstituted or substituted, aromatic or heteroaromatic radical, alk represents an...
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4507292 |
Combating pests with aryl N-oxalyl-N-methyl-carbamates
Aryl N-oxalyl-N-methyl-carbamates of the general formula ##STR1## in which X represents an alkoxy, alkenoxy, alkinoxy, aryloxy, alkylthio, alkenylthio, alkinylthio or arylthio radical, each of...
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4505923 |
Ethers of hydroxybenzothiazole-2-sulfonamide for the topical treatment of elevated intraocular pressure
Novel ethers of hydroxy-2-benzothiazolesulfonamide are useful for the topical treatment of elevated intraocular pressure. Ophthalmic compositions include drops and inserts.
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4503051 |
Substituted 3-cyclobutene-1,2-diones, pharmaceutical compositions thereof and methods of use
Compounds of the formula ##STR1## wherein R 12 is a leaving group, Z is S, O or CH 2 and A is a phenyl, furyl, thienyl or pyridyl ring substituted by a ##STR2## moiety, in which R 8 and R 9 are...
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4500528 |
N-Substituted 1,4-dihydropyridines and pharmaceutical compositions
The compounds of the formula: ##STR1## wherein each of the substituents is as defined herein are useful anti-hypertensive agents.
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4499103 |
Benzothiazole-2-sulfonamide derivatives for the topical treatment of elevated intraocular pressure
Novel 2-benzothiazolesulfonamides are useful for the topical treatment of elevated intraocular pressure. Ophthalmic compositions including drops and inserts are also disclosed, as well as methods...
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4497808 |
N-Oxide compounds useful in the treatment of cardiovascular ailments
The present invention relates to novel N-oxide compounds that have cardiovascular properties, especially antihypertensive activity, and that correspond to the formula ##STR1## in which Py...
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4490373 |
Method of treating asthma
A new method of treating asthma is provided. The method is the administration of an effective dose of a Benzoxazole-2-carboxylic acid amide.
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4485104 |
1,2,4-Triazole-3-amines and their pharmaceutical use
Compounds of the general formula (I) ##STR1## and physiologically acceptable salts, hydrates and bioprecursors thereof have been found to show pharmacological activity as selective histamine H 2 ...
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4479949 |
Benzothiazoline compounds
This invention relates to benzothiazoline derivatives of the formula [I] and salts thereof, which are useful for (i) treating cardiovascular diseases, and (ii) as the active ingredient of...
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4472418 |
Benzothiazolesulfonamide derivatives for the topical treatment of elevated intraocular pressure
Novel sulfamates of 6(or 5)-hydroxy-2-benzothiazolesulfonamide are useful for the topical treatment of elevated intraocular pressure. Ophthalmic compositions include drops and inserts.
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4468399 |
2-[2-(2-Aminoalkyl-4-thiazolylmethylthio)alkyl]-amino-5-substituted-4-pyr imidones
2-[2-(2-aminoalkyl-4-thiazolylmethylthio)-alkylene]amino-5-a
romatic-substit uted alkylene-4-pyrimidones and related compounds, H 2 receptor antagonists, useful in inhibiting gastric acid...
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4435395 |
N-Substituted 1,4-dihydropyridazines and pharmaceutical compositions
Compounds of the formula: ##STR1## which are useful as antihypertensive agents are disclosed.
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4435394 |
3-Sulfonamido-benzophenonimine derivatives useful for treating virus infections
3-Sulfonamido-benzophenonimine derivatives useful for prophylactically or therapeutically treating patients suffering from viral infections are provided from 3-sulfonamido-benzophenones.
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4424213 |
Biologically active heterobicyclic hydroximidates and thiolhydroximidates and carbamate ester derivatives thereof
Novel heterobicyclic compounds of Formula I, processes for preparing same and pesticidal compositions and methods are described. ##STR1##
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4414214 |
Benzodioxole derivatives and pharmaceutical use thereof
The invention relates to novel benzodioxole derivatives of the formula I ##STR1## in which R 1 represents an unsubstituted or substituted, aromatic or heteroaromatic radical, alk represents an...
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4414211 |
Heterocyclic derivatives of guanidine
5-Membered, 6-membered and 7-membered heterocyclic derivatives of guanidine having hypoglycemic activity.
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4409216 |
Method of treating diabetes using oxazoline or thiazoline compounds
A compound, with hypoglycaemic activity, having formula (II) or a pharmaceutically acceptable acid addition salt thereof: ##STR1## wherein X represents oxygen or sulphur; R 1 R 2 are the same...
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4400380 |
Antiviral 1-aryl-5-amino-1-penten-3-ones
Compounds of the formula ##STR1## wherein R is H, halo, C 1 -4 alkyl, C 1 -4 alkoxy, 3,4-methylenedioxy, CF 3 , NO 2 , NH 2 , N(C 1 -4 alkyl) 2 , CN, OH, --S(C 1 -4 alkyl) or --SO 2 (C 1 -4...
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4362738 |
Esters and amides containing the 1-(4-chlorobenzoyl)-5-methoxy-2-methyl-1H-indole-3-acetyl moiety
Compounds of the formula ##STR1## wherein each X, which may be identical or different from the other X, is oxygen or imino; R 1 is hydrogen, fluorine, chlorine or bromine; R 2 and R 3 ,...
