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4514411 |
Substituted 4,10-dihydro-10-oxothieno benzoxepins
This invention relates to substituted 4,10-dihydro-10-oxothieno benzoxepins of the formula, ##STR1## where R is hydrogen and lower alkyl; R 1 is ##STR2## where R 2 is hydrogen, lower alkyl and...
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4503060 |
3-Imino-3H-dibenzo-[c,f]-imidazo-[1,5-a]azepine pharmaceuticals
Compounds of the formula ##STR1## wherein R 1 , R 2 , R 3 and R 4 are each hydrogen, halogen, alkyl of 1 to 6 carbon atoms or alkoxy of 1 to 6 carbon atoms; R 5 is hydrogen, alkyl of 1 to 6...
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4492691 |
Azatetracyclic carbonitriles
Azatetracyclic carbonitriles of the formula ##STR1## in which R represents hydrogen, lower alkyl, cycloalkyl-lower alkyl having up to 10 carbon atoms, lower alkenyl, lower alkynyl or free,...
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4486433 |
Fused-ring amino-pyrazines as bradycardiacs
Compounds of the formula ##STR1## wherein A and B, which may be the same or different, each represent methylene, (alkyl of 1 to 3 carbon atoms)-methylene, ethylene or (alkyl of 1 to 3 carbon...
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4444778 |
Method and composition for treating atherosclerosis
A method of improving the arteriosclerotic condition in an animal having arteriosclerosis or having a high risk of developing arteriosclerosis, which method comprises administering an effective...
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4440779 |
Tricyclic derivatives of substituted pyrrole acids as analgesic and anti-inflammatory agents
Tricyclic derivatives of substituted pyrrole acids, e.g., substituted 4,10-dihydro-10-oxo-1H-[1]benzoxepino[4,3-b]pyrrole-2-acetic
acids or the 5-thia analogs thereof have been prepared via...
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4414225 |
Azepine derivatives and their anti-thrombotic compositions and methods
Compounds of the formula ##STR1## wherein n and m are each 1, 2 or 3, and the sum of n+m is 4; R 1 is alkyl; alkenyl; unsubstituted, mono- or di-substituted aralkyl; unsubstituted, mono- or...
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4400378 |
Pharmaceutical composition for the treatment of glaucoma
The method of treating glaucoma with compounds of the formula ##STR1## wherein R 1 is hydrogen, alkyl of 1 to 4 carbon atoms, hydroxy-(alkyl of 1 to 4 carbon atoms), benzyl, halo-benzyl,...
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4369186 |
4,5-Dichloroimidazole-2-carboxylic acid derivatives
4,5-Dichloroimidazole-2-carboxylic acid derivatives of the formula ##STR1## in which the group ##STR2## represents a carbon atom which has three bonds to hetero-atoms, and their salts with bases,...
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4362727 |
5-Substituted 9-cyanomethylene-dithieno[3,4-b:4,3-e]-azepines and therapeutic agents which contain these compounds
5-Substituted 9-cyanomethylene-dithieno[3,4-b:4',3'-e]-azepines, processes for their preparation, and therapeutic agents which contain these compounds and can be used as sedatives, hypnotic drugs,...
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4313950 |
Antireproductive tricyclic ortho-fused nitrogen containing compounds
New tricyclic ortho-fused nitrogen containing compounds of the following formula: ##STR1## wherein R and R 1 are independently selected from hydrogen, fluoro, chloro, bromo and (C 1 -C 4 )alkoxy;...
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4271178 |
1,2,3,3a,8,12b-Hexahydro-dibenzo[b,f]pyrrolo[3,4-d]azepines and pharmaceutical use thereof
The invention relates to novel dibenzo[1,2;5,6] cyclohepta pyridine or -pyrrole derivatives, dibenzo[2,3;6,7] oxepino pyridine or pyrrole derivatives, dibenzo[2,3;6,7] thiepino pyridine or pyrrole...
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4259342 |
Antianginal treatment with azepine derivatives
Antianginal pharmaceutical compositions containing as the active ingredient a compound of the formula ##STR1## wherein R 1 is hydrogen, unsubstituted or hydroxyl-substituted alkyl of 1 to 4 carbon...