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4333930 |
Orthoarylideneaminophenethylamines and pharmaceutical compositions
Compounds, exhibiting central nervous system activity, of the formula ##STR1## wherein R 1 is phenyl which is unsubstituted or substituted by at least one member selected from the group consisting...
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4308274 |
N-Alkylsulfonyl-, N-arylsulfonyl-, and N-aminosulfonylaminosulfinylcarbamate esters
A novel class of chemical compounds useful as pesticides consists of N-alkylsulfonyl-, N-arylsulfonyl-, and N-aminosulfonylaminosulfinylcarbamate esters. The preparation of these compounds and...
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4271160 |
Substituted morpholine derivatives and pharmaceutical compositions
Substituted morpholine derivatives, such as, for instance the compound 2-[α-(3,4-methylendioxy-phenoxy)-benzyl]-morpholine are disclosed. The claimed compounds are active on the central nervous...
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4258042 |
Antihypertensive pyridines and compositions
Antihypertensive compounds of the formula ##STR1## wherein R 5 is H, alkyl, aryl, halo, lower alkoxy, nitro amino, alkylmercapto, cyano, carboxy, carbalkoxy, sulfamyl, trifluoromethyl, hydroxy,...
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4256744 |
Agricultural and horticultural pesticides
This invention relates to novel compounds of the general formula (I): ##STR1## wherein A represents ##STR2## in which B represents a ring-forming residue of a 5- or 6-membered carbon-containing...
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4240821 |
Biocidally-active 1,3-benzodithiole-2-thione compounds
1,3-Benzodithiole-2-thione compounds are disclosed including the novel method of preparing said compounds and their biocidal activity.
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4217349 |
Benzisoxazole derivatives
Novel benzisoxazole compounds of the formula: ##STR1## wherein R 1 and R 2 are each hydrogen, C 1 -C 4 alkyl, C 1 -C 4 alkoxy, ar(C 1 -C 3 )alkoxy or halogen or, when taken together, they...
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4209517 |
α-Ethylenic alcohols and ketones, their preparation, and their use as medicaments
The invention provides new compounds of the formula ##STR1## in which one of the symbols R 1 and R 2 denoted a hydrogen atom and the other a hydroxyl group or, together, the two denote an oxygen...
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4206117 |
Pyridinyl aminoalkyl ethers
New pyridinyl aminoalkyl ethers, their N-oxides and their physiologically acceptable addition salts with acids, processes for their preparation and pharmaceutical formulations which contain these...
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4177270 |
Soil fungicidal (nitrogen heterocyclic)-substituted-1,3-benzodithiole-2-ones
1,3-Benzodithiole-2-one and 1,3-benzodithiole-2-thione compounds are disclosed including the novel method of preparing said compounds and their biocidal activity.
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4177271 |
Hydroxy- and oxo-substituted α-benzylidenylcycloalkanes
Hydroxy- and oxo-substituted α-benzylidenylcycloalkanes having the formula: ##STR1## Z 1 , Z 2 and Z 3 each denotes a methoxy group or Z 1 or Z 2 and Z 3 together denote a methylenedioxy...
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4163784 |
Heterocyclylcarbonyl derivatives of urea, agents for dissolution of gallstones
Heterocyclylcarbonyl derivatives of urea having the formula ##STR1## wherein R is a heterocyclyl group; R 1 is hydrogen, alkyl having up to ten carbon atoms or phenyl; R 2 is R 1 , 1-naphthyl and...
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4148895 |
Basically substituted indole derivatives
The present invention relates to basically substituted indole derivatives and to a process for their manufacture. The novel compounds are valuable medicaments which exhibit hypotensive and...
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4133880 |
N.sup.2 -Substituted-L-arginine derivatives and the pharmaceutically acceptable acid addition salts thereof
N 2 -substituted-L-arginine esters and amides, and the pharmaceutically acceptable acid addition salts thereof have been found to be effective as pharmaceutical agents for the inhibition and...
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4027037 |
N-substituted β-aminocrotonic acid esters
N-substituted β-aminocrotonic acid esters of the formula ##STR1## in which R 1 is hydrogen, or alkyl or alkenyl with up to 4 carbon atoms; R 2 is straight-chain or branched alkyl or alkenyl...
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4013768 |
Pyrimidin-6-yl acethydroxamic acids, their therapeutic application and their process of preparation
Compounds of the formula ##STR1## in which R is aminocarbonylphenyl in which amino is --NH 2 , pyrrolidino, piperidino or morpholino, and Ar is phenyl substituted with chloro, fluoro,...
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3495008 |
METHODS OF TREATMENT OF PAIN IN MAMMALS WITH SUBSTITUTED METHYLENEDIOXYBENZAMIDES
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3495007 |
METHODS OF TREATMENT OF PSYCHOSIS IN MAMMALS WITH SUBSTITUTED METHYLENEDIOXYBENZAMIDES
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3423512 |
TREATMENT OF EMESIS IN MAMMALS WITH SUBSTITUTED METHYLENEDIOXY BENZAMIDES
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3336194 |
Indolyl acid amides
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3300377 |
Biocidal quaternary ammonium aromatic cyclic imides
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3278374 |
Cyclic amidines for control of bacterial and fungal diseases in plants
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3663706 |
Title is not available
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