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4255445 |
8-Hydro xy-6,7-(2-methyl-2,3-dihydrofuro)-1-phenyl-2,3,4,5-tetrahydro-1H-3-benzaz epines
8-Hydroxy-6,7-(2,3-dihydrofuro)-1-phenyl-2,3,4,5-tetrahydro-
1H-3-benzazepin es are prepared by a reaction sequence whose key is a dual cyclization forming the 3-benzazepine ring and fused thereto...
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4247557 |
Benzopyranopyridines as antiglaucoma agents
A method of reducing intra-ocular pressure in mammalian patients comprising administering to a glaucoma patient a therapeutically effective amount of a compound of the formula ##STR1## wherein, in...
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4177275 |
Tension reducing 2,3,4,4a,9,13b-hexahydro-1H-dibenzo[b,f]pyrido[3,4-d]azepine derivatives
The invention relates to novel dibenzo[1,2;5,6]cyclohepta pyridine or -pyrrole derivatives, dibenzo[2,3;6,7]oxepino pyridine or pyrrole derivatives, dibenzo[2,3;6,7]thiepino pyridine or pyrrole...
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4165372 |
6-Carboxy-1-phenyl-2,3,4,5-tetrahydro-1H-3-benzazepine compounds and use as dopaminergic agents
A group of 1-phenyl-3-benzazepines with structures characterized by having a carboxy derived substituent at position 6 which are dopaminergic agents or are intermediates for preparing other...
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4021557 |
11-Aminoalkyl-pyridobenzodiazepinones and salts thereof
Compounds of the formula ##STR1## wherein R 1 is hydrogen, straight or branched alkyl of 1 to 3 carbon atoms or benzyl, R 2 is straight or branched alkyl of 1 to 3 carbon atoms, or R 1 and...
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3959282 |
10-Piperazino-4H-thieno[2,3-c] [1]benzazepines
This invention provides new compounds of formula I, ##SPC1## wherein R 1 is hydrogen, or alkyl, alkoxy or alkylthio of 1 to 4 carbon atoms, or trifluoromethyl, and R 2 is hydrogen, or...
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3907996 |
Pharmaceutical composition containing a 2-amino-4,5,7,8-tetrahydro-6H-thiazolo or -oxazolo 5,4-D azepine and method of use
Pharmaceutical compositions containing as an active ingredient a compound of the formula ##EQU1## wherein R 1 is hydrogen, straight or branched alkyl of 1 to 4 carbon atoms, hydroxy-alkyl of 1 to...
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3856910 |
NOVEL THIENOBENZAZEPINES AS ANTI-DEPRESSANTS
Novel 4-(alkylaminoalkyl)-[4H]-thieno-[3,2-b][f]-benzazepines of the formula ##SPC1## Wherein R 1 and R 2 are selected from the group consisting of hydrogen, halogen, --CF 3 , lower alkoxy...
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3783161 |
DERIVATIVES OF DIBENZO(B,F) PYRROLO (3,4-D)AZEPINE AS CNS - DEPRESSANTS
Compounds of the class of 1,2,3,8-tetrahydrodibenzo[b,f]pyrrolo[3,4-d]azepines which may be substituted in the 5-/ or 6-/ and/or 8-position by chlorine, the trifluoromethyl group or alkyl groups...
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3676558 |
ANOREXIGENIC COMPOSITIONS COMPRISING 6-ALKYL-1,2,3,4,5,6-HEXAHYDROAZEPINO 4,5-INDOLES AS ACTIVE INGREDIENT AND PROCESS OF TREATMENT
Compositions comprising 6-alkyl-1,2,3,4,5,6-hexahydroazepino[4,5-b]indole of the formula: ##SPC1## Wherein R and R' are selected from the group consisting of hydrogen, alkoxy and alkyl containing...
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3622673 |
4-(1,4,5,6-TETRAHYDROZEPINO 4,5-b INDOL-3(2H)-YL-BUTYROPHENON COMPOSITIONS AND PROCESS OF TREATMENT MENTAL OR EMOTIONAL DISORDERS
Compounds of the formula ##SPC1## And the pharmacologically acceptable acid addition salts thereof wherein R and R 1 are hydrogen or methoxy; R 1 is hydrogen or methyl; and R 2 is fluorine...
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3529062 |
INDOLE DERIVATIVES AS ANTITUSSIVE AGENTS
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2817623 |
Tabernanthine, ibogaine containing analgesic compositions
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3821381 |
Title is not available
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3749790 |
Title is not available
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3821409 |
Title is not available
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